Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(939 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.945 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(148 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(407 prodotti)
- Recettore dell'endotelina(76 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(31 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(165 prodotti)
- Proteina Hedgehog/Smoothened(44 prodotti)
- Recettore dell'istamina(358 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(297 prodotti)
- PAFR(11 prodotti)
- PKA(48 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
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Trovati 5352 prodotti di "Proteina G/GPCR"
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Galantide acetate
<p>Galantide acetate, a non-specific galanin receptor antagonist, is a peptide consisting of fragments of galanin and substance P.</p>Formula:C106H155N25O28SPurezza:97.8% - 97.91%Colore e forma:SolidPeso molecolare:2259.58KB-5492 FA
<p>KB-5492 FA is a selective sigma receptor inhibitor with antiulcerogenic effects.CAS 번호128-52-56-8</p>Formula:C24H32N2O8Purezza:98.12%Colore e forma:SolidPeso molecolare:476.52Setmelanotide
CAS:<p>Setmelanotide (BIM-22493) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).</p>Formula:C49H68N18O9S2Purezza:98%Colore e forma:SolidPeso molecolare:1117.31Oxmetidine
CAS:<p>Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular system and is used in the study of duodenal ulcers.</p>Formula:C19H21N5O3SPurezza:99.67%Colore e forma:SolidPeso molecolare:399.47Cetirizine D8 dihydrochloride
CAS:<p>Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.</p>Formula:C21H26Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:433.4Cetirizine Impurity C dihydrochloride
CAS:<p>Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.</p>Formula:C21H27Cl3N2O3Colore e forma:SolidPeso molecolare:461.81Galanin (1-29)(rat, mouse)
CAS:<p>Non-selective galanin agonist; Ki: GAL1-0.98, GAL2-1.48, GAL3-1.47 nM. Anticonvulsant, stops full seizures in rats.</p>Formula:C141H211N43O41Purezza:98%Colore e forma:White Lyophilized PowderPeso molecolare:3164.499FR252384
CAS:<p>FR252384 is an antagonist of the neuropeptide Y-Y5 receptor (IC50: 2.3 nM).</p>Formula:C18H17N3Purezza:98%Colore e forma:SolidPeso molecolare:275.35GLP-1R Agonist DMB
CAS:<p>GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).</p>Formula:C13H15Cl2N3O2SPurezza:99.52%Colore e forma:SolidPeso molecolare:348.25L-770644
CAS:<p>L-770644 is an agonist of B3 adrenergic receptor.</p>Formula:C30H37N7O4SColore e forma:SolidPeso molecolare:591.72Neurokinin A(4-10)
CAS:<p>Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .</p>Formula:C34H54N8O10SPurezza:98%Colore e forma:SolidPeso molecolare:766.91Calcitonin-13C6,15N4 TFA
<p>Calcitonin-13CIC6,15NIC4(salmon) (Salmon calcitonin-13CIC6,15NIC4) TFA is a version of calcitonin(salmon) labeled with carbon-13 and nitrogen-15. This hormone regulates calcium and acts dualistically as an agonist to both amylin and calcitonin receptors, promoting bone formation while inhibiting bone resorption.</p>Formula:C1401C5H240N4315NO48S2·5C2HF3O2Colore e forma:SolidPeso molecolare:4007.93γ-Glu-Abu TFA
<p>Gamma-Glu-AbuTFA is the TFA salt form of Gamma-Glu-Abu. This compound acts as an agonist for the calcium sensing receptor (CaSR), activating CaSR in HEK-293 cells with an EC50 of 0.21 μM.</p>Formula:C11H17F3N2O7Colore e forma:SolidPeso molecolare:346.26MD01-67
CAS:<p>MD01-67 is a macrocyclic compound selectively targeting the neurotensin 2 receptor (NTS2), with a Ki of 2.9 nM. It exhibits analgesic activity and reduces tactile hypersensitivity in rat models of acute, sustained, and chronic inflammatory pain.</p>Formula:C37H58N8O8Colore e forma:SolidPeso molecolare:742.91Pasireotide (diaspartate)
CAS:<p>Pasireotide diaspartate (SOM230) has high agonist activity at sst1/2/3/5, less at sst4; it's antiproliferative and proapoptotic.</p>Formula:C66H80N12O17Colore e forma:SolidPeso molecolare:1313.41BMY-14802
CAS:<p>BMY-14802 (alpha-(4-fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazine butanol) is a selective and orally active sigma-1 antagonist with an IC50 of 112 nM.</p>Formula:C18H22F2N4OPurezza:99.84%Colore e forma:SoildPeso molecolare:348.39[18F]-Labeled L-dopa precursor
CAS:<p>[18F]-Labeled L-dopa precursor is a precursor for synthesis of 18F-labeled L-dopa[1].</p>Formula:C35H36N2O7Colore e forma:SolidPeso molecolare:596.674-Butyl-α-agarofuran
CAS:<p>4-Butyl-alpha-agarofuran, a Gharu-wood derivative, is an anxiolytic, antidepressant, and aids neurological research.</p>Formula:C18H30OColore e forma:SolidPeso molecolare:262.43BAM (8-22) acetate
<p>BAM (8-22) acetate, a proenkephalin A derivative, stimulates MrgprC11, hMrgprX1, and causes scratching in mice.</p>Formula:C93H131N25O25SPurezza:98.85%Colore e forma:SolidPeso molecolare:2031.25Litoxetine HCl
<p>Litoxetine HCl, an SSRI and 5-HT antagonist, treats urinary incontinence and relaxes rat oesophageal muscles without antimuscarinic effects.</p>Formula:C16H20ClNOPurezza:99.56% - 99.75%Colore e forma:SoildPeso molecolare:277.79CB2R/FAAH modulator-3
CAS:<p>CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.</p>Formula:C22H31NO2Purezza:99.81%Colore e forma:SoildPeso molecolare:341.49N-Desmethyl Pimavanserin
CAS:<p>N-Desmethyl Pimavanserin (AC-279) is the active metabolite of Pimavanserin and is used in the treatment of insomnia and other sleep disorders.</p>Formula:C24H32FN3O2Purezza:98.02%Colore e forma:SolidPeso molecolare:413.53MLN-3897 TFA
<p>MLN-3897 TFA is a potent CCR1 antagonist that inhibits the binding of 125I-MIP-1α to THP-1 cell membranes.</p>Formula:C32H32ClF3N2O6Purezza:98.62%Colore e forma:SolidPeso molecolare:633.05Fasitibant chloride hydrochloride
CAS:<p>Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.</p>Formula:C36H50Cl4N6O6SColore e forma:SolidPeso molecolare:836.7AG 045572
CAS:<p>AG 045572 is a potent GnRH receptor antagonist that inhibits the GnRH receptor in humans and rats with Ki values of 6.0 nM and 3.8 nM, respectively.AG 045572 is</p>Formula:C30H37NO5Purezza:99.96%Colore e forma:SolidPeso molecolare:491.62SC 31391
CAS:<p>SC 31391 is a PGE1 analog.</p>Formula:C24H32O6Colore e forma:SolidPeso molecolare:416.51KSK94 FA
<p>KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity.</p>Formula:C26H28N4O3Purezza:97.51%Colore e forma:SoildPeso molecolare:444.53[Des-His1,Glu9]-Glucagon amide
CAS:<p>Glucagon blocker with pA2 of 7.2; no agonist effect. Boosts insulin; prevents glucagon-driven hyperglycemia in rabbits and diabetic rats.</p>Formula:C148H221N41O47SPurezza:98%Colore e forma:SolidPeso molecolare:3358.68CCR6 inhibitor 1
CAS:<p>CCR6 inhibitor 1 selectively blocks CCR6 (0.45 nM in monkeys, 6 nM in humans), aiding in vitro/vivo disease studies.</p>Formula:C24H23F3N4O3SPurezza:99.89%Colore e forma:SolidPeso molecolare:504.52Isoprenaline
CAS:<p>Isoprenaline is a non-selective and orally active β-adrenoceptor agonist.Isoproterenol is a potent peripheral vasodilator and bronchodilator.</p>Formula:C11H17NO3Purezza:99.31%Colore e forma:SolidPeso molecolare:211.26S1R agonist 1
CAS:<p>Compound 6b: Selective S1R agonist, K i = 0.93 nM (S1R), 72 nM (S2R); neuroprotective against ROS, NMDA toxicity.</p>Formula:C20H25NOColore e forma:SolidPeso molecolare:295.42PD-149164
CAS:<p>PD-149164 is an agonist of the CCK-A receptor.</p>Formula:C33H38FN3O5Colore e forma:SolidPeso molecolare:575.67JNJ-5207787
CAS:<p>JNJ-5207787, a blood-brain barrier-crossing Y2 receptor antagonist, is >100x selective against Y1/Y4/Y5 and inhibits human/rat Y2 with pIC50s of 7.0/7.1.</p>Formula:C32H38N4O2Purezza:98%Colore e forma:SolidPeso molecolare:510.67CRL-42872 free base
CAS:<p>CRL-42872 free base is a bioactive chemical.</p>Formula:C22H26N6O6SColore e forma:SolidPeso molecolare:502.54Vapiprost hydrochloride
CAS:<p>Vapiprost hydrochloride is a biochemicla.</p>Formula:C30H40ClNO4Colore e forma:SolidPeso molecolare:514.1SAG dihydrochloride
CAS:<p>SAG dihydrochloride: potent Smo agonist, activates Hedgehog pathway, counters Cyclopamine. EC50=3 nM, Kd=59 nM.</p>Formula:C28H30Cl3N3OSPurezza:>99.99%Colore e forma:SoildPeso molecolare:562.98Vatinoxan
CAS:<p>Vatinoxan is a peripheral α2 adrenoreceptor antagonist.</p>Formula:C20H26N4O4SPurezza:98%Colore e forma:SolidPeso molecolare:418.51CCR4 antagonist 3
CAS:<p>Orally active CCR4 antagonist with piperidinyl-azetidine; IC50: 22 nM (calcium flux), 50 nM (CTX); antitumor effects.</p>Formula:C24H27Cl2N7OColore e forma:SolidPeso molecolare:500.43SC-53116
CAS:<p>SC-53116 HCl can increase the production of serotonin in central nervous system tissues and is a psychoactive agent.</p>Formula:C16H22ClN3O2Colore e forma:SolidPeso molecolare:323.82CCR2 antagonist 1
CAS:<p>CCR2 antagonist 1 is a high-affinity and long-residence-time antagonist of CCR2 (Ki: 2.4 nM).</p>Formula:C28H32BrF3N2OColore e forma:SolidPeso molecolare:549.47Tetrapeptide-1
CAS:<p>Tetrapeptide-1 is a bioactive peptide renowned for its antioxidant properties and has been cited as an ingredient in cosmetics [1].</p>Formula:C20H36N4O6Purezza:98%Colore e forma:SolidPeso molecolare:428.52[D-Pro2] Spantide I TFA
<p>[D-Pro2] Spantide I TFA is an analog of Spantide I, a selective antagonist of the NK1 receptor [1].</p>Formula:C75H108N20O13·xC2HF3O2Purezza:98%Colore e forma:SolidRC-3095
CAS:<p>RC-3095, a selective GRPR antagonist, has been shown to have anti-inflammatory properties in different models of inflammation.</p>Formula:C56H79N15O9Purezza:98%Colore e forma:SolidPeso molecolare:1106.32Men 10208
CAS:<p>Men 10208 is an antagonist of the neurokinin A receptor.</p>Formula:C61H75N15O12Purezza:98%Colore e forma:SolidPeso molecolare:1210.36MRS7925
<p>MRS7925 (Compound 43) serves as a potent antagonist of the 5-HT2B receptor, with an inhibition constant (Ki) of 17 nM, and is utilized in the study of fibrosis</p>Formula:C20H26IN5O3Purezza:98%Colore e forma:SolidPeso molecolare:511.36FGH31
<p>FGH31 (Compound 24), a dopamine D4 agonist, exhibits potent and selective GRK2-dependency with a K i of 1.6 nM and partially activates β-arrestin [1].</p>Formula:C33H36N4O2Purezza:98%Colore e forma:SolidPeso molecolare:520.66Endolide F
<p>Endolide F (Compound 2) is a proline-containing lactone that serves as a moderate antagonist of the arginine vasopressin V1A receptor.</p>Formula:C25H32N4O6Peso molecolare:484.23218GUB03385
<p>GUB03385 is a long-acting PrRP31 analogue and an effective dual agonist for GPR10 (full agonist, EC50: 0.4 nM) and NPFF2R (partial agonist, EC50: 20 nM), with anti-obesity properties.</p>Formula:C198H322N60O52SPeso molecolare:4404.41173CB2R agonist 3
<p>CB2R agonist 3, a potent activator of cannabinoid receptor 2 (CB2R), exhibits an EC50 value of 0.37μM, indicative of its significant role in the immune system [</p>Purezza:98%Colore e forma:Odour SolidMR33317
<p>MR33317 is an inhibitor of acetylcholinesterase with an IC50 value of 41 nM. Additionally, it acts as an agonist for brain 5-HT4 receptors.</p>Formula:C22H28ClN3O2Peso molecolare:401.187Cyclic AC253
<p>Cyclic AC253 is an amylin receptor antagonist with an IC50 of 0.3 μM. It offers neuroprotective effects against Aβ toxicity and mitigates Aβ-induced impairments in hippocampal long-term potentiation. Additionally, Cyclic AC253 is capable of penetrating the blood-brain barrier.</p>Formula:C126H202N42O40S2Peso molecolare:3007.45049S1H
<p>S1H is an analog of human growth hormone (hGH) and acts as an antagonist to the human growth hormone receptor (hGHR). It inhibits the interaction between hGH and hGHR and prevents the phosphorylation of STAT5 in cells treated with hGH.</p>Formula:C94H141N23O27Peso molecolare:2024.03673MCL0129
CAS:<p>MCL0129, a selective and non-peptidergic melanocortin 4 (MC4) receptor antagonist, is a potential treatment for cachexia.</p>Formula:C34H47FN4OPurezza:98%Colore e forma:SolidPeso molecolare:546.76LHRH
CAS:<p>Luteinizing hormone-releasing hormone (LHRH) is a neuropeptide produced in the hypothalamus that plays a pivotal role in regulating reproduction and has</p>Formula:C55H74N16O14Purezza:98%Colore e forma:SolidPeso molecolare:1183.27Cinanserin hydrochloride
CAS:<p>Cinanserin hydrochloride (SQ 10643) is a 5-HT2 receptor blocker (Ki: 41 nM) and SARS-CoV 3C-like protease inhibitor.</p>Formula:C20H25ClN2OSPurezza:99.57%Colore e forma:SolidPeso molecolare:376.94TCMCB07
CAS:<p>TCMCB07, a cyclic nonapeptide, serves as an orally active, brain-penetrant antagonist of the melanocortin receptor 4 (MC4R), with significant implications in</p>Formula:C63H87N15O11Purezza:98%Colore e forma:SolidPeso molecolare:1230.46QWF
CAS:<p>Tripeptide SP antagonist (IC50: 90 μM); blocks SP-MRGPR X2 binding and mast cell degranulation; reduces 48/80-induced scratching in mice.</p>Formula:C38H43N5O8Purezza:98%Colore e forma:SolidPeso molecolare:697.78Ethylnorepinephrine hydrochloride
CAS:<p>Ethylnorepinephrine hydrochloride is a unique bronchodilator.</p>Formula:C10H16ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:233.69Vapreotide diacetate
CAS:<p>Vapreotide diacetate, a synthetic somatostatin analog, blocks NK1R to provide analgesic effects.</p>Formula:C61H78N12O13S2Purezza:98%Colore e forma:SolidPeso molecolare:1251.47L-770644 dihydrochloride
CAS:<p>L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.</p>Formula:C30H38ClN7O4SColore e forma:SolidPeso molecolare:628.19LRGILS-NH2
CAS:<p>LRGILS-NH2, reverse sequence of SLIGRL-NH2, is a control peptide for PAR2, affecting gut transit.</p>Formula:C29H56N10O7Purezza:98%Colore e forma:SolidPeso molecolare:656.82Apelin-12 acetate
<p>Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.</p>Formula:C66H107N21O16SPurezza:98.82%Colore e forma:SolidPeso molecolare:1482.75Oxaprotiline hydrochloride
CAS:<p>Oxaprotiline hydrochloride is an antidepressant.</p>Formula:C20H24ClNOPurezza:98%Colore e forma:SolidPeso molecolare:329.86Neurokinin B acetate(86933-75-7 free base)
<p>Neurokinin B acetate, a tachykinin, interacts with NK1R, NK2R, & NK3R receptors to exert biological effects.</p>Formula:C57H83N13O16S2Purezza:98.53%Colore e forma:SolidPeso molecolare:1270.48JMV-1645
CAS:<p>JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.</p>Formula:C49H69N13O12SPurezza:98%Colore e forma:SolidPeso molecolare:1064.23Azaline
CAS:<p>Azaline is a gonadorelin antagonist.</p>Formula:C74H106ClN23O12Purezza:98%Colore e forma:SolidPeso molecolare:1545.26Ecraprost
CAS:<p>Ecraprost is used as a prodrug of prostaglandin E1.</p>Formula:C28H48O6Colore e forma:SolidPeso molecolare:480.68LEK 8804
CAS:<p>LEK 8804 is a 5-HT(2) receptor antagonist and 5-HT(1A) receptor agonist.</p>Formula:C19H19N3OColore e forma:SolidPeso molecolare:305.37Clopidogrel-related Compound B hydrochloride
CAS:<p>Clopidogrel Related Compound B is a useful organic compound for research related to life sciences.</p>Formula:C16H17Cl2NO2SColore e forma:SolidPeso molecolare:358.28A 76154
CAS:<p>A 76154 is an antagonist of leutenizing hormone releasing hormone (LHRH).</p>Formula:C70H93FN12O12Colore e forma:SolidPeso molecolare:1313.584R 50595
CAS:<p>R 50595 is a selective non-competitive cisapride antagonist.</p>Formula:C30H35Cl2F2N3O3Purezza:98%Colore e forma:SolidPeso molecolare:594.52PSB-22269
<p>PSB-22269 is identified as a GPR17 antagonist with a Ki value of 8.91 nM. It exhibits significant inhibitory effects in cAMP and G protein activation assays. Molecular docking studies indicate that the binding site of PSB-22269 includes positively charged arginine residues and a hydrophobic pocket. PSB-22269 promotes myelin regeneration strategies, offering potential for multiple sclerosis research.</p>Formula:C26H21NO6Colore e forma:SolidPeso molecolare:443.45Galanin-Like Peptide (rat)
CAS:<p>Galanin-Like Peptide (rat), a neuropeptide comprising 60 amino acids, plays a crucial role in regulating feeding, body weight, and energy metabolism [1].</p>Formula:C288H461N87O83SPurezza:98%Colore e forma:SolidPeso molecolare:6502.34A3AR agonist 1
<p>A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effective</p>Formula:C28H34N6O6Purezza:98%Colore e forma:SolidPeso molecolare:550.61Lys-(Des-Arg9,Leu8)-Bradykinin
CAS:<p>Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].</p>Formula:C47H75N13O11Purezza:98%Colore e forma:SolidPeso molecolare:998.18Spns2-IN-1
<p>Spns2-IN-1 is a potent Spns2 inhibitor, effectively impeding Spns2-dependent S1P transport with an IC50 value of 1.4±0.3 μM, crucial for modulating the immune</p>Purezza:98%Colore e forma:Odour SolidHuman growth hormone-releasing factor
CAS:<p>GHRH from the hypothalamus prompts the pituitary to produce/release GH by attaching to the GHRHR.</p>Formula:C215H358N72O66SPurezza:98%Colore e forma:SolidPeso molecolare:5039.65Albenatide
CAS:<p>Albenatide is a modified analog of exendin 4 conjugated to recombinant human albumin.</p>Formula:C26H47N7O9SPurezza:98%Colore e forma:SolidPeso molecolare:633.76Cortistatin-29 (rat) (trifluoroacetate salt)
CAS:<p>Cortistatin-29, similar to somatostatin-28, derives from preprocortistatin and binds to SST receptors 1-5 with varying IC50 values.</p>Formula:C161H240N46O41S2Colore e forma:SolidPeso molecolare:3540.09LY-53857 free base
CAS:<p>LY-53857 free base is a bioactive chemical.</p>Formula:C23H32N2O3Colore e forma:SolidPeso molecolare:384.51[Deamino-Pen1,Val4,D-Arg8]-vasopressin
CAS:<p>[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an antagonist of arginine-vasopressin (AVP).</p>Formula:C48H69N13O11S2Purezza:98%Colore e forma:SolidPeso molecolare:1068.27[Des-Arg9]-Bradykinin
CAS:<p>[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.</p>Formula:C44H61N11O10Purezza:98%Colore e forma:SolidPeso molecolare:904.02Latanoprost lactone diol
CAS:<p>Latanoprost lactone diol, a key intermediate for synthesizing Latanoprost (a prostaglandin F2α analogue), lowers IOP by activating FP receptors.</p>Formula:C18H24O4Purezza:98%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:304.38Misoprostol acid
CAS:<p>Misoprostol acid is an active metabolite of Misoprostol,can be used for non-steroidal anti-inflammatory drug-induced (NSAID) gastric ulcers.</p>Formula:C21H36O5Purezza:98%Colore e forma:SolidPeso molecolare:368.51IRL-3630
CAS:<p>IRL 3460 is an enantiomer.</p>Formula:C31H40N4O6SPurezza:98%Colore e forma:SolidPeso molecolare:596.74Pal-Glu(OSu)-OH
CAS:<p>Pal-Glu(OSu)-OH is a Liraglutide side chain, a GLP-1 agonist for type 2 diabetes study.</p>Formula:C25H42N2O7Colore e forma:SolidPeso molecolare:482.618(D-Arg8)-Inotocin
CAS:<p>'(D-Arg8)-Inotocin is a potent, selective, and competitive antagonist of the vasopressin receptor (V 1a R), exhibiting a binding affinity (K i) of 1.3 nM.</p>Formula:C39H68N14O11S2Purezza:98%Colore e forma:SolidPeso molecolare:973.17MLS1082
CAS:<p>MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.</p>Formula:C24H23N3O2Purezza:99.53%Colore e forma:SolidPeso molecolare:385.46Pancreatic Polypeptide, bovine
CAS:<p>Agonist at Y4 neuropeptide Y receptors.</p>Formula:C186H287N53O56S2Purezza:98%Colore e forma:SolidPeso molecolare:4225.78Prostaglandin K1
CAS:<p>Prostaglandin K1 (compound 46) is a structurally modified prostanoid analog with an EC50 and Ki of 2800 nM for the EP1 receptor.</p>Formula:C20H32O5Colore e forma:SolidPeso molecolare:352.475-HT2A receptor agonist-6
CAS:<p>5-HT2A receptor agonist-6 (compound 47) is a selective agonist of the 5-HT2A receptor with a pEC50 value of 6.58.</p>Formula:C18H19N3O3Colore e forma:SolidPeso molecolare:325.36YM 16638
CAS:<p>YM 16638 is an LT antagonist that can be used to study antigen-induced early and late airway responses in allergic sheep.</p>Formula:C18H22N2O5S3Purezza:99.18%Colore e forma:SolidPeso molecolare:442.574-Hydroxy MPT
CAS:<p>4-Hydroxy MPT (4-OH-MPT) is a serotonin-active compound that acts as an agonist for 5-HT2A and 5-HT2B receptors, with EC50 values of 3.82 nM and 3.4 nM, respectively.</p>Formula:C14H20N2OColore e forma:SolidPeso molecolare:232.32exo-Tetrahydrocannabivarin
CAS:<p>exo-Tetrahydrocannabivarin (Compound 12) is an analog of Δ9,11-THC. It weakly binds to cannabinoid receptors (CB) with an IC50 of 1.4 μM. In mice, exo-Tetrahydrocannabivarin exhibits activity related to both motor function and analgesia.</p>Formula:C19H26O2Colore e forma:SolidPeso molecolare:286.41Afubiata
CAS:<p>ADB-FUBIATA is a synthetic cannabinoid studied for its metabolic profile, along with AFUBIATA, CH-FUBIATA, and CH-PIATA. This in vitro analysis by Watanabe S, et al., examines these compounds, as published in "Arch Toxicol," 2023 Dec;97(12):3085-3094.</p>Formula:C27H29FN2OColore e forma:SolidPeso molecolare:416.5317-phenyl trinor Prostaglandin F2α cyclopropyl amide
CAS:<p>17-phenyl trinor Prostaglandin F2α cyclopropyl amide (17-phenyl trinor PGF2α cyclopropyl amide) is a novel analog of 17-phenyl trinor PGF2α ethyl amide.</p>Formula:C26H37NO4Colore e forma:SolidPeso molecolare:427.585SHU 9119
CAS:<p>SHU 9119 is a potent antagonist for human MC3R/MC4R and partial agonist for MC5R with IC50 values of 0.23, 0.06, 0.09 nM.</p>Formula:C54H71N15O9Purezza:98%Colore e forma:SolidPeso molecolare:1074.258PSB-SB-1203
CAS:<p>PSB-SB-1203 (Compound 25b) is a dual CB1/CB2 ligand that blocks the CB1 receptor and activates the CB2 receptor with a CB1 Ki of 0.244 μM, a CB2 Ki of 0.210 μM, and an EC50 of 0.054 μM. It shows potential for research in obesity and cancer.</p>Formula:C25H30O4Colore e forma:SolidPeso molecolare:394.5Sulfatroxazole
CAS:<p>Sulfatroxazole (Isosulfafurazole) (compound 12) is a selective antagonist of the ETA receptor with an IC50 of 0.26 μM.</p>Formula:C11H13N3O3SColore e forma:SolidPeso molecolare:267.3Vazegepant
CAS:<p>Vazegepant is an intranasal CGRP receptor antagonist utilized for conducting acute migraine research.</p>Formula:C36H46N8O3Purezza:98.61%Colore e forma:SolidPeso molecolare:638.80Neuropeptide S(Rat)
CAS:<p>Potent endogenous neuropeptide S receptor (NSPR) agonist (EC50 = 3.2 nM).</p>Formula:C95H160N34O27Purezza:98%Colore e forma:SolidPeso molecolare:2210.52CACPD2011a-0001278239
CAS:<p>CACPD2011a-0001278239 is a β2AR hybrid agonist with high affinity binding to both the wild-type and T164I β2AR variants. It exhibits neither cytotoxicity nor mutagenicity, making it suitable for asthma research.</p>Formula:C21H22N4O4Colore e forma:SolidPeso molecolare:394.42Cannabidivarinic acid
CAS:<p>Cannabidivarinic acid (CBDVA), the carboxylic acid precursor to cannabidivarin (CBDV), is a non-psychoactive cannabinoid found in Cannabis and known for its anti-inflammatory properties.</p>Formula:C20H26O4Colore e forma:SolidPeso molecolare:330.42RFRP-3(human)
CAS:<p>NPFF1 receptor agonist, IC50 0.7 nM, blocks cAMP by forskolin. A GnIH homolog, it inhibits GnRH neuron activity.</p>Formula:C45H72N14O10Purezza:98%Colore e forma:SolidPeso molecolare:969.15Esmolol acid hydrochloride
CAS:<p>Esmolol acid (ASL-8123) hydrochloride is a mild antagonist of β-adrenergic receptors. It inhibits the heart rate and diastolic pressure responses induced by Isoproterenol in a dose-dependent manner and is applicable for renal failure research.</p>Formula:C15H24ClNO4Colore e forma:SolidPeso molecolare:317.81Semaglutide TFA
<p>Semaglutide TFA is a glucagon-like peptide-1 congener that induces weight loss, lowers blood glucose levels and reduces cardiovascular risk in diabetic patients</p>Formula:C189H290F3N45O61Purezza:99.69%Colore e forma:SolidPeso molecolare:4225.6482ATMW-2
<p>ATMW-2 is an antagonist engineered using NeuralGenThesis (NGT) technology, specifically targeting the melanocortin 2 receptor (MC2R).</p>Formula:C27H29ClN2O4Colore e forma:SolidPeso molecolare:480.98Moperone
CAS:<p>Moperone (R 1658) is an antagonist of both the D2 dopamine receptor (D2 dopamine receptor) and the D3 dopamine receptor (D3 dopamine receptor), with IC50 values for each of 1.0 nM.</p>Formula:C22H26FNO2Colore e forma:SolidPeso molecolare:355.457-Methyl DMT
CAS:<p>7-Methyl DMT (7-TMT) acts as a 5-HT2 receptor agonist. Structurally, it is a tryptamine derivative and serves as an analytical reference for the psychoactive substance DOM. It is also applicable in research related to neurological disorders.</p>Formula:C13H18N2Colore e forma:SolidPeso molecolare:202.3Stressin I
<p>Potent CRF1 agonist; Ki: 1.5 nM (CRF1), 224 nM (CRF2). Boosts ACTH, enhances stool frequency after i.p. administration.</p>Formula:C203H337N57O56Purezza:98%Colore e forma:SolidPeso molecolare:4472.244-Iodoamphetamine hydrochloride
CAS:<p>4-Iodoamphetamine (p-Iodoamphetamine) hydrochloride is a halogenated phenethylamine characterized by the presence of an iodine atom at the para position of the phenyl group. It selectively induces serotonin release and inhibits reuptake in rat brain synaptosomes.</p>Formula:C9H13ClINColore e forma:SolidPeso molecolare:297.56Δ8-THC methyl ether
CAS:<p>Δ8-THC methyl ether (compound 3) demonstrates a strong docking score of -10.167 kcal/mol for the CB2 receptor. Additionally, Δ8-THC methyl ether exhibits antinociceptive activity in mice.</p>Formula:C22H32O2Colore e forma:SolidPeso molecolare:328.494-hydroxy DiPT hydrochloride
CAS:<p>4-hydroxy DiPT (hydrochloride) is a 5-HT2A agonist that can induce head twitch response (HTR) in mice, indicating its hallucinogenic potential. This compound holds promise for research into hallucinogens.</p>Formula:C16H25ClN2OColore e forma:SolidPeso molecolare:296.84QWF acetate
<p>QWF acetate is a Substance P antagonist peptide that specifically inhibits the binding to its receptor, NK1, and inhibits the activation of MRGPRX2.</p>Formula:C40H47N5O10Purezza:96.65%Colore e forma:SolidPeso molecolare:757.84Pobilukast
CAS:<p>Pobilukast (SKF 104353) is a cysteinyl leukotriene receptor antagonist that can be used to study limiting myocardial injury in MI/R rats.</p>Formula:C26H34O5SPurezza:99.65% - 99.84%Colore e forma:SolidPeso molecolare:458.61Prolactin Releasing Peptide (1-31), human
CAS:<p>Human Prolactin Releasing Peptide (1-31) is a potent GPR10 agonist; Ki values are 1.03 nM (human) and 0.33 nM (rat).</p>Formula:C160H252N56O42SPurezza:98%Colore e forma:SolidPeso molecolare:3664.15Ceruletide Ammonium Salt
<p>Ceruletide Ammonium Salt is a decapeptide, originating from the skin of tropical frogs, which is a potent cholecystokinin receptor agonist and a safe and</p>Formula:C58H77N14O21S2Purezza:98.47% - 98.54%Colore e forma:SoildPeso molecolare:1370.44GR 82334
CAS:<p>Tachykinin NK1 receptor antagonist.</p>Formula:C69H91N15O16Purezza:98%Colore e forma:SolidPeso molecolare:1386.57Quinelorane
CAS:<p>Quinelorane is dextrorotary isomer.</p>Formula:C14H22N4Colore e forma:SolidPeso molecolare:246.3516-phenoxy tetranor Prostaglandin F2α isopropyl ester
CAS:<p>Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor.</p>Formula:C25H36O6Colore e forma:SolidPeso molecolare:432.557RVD-Hpα
CAS:<p>N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.</p>Formula:C65H105N19O17Purezza:98%Colore e forma:SolidPeso molecolare:1424.66NXT-10796
<p>NXT-10796 is an orally active, intestinally restricted agonist of the EP4 receptor [1].</p>Formula:C23H31N3O6Purezza:98%Colore e forma:SolidPeso molecolare:445.514-Methylhistamine
CAS:<p>4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for research into immune-related diseases, including cancer and</p>Formula:C6H11N3Purezza:98%Colore e forma:SolidPeso molecolare:125.17Conopeptide rho-TIA
CAS:<p>Conopeptide rho-TIA, a peptide from Conus tulipa venom, acts as a selective, noncompetitive inhibitor at the human α1B-Adrenergic Receptor and as a competitive</p>Formula:C105H160N36O21S4Purezza:98%Colore e forma:SolidPeso molecolare:2390.88SphK1&2-IN-1
CAS:<p>SphK1&2-IN-1 is a sphingosine kinase inhibitor with anti-inflammatory, antitumor and hemostatic effects.</p>Formula:C14H14N2O3SPurezza:99.59%Colore e forma:SolidPeso molecolare:290.34Atrial natriuretic peptide (3-28) (human)
CAS:<p>Atrial natriuretic peptide (3-28) (human) (ANP (3-28) (human)), a peptide hormone produced by the atrial myocardium, plays a critical role in the regulation of</p>Formula:C118H187N43O36S3Purezza:98%Colore e forma:SolidPeso molecolare:2880.21ACTH (7-38) (human)
CAS:<p>ACTH (7-38) (human) is a fragment (7-38) of the full human adrenocorticotropic hormone (ACTH (1-39)), also referred to as corticotropin inhibitory peptide (CIP</p>Formula:C167H257N47O46Purezza:98%Colore e forma:SolidPeso molecolare:3659.11FLLRN
CAS:<p>FLLRN is a biologically active peptide serving as a PAR1-specific antagonist.</p>Formula:C31H51N9O7Colore e forma:SolidPeso molecolare:661.79Parstatin(human) TFA
<p>Parstatin(human) TFA, a cell-penetrating PAR-1 thrombin receptor agonist peptide, effectively inhibits angiogenesis, as indicated by studies [1] [2].</p>Formula:C193H331F3N64O55S3Colore e forma:SolidPeso molecolare:4581.28SFNGGP-NH2
CAS:SFNGGP-NH2 is a biologically active peptide that interacts with Protease-Activated Receptor 3 (PAR-3), a high-affinity thrombin receptor.Formula:C25H36N8O8Colore e forma:SolidPeso molecolare:576.617-trifluoromethylphenyl-13,14-dihydro trinor Prostaglandin F2α
CAS:<p>A number of 17-phenyl trinor prostaglandin F2α(17-phenyl trinor PGF2α) derivatives have been approved for the treatment of glaucoma.1,2,3Of these, the ones</p>Formula:C24H33F3O5Colore e forma:SolidPeso molecolare:458.518Dolcanatide
CAS:<p>Dolcanatide: oral GC-C agonist with laxative, pain-relief, and anti-inflammatory properties for IBD research.</p>Formula:C65H104N18O26S4Colore e forma:SolidPeso molecolare:1681.89PZ-1922
<p>PZ-1922 (Compound 16), able to cross the blood-brain barrier, is a dual antagonist for 5-HT6R and 5-HT3R with K i values of 17 nM and 0.45 nM, respectively.</p>Purezza:98%Colore e forma:Odour SolidTRAP-5 amide
CAS:<p>TRAP-5 amide is a peptide agonist for protease-activated receptor 1 (PAR 1) [1].</p>Formula:C30H51N9O6Colore e forma:SolidPeso molecolare:633.78Levocarnitine propionate hydrochloride
CAS:<p>Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.</p>Formula:C10H20ClNO4Purezza:90% - 99.77%Colore e forma:SolidPeso molecolare:253.72TGR5 agonist 1
<p>Compound 18 (TGR5 agonist 1) is a potent agonist of TGR5, exhibiting an EC50 value of 0.31 µM [1].</p>Formula:C28H48NNaO6SColore e forma:SolidPeso molecolare:549.74Olcegepant hydrochloride
CAS:<p>Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a selective calcitonin gene-related peptide 1 (CGRP1) receptor antagonist.</p>Formula:C38H48Br2ClN9O5Purezza:99.69%Colore e forma:SolidPeso molecolare:906.11LysoPalloT-NH-amide-C3-ph-m-O-C11
CAS:<p>LysoPalloT-NH-amide-C3-ph-m-O-C11 is an agonist of the GPR174 receptor with an EC50 value of 34 nM.</p>Formula:C27H47N2O9PColore e forma:SolidPeso molecolare:574.645-trans Latanoprost (free acid)
CAS:<p>Latanoprost, a prodrug eye drop, turns into active acid inside the body and treats high eye pressure. Its trans isomer also likely reduces eye pressure.</p>Formula:C23H34O5Colore e forma:SolidPeso molecolare:390.525-methoxy-α-Ethyltryptamine
CAS:<p>5-Methoxy-alpha-ethyltryptamine is a psychoactive substance that can cause various effects. It belongs to the tryptamine chemical class and can be used for various psychoactive and stimulant effects. </p>Formula:C13H18N2OPurezza:98.25%Colore e forma:SolidPeso molecolare:218.29ent-Prostaglandin E2
CAS:<p>Enzymatic PGE2 is optically pure; radical peroxidation makes it racemic. In oxidative stress, rac-PGE2 forms via 15-E2t-isoprostane.</p>Formula:C20H32O5Colore e forma:SolidPeso molecolare:352.471Nα-Methylhistamine FA
<p>Nα-Methylhistamine FA is a histamine H3 receptor agonist</p>Formula:C7H13N3O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:171.2[Ala11,D-Leu15]-Orexin B acetate
<p>[Ala11,D-Leu15]-Orexin B acetate is a selective agonist of orexin-2 receptor (OX2) with an EC50 of 0.13 nM, showing 400-fold selectivity over OX1 (52 nM).</p>Formula:C122H210N44O37SPurezza:98.18%Colore e forma:SolidPeso molecolare:2917.31Tizanidine
CAS:<p>Tizanidine, an α2-adrenergic receptor agonist, suppresses the release of neurotransmitters from central nervous system (CNS) noradrenergic neurons.</p>Formula:C9H8ClN5SPurezza:99.11%Colore e forma:White SolidPeso molecolare:253.71Femoxetine
CAS:<p>Femoxetine: antidepressant, enhances morphine, inhibits MAO-A/B, boosts mice's exercise capacity.</p>Formula:C20H25NO2Purezza:99.1% - 99.35%Colore e forma:SolidPeso molecolare:311.42Substance P(1-7)
CAS:<p>Substance P(1-7) is a bioactive metabolite of tachykinin SP with anti-inflammatory and analgesic properties.</p>Formula:C41H65N13O10Purezza:98%Colore e forma:SolidPeso molecolare:900.04TAK-448 acetate
CAS:<p>TAK-448 acetate (MVT-602 acetate) is a KISS1R agonist, a synthetic peptide similar to kisspeptin.</p>Formula:C60H84N16O16Purezza:99.88%Colore e forma:SolidPeso molecolare:1285.41PACAP-38 (31-38), human, mouse, rat acetate
<p>PACAP-38 (31-38) acetate stimulates PAC1 receptor and boosts NPY and catecholamine in sympathetic neurons.</p>Formula:C49H87N17O13Purezza:99.92%Colore e forma:SolidPeso molecolare:1122.32PACAP-related Peptide (human) (trifluoroacetate salt)
<p>Endogenous 29-amino acid PRP belongs to secretin/glucagon family, found in pancreas, adrenal glands, and some VIP tumors; secreted by CHO-K1 cells.</p>Colore e forma:LiquidNeuropeptide Y 13-36 (porcine)
CAS:<p>Neuropeptide Y 13-36 (porcine) is a selective neuropeptide Y2 receptor agonist.</p>Formula:C135H209N41O36Colore e forma:SolidPeso molecolare:2982.408GLP-1 receptor agonist 4
CAS:<p>GLP-1 receptor agonist 4 targets GLP-1R, EC50 64.5 nM, potential diabetes treatment research.</p>Formula:C51H44Cl2N4O6Purezza:98%Colore e forma:SolidPeso molecolare:879.82mPGES-1/sEH-IN-1
<p>mPGES-1/sEH-IN-1 (compound 1f) is an sEH inhibitor with an IC50 value of 5 μM. It also exhibits antitumor activity by inhibiting mPGES-1, with an IC50 value of 25 µM.</p>Formula:C20H16F3N3O2Colore e forma:SolidPeso molecolare:387.355GSK-3050002
<p>GSK-3050002 (HGS-1035) is a humanized IgG1 antibody that targets and binds to CCL20. It holds potential for inflammation research. For isotype control, refer to Human IgG1 kappa, Isotype Control.</p>Colore e forma:Odour LiquidAmylin (1-37), human acetate
<p>Amylin (1-37), human acetate, a peptide hormone containing 37 amino acids secreted by the pancreas in conjunction with insulin, inhibits glucagon secretion.</p>Purezza:96.21%Colore e forma:Odour SolidGLP-1R agonist 4
CAS:<p>GLP-1R agonist 4, potentially for diabetes research, is a potent GLP-1R stimulator linked to hypoglycemia.</p>Formula:C32H30ClF2N3O5Colore e forma:SolidPeso molecolare:610.05Upacicalcet HCl
<p>Upacicalcet HCl, a calcium mimetic, reduces blood PTH by targeting parathyroid receptors; treats secondary hyperparathyroidism.</p>Formula:C11H15Cl2N3O6SPurezza:98.56%Colore e forma:SoildPeso molecolare:388.22Lintitript
CAS:<p>Lintitript (SR 27897) is a selective antagonist of CCK1 with EC50s of 6 nM and 200 nM for CCK1 and CCK2. The Ki value is 0.2 nM for CCK1.</p>Formula:C20H14ClN3O3SPurezza:99.28%Colore e forma:SolidPeso molecolare:411.86[Gln8]-C517 (LH-RH), chicken
CAS:[Gln8] LH-RH: Avian hypothalamic peptide; prompts anterior pituitary to release gonadotropins, controlling reproduction.Formula:C54H71N15O14Purezza:98%Colore e forma:SolidPeso molecolare:1154.23Onvitrelin ucalontide
CAS:Onvitrelin ucalontide is a LHRH analogue with anticancer effect; halts breast, ovarian, and prostate tumors in mice.Formula:C163H243N43O32Peso molecolare:3316.94PF-232798
CAS:<p>PF-232798 is a second generation oral CCR5 antagonist with potent broad-spectrum anti-HIV-1 activity.</p>Formula:C29H40FN5O2Colore e forma:SolidPeso molecolare:509.66(Des-Bromo)-Neuropeptide B (1-23) (human)
CAS:'(Des-Bromo)-Neuropeptide B (1-23) (human)' is an agonist for orphan G-protein-coupled receptors, exhibiting a K i of 1.2 nM for GPR7 (NPBW1) and 341 nM forFormula:C107H162N30O30Peso molecolare:2348.61Semaglutide, FITC labeled
Semaglutide (FITC-labeled Semaglutide) is a long-acting analog of human glucagon-like peptide-1, functioning as an agonist of the GLP-1 receptor. It shows potential for research related to type 2 diabetes.Formula:C209H304N46O63SPeso molecolare:4498.17191Suntinorexton
CAS:<p>Suntinorexton (TAK 861) is an orexin type 2 receptor (OX2R) agonist used in the study of neurologic disorders.</p>Formula:C23H28F2N2O4SPurezza:99.89%Colore e forma:SolidPeso molecolare:466.54ACTH (34-39)
CAS:ACTH (34-39) is an adrenocorticotropic hormone fragment.Formula:C37H50N6O9Purezza:98%Colore e forma:SolidPeso molecolare:722.831-Octadecyl Lysophosphatidic Acid
CAS:<p>1-Octadecyl LPA, an LPA analog with stearic acid at sn-1, has strong platelet aggregation (EC50=9 nM) via G protein receptors.</p>Formula:C21H45O6PColore e forma:SolidPeso molecolare:424.559Vilanterol
CAS:<p>Vilanterol is a selective long-acting beta2-adrenergic agonist (LABA) used in the treatment of COPD and asthma.</p>Formula:C24H33Cl2NO5Purezza:97.47% - 99.46%Colore e forma:SolidPeso molecolare:486.43Neuronostatin-13 (human)
CAS:<p>Neuronostatin-13: human-conserved, 13-amino-acid peptide with amidated C-terminus.</p>Formula:C64H110N20O16Purezza:98%Colore e forma:SolidPeso molecolare:1415.68PG106 TFA
<p>PG106 TFA is a potent hMC3 antagonist (IC50=210 nM), inactive at hMC4 (EC50=9900 nM) and hMC5 receptors.</p>Formula:C53H70F3N13O11Colore e forma:SolidPeso molecolare:1122.2GHRF, porcine
CAS:<p>GHRF, porcine, a growth hormone releasing factor (GHRF) peptide (porcine), binds to the growth hormone secretagogue receptor (GHSR), thereby inducing the</p>Formula:C219H365N73O66SColore e forma:SolidPeso molecolare:5108.76α-Helical CRF(9-41) TFA
<p>α-Helical CRF(9-41) TFA acts as a competitive antagonist for the CRF2 receptor, possessing a binding constant (K B) of approximately 100 nM.</p>Formula:C168H275F3N46O55S2Colore e forma:SolidPeso molecolare:3940.42Corazonin
CAS:<p>Corazonin, a neuropeptide in insects, regulates caste identity and behavior, mainly in workers/foragers.</p>Formula:C62H83N17O19Colore e forma:SolidPeso molecolare:1370.42dCNP
<p>dCNP binds to NPR-B/C receptors (NPR-B/C receptor), initiating the cGMP signaling pathway and regulating vascular function. It exhibits anti-hypoxic effects by downregulating hypoxia-related genes such as HIF1α and HIF2α. Additionally, dCNP inhibits tumor stroma induction, demonstrating antifibrotic properties. It also enhances immune response by upregulating CTL, NK cells, and conventional type 1 dendritic cells in tumors.</p>Formula:C141H248N38O36S3Colore e forma:SolidPeso molecolare:3147.91Utreglutide
CAS:<p>Utreglutide is a potent glucagon-like peptide 1 (GLP-1) receptor agonit [1] .</p>Formula:C191H298N46O58Colore e forma:SolidPeso molecolare:4166.67Substance P (4-11)
CAS:Substance P (4-11), a C-terminal fragment of Substance P, acts as a highly selective agonist for NK1 receptors, demonstrating specificity in its interaction.Formula:C46H67N11O10SColore e forma:SolidPeso molecolare:966.16MLGFFQQPKPR-NH2
CAS:<p>MLGFFQQPKPR-NH2 is a reversed Substance P peptide. Substance P is a neuropeptide [1] .</p>Formula:C63H98N18O13SColore e forma:SolidPeso molecolare:1347.63Neuropeptide W-30 (rat)
CAS:<p>Neuropeptide W-30 (rat) acts as a crucial stress mediator within the central nervous system, influencing the hypothalamus-pituitary-adrenal (HPA) axis and sympathetic outflow. It serves as an endogenous ligand for the two related orphan G-protein-coupled receptors (GPCRs), GPR7 and GPR8. NPW-30 binds and activates both GPR7 and GPR8 at comparable effective doses [1] [2] [3].</p>Formula:C165H249N49O38SColore e forma:SolidPeso molecolare:3559.11Selepressin acetate
<p>Selepressin acetate is a useful organic compound for research related to life sciences and the catalog number is T73654.</p>Formula:C48H77N13O13S2Colore e forma:SolidPeso molecolare:1108.33[Ala2] Endothelin-3, human
CAS:<p>[Ala2] Endothelin-3, a linear ET-3 analog with Ala replacing Cys, stimulates endothelial cell migration.</p>Formula:C120H166N26O32S4Colore e forma:SolidPeso molecolare:2613.02Dotanoc
CAS:<p>Dotanoc is a ligand to make gallium Ga 68-DOTANOC, which is a gallium Ga 68-radiolabeled analog of somatostatin.</p>Formula:C69H94N14O17S2Colore e forma:SolidPeso molecolare:1455.71Gastrin I, rat
CAS:<p>Gastrin I, rat is a peptide hormone that effectively stimulates gastric acid secretion.</p>Formula:C94H128N22O31S2Colore e forma:SolidPeso molecolare:2126.3Neuropeptide Y (3-36) (porcine)
CAS:<p>Neuropeptide Y (3-36) (porcine) is a potent, selective agonist at NPY Y2 receptors, increasing feeding in rats.</p>Formula:C176H271N53O54Colore e forma:SolidPeso molecolare:3993.36Kisspeptin-54(human) TFA
<p>Endogenous kisspeptin-54(human) TFA targets KISS1/GPR54 receptors; Ki: 1.81 nM (rat), 1.45 nM (human); inhibits metastasis, boosts gonadotropin.</p>Formula:C258H401N79O78·C2HF3O2Colore e forma:SolidPeso molecolare:5971.45Cyclic SSTR agonist octreotide
<p>Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .</p>Formula:C53H71N11O14S2Colore e forma:SolidPeso molecolare:1150.33[Asu1,6-Arg8]Vasopressin
CAS:<p>[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.</p>Formula:C48H68N14O12Colore e forma:SolidPeso molecolare:1033.14(2R,2R)-PF-07258669
CAS:<p>(2R,2R)-PF-07258669' is an antagonist for the MC4R (melanocortin 4 receptor), primarily studied for its role in regulating appetite and energy expenditure.</p>Formula:C25H27FN6O2Colore e forma:SolidPeso molecolare:462.52Melanostatin, frog
CAS:<p>Melanostatin, frog, is an inhibitor of α-melanocyte-stimulating hormone (α-MSH) release, with an IC50 of 60 nM [1] [2].</p>Formula:C189H285N53O57SColore e forma:SolidPeso molecolare:4243.67α-CGRP(human) TFA
<p>α-CGRP(human) TFA is a 37-amino acid regulatory neuropeptide that is extensively located within the central and peripheral nervous system, functioning as a</p>Formula:C165H268F3N51O51S2Colore e forma:SolidPeso molecolare:3903.33Neuropeptide Y (3-36) (human, rat)
CAS:<p>Neuropeptide Y (3-36) is a Y2 receptor agonist that limits norepinephrine release, produced by DPP4 from NPY.</p>Formula:C175H269N53O54SColore e forma:SolidPeso molecolare:4011.5[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH
CAS:<p>[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH is a synthetic LHRH analog and a GnRH receptor antagonist.</p>Formula:C67H84N16O13Colore e forma:SolidPeso molecolare:1321.48Cenderitide
CAS:<p>Cenderitide fuses CNP with DNP, stimulates pGC-A/B, ups cGMP, curbs aldosterone, and aids GFR, not affecting BP—used in heart failure studies.</p>Formula:C158H263N49O50S3Colore e forma:SolidPeso molecolare:3745.27Chemerin-9, Mouse
CAS:<p>Chemokine-like receptor 1 (CMKLR1) agonist (EC50 = 42 nM). Corresponds to C-terminal of full length mouse Chemerin, amino acids 148 - 156.</p>Formula:C51H68N10O12Colore e forma:SolidPeso molecolare:1013.163Urocortin III (human)
CAS:<p>Urocortin III, a human peptide, binds CRF-R2, affecting insulin via somatostatin feedback with K i values 13.5-100+ nM.</p>Formula:C185H307N53O50S2Colore e forma:SolidPeso molecolare:4137.93Kadsurenin B
CAS:<p>Kadsurenin B, a platelet-activating factor (PAF) antagonist, exhibits neuroprotective properties and has a broad spectrum of pharmacological research</p>Formula:C20H22O5Colore e forma:SolidPeso molecolare:342.39(Phe2,Orn8)-Oxytocin
CAS:<p>(Phe2,Orn8)-Oxytocin: Selective V1 agonist, induces rabbit epididymis contractility, EC50=280 nM.</p>Formula:C42H65N13O11S2Colore e forma:SolidPeso molecolare:992.18AC 187 TFA
<p>AC 187 TFA, a potent and orally active amylin receptor antagonist, exhibits an IC50 of 0.48 nM and a Ki of 0.275 nM.</p>Formula:C129H206F3N37O42Colore e forma:SolidPeso molecolare:3004.27ORG 2766
CAS:<p>ORG 2766 is an ACTH 4-9 (H-Met(O)-Glu-His-Phe-D-Lys-Phe-OH) analog and neurotrophic peptide.</p>Formula:C40H55N9O11SColore e forma:SolidPeso molecolare:869.99Kisspeptin-10, rat TFA
<p>Kisspeptin-10, a rat TFA, constricts blood vessels, inhibits vessel growth, and counters Methotrexate reproductive toxicity.</p>Formula:C65H84F3N17O17Colore e forma:SolidPeso molecolare:1432.46Guanylin(human) TFA
<p>Guanylin (human) TFA, a 15-amino acid peptide, activates intestinal guanylate cyclase, regulating electrolyte and water transport via cGMP.</p>Colore e forma:LiquidZebrafish Kisspeptin-1
CAS:<p>Zebrafish Kisspeptin-1 is the core sequence of the neuropeptide kisspeptin-1, which plays a crucial role in regulating the release of gonadotropin-releasing hormone (GnRH) and modulating the reproductive system.</p>Formula:C58H84N16O15Colore e forma:SolidPeso molecolare:1245.39Biotin-NeurokininA
<p>Biotin-NeurokininA: biotinylated peptide, NK-2 receptor agonist, key in human airway and gut function.</p>Formula:C60H94N16O16S2Colore e forma:SolidPeso molecolare:1359.61
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