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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

Mostrare 18 più sottocategorie

Trovati 5745 prodotti di "Proteina G/GPCR"

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  • Blonanserin
    Targetmol
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    Blonanserin

    CAS:
    Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.
    Formula:C23H30FN3
    Purezza:99.85%
    Colore e forma:Solid
    Peso molecolare:367.5

    Ref: TM-T1180

  • KGA-2727
    Targetmol
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    KGA-2727

    CAS:
    KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.
    Formula:C26H40N4O8
    Purezza:98.46%
    Colore e forma:Solid
    Peso molecolare:536.62

    Ref: TM-T15656

  • (3aR,9aR)-Fluparoxan
    Targetmol
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    (3aR,9aR)-Fluparoxan

    CAS:
    <p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Formula:C10H10FNO2
    Purezza:97.82%
    Colore e forma:Soild
    Peso molecolare:195.19

    Ref: TM-T77566

  • Azatadine dimaleate
    Targetmol
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    Azatadine dimaleate

    CAS:
    <p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine（IC50=6.5 nM） and cholinergic（IC50=10 nM）.</p>
    Formula:C28H30N2O8
    Purezza:99.7% - >99.99%
    Colore e forma:Powder
    Peso molecolare:522.55

    Ref: TM-T0236

  • Zolmitriptan
    Targetmol
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    Zolmitriptan

    CAS:
    <p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>
    Formula:C16H21N3O2
    Purezza:99.69% - 99.91%
    Colore e forma:White Or Kind Of White Powder
    Peso molecolare:287.36

    Ref: TM-T1092

  • Brefonalol HCl
    Targetmol
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    Brefonalol HCl

    Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.
    Formula:C22H29ClN2O2
    Purezza:99.98%
    Colore e forma:Solid
    Peso molecolare:388.93

    Ref: TM-T30586L

  • AH 6809
    Targetmol
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    AH 6809

    CAS:
    <p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>
    Formula:C17H14O5
    Purezza:97.59%
    Colore e forma:Solid
    Peso molecolare:298.29

    Ref: TM-T14148

  • Dopexamine hydrochloride
    Targetmol
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    Dopexamine hydrochloride

    CAS:
    Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.
    Formula:C22H34Cl2N2O2
    Purezza:98.55%
    Colore e forma:Solid
    Peso molecolare:429.42

    Ref: TM-T11318

  • Noradrenaline bitartrate
    Targetmol
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    Noradrenaline bitartrate

    CAS:
    <p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>
    Formula:C12H19NO10
    Purezza:99.53% - >99.99%
    Colore e forma:Solid
    Peso molecolare:337.28

    Ref: TM-T0871

  • Antazoline hydrochloride
    Targetmol
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    Antazoline hydrochloride

    CAS:
    Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous
    Formula:C17H19N3·HCl
    Purezza:98% - 99.53%
    Colore e forma:White Or Almost White Crystalline Powder
    Peso molecolare:301.82

    Ref: TM-T0092

  • Mifentidine
    Targetmol
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    Mifentidine

    CAS:
    <p>Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.</p>
    Formula:C13H16N4
    Purezza:98.34% - 99.73%
    Colore e forma:Solid
    Peso molecolare:228.29

    Ref: TM-T68100

  • Bambuterol hydrochloride
    Targetmol
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    Bambuterol hydrochloride

    CAS:
    Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.
    Formula:C18H30ClN3O5
    Purezza:99.53% - 99.61%
    Colore e forma:White Solid
    Peso molecolare:403.91

    Ref: TM-T1446

  • Ticlopidine hydrochloride
    Targetmol
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    Ticlopidine hydrochloride

    CAS:
    <p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>
    Formula:C14H15Cl2NS
    Purezza:99.85% - >99.99%
    Colore e forma:White Powder
    Peso molecolare:300.25

    Ref: TM-T0362

  • Senktide acetate
    Targetmol
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    Senktide acetate

    <p>Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM and can be used to study Alzheimer's disease.</p>
    Formula:C42H59N7O13S
    Purezza:98.26%
    Colore e forma:Solid
    Peso molecolare:902.02

    Ref: TM-T7633L

  • (R)-Elagolix
    Targetmol
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    (R)-Elagolix

    CAS:
    (R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.
    Formula:C32H30F5N3O5
    Purezza:99.08%
    Colore e forma:Solid
    Peso molecolare:631.59

    Ref: TM-T11174

  • LCKLSL hydrochloride
    Targetmol
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    LCKLSL hydrochloride

    <p>LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.</p>
    Formula:C30H58ClN7O8S
    Purezza:98.02% - 99.31%
    Colore e forma:Solid
    Peso molecolare:712.34

    Ref: TM-T78015

  • Flopropione
    Targetmol
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    Flopropione

    CAS:
    <p>Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.</p>
    Formula:C9H10O4
    Purezza:99.93%
    Colore e forma:Solid
    Peso molecolare:182.17

    Ref: TM-T0525

  • YNT-185
    Targetmol
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    YNT-185

    CAS:
    YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,
    Formula:C33H37N5O5S
    Purezza:99.67%
    Colore e forma:Solid
    Peso molecolare:615.74

    Ref: TM-T39229

  • Ziprasidone hydrochloride
    Targetmol
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    Ziprasidone hydrochloride

    CAS:
    <p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>
    Formula:C21H22CL2N4OS
    Purezza:97.97% - 99.82%
    Colore e forma:Solid
    Peso molecolare:449.4

    Ref: TM-T0031L

  • Ifenprodil Tartrate
    Targetmol
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    Ifenprodil Tartrate

    CAS:
    <p>Ifenprodil is a selective NMDA receptor (glutamate) antagonist.</p>
    Formula:C21H27NO2C4H6O6
    Purezza:99.02% - 99.55%
    Colore e forma:Solid
    Peso molecolare:400.49

    Ref: TM-T1186