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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5838 prodotti di "Proteina G/GPCR"

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  • Logo CymitQuimica
    Targetmol
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    Secretin (28-54), human TFA

    <p>Secretin (28-54), human TFA is a 27-amino acid peptide that works on the human Secretin receptor.</p>
    Formula:C132H221N44F3O42
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3153.48

    Ref: TM-TP1135

  • JNJ-39933673
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    JNJ-39933673

    CAS:
    JNJ-39933673 is a bio-active chemical.
    Formula:C48H54F2N2O11
    Colore e forma:Solid
    Peso molecolare:872.96

    Ref: TM-T32305

  • Cortistatin 14, human, rat acetate
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    Cortistatin 14, human, rat acetate

    Cortistatin 14, human, rat acetate is a neuropeptide having structural similarity to somatostatin-14 and shows anticonvulsive, neuroprotective effects and
    Formula:C80H112N18O19S2
    Purezza:97.86%
    Colore e forma:Solid
    Peso molecolare:1693.98

    Ref: TM-TP1188L

  • [cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide
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    [cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide

    CAS:
    Potent, selective NPY Y5 receptor agonist; IC50: 0.24 nM (Y5), >500 nM (Y2), 530 nM (Y1), 51 nM (Y4); Ki: 0.1-0.15 nM (Y5); increases food intake in vivo.
    Formula:C183H281N57O54S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:4207.67

    Ref: TM-TP1963

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    Sigma-1 receptor antagonist 4

    <p>Sigma-1 receptor antagonist 4 (Compound 32) is a potent σ1R antagonist that significantly enhances morphine's analgesic effects and reverses morphine-induced</p>
    Formula:C22H26N2O
    Colore e forma:Solid
    Peso molecolare:334.45

    Ref: TM-T74813

  • HS014
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    HS014

    CAS:
    Potent MC4 antagonist; Ki: 3.16 nM (MC4), 108 (MC1), 54.4 (MC3), 694 (MC5). Boosts rat appetite, mouse pain, blocks IL-1β Fos in hypothalamus.
    Formula:C71H94N20O17S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1563.77

    Ref: TM-TP2015

  • (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
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    (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin

    CAS:
    V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.
    Formula:C52H74N14O12S2
    Purezza:98%
    Colore e forma:White Lyophilized Powder
    Peso molecolare:1151.38

    Ref: TM-TP2136

  • CAY10597
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    CAY10597

    CAS:
    <p>PGD2 effects via DP1/CRTH2/DP2 receptors; CAY10597 blocks CRTH2/DP2 (Ki=37nM), R enantiomer stronger (Ki=23-22nM), inhibits eosinophil migration (IC50=40nM).</p>
    Formula:C20H14ClFN2O5
    Colore e forma:Solid
    Peso molecolare:416.79

    Ref: TM-T38365

  • Hemokinin 1, human
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    Hemokinin 1, human

    CAS:
    Endogenous P-like compound, NK1 receptor agonist; IC50: NK1-1.8 nM, NK3-370 nM, NK2-480 nM; boosts B-cell growth, antiapoptotic, lowers blood pressure in vivo.
    Formula:C54H84N14O14S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1185.4

    Ref: TM-TP1899

  • Adrenomedullin (AM) (22-52), human acetate
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    Adrenomedullin (AM) (22-52), human acetate

    Adrenomedullin (AM) (22-52), human acetate is an antagonist of calcitonin generelated peptide receptor in the hindlimb vascular bed of the cat and an
    Formula:C161H256N46O50
    Purezza:99.42%
    Colore e forma:Solid
    Peso molecolare:3636.09

    Ref: TM-TP1257L

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    Liraglutide acetate

    CAS:
    Liraglutide acetate is the acetate salt form of Liraglutide, which is a glucagon-like peptide-1 (GLP-1) receptor agonist, utilized in the study of type 2 diabetes.
    Formula:C172H265N43O51·xC2H4O2
    Peso molecolare:3751.20 (free base)

    Ref: TM-TP3096

  • Thiothixene
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    Thiothixene

    CAS:
    Thiothixene has a wide range of applications in life science related research.
    Formula:C23H29N3O2S2
    Colore e forma:Solid
    Peso molecolare:443.62

    Ref: TM-T38200

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    Urocortin II, human acetate

    Urocortin II, human acetate, is a selective endogenous peptide agonist of type 2 corticotropin-releasing factor (CRF2) receptors, used to study the role of CRF2 receptors in feeding behavior.
    Colore e forma:Odour Solid

    Ref: TM-TP3688

  • INCB3344 R-isomer
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    INCB3344 R-isomer

    <p>INCB3344 is a potent CCR2 antagonist. INCB3344 R-isomer is the R-isomer of INCB3344.</p>
    Formula:C29H34F3N3O6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:577.59

    Ref: TM-T11650

  • 15-keto-17-phenyl trinor Prostaglandin F2α ethyl amide
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    15-keto-17-phenyl trinor Prostaglandin F2α ethyl amide

    CAS:
    Bimatoprost is the Allergan trade name for 17-phenyl trinor prostaglandin F2α ethyl amide (17-phenyl trinor PGF2α ethyl amide), an F-series PG analog which has
    Formula:C25H35NO4
    Colore e forma:Solid
    Peso molecolare:413.558

    Ref: TM-T35944

  • Cortistatin-8 acetate
    Targetmol
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    Cortistatin-8 acetate

    <p>Cortistatin-8 acetate: synthetic corticosteroid analog, GHS-R antagonist; doesn't affect acyl GH release or hesperidin response.</p>
    Formula:C49H72N12O11S2
    Purezza:99.01%
    Colore e forma:Soild
    Peso molecolare:1069.3

    Ref: TM-TP2236L

  • Bucindolol Formate
    Targetmol
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    Bucindolol Formate

    Bucindolol is a β1-adrenergic blocker with sympathomimetic activity, used in heart failure research.
    Formula:C23H27N3O4
    Purezza:99.76% - 99.88%
    Colore e forma:Solid
    Peso molecolare:409.48

    Ref: TM-T10631L

  • Pobilukast
    Targetmol
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    Pobilukast

    CAS:
    Pobilukast (SKF 104353) is a cysteinyl leukotriene receptor antagonist that can be used to study limiting myocardial injury in MI/R rats.
    Formula:C26H34O5S
    Purezza:99.65% - 99.84%
    Colore e forma:Solid
    Peso molecolare:458.61

    Ref: TM-T68130

  • Gemeprost
    Targetmol
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    Gemeprost

    CAS:
    Gemeprost treats obstetric bleeding and induces abortion up to 24 weeks when used with mifepristone.
    Formula:C23H38O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:394.54

    Ref: TM-T20855

  • [D-p-Cl-Phe6,Leu17]-VIP
    Targetmol
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    [D-p-Cl-Phe6,Leu17]-VIP

    CAS:
    Selective vasoactive intestinal peptide (VIP) receptor antagonist (IC50 = 125.8 nM). Displays no activity on glucagon, secretin or GRF receptors.
    Formula:C148H239ClN44O42
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3342.24

    Ref: TM-TP2103