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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5378 prodotti di "Proteina G/GPCR"

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  • LY 306669

    CAS:
    LY 306669 is an antagonist of leukotriene B4 receptor.
    Formula:C23H29FN4NaO2
    Colore e forma:Solid
    Peso molecolare:435.499
  • Protokylol

    CAS:
    <p>Protokylol is a β-adrenergic receptor agonist.</p>
    Formula:C18H21NO5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:331.36
  • Ono 6240

    CAS:
    <p>Ono 6240 is an antagonist of platelet-activating factor. Ono 6240 prevents airway eosinophilia by inhibiting production of IL-2 and IL-5.</p>
    Formula:C32H63NO6S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:621.98
  • ASP7657

    CAS:
    <p>ASP7657 is a novel, potent, and selective prostaglandin EP4 receptor antagonist.</p>
    Formula:C28H26F3N3O3
    Colore e forma:Solid
    Peso molecolare:509.52
  • ADRA1D receptor antagonist 1 free base

    CAS:
    <p>ADRA1D antagonist blocks bladder contractions; Ki=1.6 nM, IC30=15 nM, useful in overactive bladder research.</p>
    Formula:C15H13ClN4O
    Colore e forma:Solid
    Peso molecolare:300.74
  • 5-HT2A receptor agonist-2

    CAS:
    <p>Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.</p>
    Formula:C20H21ClN2O3
    Colore e forma:Solid
    Peso molecolare:372.85
  • A 69024

    CAS:
    <p>A 69024 is a highly selective antagonist of dopamine D-1 receptor.</p>
    Formula:C20H24BrNO4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:422.31
  • RS 64459-193

    CAS:
    <p>RS 64459-193 has a high affinity for the 5-HT1A binding site.</p>
    Formula:C26H36Cl2N2O2
    Colore e forma:Solid
    Peso molecolare:479.48
  • MAT2A-IN-3

    CAS:
    <p>MAT2A-IN-3: potent MAT2A inhibitor, hinders MTAP-deficient cancer cell growth, potential for cancer research.</p>
    Formula:C24H16F5N5O3
    Colore e forma:Solid
    Peso molecolare:517.41
  • AHR-13268D

    CAS:
    <p>AHR-13268D is a new agent of antiallergic/antihistaminic.</p>
    Formula:C28H29F2NNaO4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:504.53
  • ABT-239

    CAS:
    <p>ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.</p>
    Formula:C22H22N2O
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:330.42
  • TSHR antagonist S37b

    CAS:
    <p>S37b, a less effective enantiomer of TSHR antagonist S37a, offers minor thyrotropin receptor inhibition, useful for thyroid research.</p>
    Formula:C25H20N2O3S2
    Colore e forma:Solid
    Peso molecolare:460.57
  • DH97

    CAS:
    <p>MT2 melatonin receptor antagonist</p>
    Formula:C22H26N2O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:334.45
  • GSK1059865

    CAS:
    GSK1059865 is a potent antagonist of the orexin 1 receptor.
    Formula:C20H23BrFN3O2
    Colore e forma:Solid
    Peso molecolare:436.32
  • Metazosin

    CAS:
    <p>Metazosin is an antihypertensive agent that replaces 3H-prazosin from its bond to alpha-1 receptors of the cerebral cortex.</p>
    Formula:C18H25N5O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:375.42
  • LY 302148

    CAS:
    <p>LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.</p>
    Formula:C19H23FN4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:326.41
  • SB-269970

    CAS:
    SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).
    Formula:C18H28N2O3S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:352.49
  • Remogliflozin

    CAS:
    <p>Remogliflozin is an effective sodium-glucose transporter 2 inhibitor (Kis = 12.4 and 26 nM for human and rat SGLT2, respectively).</p>
    Formula:C23H34N2O7
    Colore e forma:Solid
    Peso molecolare:450.53
  • Etersalate

    CAS:
    <p>Etersalate inhibits platelet function. It also reduces thromboxane A2 (TXA2) levels.</p>
    Formula:C19H19NO6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:357.36
  • CCG-224406

    CAS:
    <p>CCG-22440 is a Highly Selective and Potent Inhibitor of G Protein-Coupled Receptor Kinase 2.</p>
    Formula:C29H27FN6O5
    Colore e forma:Solid
    Peso molecolare:558.56
  • GB83

    CAS:
    GB83 is a selective human protease activated receptor 2 (PAR2) antagonist.
    Formula:C32H44N4O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:548.72
  • A1AR antagonist 3

    CAS:
    <p>Compound 13: selective A1AR antagonist, Ki human A1: 9.69 nM, rat A1: 0.529 nM, useful for neurological research.</p>
    Formula:C25H20N2O3S
    Colore e forma:Solid
    Peso molecolare:428.5
  • Usmarapride

    CAS:
    <p>Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.</p>
    Formula:C23H31N5O6
    Colore e forma:Solid
    Peso molecolare:473.53
  • PD-135666

    CAS:
    <p>PD-135666 is an antagonist of CCK receptor.</p>
    Formula:C33H39N3O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:557.68
  • Levobunolol hydrochloride

    CAS:
    <p>Levobunolol hydrochloride 是一种非选择性的 β-肾上腺素受体阻滞剂,可用于治疗青光眼和上斜肌肌障碍的研究。</p>
    Formula:C17H26ClNO3
    Purezza:98.49% - >99.99%
    Colore e forma:Solid
    Peso molecolare:327.85
  • FRG8701

    CAS:
    <p>FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.</p>
    Formula:C22H30N2O4S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:418.55
  • A 55453

    CAS:
    <p>A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.</p>
    Formula:C25H32N6O3
    Colore e forma:Solid
    Peso molecolare:464.56
  • Zicronapine

    CAS:
    <p>Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.</p>
    Formula:C22H27ClN2
    Colore e forma:Solid
    Peso molecolare:354.92
  • SMANT hydrochloride

    CAS:
    SMANT hydrochloride (N-(4-bromophenyl)-3-(3,5-dimethylpiperidin-1-yl)propanamide hydrochloride) is an antagonist of Smoothened accumulation.
    Formula:C16H24BrClN2O
    Purezza:99.81%
    Colore e forma:Solid
    Peso molecolare:375.73
  • LG 82-4-00

    CAS:
    <p>LG 82-4-00 is an inhibitor of thromboxane.</p>
    Formula:C10H11ClN2O3S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:274.72
  • SKF-75670 Hydrobromide

    CAS:
    <p>SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.</p>
    Formula:C17H20BrNO2
    Colore e forma:Solid
    Peso molecolare:350.25
  • TBC3711

    CAS:
    <p>TBC3711 is an endothelin receptor modulator. It is used for the research of endothelin-mediated disorders.</p>
    Formula:C20H21N3O5S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:447.53
  • OPC-14523 free base

    CAS:
    OPC-14523, a 5-HT1A receptor agonist, is used potentially for the treatment of depression and neuropathic pain.
    Formula:C23H28ClN3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:413.94
  • A-304121

    CAS:
    <p>A-304121 is a histamine H(3) receptor.</p>
    Formula:C20H29N3O3
    Colore e forma:Solid
    Peso molecolare:359.46
  • Org-12962 hydrochloride

    CAS:
    <p>Org-12962 hydrochloride is a 5-HT2C receptor agonist.</p>
    Formula:C10H12Cl2F3N3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:302.12
  • Mrgx2 antagonist-1

    CAS:
    Mrgx2 antagonist-1 is a potent antagonist of Mrgx2 (Mas-related Gene X2) and can be used to study Mrgx2-mediated diseases and disorders.
    Formula:C23H26F5N5O3
    Colore e forma:Solid
    Peso molecolare:515.48
  • A1AR antagonist 4

    CAS:
    <p>Compound 22: A1AR antagonist, pIC50 5.51, pKi 6.29, potent and selective.</p>
    Formula:C23H25N3O2
    Colore e forma:Solid
    Peso molecolare:375.46
  • SB 207710

    CAS:
    SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.
    Formula:C19H27IN2O4
    Colore e forma:Solid
    Peso molecolare:474.33
  • ASP1126

    CAS:
    <p>ASP1126 is a selective and orally active sphingosine-1-phosphate (S1P) agonist (EC50s: 7.12 nM, 517 nM for hS1P1 and hS1P3).</p>
    Formula:C26H26ClF6NO5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:581.93
  • AHR-14310C

    CAS:
    <p>AHR-14310C is a long-acting and nonsedating H1-antihistamine.</p>
    Formula:C24H28F2N2O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:430.49
  • Fluprostenol methyl ester

    CAS:
    <p>Fluprostenol, a vet-approved luteolytic, has an isopropyl ester, travoprost, used as an eye pressure reducer. CAY10532 is its methyl ester form.</p>
    Formula:C24H31F3O6
    Colore e forma:Solid
    Peso molecolare:472.49
  • Arbutamine hydrochloride

    CAS:
    <p>Arbutamine hydrochloride is a catecholamine which acts as a cardiac stimulant.</p>
    Formula:C18H24ClNO4
    Colore e forma:Solid
    Peso molecolare:353.84
  • Org41841

    CAS:
    Org41841 is an agonist of luteinising hormone/chorionic gonadotropin receptor and thyroid stimulating hormone receptor and can be used to study hyperthyroidism.
    Formula:C19H22N4O2S2
    Purezza:99.46% - 99.92%
    Colore e forma:Solid
    Peso molecolare:402.53
  • Denopamine

    CAS:
    <p>Denopamine is an agonist of 1-Adrenoceptor.</p>
    Formula:C18H23NO4
    Colore e forma:Solid
    Peso molecolare:317.38
  • hBChE-IN-2

    CAS:
    <p>hBChE-IN-2 is a BChE inhibitor and CB2R agonist with neuroprotective activity for the study of Alzheimer's disease-like neurological disorders.</p>
    Formula:C27H36N4O3
    Purezza:99.60% - 99.83%
    Colore e forma:Soild
    Peso molecolare:464.6
  • LP 20 hydrochloride

    CAS:
    <p>ligand of the 5-HT7 receptor</p>
    Formula:C17H21ClN2O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:304.81
  • LY314228

    CAS:
    <p>LY314228 is an antagonist of 5-HT2A receptor.</p>
    Formula:C20H24N4O3
    Colore e forma:Solid
    Peso molecolare:368.43
  • L748337

    CAS:
    <p>L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective effects of CL316243.</p>
    Formula:C26H31N3O5S
    Purezza:99.67% - >99.99%
    Colore e forma:Solid
    Peso molecolare:497.61
  • FR-171113

    CAS:
    <p>Protease-activated receptor 1 antagonist</p>
    Formula:C19H11Cl3N2O4S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:469.73
  • LY 25648

    CAS:
    <p>LY 25648 is an antagonist of leukotriene B4.</p>
    Formula:C19H27NO2S
    Colore e forma:Solid
    Peso molecolare:333.49
  • ADR-851 HCl

    CAS:
    ADR-851 HCl is an HT3 receptor antagonist. It works against mechanical, acute thermal, and formalin-induced inflammatory pain.
    Formula:C14H19Cl2N3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:332.23
  • FR 139317

    CAS:
    <p>highly potent and selective ETA endothelin receptor antagonist</p>
    Formula:C33H44N6O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:604.74
  • OPC-14523 hydrochloride

    CAS:
    <p>OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.</p>
    Formula:C23H29Cl2N3O2
    Purezza:99.60%
    Colore e forma:Solid
    Peso molecolare:450.4
  • Asperlicin D

    CAS:
    <p>Asperlicin D is a cholecystokinin antagonist agent.</p>
    Formula:C25H18N4O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:406.44
  • JTH-601 free base

    CAS:
    <p>JTH-601 free base is an antagonist of alpha 1 adrenergic receptor.</p>
    Formula:C24H35NO4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:401.54
  • AZ-GHS-22

    CAS:
    <p>AZ-GHS-22, an inverse agonist for GHS-R1a (ghrelin receptor), binds with 0.77 nM IC50, cutting mice food intake by 54% at 100 mg/kg.</p>
    Formula:C27H33ClN6O5S2
    Colore e forma:Solid
    Peso molecolare:621.17
  • Fenethazine

    CAS:
    <p>Fenethazine is an effective antihistamine used as an antiallergic drug.</p>
    Formula:C16H18N2S
    Colore e forma:Solid
    Peso molecolare:270.39
  • Vapitadine dihydrochloride

    CAS:
    <p>Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.</p>
    Formula:C17H22Cl2N4O
    Purezza:98.28% - 99.30%
    Colore e forma:Solid
    Peso molecolare:369.29
  • SORT-PGRN interaction inhibitor 3

    CAS:
    <p>SORT-PGRN Interaction Inhibitor 3 (Compound 13), with an IC50 value of 0.17 μM, acts as an inhibitor of the SORT-PGRN interaction, and is utilized in the study</p>
    Formula:C15H19Cl2NO3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:332.22
  • Nafadotride

    CAS:
    <p>Nafadotride is a dopamine D3 receptor antagonist.</p>
    Formula:C22H27N3O2
    Colore e forma:Solid
    Peso molecolare:365.47
  • Midodrine D6 hydrochloride

    CAS:
    <p>Midodrine D6 hydrochloride is a vasopressor/antihypotensive agent.</p>
    Formula:C12H19ClN2O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:296.78
  • Meseclazone

    CAS:
    <p>Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP aggregation.</p>
    Formula:C11H10ClNO3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:239.65
  • ATC0065 HCl

    CAS:
    <p>ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.</p>
    Formula:C25H31BrCl2F3N5O
    Colore e forma:Solid
    Peso molecolare:625.35
  • LEK 8841

    CAS:
    <p>LEK 8841 is an ergoline derivative that is a potential antipsychotic.</p>
    Formula:C21H24BrN3O4S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:494.4
  • L 659989

    CAS:
    <p>L 659989 is an antagonist of the Platelet-activating factor receptor.</p>
    Formula:C24H32O8S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:480.57
  • 12(S)-hydroxy-16-Heptadecynoic Acid

    CAS:
    <p>The compound is a mechanism-based inhibitor of cytochrome P450 ω-hydroxylase.</p>
    Formula:C17H30O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:282.42
  • Lofepramine hydrochloride

    CAS:
    <p>Lofepramine is a serotonin and norepinephrine reuptake inhibitor. Lofepramine is also a psychotropic IMIPRAMINE derivative.</p>
    Formula:C26H28Cl2N2O
    Purezza:98%
    Colore e forma:Off-White Solid
    Peso molecolare:455.42
  • FMS586

    CAS:
    <p>FMS586 is a selective antagonist of neuropeptide Y Y5 receptor with oral activity.</p>
    Formula:C24H30N4O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:390.52
  • BMS-192364

    CAS:
    <p>BMS-192364 is a bio-active chemical.</p>
    Formula:C15H9ClF3N3O2
    Colore e forma:Solid
    Peso molecolare:355.70
  • Clencyclohexerol

    CAS:
    <p>Clencyclohexerol, like clenbuterol, is a β-adrenoceptor agonist with potential in muscle disorders but poses cardiovascular risks at high doses.</p>
    Formula:C14H20Cl2N2O2
    Colore e forma:Solid
    Peso molecolare:319.23
  • L 657925

    CAS:
    <p>L 657925 is an antagonist of the thromboxane A2 receptor.</p>
    Formula:C21H21ClFNO2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:373.85
  • L 648051

    CAS:
    <p>L 648051 is a leukotriene D4 receptor antagonist.</p>
    Formula:C24H28O8S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:476.54
  • Delequamine HCl

    CAS:
    <p>Delequamine HCl: potent, selective alpha 2-adrenoceptor blocker; pKi 9.45 in rat cortex, pA2 9.72 in guinea-pig ileum.</p>
    Formula:C18H27ClN2O3S
    Colore e forma:Solid
    Peso molecolare:386.94
  • Talipexole

    CAS:
    <p>Talipexole (B-HT920) is an agonist of dopamine, and is an antiparkinsonian agent.</p>
    Formula:C10H15N3S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:209.31
  • MRS1067

    CAS:
    <p>MRS1067 is an antagonist of A3 adenosine receptor.</p>
    Formula:C19H16Cl2O3
    Colore e forma:Solid
    Peso molecolare:363.23
  • (Rac)-SEP-363856

    CAS:
    <p>(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a unique</p>
    Formula:C9H13NOS
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:183.27
  • N-0861 racemate

    CAS:
    <p>N-0861 racemate is the racemate of N-0861.</p>
    Formula:C13H17N5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:243.31
  • Ifoxetine sulfate

    CAS:
    <p>Ifoxetine sulfate, an atypical 5-HT inhibitor, may show unique therapeutic effects and side-effects.</p>
    Formula:C13H19NO2H2O4S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:270.34
  • 8-M-PDOT

    CAS:
    <p>8-M-PDOT (AH-002) is an MT2 receptor agonist that inhibits MT1.8-M-PDOT has anxiolytic activity and may be used in the study of neuropathic pain.</p>
    Formula:C14H19NO2
    Purezza:99.54% - 99.54%
    Colore e forma:Solid
    Peso molecolare:233.31
  • A412997

    CAS:
    <p>A412997 is a selective agonist of dopamine D4 receptor.</p>
    Formula:C19H23N3O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:309.41
  • Pronethalol hydrochloride

    CAS:
    <p>β-adrenergic antagonist</p>
    Formula:C15H20ClNO
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:265.78
  • Naminterol

    CAS:
    <p>Naminterol is a phenethanolamine derivative is an agonist of β2 adrenoceptor with bronchodilatory properties, and used for treatment of asthma.</p>
    Formula:C19H26N2O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:330.42
  • Amitriptylinoxide

    CAS:
    <p>Amitriptylinoxide is an antidepressant.</p>
    Formula:C20H23NO
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:293.4
  • Chlorazanil

    CAS:
    <p>Chlorazanil is a triazine-based, orally active diuretic that blocks Na+ and Cl– reabsorption in distal tubules, increases renal prostaglandin.</p>
    Formula:C9H8ClN5
    Purezza:98.89%
    Colore e forma:Solid
    Peso molecolare:221.65
  • WB 4101 hydrochloride

    CAS:
    <p>α1A-adrenergic antagonist</p>
    Formula:C19H24ClNO5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:381.85
  • Captodiame

    CAS:
    <p>Captodiame is an antihistamine agent.</p>
    Formula:C21H29NS2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:359.59
  • Hedgehog IN-3

    CAS:
    <p>Hedgehog IN-3 (compound 3), with an IC50 value of 0.01 µM, serves as a hedgehog pathway inhibitor, proving beneficial for cancer research applications [1].</p>
    Formula:C18H13ClF3N5O
    Colore e forma:Solid
    Peso molecolare:407.78
  • (Rac)-E1R

    CAS:
    <p>(Rac)-E1R is the racemate of E1R. (Rac)-E1R is a sigma-1 receptor positive allosteric (Sig1R PAM) modulator of for the treatment of cognition/memory disorders.</p>
    Formula:C13H16N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:232.28
  • Thioproperazine

    CAS:
    <p>Thioproperazine (RP 7843) is an orally effective antipsychotic schizophrenia and bipolar disorder, histamine and adrenergic receptor blocker.</p>
    Formula:C22H30N4O2S2
    Purezza:99.45%
    Colore e forma:Solid
    Peso molecolare:446.63
  • TCV-309 chloride

    CAS:
    TCV-309 chloride is an antagonist of platelet activating factor (PAF).
    Formula:C30H34BrClN4O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:629.97
  • GSK 189254 HCl

    CAS:
    <p>GSK 189254A: histamine H3 antagonist, treats narcolepsy, may improve cognition and help with dementia, neuropathic pain.</p>
    Formula:C21H26ClN3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:387.9
  • BN 52111

    CAS:
    <p>BN 52111 is a platelet activating factor antagonist.</p>
    Formula:C33H58BrNO4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:612.734
  • RS 23597-190 hydrochloride

    CAS:
    <p>RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.</p>
    Formula:C16H24Cl2N2O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:363.28
  • MK-0249

    CAS:
    <p>MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).</p>
    Formula:C23H24F3N3O2
    Purezza:99.90%
    Colore e forma:Solid
    Peso molecolare:431.45
  • L659989

    CAS:
    <p>L659989 is an antagonist of PAF receptor.</p>
    Formula:C24H32O8S
    Colore e forma:Solid
    Peso molecolare:480.57
  • Falintolol, (Z)-

    CAS:
    Falintolol, (Z)-, is a novel β-adrenergic antagonist compound distinguished by the inclusion of an oxime moiety.
    Formula:C12H24N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:228.33
  • 2-Methylthio-AMP diTEA

    CAS:
    <p>2-MeSAMP diTEA blocks P2Y12 receptor, inhibits ADP platelet clumping.</p>
    Formula:C23H46N7O7PS
    Colore e forma:Solid
    Peso molecolare:595.69
  • Tropodifene

    CAS:
    <p>Tropodifene is an inhibitor of the α-Adrenergic receptor.</p>
    Formula:C25H29NO4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:407.5
  • Zimelidine dihydrochloride

    CAS:
    <p>5-HT re-uptake inhibitor</p>
    Formula:C16H18BrClN2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:353.69
  • Adenosine receptor inhibitor 2

    CAS:
    <p>Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.</p>
    Formula:C17H20BrN5O2
    Colore e forma:Solid
    Peso molecolare:406.28
  • Dopamine D2 receptor antagonist-1

    CAS:
    <p>Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity.</p>
    Formula:C14H17N3S
    Purezza:99.86%
    Colore e forma:Solid
    Peso molecolare:259.37
  • Cicloprolol hydrochloride

    CAS:
    <p>Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.</p>
    Formula:C18H30ClNO4
    Purezza:97.26%
    Colore e forma:Solid
    Peso molecolare:359.89
  • Bamirastine

    CAS:
    <p>Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on</p>
    Formula:C31H37N5O3
    Purezza:96.68%
    Colore e forma:Solid
    Peso molecolare:527.66
  • S-3608

    CAS:
    <p>S-3608 is an atypical dopamine agonist.</p>
    Formula:C16H20ClN3OS
    Colore e forma:Solid
    Peso molecolare:337.87
  • CP-66948

    CAS:
    <p>CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.</p>
    Formula:C13H20N6S
    Purezza:99.14%
    Colore e forma:Solid
    Peso molecolare:292.4
  • Indanidine

    CAS:
    Indanidine is a highly selective and potent α-adrenergic agonist with antihypertensive activity.Indanidine is an α-adrenergic antagonist that can be used in the
    Formula:C11H13N5
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:215.25
  • RS-601

    CAS:
    <p>RS-601 is a potent dual leukotriene D4/thromboxane A2 inhibitor that inhibits antigen-induced airway hyperresponsiveness (AHR) and shows asthmatic effects in a</p>
    Formula:C22H23F6NO4S
    Purezza:99.31%
    Colore e forma:Solid
    Peso molecolare:511.48
  • ANEB-001

    CAS:
    <p>ANEB-001 is an orally active CB1 inhibitor that can be used in studies of acute cannabinoid intoxication.</p>
    Formula:C22H24ClF3N2O2
    Colore e forma:Solid
    Peso molecolare:440.89
  • PGN36

    CAS:
    <p>PGN36 (Compound 18) is a potent CB2 receptor antagonist with a high affinity (Ki=0.09 μM).</p>
    Formula:C21H23N3O3
    Colore e forma:Solid
    Peso molecolare:365.43
  • Napitane

    CAS:
    <p>napitane (A 75200) is a novel catecholamine uptake inhibitor with inhibitory effects on α-adrenergic receptors and potential antidepressant activity for the</p>
    Formula:C22H25NO2
    Purezza:99.77% - 99.89%
    Colore e forma:Solid
    Peso molecolare:335.44
  • J-2156

    CAS:
    <p>J-2156, a potent SST4 agonist, has ED50s of 3.7 mg/kg for allodynia and 8.0 mg/kg for hyperalgesia in rats; IC50s are 0.05/0.07 nM in human/rat receptors.</p>
    Formula:C24H28N4O4S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:468.57
  • Phenindamine

    CAS:
    <p>Phenindamine (Nu 1504) is an H1-receptor antagonist which is antihistamine[1].</p>
    Formula:C19H19N
    Colore e forma:Solid
    Peso molecolare:261.36
  • Daledalin tosylate

    CAS:
    Daledalin tosylate is an antidepressant.
    Formula:C26H32N2O3S
    Colore e forma:Solid
    Peso molecolare:452.61
  • Eplivanserin hemifumarate

    CAS:
    <p>Eplivanserin is an inverse agonist of 5-HT2A.</p>
    Formula:C23H25FN2O6
    Colore e forma:Solid
    Peso molecolare:444.45
  • Trebenzomine

    CAS:
    Trebenzomine is apsychotropic agent with potential as an antidepressant and an antipsychotic.
    Formula:C12H17NO
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:191.27
  • Argtide

    CAS:
    <p>Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.</p>
    Formula:C80H104ClN21O14
    Colore e forma:Solid
    Peso molecolare:1619.27
  • Argiprestocin

    CAS:
    Argiprestocin: antidiuretic, regulates osmolality, neurohypophysial hormone, vasoconstrictor.
    Formula:C43H67N15O12S2
    Purezza:99.34%
    Colore e forma:Solid
    Peso molecolare:1050.22
  • Blonanserin HCl

    CAS:
    Blonanserin is an antagonist of dopamine-D2 and serotonin-S2.
    Formula:C23H32Cl2FN3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:440.42
  • CCK-B Receptor Antagonist 2

    CAS:
    <p>CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin/CCK-B (IC50: 0.43 nM). It also inhibits gastrin/CCK-A activity (IC50: 1.82 μM).</p>
    Formula:C27H28N6O3
    Colore e forma:Solid
    Peso molecolare:484.55
  • IMMH001

    CAS:
    <p>IMMH001/SYL930: Oral S1P1 receptor agonist; lowers IL-1β, IL-5, IL-18, IP10, CCL3, CCL5; for RA research.</p>
    Formula:C23H28N2O3
    Colore e forma:Solid
    Peso molecolare:380.48
  • Methapyrilene

    CAS:
    <p>Methapyrilene is a histamine H1 antagonist with sedative action.</p>
    Formula:C14H19N3S
    Colore e forma:Liquid Physical Description Clear Colorless Liquid (Ntp 1992)
    Peso molecolare:261.39
  • L-902688

    CAS:
    <p>L-902688 is an orally active EP4 receptor agonist (Ki: 0.38 nM; EC50: 0.6 nM).</p>
    Formula:C21H27F2N5O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:419.47
  • LPA2 antagonist 2

    CAS:
    LPA2 antagonist 2 is an and LPA2 antagonist (IC50: 28.3 nM) with potential anticancer activity, inhibits LPA3, and can be used for cancer research.
    Formula:C20H16N2O6
    Purezza:96.13%
    Colore e forma:Solid
    Peso molecolare:380.35
  • CAY10680

    CAS:
    <p>CAY10680 inhibits MAO-B (IC50=34.9 nM) &amp; A2A receptors (Ki=39.5 nM), sparing other adenosine types &amp; MAO-A, may treat Parkinson's.</p>
    Formula:C18H16N2O2S
    Colore e forma:Solid
    Peso molecolare:324.4
  • Immepip

    CAS:
    <p>Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.</p>
    Formula:C9H15N3
    Colore e forma:Solid
    Peso molecolare:165.24
  • Seliforant

    CAS:
    <p>Seliforant is a histamine H4 receptor antagonist.</p>
    Formula:C12H21N5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:235.33
  • Phenyltoloxamine

    CAS:
    <p>Phenyltoloxamine (Bistrimin): antihistamine with sedative, analgesic properties, and Sigma-1 receptor affinity (Ki=160 nM).</p>
    Formula:C17H21NO
    Colore e forma:Solid
    Peso molecolare:255.35
  • VUF 5681 dihydrobromide

    CAS:
    <p>histamine H3 receptor silent antagonist</p>
    Formula:C11H21Br2N3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:355.11
  • COR167

    CAS:
    <p>COR167 is a CB2 agonist with immunomodulatory effects, protective brain properties, and antinociception.</p>
    Formula:C28H38N2O2
    Colore e forma:Solid
    Peso molecolare:434.61
  • BAY 1214784

    CAS:
    <p>BAY 1214784: potent, oral hGnRH-R antagonist, reduces LH levels, low variability, good tolerance, may research uterine fibroids.</p>
    Formula:C29H26ClF4N3O5S2
    Colore e forma:Solid
    Peso molecolare:672.11
  • L-692585

    CAS:
    <p>ghrelin receptor (GHS-R1a) agonist</p>
    Formula:C32H37N7O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:567.68
  • GRK5-IN-3

    CAS:
    <p>GRK5-IN-3 is a covalent inhibitor of G protein-coupled receptor kinase 5 (GRK5).GRK5-IN-3 significantly inhibits GRK5 (IC50: 0.22 μM) and GRK6 (IC50: 0.41 μM).</p>
    Formula:C23H21N7O3
    Colore e forma:Solid
    Peso molecolare:443.46
  • RS 39604

    CAS:
    <p>potent and selective 5-HT4 antagonist</p>
    Formula:C26H37Cl2N3O6S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:590.56
  • CP-809101

    CAS:
    CP-809101 is an effective and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).
    Formula:C15H17ClN4O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:304.77
  • ASP-4058 hydrochloride

    CAS:
    <p>ASP-4058 hydrochloride: selective oral S1P1/S1P5 agonist, safe, mitigates mouse autoimmune encephalomyelitis.</p>
    Formula:C19H13ClF6N4O2
    Colore e forma:Solid
    Peso molecolare:478.78
  • KW-8232 free base

    CAS:
    <p>KW-8232 free base can reduces the biosynthesis of PGE2, is an anti-osteoporotic agent.</p>
    Formula:C36H37ClN4O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:609.16
  • GCGR antagonist 2

    CAS:
    <p>Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.</p>
    Formula:C28H26N4O2
    Colore e forma:Solid
    Peso molecolare:450.53
  • Belaperidone

    CAS:
    <p>Belaperidone, an antipsychotic, resembles clozapine, binds D(4) and 5-HT(2A) receptors, minimally extends Q-T without causing arrhythmias.</p>
    Formula:C22H22FN3O2
    Colore e forma:Solid
    Peso molecolare:379.43
  • DuP 734

    CAS:
    <p>DuP 734 is a potent and selective sigma receptor antagonist, functioning as a ligand for both sigma and 5-HT2 receptors, and exhibiting weak affinity towards D2 receptors. It possesses potential antipsychotic activity, potentially devoid of the motor side effects commonly observed with neuroleptics[1][2][3].</p>
    Formula:C17H23BrFNO
    Colore e forma:Solid
    Peso molecolare:356.279
  • AM-6538

    CAS:
    <p>AM6538: long-acting, high-affinity CB antagonist similar to rimonabant, useful for studying cannabinoid agonists.</p>
    Formula:C26H25Cl2N5O4
    Colore e forma:Solid
    Peso molecolare:542.41
  • Cyclazosin HCl

    CAS:
    <p>Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.</p>
    Formula:C23H28ClN5O4
    Purezza:99.10%
    Colore e forma:Solid
    Peso molecolare:473.95
  • CB1-IN-2

    CAS:
    <p>CB1-IN-2 (4g) inhibits CB1 receptor with 0.644 μM IC50; crosses blood-brain barrier, may cause CNS side effects like Rimonabant.</p>
    Formula:C17H19Cl2N5O
    Colore e forma:Solid
    Peso molecolare:380.27
  • BX 667

    CAS:
    <p>BX 667, a P2Y12 antagonist, inhibits ADP-induced platelet clumping in humans, dogs, rats with IC50s: 97, 317, 3000 nM.</p>
    Formula:C29H38N4O9
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:586.63
  • Methyldopa hydrochloride

    CAS:
    <p>L-(-)-α-Methyldopa HCl: alpha-adrenergic agonist, antihypertensive, inhibits DOPA decarboxylase.</p>
    Formula:C10H14ClNO4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:247.68
  • Ko-3290

    CAS:
    <p>Ko-3290 is a cardioselective antagonist of β-adrenoceptors known for its antilipolytic effects in animals.</p>
    Formula:C19H25N3O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:343.42
  • SKF 83959 hydrobromide

    CAS:
    SKF 83959 hydrobromide is a Dopamine D1-like receptor partial agonist.
    Formula:C18H21BrClNO2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:398.72
  • Bopindolol fumarate

    CAS:
    <p>Bopindolol fumarate: non-selective β1/β2-adrenoceptor blocker, partial agonist, low β3 affinity, treats hypertension.</p>
    Formula:C27H32N2O7
    Colore e forma:Solid
    Peso molecolare:496.56
  • Orexin receptor antagonist 2

    CAS:
    <p>Compound 30, potent orexin antagonist with pKis of 7.69/9.78, potential for insomnia research.</p>
    Formula:C25H31N5O2
    Colore e forma:Solid
    Peso molecolare:433.55
  • 6-Chloromelatonin

    CAS:
    <p>6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.</p>
    Formula:C13H15ClN2O2
    Purezza:98.01% - 99.25%
    Colore e forma:Solid
    Peso molecolare:266.72
  • SR-31747

    CAS:
    SR-31747 blocks cell proliferation by inhibiting sterol isomerase. SR-31747 is a sigma ligand. It has immunosuppressive and anti-inflammatory properties.
    Formula:C23H35Cl2N
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:396.44
  • Landiolol

    CAS:
    <p>Landiolol is used as a highly cardioselective ultra short-acting beta-blocker.</p>
    Formula:C25H39N3O8
    Purezza:98%
    Colore e forma:White Crystalline Powder
    Peso molecolare:509.59
  • UNC9975

    CAS:
    <p>UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.</p>
    Formula:C23H28Cl2N4O2
    Purezza:98.78% - 98.78%
    Colore e forma:Solid
    Peso molecolare:463.4
  • I-SAP

    CAS:
    <p>I-SAP: TP receptor blocker, alters platelet shape without causing clumping, EC50 9.7 nM, max binding pH 6.5-7.4, Kd 468-490 pM.</p>
    Formula:C22H30INO4S
    Colore e forma:Solid
    Peso molecolare:531.45
  • BGC-20-1531 free base

    CAS:
    <p>BGC-20-1531 (PGN 1531) free base is a selective and potent prostaglandin EP4 receptor antagonist (pKB: 7.6) that exhibits potential for migraine research.</p>
    Formula:C26H24N2O6S
    Colore e forma:Solid
    Peso molecolare:492.54
  • Modipafant

    CAS:
    <p>Modipaafant is a potent dihydropyridine PAF (platelet activating factor) antagonist.</p>
    Formula:C34H29ClN6O3
    Colore e forma:Solid
    Peso molecolare:605.09
  • A 68930 hydrochloride

    CAS:
    <p>A68930 hydrochloride is a dopamine D1 receptor agonist which can be used for the research of bronchiectasis [1].</p>
    Formula:C16H18ClNO3
    Colore e forma:Off-White Solid
    Peso molecolare:307.77
  • Sinitrodil

    CAS:
    Sinitrodil (ITF-296) is a guanylate cyclase stimulant that may be used in the treatment of myocardial ischemia and angina pectoris.
    Formula:C10H10N2O5
    Purezza:97.03%
    Colore e forma:Solid
    Peso molecolare:238.2
  • Ticolubant

    CAS:
    <p>Ticolubant: Oral LTB4 antagonist, Ki=0.78 nM; blocks Ca2+ migration, IC50=6.6 nM; anti-inflammatory in mice.</p>
    Formula:C23H19Cl2NO3S
    Purezza:99.59%
    Colore e forma:Solid
    Peso molecolare:460.37
  • Isbogrel

    CAS:
    <p>Isbogrel (CV4151) is a TXA2 synthase inhibitor for researching arrhythmias, ischemic attacks, and thrombosis.</p>
    Formula:C18H19NO2
    Purezza:99.58%
    Colore e forma:Solid
    Peso molecolare:281.35
  • RLX-33

    CAS:
    <p>RLX-33 blocks RXFP3 and relaxin 3 effects, controls food intake in rats, and may help study metabolic syndrome.</p>
    Formula:C24H19ClN4O4
    Purezza:99.89%
    Colore e forma:Solid
    Peso molecolare:462.89
  • Olorinab

    CAS:
    <p>Olorinab (APD 371) (APD 371) is a highly potent, selective and fully efficacious cannabinoid receptor type 2 (CB2) agonist. With an EC50 of 6.2 nM for hCB2.</p>
    Formula:C18H23N5O3
    Purezza:97.67% - 98.47%
    Colore e forma:Solid
    Peso molecolare:357.41
  • Piromelatine

    CAS:
    <p>Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity with</p>
    Formula:C17H16N2O4
    Purezza:99.89%
    Colore e forma:Solid
    Peso molecolare:312.32
  • Butofilolol

    CAS:
    <p>Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.</p>
    Formula:C17H26FNO3
    Purezza:98.96% - >99.99%
    Colore e forma:Solid
    Peso molecolare:311.392
  • SLP9101555


    <p>SLP9101555 is a potent and selective sphingosine kinase 2 (SphK2) inhibitor with a Ki of 90 nM.SLP9101555 has a high affinity for SphK2, which is 200-fold</p>
    Formula:C16H22BrClN2
    Purezza:99.45%
    Colore e forma:Solid
    Peso molecolare:357.72
  • KP136

    CAS:
    <p>KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 ug/mL for degranulation).</p>
    Formula:C16H18N4O3
    Purezza:98.3% - 98.61%
    Colore e forma:Solid
    Peso molecolare:314.34
  • U 99194 maleate

    CAS:
    <p>U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.</p>
    Formula:C21H31NO6
    Purezza:99.45%
    Colore e forma:Solid
    Peso molecolare:393.47
  • JTE-907

    CAS:
    <p>JTE-907 是一种具有高度选择性和口服活性的 CB2 受体反向激动剂。JTE-907在体内展现出抗炎活性。</p>
    Formula:C24H26N2O6
    Purezza:99.93%
    Colore e forma:Solid
    Peso molecolare:438.47
  • 2'-MeCCPA

    CAS:
    2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.
    Formula:C16H22ClN5O4
    Purezza:99.93%
    Colore e forma:Solid
    Peso molecolare:383.83
  • Ticalopride

    CAS:
    <p>Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.</p>
    Formula:C14H20ClN3O3
    Purezza:99.51%
    Colore e forma:Solid
    Peso molecolare:313.78
  • Antalarmin hydrochloride

    CAS:
    Antalarmin hydrochloride, a CRF1 antagonist, offers anti-inflammatory benefits and prevents stress ulcers in IBS.
    Formula:C24H35ClN4
    Purezza:99.84% - 99.85%
    Colore e forma:Solid
    Peso molecolare:415.02
  • Liafensine

    CAS:
    Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.
    Formula:C24H22N4
    Purezza:99.91%
    Colore e forma:Solid
    Peso molecolare:366.46
  • Seridopidine

    CAS:
    <p>Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy for schizophrenia, Parkinson's disease, and Tourette's syndrome.</p>
    Formula:C14H20FNO2S
    Purezza:99.65%
    Colore e forma:Solid
    Peso molecolare:285.38
  • Roxindole

    CAS:
    Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.
    Formula:C23H26N2O
    Purezza:98.03% - 98.93%
    Colore e forma:Solid
    Peso molecolare:346.47
  • OPC-51803

    CAS:
    <p>OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.</p>
    Formula:C26H32ClN3O2
    Purezza:98.93% - >99.99%
    Colore e forma:Solid
    Peso molecolare:454
  • Adenosine antagonist-1

    CAS:
    <p>Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.</p>
    Formula:C18H13N7S
    Purezza:99.28% - 99.95%
    Colore e forma:Solid
    Peso molecolare:359.41
  • Anpirtoline hydrochloride

    CAS:
    <p>Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.</p>
    Formula:C10H14Cl2N2S
    Purezza:>99.99% - >99.99%
    Colore e forma:Solid
    Peso molecolare:265.20
  • 4-PPBP maleate

    CAS:
    <p>4-PPBP maleate: potent σ1 agonist, selective NR1a/2B NMDA antagonist, neuroprotective.</p>
    Formula:C25H31NO4
    Purezza:99.88%
    Colore e forma:Solid
    Peso molecolare:409.52
  • SB-277011

    CAS:
    <p>SB-277011A: dopamine D3 antagonist, pKi 8.0 (D3), 6.0 (D2), 5.0 (5-HT1D), &lt;5.2 (5-HT1B).</p>
    Formula:C28H30N4O
    Purezza:99.39%
    Colore e forma:Solid
    Peso molecolare:438.56
  • CyPPA

    CAS:
    <p>CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.</p>
    Formula:C16H23N5
    Purezza:99.88%
    Colore e forma:Solid
    Peso molecolare:285.39
  • Rilapine

    CAS:
    <p>Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.</p>
    Formula:C22H20ClN3
    Purezza:97.76% - 99.20%
    Colore e forma:Solid
    Peso molecolare:361.87
  • ReN-1869

    CAS:
    <p>ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseases</p>
    Formula:C24H27NO2
    Purezza:99.83% - 99.98%
    Colore e forma:Solid
    Peso molecolare:361.48
  • Milenperone

    CAS:
    <p>Milenperone (R 34009) is a novel anti-invasive compound for the control of behavioral disorders in patients with epilepsy and alcoholism.</p>
    Formula:C22H23ClFN3O2
    Purezza:98.09% - 99.84%
    Colore e forma:Solid
    Peso molecolare:415.89
  • UNC0006

    CAS:
    <p>UNC0006 is a β-arrestin-biased dopamine D2 ligand.</p>
    Formula:C24H29Cl2N3O2
    Purezza:99.35% - 99.97%
    Colore e forma:Solid
    Peso molecolare:462.41
  • GSK299115A

    CAS:
    <p>GSK299115A (GSK-299115A) is a selective ROCK1 Inhibitor. GSK299115A exhibits IC50 of 8nM, 620nM, 560nM for ROCK1, RSK1, p70S6K, respectively.</p>
    Formula:C20H16Cl2N4O2
    Purezza:99.81%
    Colore e forma:Solid
    Peso molecolare:415.27
  • cis-Urocanic acid

    CAS:
    <p>cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).</p>
    Formula:C6H6N2O2
    Purezza:99.81%
    Colore e forma:Solid
    Peso molecolare:138.12
  • AS-35

    CAS:
    <p>AS-35, an oral selective leukotriene antagonist, counters ileum contractions with IC50: 8 nM (LTC4), 4 nM (LTD4), 3 nM (LTE4); shows antiallergic effects.</p>
    Formula:C21H20N6O4
    Purezza:96.69%
    Colore e forma:Solid
    Peso molecolare:420.42
  • BMS CCR2 22

    CAS:
    BMS CCR2 22 is a potent and selective antagonist of CCR2 with calcium flux IC50 of 18 nM, chemotaxis IC50 of 1 nM, and binding IC50 of 5.1 nM.
    Formula:C28H34F3N5O4S
    Purezza:99.65%
    Colore e forma:Solid
    Peso molecolare:593.66
  • L 674573

    CAS:
    <p>L 674573 is an inhibitor of leukotriene biosynthesis.</p>
    Formula:C28H27NO3S
    Purezza:99.51%
    Colore e forma:Solid
    Peso molecolare:457.58
  • GR 46611

    CAS:
    GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.
    Formula:C23H27N3O2
    Purezza:99.75%
    Colore e forma:Solid
    Peso molecolare:377.48
  • Nonabine

    CAS:
    <p>Nonabine is a compound with strong antiemetic properties that can be used to prevent nausea and vomiting associated with cancer chemotherapy.</p>
    Formula:C25H33NO2
    Purezza:99.46% - 99.95%
    Colore e forma:Solid
    Peso molecolare:379.54
  • GW-493838

    CAS:
    <p>GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia</p>
    Formula:C21H21ClFN7O4
    Purezza:99.11% - 99.58%
    Colore e forma:Solid
    Peso molecolare:489.89
  • CYM5181

    CAS:
    <p>CYM5181 is related to the body's immune system and can be used to study multiple sclerosis, transplant rejection, and adult respiratory distress syndrome.</p>
    Formula:C17H17N3O3
    Purezza:99.51%
    Colore e forma:Solid
    Peso molecolare:311.34
  • Lecozotan HCl

    CAS:
    <p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>
    Formula:C28H30ClN5O3
    Purezza:99.04%
    Colore e forma:Solid
    Peso molecolare:520.02
  • Halopemide

    CAS:
    Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).
    Formula:C21H22ClFN4O2
    Purezza:96.57%
    Colore e forma:Solid
    Peso molecolare:416.88
  • D18024

    CAS:
    <p>D18024 is a phthalazinonderivat with anti-allergic and anti-histamine effect.</p>
    Formula:C29H31ClFN3O
    Purezza:99.86%
    Colore e forma:Solid
    Peso molecolare:492.03
  • JP1302

    CAS:
    <p>JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.</p>
    Formula:C24H24N4
    Purezza:99.96%
    Colore e forma:Solid
    Peso molecolare:368.47
  • GS-9667

    CAS:
    <p>GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia via</p>
    Formula:C21H24FN5O4S
    Purezza:99.76% - 99.77%
    Colore e forma:Solid
    Peso molecolare:461.51
  • ABT-080

    CAS:
    <p>ABT-080 (VML 530), a leukotriene synthesis inhibitor, is used potentially for treatment of asthma.</p>
    Formula:C37H31N2NaO4
    Purezza:98.42%
    Colore e forma:Solid
    Peso molecolare:590.64
  • Linetastine

    CAS:
    Linetastine (TMK-688) inhibits 5-LOX, blocks leukotrienes, counters histamine; researched for asthma, atherosclerosis, ulcers.
    Formula:C35H40N2O6
    Purezza:99.76%
    Colore e forma:Solid
    Peso molecolare:584.7
  • Rafabegron

    CAS:
    <p>Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.</p>
    Formula:C21H23ClN2O4
    Purezza:99.21%
    Colore e forma:Solid
    Peso molecolare:402.87