Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(939 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.945 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(148 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(407 prodotti)
- Recettore dell'endotelina(76 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(31 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(165 prodotti)
- Proteina Hedgehog/Smoothened(44 prodotti)
- Recettore dell'istamina(358 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(297 prodotti)
- PAFR(11 prodotti)
- PKA(48 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5352 prodotti di "Proteina G/GPCR"
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GSK2239633A
CAS:<p>GSK2239633A is an allosteric antagonist of CC-chemokine receptor 4 (CCR4) with a pIC50 of 7.96 for the binding of [125I]-TARC to human CCR4.</p>Formula:C24H25ClN4O5S2Purezza:99.82%Colore e forma:SolidPeso molecolare:549.06(Z)-Thiothixene
CAS:<p>(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.</p>Formula:C23H29N3O2S2Purezza:99.21%Colore e forma:Yellow To Yellow With A Tan Cast PowderPeso molecolare:443.63Safotibant
CAS:<p>Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edema</p>Formula:C25H34N4O5SPurezza:99.62% - 99.67%Colore e forma:SolidPeso molecolare:502.63Landipirdine
CAS:<p>Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.</p>Formula:C18H19FN2O3SPurezza:97.61% - 99.37%Colore e forma:SolidPeso molecolare:362.42APNEA
CAS:APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.Formula:C18H22N6O4Purezza:99.88%Colore e forma:SolidPeso molecolare:386.41AM-1235
CAS:<p>AM-1235 is a potent and selective cannabinoid receptor CB1 agonist.</p>Formula:C24H21FN2O3Purezza:97.77%Colore e forma:SolidPeso molecolare:404.43Octimibate
CAS:<p>Octimibate: non-prostaglandin antiplatelet, treats cardiovascular disease, aids atherosclerosis/thrombosis research.</p>Formula:C29H30N2O3Purezza:99.51%Colore e forma:SolidPeso molecolare:454.56Rilapine
CAS:<p>Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.</p>Formula:C22H20ClN3Purezza:97.76% - 99.20%Colore e forma:SolidPeso molecolare:361.87CCR2 antagonist 5
CAS:<p>JNJ-41443532: oral hCCR2 antagonist, IC50=37 nM, anti-chemotaxis, treats inflammation & diabetes.</p>Formula:C22H25F3N4O3SPurezza:99.09%Colore e forma:SolidPeso molecolare:482.52SCH-336
CAS:<p>SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 preference, reduces leukocyte migration and eosinophilia.</p>Formula:C23H25NO8S3Purezza:95.01%Colore e forma:SolidPeso molecolare:539.64CMF019
CAS:<p>CMF019 is a potent agonist of the Apelin receptor (APJ) with G protein bias. CMF019 binds to APJ (pKis: 8.58, 8.49, and 8.71 for the human, rat, and mouse).</p>Formula:C25H33N3O3SPurezza:99.5%Colore e forma:SolidPeso molecolare:455.615-HT2 antagonist 1
CAS:<p>5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.</p>Formula:C22H29FN4O2Purezza:99.76%Colore e forma:SolidPeso molecolare:400.49Sitaxsentan
CAS:<p>Sitaxsentan (TBC-11251), a selective ETA receptor antagonist, prevents vasoconstriction by blocking endothelin.</p>Formula:C18H15ClN2O6S2Purezza:97.99% - 98.71%Colore e forma:SolidPeso molecolare:454.9H-9 dihydrochloride
CAS:<p>H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.</p>Formula:C11H15Cl2N3O2SPurezza:97.3%Colore e forma:SolidPeso molecolare:324.23Cilansetron
CAS:<p>Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.</p>Formula:C20H21N3OPurezza:99.82% - 99.98%Colore e forma:SolidPeso molecolare:319.4CB1 agonist 1
CAS:<p>CB1 agonist 1 is a potent CB1 agonist with a pIC50 value of 5.7 for CB1 receptors.CB1 agonist 1 can be used to study brain disorders, pain, and inflammation.</p>Formula:C24H24N2O5SPurezza:98.56%Colore e forma:SolidPeso molecolare:452.52Bavisant
CAS:<p>Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.</p>Formula:C19H27N3O2Purezza:99.21% - 99.65%Colore e forma:SolidPeso molecolare:329.44Taprizosin
CAS:<p>Taprizosin（UK-338003） is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.</p>Formula:C25H26N6O4SPurezza:96.34% - 99.11%Colore e forma:SolidPeso molecolare:506.58Clemastine
CAS:<p>Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.</p>Formula:C21H26ClNOPurezza:99.21%Colore e forma:SolidPeso molecolare:343.89JZP-361
CAS:<p>JZP-361: selective MAGL inhibitor (IC50 = 46 nM); weaker on FAAH, hABHD6; anti-histamine; for asthma research.</p>Formula:C22H20ClN5OPurezza:99.82%Colore e forma:SolidPeso molecolare:405.88PF-00217830
CAS:<p>PF-00217830: agonist at serotonin 1A & dopamine D2, antagonist at serotonin 2A, potential schizophrenia study drug.</p>Formula:C26H30N4O2Purezza:98.72%Colore e forma:SolidPeso molecolare:430.54Teniloxazine
CAS:<p>Teniloxazine is an orally available antidepressant compound with anti-hypoxic properties.</p>Formula:C16H19NO2SPurezza:99.23%Colore e forma:SolidPeso molecolare:289.39UNC0006
CAS:<p>UNC0006 is a β-arrestin-biased dopamine D2 ligand.</p>Formula:C24H29Cl2N3O2Purezza:99.35% - 99.97%Colore e forma:SolidPeso molecolare:462.41CV-6209
CAS:<p>CV-6209 is a potent antagonist of the platelet-activating factor (PAF) receptor.</p>Formula:C34H60ClN3O6Purezza:>99.99% - >99.99%Colore e forma:SolidPeso molecolare:642.31SF-22
CAS:<p>SF-22 is a Y2R antagonist with potential anti-inflammatory activity that can be used to study diseases associated with neurological disorders.</p>Formula:C28H26N2O3SPurezza:99.09%Colore e forma:SolidPeso molecolare:470.58NGD 94-1
CAS:<p>NGD 94-1 is a D4 receptor antagonist that can be used to study psychiatric disorders such as cognitive impairment.</p>Formula:C18H20N6Purezza:99.61%Colore e forma:SolidPeso molecolare:320.39Bedoradrine sulfate
CAS:<p>Bedoradrine sulfate (MN-221 sulfate) is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.</p>Formula:C24H32N2O5H2O4SPurezza:99.31%Colore e forma:SolidPeso molecolare:477.56RLX-33
CAS:<p>RLX-33 blocks RXFP3 and relaxin 3 effects, controls food intake in rats, and may help study metabolic syndrome.</p>Formula:C24H19ClN4O4Purezza:99.89%Colore e forma:SolidPeso molecolare:462.89Remoxipride hydrochloride
CAS:<p>Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, ＞100 μM and 42 μM for D2 receptor, D1 receptor and α1-</p>Formula:C16H24BrClN2O3Purezza:99.88%Colore e forma:SolidPeso molecolare:407.73NE-100 hydrochloride
CAS:<p>NE-100 hydrochloride (NE-100 HCl) is a potent and selective antagonist of σ1 (IC50 = 4.16 nM) with antipsychotic activity.</p>Formula:C23H34ClNO2Purezza:99.76%Colore e forma:SolidPeso molecolare:391.98SLF1081851
CAS:<p>SLF1081851 is a Spns2 inhibitor. SLF1081851 inhibits S1P release with IC50 of 1.93 μM.</p>Formula:C21H33N3OPurezza:99.26%Colore e forma:SolidPeso molecolare:343.51PNU-282987 free base
CAS:<p>PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.</p>Formula:C14H17ClN2OPurezza:99.64%Colore e forma:SolidPeso molecolare:264.75Noberastine
CAS:<p>Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.</p>Formula:C17H21N5OPurezza:99.72% - >99.99%Colore e forma:SolidPeso molecolare:311.38SDZ-62-434
CAS:<p>SDZ-62-434 is a platelet-activating factor inhibitor with antitumor activity and may be used in the study of leukemia.</p>Formula:C23H27Cl2N3Purezza:98.38%Colore e forma:SolidPeso molecolare:416.39BMY-14802 hydrochloride
CAS:<p>BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.</p>Formula:C18H23ClF2N4OPurezza:99.97%Colore e forma:SolidPeso molecolare:384.85Compound C108
CAS:<p>Compound C108 is an inhibitor of GTPase-activating protein SH3 domain-binding protein 2 (G3BP2).</p>Formula:C15H14N2O3Purezza:99.77%Colore e forma:SolidPeso molecolare:270.28Lensiprazine
CAS:<p>Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder and</p>Formula:C24H27FN4O2Purezza:98.04%Colore e forma:SolidPeso molecolare:422.5CYM5181
CAS:<p>CYM5181 is related to the body's immune system and can be used to study multiple sclerosis, transplant rejection, and adult respiratory distress syndrome.</p>Formula:C17H17N3O3Purezza:99.51%Colore e forma:SolidPeso molecolare:311.34E6801
CAS:<p>E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.</p>Formula:C17H18ClN5O2S2Purezza:96.32% - 99.53%Colore e forma:SolidPeso molecolare:423.94PSB-16133 sodium
CAS:<p>PSB-16133 sodium is a selective P2Y purine receptor variant antagonist with an IC of 233 nM.</p>Formula:C28H21N2NaO5S2Purezza:98.03% - 98.93%Colore e forma:SolidPeso molecolare:552.60LY266097 hydrochloride
CAS:<p>LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.</p>Formula:C21H24Cl2N2O2Purezza:98.58%Colore e forma:SolidPeso molecolare:407.33Soquinolol
CAS:<p>Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a long</p>Formula:C17H26N2O3Purezza:97.48% - 98.63%Colore e forma:SolidPeso molecolare:306.4Proxyfan
CAS:<p>Proxyfan is a high-affinity protean antagonist/agonist of H3 receptors from full agonist to full inverse agonist, depending on given tissue or brain region.</p>Formula:C13H16N2OPurezza:99.68%Colore e forma:SolidPeso molecolare:216.28Nonabine
CAS:<p>Nonabine is a compound with strong antiemetic properties that can be used to prevent nausea and vomiting associated with cancer chemotherapy.</p>Formula:C25H33NO2Purezza:99.46% - 99.95%Colore e forma:SolidPeso molecolare:379.54Perphenazine dihydrochloride
CAS:<p>Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.</p>Formula:C21H28Cl3N3OSPurezza:99.67%Colore e forma:SolidPeso molecolare:476.89FPL 55712
CAS:<p>FPL 55712 is a leukotriene receptor and SRS-A antagonist that inhibits bronchoconstriction and can be used in studies of asthma and coronary artery thrombosis.</p>Formula:C27H30O9Purezza:98.15% - 99.8%Colore e forma:SolidPeso molecolare:498.52CB2R PAM
CAS:<p>CB2R PAM, an oral drug, boosts CB2 receptor response to specific agonists, showing potential in neuropathic pain relief.</p>Formula:C21H24BrFN2O2Purezza:99.09%Colore e forma:SolidPeso molecolare:435.33Egis-11150
CAS:<p>Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.</p>Formula:C19H21ClFN5O2Purezza:97.49% - >99.99%Colore e forma:SolidPeso molecolare:405.85RS 67333 hydrochloride
CAS:<p>RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.</p>Formula:C19H30Cl2N2O2Purezza:98.78%Colore e forma:SolidPeso molecolare:389.36LAS38096
CAS:<p>LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .</p>Formula:C17H12N6OPurezza:99.18% - 99.95%Colore e forma:SolidPeso molecolare:316.32Remogliflozin etabonate
CAS:<p>Remogliflozin etabonate is a prodrug SGLT2 inhibitor; Ki for hSGLT2: 1.95μM, rSGLT2: 2.14μM, rSGLT1: 8.57μM, hSGLT1: 43.1μM.</p>Formula:C26H38N2O9Purezza:98.98%Colore e forma:SolidPeso molecolare:522.59Ensaculin
CAS:<p>Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.</p>Formula:C26H32N2O5Purezza:99.17% - 99.67%Colore e forma:SolidPeso molecolare:452.54Antalarmin hydrochloride
CAS:<p>Antalarmin hydrochloride, a CRF1 antagonist, offers anti-inflammatory benefits and prevents stress ulcers in IBS.</p>Formula:C24H35ClN4Purezza:99.84% - 99.85%Colore e forma:SolidPeso molecolare:415.02Femoxetine hydrochloride
CAS:<p>Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.</p>Formula:C20H26ClNO2Purezza:99.63%Colore e forma:SolidPeso molecolare:347.88SR144528
CAS:<p>SR144528 is an antagonist of the CB2 receptor (Ki = 0.6 nM) and inhibits microsomal ACAT activity (IC50 = 3.6 μM).</p>Formula:C29H34ClN3OPurezza:99.63%Colore e forma:SolidPeso molecolare:476.05Regrelor disodium
CAS:<p>Regrelor disodium (INS 50589) is a p2y12 receptor antagonist that prevents thrombosis, effectively inhibits vascular smooth muscle cell contraction, inhibits</p>Formula:C22H23N6Na2O8PPurezza:99.95%Colore e forma:SolidPeso molecolare:576.41BP14979
CAS:<p>BP14979 is D3R-selective partial agonist.</p>Formula:C23H34N4O2Purezza:98.29% - 99.73%Colore e forma:SolidPeso molecolare:398.54AZ-1355
CAS:<p>AZ-1355 is a novel dibenzoxepine derivative with lipid-lowering properties.</p>Formula:C17H17NO4Purezza:>99.99%Colore e forma:SolidPeso molecolare:299.32Efletirizine
CAS:<p>Efletirizine (UCB-28754), a histamine blocker and 5-LO inhibitor, aids in topical allergy treatment.</p>Formula:C21H24F2N2O3Purezza:99.39%Colore e forma:SolidPeso molecolare:390.42SPD-473 citrate
CAS:<p>SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.</p>Formula:C23H31Cl2NO8SPurezza:99.37%Colore e forma:SolidPeso molecolare:552.47ST-1535
CAS:<p>ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.</p>Formula:C12H16N8Purezza:99.64% - 99.69%Colore e forma:SolidPeso molecolare:272.31Litoxetine
CAS:<p>Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.</p>Formula:C16H19NOPurezza:99.47%Colore e forma:SolidPeso molecolare:241.33Bedoradrine
CAS:<p>Bedoradrine (MN-221) free base is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.</p>Formula:C24H32N2O5Purezza:>99.99%Colore e forma:SolidPeso molecolare:428.52Ronacaleret HCl
CAS:<p>Ronacaleret HCl (SB-751689) is a small molecule CaSR antagonist for the treatment of endocrine and metabolic diseases, skin and musculoskeletal disorders.</p>Formula:C25H32ClF2NO4Purezza:99.97%Colore e forma:SolidPeso molecolare:483.98N 0861
CAS:<p>N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.</p>Formula:C13H17N5Purezza:98.78%Colore e forma:SolidPeso molecolare:243.31Crinecerfont
CAS:<p>Crinecerfont (SSR-125543) is a CRF1 antagonist, useful in congenital adrenal hyperplasia research.</p>Formula:C27H28ClFN2OSPurezza:98.01% - 98.55%Colore e forma:SolidPeso molecolare:483.04Pirmagrel
CAS:<p>pirmagrel is a potent thromboxane synthase inhibitor.</p>Formula:C13H16N2O2Purezza:98.02%Colore e forma:SolidPeso molecolare:232.28Spizofurone
CAS:<p>Spizofurone (Espizofurona) has anti-ulcer activity, protective effect on the gastric mucosa of rats and can increase alkaline secretion.</p>Formula:C12H10O3Purezza:>99.99%Colore e forma:SolidPeso molecolare:202.21SMO-IN-2
CAS:<p>SMO-IN-2 is a SMO inhibitor with antiproliferative activity and anticancer activity and inhibits Hh signaling.SMO-IN-2 can be used in the study of cancer.</p>Formula:C25H25F4N5O2Purezza:98.64%Colore e forma:SolidPeso molecolare:503.49LX-2931
CAS:<p>LX-2931(LX-3305) is a sphingosine-1-phosphate cleavage enzyme (S1P) inhibitor for the treatment of rheumatoid arthritis.</p>Formula:C9H15N3O5Purezza:98.85% - 99.83%Colore e forma:SolidPeso molecolare:245.23Impromidine hydrochloride
CAS:<p>Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.</p>Formula:C14H26Cl3N7SPurezza:99.82%Colore e forma:SolidPeso molecolare:430.83L-161982
CAS:<p>L-161982 is a selective EP4 receptor antagonist that inhibits PGE2-induced ERK phosphorylation and cell proliferation in HCA-7 cells.Cost-effective and quality-assured.</p>Formula:C32H29F3N4O4S2Purezza:99.58% - 99.6%Colore e forma:SolidPeso molecolare:654.72NNC 92-1687
CAS:<p>NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.</p>Formula:C15H12N2O3SPurezza:98.70% - 99.70%Colore e forma:SolidPeso molecolare:300.33LY 272015 hydrochloride
CAS:<p>LY 272015 hydrochloride is a 5-HT2B receptor antagonist.</p>Formula:C21H25ClN2O2Purezza:99.47%Colore e forma:SolidPeso molecolare:372.895HT6-ligand-1
CAS:<p>5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).</p>Formula:C20H22BrN3O2SPurezza:99.24% - 99.93%Colore e forma:SolidPeso molecolare:448.38Ticolubant
CAS:<p>Ticolubant: Oral LTB4 antagonist, Ki=0.78 nM; blocks Ca2+ migration, IC50=6.6 nM; anti-inflammatory in mice.</p>Formula:C23H19Cl2NO3SPurezza:99.59%Colore e forma:SolidPeso molecolare:460.37CCR1 antagonist 6
CAS:<p>CCR1 antagonist 6 is a CCR1 antagonist (IC50: 3 nM).</p>Formula:C21H23ClN4O3SPurezza:99.02% - 99.15%Colore e forma:SolidPeso molecolare:446.95Ricasetron
CAS:<p>Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.</p>Formula:C19H27N3OPurezza:99.52%Colore e forma:SolidPeso molecolare:313.44AZD1940
CAS:<p>AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.</p>Formula:C20H29F2N3O2SPurezza:98.68%Colore e forma:SolidPeso molecolare:413.52Thiethylperazine dimaleate
CAS:<p>Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor.</p>Formula:C30H37N3O8S2Purezza:99.07%Colore e forma:SolidPeso molecolare:631.76FK-453
CAS:<p>FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.</p>Formula:C23H25N3O2Purezza:99.44%Colore e forma:SolidPeso molecolare:375.46Medifoxamine
CAS:<p>Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition of 5 HT reuptake.Medifoxamine</p>Formula:C16H19NO2Purezza:97.14%Colore e forma:SolidPeso molecolare:257.33Anpirtoline hydrochloride
CAS:<p>Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.</p>Formula:C10H14Cl2N2SPurezza:>99.99% - >99.99%Colore e forma:SolidPeso molecolare:265.20Tiopinac
CAS:<p>Tiopinac: tricyclic with anti-inflammatory, analgesic, antipyretic properties; inhibits prostaglandin synthesis; mild anti-platelet effects in humans.</p>Formula:C16H12O3SPurezza:>99.99%Colore e forma:SolidPeso molecolare:284.33BL-1020 Mesylate
CAS:<p>BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.</p>Formula:C28H45ClN4O11S4Purezza:>99.99%Colore e forma:SolidPeso molecolare:777.39NP10679
CAS:<p>NP10679 is a N-methyl-D-aspartate (NMDA) receptor inhibitor of the GluN2B subunit that inhibits histamine H1, hERG channels, and CYPase.</p>Formula:C23H26F3N3O3Purezza:99.43%Colore e forma:SolidPeso molecolare:449.47ML 10302 hydrochloride
CAS:<p>ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.</p>Formula:C15H22Cl2N2O3Purezza:99.99%Colore e forma:SolidPeso molecolare:349.25Masupirdine free base
CAS:<p>Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.</p>Formula:C21H24BrN3O3SPurezza:98.36% - 99.65%Colore e forma:SolidPeso molecolare:478.4CB1R antagonist 1
CAS:<p>CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.</p>Formula:C18H23F3N2O3SPurezza:99.65%Colore e forma:SolidPeso molecolare:404.45Sergliflozin etabonate
CAS:<p>Sergliflozin etabonate (KGT-1251) is an inhibitor of SGLT2 and can be used in studies about type 2 diabetes and obesity.</p>Formula:C23H28O9Purezza:97.88%Colore e forma:SolidPeso molecolare:448.46Sarizotan HCl
CAS:<p>Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.</p>Formula:C22H22ClFN2OPurezza:96%Colore e forma:SolidPeso molecolare:384.87ST 91
CAS:<p>ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.</p>Formula:C13H20ClN3Purezza:99.83%Colore e forma:SolidPeso molecolare:253.77O-1602
CAS:<p>O-1602 is a novel GPR55 agonist, an atypical cannabinoid associated with the central nervous system and obesity, and is a candidate compound for the treatment</p>Formula:C17H22O2Purezza:99.85%Colore e forma:SolidPeso molecolare:258.36ASP-4058
CAS:<p>ASP-4058: Safe, oral S1P1/S1P5 agonist; improves autoimmune encephalomyelitis in mice.</p>Formula:C19H12F6N4O2Purezza:99.30% - 99.53%Colore e forma:SolidPeso molecolare:442.31Selodenoson
CAS:<p>Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.</p>Formula:C17H24N6O4Purezza:99.52%Colore e forma:SolidPeso molecolare:376.41Benperidol
CAS:<p>Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.</p>Formula:C22H24FN3O2Purezza:99.91%Colore e forma:SolidPeso molecolare:381.44N-[(4-Aminophenyl)methyl]adenosine
CAS:<p>N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).</p>Formula:C17H20N6O4Purezza:98.75%Colore e forma:SolidPeso molecolare:372.38ML-354
CAS:<p>ML354 is a selective antagonist of PAR4 with an IC 50 of 140 nM [1].</p>Formula:C16H14N2O3Purezza:99.44%Colore e forma:SolidPeso molecolare:282.29MLS1547
CAS:<p>MLS1547 is a potent D2 receptor G protein-biased agonist (Ki=1.2 μM, EC50=0.37 μM in Ca2+ assay).</p>Formula:C19H19ClN4OPurezza:99.64%Colore e forma:SolidPeso molecolare:354.83Tildacerfont
CAS:<p>Tildacerfont inhibits CRF1, lowers ACTH/adrenal androgens, and aids in congenital adrenal hyperplasia research.</p>Formula:C20H26ClN5OSPurezza:>99.99%Colore e forma:SolidPeso molecolare:419.97BAY 60-6583
CAS:<p>BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3</p>Formula:C19H17N5O2SPurezza:98.46% - 99.8%Colore e forma:SolidPeso molecolare:379.44MRS1220
CAS:<p>MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeutic</p>Formula:C21H14ClN5O2Purezza:98.43%Colore e forma:SolidPeso molecolare:403.82SLP9101555
<p>SLP9101555 is a potent and selective sphingosine kinase 2 (SphK2) inhibitor with a Ki of 90 nM.SLP9101555 has a high affinity for SphK2, which is 200-fold</p>Formula:C16H22BrClN2Purezza:99.45%Colore e forma:SolidPeso molecolare:357.72Terbogrel
CAS:<p>Terbogrel is an antiplatelet drug, blocking thromboxane A2 receptor/synthase. Helps prevent clots.</p>Formula:C23H27N5O2Purezza:98.95%Colore e forma:SolidPeso molecolare:405.49Runcaciguat
CAS:<p>Runcaciguat, a soluble guanylate cyclase stimulator, aids in cardiovascular and renal research.</p>Formula:C23H22Cl2F3NO3Purezza:99.17%Colore e forma:SolidPeso molecolare:488.33VA-K-14 hydrochloride
CAS:<p>VA-K-14 hydrochloride（VAK14 HCl） is a selective thyrotropin receptor (TSHR) antagonist (IC50= 12.3 μM) that inhibits TSHR stimulation by serum and monoclonal</p>Formula:C18H16ClN3SPurezza:97.15%Colore e forma:SolidPeso molecolare:341.86Butofilolol
CAS:<p>Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.</p>Formula:C17H26FNO3Purezza:98.96% - >99.99%Colore e forma:SolidPeso molecolare:311.392YIL 781
CAS:<p>YIL 781 is a selective ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM), showing a weak affinity for kinesin receptors (K = 6 μM).</p>Formula:C24H28FN3O2Purezza:98.8%Colore e forma:SolidPeso molecolare:409.5RG 7152
CAS:<p>RG 7152 is a leukotriene D4 antagonist with anti-asthmatic properties and can be used in the study of asthma.</p>Formula:C20H19N5O2Purezza:98.45%Colore e forma:SolidPeso molecolare:361.4Parogrelil Free Base
CAS:<p>Parogrelil Free Base is a phosphodiesterase inhibitor, improves claudication-limited exercise performance in patients with peripheral arterial disease.</p>Formula:C19H18BrClN4O2Purezza:99.16% - 99.17%Colore e forma:SolidPeso molecolare:449.732'-MeCCPA
CAS:2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.Formula:C16H22ClN5O4Purezza:99.93%Colore e forma:SolidPeso molecolare:383.83Camonagrel
CAS:<p>Camonagrel is a compound that has inhibitory effects on Prostaglandin E2.</p>Formula:C15H16N2O3Purezza:98.71% - 99.25%Colore e forma:SolidPeso molecolare:272.3RO3244794
CAS:<p>RO3244794 is a selective prostacyclin (IP) receptor antagonist that can be used to study liver injury.</p>Formula:C25H19F2NO5Purezza:99.36%Colore e forma:SolidPeso molecolare:451.42Rezatomidine
CAS:<p>Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.</p>Formula:C13H16N2SPurezza:98.34%Colore e forma:SolidPeso molecolare:232.34Dimethindene maleate
CAS:<p>Dimethindene maleate (SU 6518) is a histamine H1 antagonist and can be used in studies about the treatment of hypersensitivity reactions, pruritus and rhinitis.</p>Formula:C24H28N2O4Purezza:99.79%Colore e forma:SolidPeso molecolare:408.49Sinitrodil
CAS:<p>Sinitrodil (ITF-296) is a guanylate cyclase stimulant that may be used in the treatment of myocardial ischemia and angina pectoris.</p>Formula:C10H10N2O5Purezza:98.98%Colore e forma:SolidPeso molecolare:238.2PPTN hydrochloride
CAS:<p>PPTN hydrochloride is a potent, high-affinity, competitive, highly selective P2Y14 receptor antagonist (KB: 434 pM), but no agonist or antagonist activity at</p>Formula:C29H25ClF3NO2Purezza:99.80%Colore e forma:SolidPeso molecolare:511.96Aplindore Fumarate
CAS:<p>Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.</p>Formula:C22H22N2O7Purezza:>99.99%Colore e forma:SolidPeso molecolare:426.42Oxyfedrine L-form HCl
CAS:<p>Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent.</p>Formula:C19H24ClNO3Purezza:99.5% - 99.57%Colore e forma:SolidPeso molecolare:349.85CCG 203769
CAS:<p>CCG 203769 (Thiadiazolidinone (TDZD) deriv. 6) is a selective inhibitor of RGS4 with an IC50 of 17 nM for the RGS4-Gαo protein-protein interaction.</p>Formula:C8H14N2O2SPurezza:99.88%Colore e forma:SolidPeso molecolare:202.27Nexopamil
CAS:<p>Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.</p>Formula:C24H40N2O3Purezza:97.87% - >99.99%Colore e forma:SolidPeso molecolare:404.59BMS CCR2 22
CAS:BMS CCR2 22 is a potent and selective antagonist of CCR2 with calcium flux IC50 of 18 nM, chemotaxis IC50 of 1 nM, and binding IC50 of 5.1 nM.Formula:C28H34F3N5O4SPurezza:99.65%Colore e forma:SolidPeso molecolare:593.66Ecastolol
CAS:<p>Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.</p>Formula:C26H33N3O6Purezza:99.89%Colore e forma:SolidPeso molecolare:483.56OPC-51803
CAS:<p>OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.</p>Formula:C26H32ClN3O2Purezza:98.93% - >99.99%Colore e forma:SolidPeso molecolare:454Itriglumide
CAS:<p>Itriglumide, a CCK2 receptor antagonist, is used potentially for the treatment of peptic ulcers, dyspepsia, and gastroesophageal reflux disease (GERD).</p>Formula:C33H38N2O4Purezza:99.95%Colore e forma:SolidPeso molecolare:526.67SB-215505
CAS:<p>SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, 5-HT2A - 6.77).</p>Formula:C19H16ClN3OPurezza:98.33%Colore e forma:SolidPeso molecolare:337.8Halopemide
CAS:<p>Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).</p>Formula:C21H22ClFN4O2Purezza:96.57%Colore e forma:SolidPeso molecolare:416.8848740 RP
CAS:<p>48740 RP (RP 55779) is an antagonist of platelet-activating factor.</p>Formula:C12H11N3OSPurezza:99.79%Colore e forma:SolidPeso molecolare:245.3Milenperone
CAS:<p>Milenperone (R 34009) is a novel anti-invasive compound for the control of behavioral disorders in patients with epilepsy and alcoholism.</p>Formula:C22H23ClFN3O2Purezza:98.09% - 99.84%Colore e forma:SolidPeso molecolare:415.89Lorglumide sodium salt
CAS:<p>Lorglumide sodium salt (CR-1409 sodium salt) is an antagonist of cholecystokinin receptors (CCK).</p>Formula:C22H31Cl2N2NaO4Purezza:99.32%Colore e forma:SolidPeso molecolare:481.39Repinotan
CAS:<p>Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic stroke studies.</p>Formula:C21H24N2O4SPurezza:99%Colore e forma:SolidPeso molecolare:400.49TC LPA5 4
CAS:<p>TC LPA5 4 is a LPA5 receptor antagonist.</p>Formula:C23H23ClN2O3Purezza:99.93%Colore e forma:SolidPeso molecolare:410.89Lecozotan HCl
CAS:<p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>Formula:C28H30ClN5O3Purezza:99.04%Colore e forma:SolidPeso molecolare:520.02Piromelatine
CAS:<p>Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity with</p>Formula:C17H16N2O4Purezza:99.89%Colore e forma:SolidPeso molecolare:312.32AS-35
CAS:<p>AS-35, an oral selective leukotriene antagonist, counters ileum contractions with IC50: 8 nM (LTC4), 4 nM (LTD4), 3 nM (LTE4); shows antiallergic effects.</p>Formula:C21H20N6O4Purezza:96.69%Colore e forma:SolidPeso molecolare:420.42N6-(2-Phenylethyl)adenosine
CAS:<p>N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for</p>Formula:C18H21N5O4Purezza:99.83%Colore e forma:SolidPeso molecolare:371.39GS-9667
CAS:<p>GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia via</p>Formula:C21H24FN5O4SPurezza:99.76% - 99.77%Colore e forma:SolidPeso molecolare:461.51MrgprX2 antagonist-8
CAS:<p>MrgprX2 antagonist-8 is an MrgprX2 antagonist that can be used to study inflammatory diseases.</p>Formula:C24H24ClF3N4O3SPurezza:98.61%Colore e forma:SolidPeso molecolare:540.99Irdabisant
CAS:<p>Irdabisant (CEP-26401) is an H3R antagonist/inverse agonist, BBB permeable, with cognition-enhancing effects for schizophrenia/cognitive research.</p>Formula:C18H23N3O2Purezza:99.96%Colore e forma:SolidPeso molecolare:313.39AZD8542
CAS:<p>AZD8542 is an antagonist of Smoothened (SMO) with potential as an oncology therapeutic.</p>Formula:C25H24N4O2Purezza:99.96%Colore e forma:SolidPeso molecolare:412.485-HT6/7 antagonist 1
CAS:<p>5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.</p>Formula:C22H20FN3O3Purezza:98.78% - 99.26%Colore e forma:SolidPeso molecolare:393.41Adoprazine
CAS:<p>Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.</p>Formula:C24H24FN3O2Purezza:99.83%Colore e forma:SolidPeso molecolare:405.46Ordopidine
CAS:<p>Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during inactivity.</p>Formula:C14H20FNO2SPurezza:99.39%Colore e forma:SolidPeso molecolare:285.38Rocepafant
CAS:<p>Rocepafant (LAU8080), a PAF antagonist, reduces neonatal rat brain damage and inhibits TNF-α toxicity in L929 cells.</p>Formula:C26H23ClN6OS2Purezza:97.31% - 98.95%Colore e forma:SolidPeso molecolare:535.08Pirodomast
CAS:<p>Pirodomast is a thromboxane A (TXA2) synthase inhibitor.</p>Formula:C18H17N3O2Purezza:99.64%Colore e forma:SolidPeso molecolare:307.35SB-277011
CAS:<p>SB-277011A: dopamine D3 antagonist, pKi 8.0 (D3), 6.0 (D2), 5.0 (5-HT1D), <5.2 (5-HT1B).</p>Formula:C28H30N4OPurezza:99.39%Colore e forma:SolidPeso molecolare:438.56JTE-907
CAS:<p>JTE-907 是一种具有高度选择性和口服活性的 CB2 受体反向激动剂。JTE-907在体内展现出抗炎活性。</p>Formula:C24H26N2O6Purezza:99.93%Colore e forma:SolidPeso molecolare:438.47ReN-1869
CAS:<p>ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseases</p>Formula:C24H27NO2Purezza:99.83% - 99.98%Colore e forma:SolidPeso molecolare:361.48Pimethixene maleate
CAS:<p>Pimethixene maleate (Pimetixene maleate) is a 5-HT2B receptor antagonist with sedative activity that can be used to study dry cough in children.</p>Formula:C23H23NO4SPurezza:99.55%Colore e forma:SolidPeso molecolare:409.5Roxindole
CAS:<p>Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.</p>Formula:C23H26N2OPurezza:98.03% - 98.93%Colore e forma:SolidPeso molecolare:346.47BMS-470539 dihydrochloride
CAS:BMS-470539 dihydrochloride is a MC-1 R agonist with anti-inflammatory activity.Formula:C32H43Cl2N5O4Purezza:>99.99%Colore e forma:SolidPeso molecolare:632.62KSK68
CAS:<p>KSK68 is a sigma-1 and histamine H3 receptor antagonist with analgesic activity, inhibits H3 receptors and can be used to study pain.</p>Formula:C23H28N2O2Purezza:99.11%Colore e forma:SolidPeso molecolare:364.487-Hydroxy-DPAT hydrobromide
CAS:<p>7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.</p>Formula:C16H26BrNOPurezza:99.73%Colore e forma:SolidPeso molecolare:328.29JP1302
CAS:<p>JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.</p>Formula:C24H24N4Purezza:99.96%Colore e forma:SolidPeso molecolare:368.478-OH-Dpat
CAS:<p>8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.</p>Formula:C16H25NOPurezza:98%Colore e forma:SolidPeso molecolare:247.38Neldazosin
CAS:<p>Neldazosin is used as a potent α1-adrenoceptor antagonist.</p>Formula:C18H25N5O4Purezza:99.74% - 99.76%Colore e forma:SolidPeso molecolare:375.42MK-0686
CAS:<p>MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.</p>Formula:C22H19ClF4N2O4Purezza:99.88%Colore e forma:SolidPeso molecolare:486.84Seridopidine
CAS:<p>Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy for schizophrenia, Parkinson's disease, and Tourette's syndrome.</p>Formula:C14H20FNO2SPurezza:99.65%Colore e forma:SolidPeso molecolare:285.38ANR 94
CAS:<p>ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.</p>Formula:C9H13N5OPurezza:98.9%Colore e forma:SolidPeso molecolare:207.23L 674573
CAS:<p>L 674573 is an inhibitor of leukotriene biosynthesis.</p>Formula:C28H27NO3SPurezza:99.51%Colore e forma:SolidPeso molecolare:457.58LTB4-IN-1
CAS:<p>LTB4-IN-1 (Anti-inflammatory agent 2) with IC50 of 70 nM is an inhibitor of leukotriene synthesis (LTB4).</p>Formula:C26H30N2O4SPurezza:99.93%Colore e forma:SolidPeso molecolare:466.59Eclazolast
CAS:<p>Eclazolast (RHC 2871), a lipophilic anti-allergic, inhibits mast cell mediator release by affecting Fc(epsilon)RI-related processes, dose-dependently.</p>Formula:C12H12ClNO4Purezza:98.36% - 98.58%Colore e forma:SolidPeso molecolare:269.68SK609 HCl
CAS:<p>SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.</p>Formula:C10H15Cl2NPurezza:99.02%Colore e forma:SolidPeso molecolare:220.14A2A receptor antagonist 1
CAS:<p>A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.</p>Formula:C16H12FN5OPurezza:99.52% - 99.93%Colore e forma:SolidPeso molecolare:309.3Upacicalcet
CAS:<p>Upacicalcet (AJT-240) is a calcium mimetic for SHPT in dialysis, reducing PTH by targeting parathyroid receptors.</p>Formula:C11H14ClN3O6SPurezza:99.83%Colore e forma:SolidPeso molecolare:351.76SB-209670
CAS:<p>SB-209670 is a selective endothelin receptor antagonist that inhibits the activity of ET(B) receptors in rat vascular endothelium and vascular smooth muscle.</p>Formula:C29H28O9Purezza:97.80% - 99.40%Colore e forma:SolidPeso molecolare:520.53Antihistamine-1
CAS:<p>Antihistamine-1 是能够渗透血脑屏障的 H1-抗组胺药 (Ki=6.9 nM), 它也是 CYP2D6 和 hERG 通道的抑制剂，其 IC50 值分别为 5.4 和 0.8 μM。</p>Formula:C23H24FN5Purezza:99.69%Colore e forma:SolidPeso molecolare:389.47U 99194 maleate
CAS:<p>U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.</p>Formula:C21H31NO6Purezza:99.45%Colore e forma:SolidPeso molecolare:393.47KI-7
CAS:<p>KI-7 is an adenosine A2B receptor positive allosteric modulator.</p>Formula:C23H18N2O2Purezza:98.33%Colore e forma:SolidPeso molecolare:354.4Rafabegron
CAS:<p>Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.</p>Formula:C21H23ClN2O4Purezza:99.21%Colore e forma:SolidPeso molecolare:402.87GW-493838
CAS:<p>GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia</p>Formula:C21H21ClFN7O4Purezza:99.11% - 99.58%Colore e forma:SolidPeso molecolare:489.89Linetastine
CAS:<p>Linetastine (TMK-688) inhibits 5-LOX, blocks leukotrienes, counters histamine; researched for asthma, atherosclerosis, ulcers.</p>Formula:C35H40N2O6Purezza:99.76%Colore e forma:SolidPeso molecolare:584.7Sonedenoson
CAS:<p>Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase.</p>Formula:C18H20ClN5O5Purezza:99.79%Colore e forma:SolidPeso molecolare:421.84Thonzylamine hydrochloride
CAS:<p>Thonzylamine hydrochloride (Resistab) is an anticholinergic and antihistamine used as an antipruritic.</p>Formula:C16H23ClN4OPurezza:99.67%Colore e forma:White Crystalline PowderPeso molecolare:322.83BMS-817399
CAS:<p>BMS-817399: oral CCR1 antagonist with binding and chemotaxis inhibition IC50s, potential for rheumatoid arthritis research.</p>Formula:C23H36ClN3O4Purezza:99.7%Colore e forma:SolidPeso molecolare:454DF-1111301
CAS:<p>DF-1111301 is a novel anti-allergic compound with anti-histamine H1 and anti-PAF activity.</p>Formula:C15H25Cl2N3OPurezza:99.17%Colore e forma:SolidPeso molecolare:334.29Besipirdine
CAS:<p>Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.</p>Formula:C16H17N3Purezza:97.15% - 98.85%Colore e forma:SolidPeso molecolare:251.33Imiloxan
CAS:<p>Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.</p>Formula:C14H16N2O2Purezza:98.13% - 99.8%Colore e forma:SolidPeso molecolare:244.29KP136
CAS:<p>KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 ug/mL for degranulation).</p>Formula:C16H18N4O3Purezza:98.3% - 98.61%Colore e forma:SolidPeso molecolare:314.34Abt-288
CAS:<p>ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.</p>Formula:C23H24N4OPurezza:98.17% - 98.49%Colore e forma:SolidPeso molecolare:372.46Tedatioxetine
CAS:<p>Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.</p>Formula:C18H21NSPurezza:99.76% - >99.99%Colore e forma:SolidPeso molecolare:283.43D18024
CAS:<p>D18024 is a phthalazinonderivat with anti-allergic and anti-histamine effect.</p>Formula:C29H31ClFN3OPurezza:99.86%Colore e forma:SolidPeso molecolare:492.03ABT-080
CAS:<p>ABT-080 (VML 530), a leukotriene synthesis inhibitor, is used potentially for treatment of asthma.</p>Formula:C37H31N2NaO4Purezza:98.42%Colore e forma:SolidPeso molecolare:590.64GSK299115A
CAS:<p>GSK299115A (GSK-299115A) is a selective ROCK1 Inhibitor. GSK299115A exhibits IC50 of 8nM, 620nM, 560nM for ROCK1, RSK1, p70S6K, respectively.</p>Formula:C20H16Cl2N4O2Purezza:99.81%Colore e forma:SolidPeso molecolare:415.27CYM50374
CAS:<p>CYM50374 inhibits Sphingosine-1-phosphate receptor 4 (S1P4 ) with an IC50 of µM.</p>Formula:C19H19NO3SPurezza:98.35% - 98.4%Colore e forma:SolidPeso molecolare:341.42GP2-114
CAS:<p>GP2-114 is a catecholamine motility mimetic that produces current-dependent cardiovascular effects.Cost-effective and quality-assured.</p>Formula:C19H24N2O4Purezza:99.32%Colore e forma:SolidPeso molecolare:344.4Liafensine
CAS:<p>Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.</p>Formula:C24H22N4Purezza:99.91%Colore e forma:SolidPeso molecolare:366.46Ancriviroc
CAS:<p>Ancriviroc (SCH-351125) is an orally bioavailable small molecule chemokine receptor CCR5 antagonist.Cost-effective and quality-assured.</p>Formula:C28H37BrN4O3Purezza:99.76% - 99.82%Colore e forma:SolidPeso molecolare:557.52Opigolix
CAS:<p>Opigolix is a Gonadotropin-releasing hormone receptor antagonist.</p>Formula:C25H19F3N4O5SPurezza:98.60% - 98.97%Colore e forma:SolidPeso molecolare:544.5PD 168568 dihydrochloride
CAS:<p>PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).</p>Formula:C22H29Cl2N3OPurezza:99.71%Colore e forma:SolidPeso molecolare:422.39Felcisetrag
CAS:<p>Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.</p>Formula:C25H37N5O3Purezza:99.99%Colore e forma:SolidPeso molecolare:455.59Masilukast
CAS:Masilukast(MCC-847) is an oral leukotriene D4 (LTD4) receptor antagonist for the study of diseases associated with inflammation.Formula:C31H32F3N3O5SPurezza:99.23% - 99.62%Colore e forma:SolidPeso molecolare:615.66Cyamemazine
CAS:<p>Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.</p>Formula:C19H21N3SPurezza:97.01%Colore e forma:SolidPeso molecolare:323.46Amosulalol
CAS:<p>Amosulalol is a combined alpha and beta adrenoceptor antagonist.</p>Formula:C18H24N2O5SPurezza:99.5%Colore e forma:SolidPeso molecolare:380.46Enerisant hydrochloride
CAS:<p>Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteins</p>Formula:C22H31ClN4O3Purezza:99.95%Colore e forma:SolidPeso molecolare:434.96Macimorelin acetate
CAS:<p>Macimorelin acetate (EP-1572) is an oral GHSR agonist for AGHD and CACS research.</p>Formula:C28H34N6O5Colore e forma:SolidPeso molecolare:534.61cis-J-113863
CAS:<p>Cis-J-113863 is a competitive antagonist for the chemokine receptor 1 (CCR1), demonstrating inhibitory concentration 50 (IC50) values of 0.9 nM for human CCR1 receptors and 5.8 nM for mouse CCR1 receptors, respectively [1].</p>Formula:C30H37Cl2IN2O2Colore e forma:SolidPeso molecolare:655.445-HT2C agonist-3
CAS:<p>5-HT2C agonist-3 ((+)-19), a selective 5-HT2C agonist (EC 50: 24 nM, Ki: 78 nM), exhibits antipsychotic-like activity by blocking amphetamine-induced</p>Formula:C19H23ClFNO2Purezza:98%Colore e forma:SolidPeso molecolare:351.84(S)-Bexicaserin
CAS:<p>(S)-Bexcaserin (compound 2) serves as a 5-HT2C receptor agonist, presenting research possibilities in obesity and psychiatric disorders [1].</p>Formula:C15H19F2N3OPurezza:98%Colore e forma:SolidPeso molecolare:295.332-Thio-UTP tetrasodium
CAS:<p>2-Thio-UTP tetrasodium, a potent agonist for P2Y2, P2Y4, and P2Y6 receptors, serves as a crucial compound in cancer research [1].</p>Formula:C9H11N2Na4O14P3SColore e forma:SolidPeso molecolare:588.13
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