Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(942 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.949 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(149 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(410 prodotti)
- Recettore dell'endotelina(75 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(32 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(166 prodotti)
- Proteina Hedgehog/Smoothened(45 prodotti)
- Recettore dell'istamina(359 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(298 prodotti)
- PAFR(11 prodotti)
- PKA(49 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
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Trovati 5378 prodotti di "Proteina G/GPCR"
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BAM(8-22) TFA
<p>BAM(8-22) TFA activates Mrgprs, induces mouse scratching, and is a proenkephalin A derivative.</p>Formula:C93H128F3N25O25SColore e forma:SolidPeso molecolare:2085.22CART(55-102)(rat) TFA
<p>Rat CART(55-102) TFA suppresses appetite, links to leptin/neuropeptide Y, and may induce anxiety/stress.</p>Formula:C228H368F3N65O67S7Colore e forma:SolidPeso molecolare:5373.2(R)-Zevaquenabant
<p>(R)-Zevaquenabant ((R)-MRI-1867) is the enantiomer of Zevaquenabant. Zevaquenabant ((S)-MRI-1867) is a peripherally restricted, orally bioavailable dual antagonist of the cannabinoid CB1 receptor and inducible nitric oxide synthase (iNOS). It is beneficial in improving chronic kidney disease (CKD) caused by obesity.</p>Colore e forma:Odour SolidCGRP antagonist 6
<p>CGRP Antagonist 6 (Compound 23) is a potent CGRP receptor antagonist (Ki: 0.84 nM). It is utilized in the study of migraines.</p>Colore e forma:Odour SolidTGR5 agonist 1
<p>Compound 18 (TGR5 agonist 1) is a potent agonist of TGR5, exhibiting an EC50 value of 0.31 µM [1].</p>Formula:C28H48NNaO6SColore e forma:SolidPeso molecolare:549.74Heterobivalent ligand-1
<p>Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.</p>Formula:C86H115FN16O21Colore e forma:SolidPeso molecolare:1727.93Linzagolix choline
CAS:<p>Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.</p>Formula:C27H28F3N3O8SPurezza:99.64%Colore e forma:SolidPeso molecolare:611.598-iso Prostaglandin E1
CAS:<p>8-iso Prostaglandin E1 causes spasm in the pulmonary veins of dogs and also acts as a vasodilator.</p>Formula:C20H34O5Colore e forma:Light Yellow Crystalline SolidPeso molecolare:354.48Benzomalvin B
CAS:<p>Benzomalvin B, a metabolite from Penicillium, blocks 24% NK1 receptor binding at 100 μg/ml.</p>Formula:C24H17N3O2Colore e forma:SolidPeso molecolare:379.419Cetirizine methyl ester
CAS:<p>Cetirizine methyl ester is a Cetirizine impurity, a long-acting, oral H1-antihistamine and hydroxyzine metabolite.</p>Formula:C22H27ClN2O3Colore e forma:SolidPeso molecolare:402.91CCK Octapeptide, non-sulfated acetate
<p>CCK Octapeptide, non-sulfated acetate is a synthetic desulfated peptide of cholecystokinin.</p>Formula:C51H66N10O15S2Purezza:98.9700%Colore e forma:SolidPeso molecolare:1123.26α-Helical CRF(9-41)
CAS:<p>Corticotropin-releasing factor receptor antagonist (Ki values are 17, 5 and 0.97 at human CRF1, rat CRF2α and mouse CRF2β receptors respectively).</p>Formula:C166H274N46O53S2Purezza:98%Colore e forma:SolidPeso molecolare:3827GRPP (human)
CAS:<p>GRPP (human), a 30-amino-acid peptide derived from Gcg, modestly elevates plasma insulin levels while reducing plasma glucagon concentrations.</p>Formula:C136H215N41O58SColore e forma:SolidPeso molecolare:3384.47NPS ALX Compound 4a hydrochloride(1:1)
<p>NPS ALX Compound 4a hydrochloride(1:1) is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with an IC50 of 7.2 nM and a Ki of 0.2 nM.</p>Formula:C25H26ClN3O2SPurezza:99.84%Colore e forma:SoildPeso molecolare:468.01Ro 25-1553
CAS:<p>Ro 25-1553 is a 31-amino acid analog of vasoactive intestinal peptide (VIP) that functions as an agonist for the VIP2 receptor (VPAC2 receptor). In guinea pig models, Ro 25-1553 exhibits bronchodilator effects on tracheal smooth muscle contraction induced by neural stimuli or Carbachol.</p>Formula:C160H258N46O46Colore e forma:SolidPeso molecolare:3562.04MM 07
CAS:<p>Biased agonist for apelin/G protein pathway, enhances eNOS and cell growth, reduces apoptosis, improves heart function, and dilates vessels.</p>Formula:C67H106N22O14S3Purezza:98%Colore e forma:SolidPeso molecolare:1539.9Galanin (1-30), human
CAS:Galanin (1-30), human is a neuropeptide agonist for GalR1/R2 receptors with 1 nM affinity, influencing endocrine, metabolism, and neurotransmission.Formula:C139H210N42O43Purezza:98%Colore e forma:SolidPeso molecolare:3157.46Lanepitant
CAS:<p>Lanepitant (LY303870) is a non-peptide neurokinin-1 (NK-1) antagonist with analgesic activity for the prevention of migraine.</p>Formula:C33H45N5O3Purezza:97.71%Colore e forma:SolidPeso molecolare:559.74LH-RH (7-10)
CAS:LH-RH (7-10), a tetrapeptide, is a key LHRH degradation product found in macrophages and pneumocytes.Formula:C19H36N8O4Colore e forma:SolidPeso molecolare:440.54MrgprX2 antagonist-4
CAS:<p>MrgprX2 antagonist-4, from patent US20210128561A1, inhibits MrgprX2 receptor; useful for skin inflammation studies.</p>Formula:C16H19N3OColore e forma:SolidPeso molecolare:269.3484-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1A)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-N-(2-propyn-1-yl)-2-thiazolamine
CAS:<p>4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1A)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-N-(2-propyn-1-yl)-2-thiazolamine is an enantiomeric</p>Formula:C27H28ClFN2OSPurezza:99.02%Colore e forma:SoildPeso molecolare:483.04MAO-B-IN-3
<p>MAO-B-IN-3 is a reversible, selective inhibitor of monoamine oxidase B (MAO-B) with an IC50 of 96 nM and demonstrates affinity for the 5-HT6 receptor with a Ki</p>Formula:C24H25N3O2Purezza:98%Colore e forma:SolidPeso molecolare:387.47PG106 TFA
<p>PG106 TFA is a potent hMC3 antagonist (IC50=210 nM), inactive at hMC4 (EC50=9900 nM) and hMC5 receptors.</p>Formula:C53H70F3N13O11Colore e forma:SolidPeso molecolare:1122.2LE 300
CAS:<p>LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.</p>Formula:C20H22N2Purezza:97.91% - 98.79%Colore e forma:SolidPeso molecolare:290.4TRPV1/CB2 agonist 1
<p>TRPV1/CB2 agonist 1 (compound 41) is a dual agonist targeting hTRPV1 and CB2 receptors, with an EC50 value of 26.8 μM for hTRPV1. It is applicable in research related to the nervous system.</p>Colore e forma:Odour SolidSB234551
CAS:<p>SB234551 is a selective antagonist of endothelin ETA receptor.</p>Formula:C34H34N2O9Colore e forma:SolidPeso molecolare:614.64GHRF, porcine
CAS:<p>GHRF, porcine, a growth hormone releasing factor (GHRF) peptide (porcine), binds to the growth hormone secretagogue receptor (GHSR), thereby inducing the</p>Formula:C219H365N73O66SColore e forma:SolidPeso molecolare:5108.76(3R,5R,6S)-Atogepant
<p>(3R,5R,6S)-Atogepant (MK-8031) is a CGRP antagonist enantiomer used in migraine research.</p>Formula:C29H23F6N5O3Colore e forma:SolidPeso molecolare:603.52PZ-128
CAS:PZ-128, a PAR1 antagonist, is used potentially for the treatment of thrombosis.Formula:C55H99N13O9Purezza:98%Colore e forma:SolidPeso molecolare:1086.46Tiaprost
CAS:Tiaprost is a analog of prostaglandin F2α .Formula:C20H28O6SPurezza:98%Colore e forma:SolidPeso molecolare:396.5DOAM
CAS:<p>DOAM is an antagonist of the 5-HT2 receptor.</p>Formula:C16H27NO2Colore e forma:SolidPeso molecolare:265.39Pancreatic Polypeptide, rat
CAS:<p>Rat Pancreatic Polypeptide: 36-amino acid peptide, NPYR4 agonist, secreted by islet PP cells.</p>Formula:C195H298N58O57SPurezza:98%Colore e forma:SolidPeso molecolare:4398.87Corazonin
CAS:<p>Corazonin, a neuropeptide in insects, regulates caste identity and behavior, mainly in workers/foragers.</p>Formula:C62H83N17O19Colore e forma:SolidPeso molecolare:1370.42Eledoisin Related Peptide
CAS:<p>Eledoisin Related Peptide (Eledoisin RP) is a tachykinin receptor ligand.</p>Formula:C34H58N8O6SPurezza:98%Colore e forma:SolidPeso molecolare:706.94BIM-23190 hydrochloride
<p>BIM-23190 hydrochloride, somatostatin analog, SSRT2/5 agonist, Ki: 0.34 nM (SSTR2), 11.1 nM (SSTR5). Used in cancer, acromegaly research.</p>Colore e forma:LiquidBrexpiprazole S-oxide
CAS:<p>Brexpiprazole S-oxide is the main metabolite of Brexpiprazole, a human 5-HT1A and dopamine receptor partial agonist (Ki: 0.12, 0.3 nM).</p>Formula:C25H27N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:449.57HAEGTFTSDVS acetate
<p>HAEGTFTSDVS acetate is the first N-terminal 1-11 residues of GLP-1 which stimulates insulin secretion from pancreatic β-cells.</p>Formula:C50H75N13O22Purezza:97.47%Colore e forma:SolidPeso molecolare:1210.2JNJ-40929837 succinate
CAS:<p>JNJ-40929837 succinate is a selective, orally active inhibitor of LTA 4 H (leukotriene A 4 hydrolase). This compound effectively inhibits aminopeptidase activity, leading to the accumulation of Pro-Gly-Pro in serum, and can be utilized in asthma research [1].</p>Formula:C22H24N4O2S·xC4H6O4Colore e forma:SolidHS024 TFA
<p>HS024, a selective MC4 receptor antagonist, exhibits affinity with Ki values of 0.29, 3.29, 5.45, and 18.6 nM for MC4, MC5, MC3, and MC1 receptors, respectively</p>Formula:C60H80F3N19O12S2Colore e forma:SolidPeso molecolare:1380.52(Ala13)-Apelin-13
CAS:(Ala13)-Apelin-13 is a useful organic compound for research related to life sciences. The catalog number is T35374 and the CAS number is 568565-11-7.Formula:C63H107N23O16SPurezza:98%Colore e forma:SolidPeso molecolare:1474.75GLP-1R agonist 15
CAS:<p>GLP-1R agonist 15 (Compound 101) is a GLP-1 receptor agonist [1] .</p>Formula:C46H47FN8O7SColore e forma:SolidPeso molecolare:874.98Hemokinin 1, human TFA
<p>Hemokinin-1 is a human TFA and selective NK1 agonist; also activates NK2 & NK3 and induces opioid-independent analgesia.</p>Formula:C56H85F3N14O16SColore e forma:SolidPeso molecolare:1299.42S 16474
CAS:S 16474 is an antagonist of Neurokinin-1 Receptor.Formula:C44H48N6NaO8Purezza:98%Colore e forma:SolidPeso molecolare:811.8925-HT2C agonist-4
CAS:<p>Compound 3i, a 5-HT2C agonist-4, acts as an agonist for the 5-HT2C receptor with an EC50 of 5.7 nM. It is capable of reducing locomotor activity in zebrafish larvae.</p>Formula:C24H25N5OColore e forma:SolidPeso molecolare:399.49Secretin (28-54), human
CAS:Secretin (28-54), human, is a 27-amino acid residue peptide with a C-terminal amidation, acting on human secretin receptors.Formula:C130H220N44O40Purezza:98%Colore e forma:PowderPeso molecolare:3039.46GLP-1(28-36)amide TFA
<p>GLP-1(28-36)amide TFA, a nonapeptide cleavage product of GLP-1, shows antioxidant properties with anti-diabetic and cardioprotective effects.</p>Formula:C56H86F3N15O11Colore e forma:SolidPeso molecolare:1202.37α-Helical CRF(9-41) TFA
<p>α-Helical CRF(9-41) TFA acts as a competitive antagonist for the CRF2 receptor, possessing a binding constant (K B) of approximately 100 nM.</p>Formula:C168H275F3N46O55S2Colore e forma:SolidPeso molecolare:3940.42LRGILS-NH2
CAS:<p>LRGILS-NH2, reverse sequence of SLIGRL-NH2, is a control peptide for PAR2, affecting gut transit.</p>Formula:C29H56N10O7Purezza:98%Colore e forma:SolidPeso molecolare:656.82(-)-Eseroline fumarate
CAS:<p>(-)-Eseroline fumarate, a Physostigmine metabolite and AChE inhibitor, triggers cancer cell LDH release and neuronal cell death.</p>Formula:C17H22N2O5Colore e forma:SolidPeso molecolare:334.37Bombinakinin M
CAS:<p>Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.</p>Formula:C100H159N31O24Purezza:98%Colore e forma:SolidPeso molecolare:2179.55Luseogliflozin hydrate
CAS:<p>Luseogliflozin hydrate: SGLT2 inhibitor, IC50 2.26 nM, oral, for type 2 diabetes research.</p>Formula:C23H32O7SColore e forma:SolidPeso molecolare:452.56PROTAC(H-PGDS)-8
CAS:<p>PROTAC(H-PGDS)-8 is a PROTAC degrader targeting Hematopoietic prostaglandin D synthase (H-PGDS), exhibiting an IC50 of 0.14 μM [1].</p>Formula:C41H40N8O7Colore e forma:SolidPeso molecolare:756.811a,1b-dihomo Prostaglandin E1
CAS:<p>1a,1b-dihomo Prostaglandin E1 is a class of prostaglandin compounds.</p>Formula:C22H38O5Colore e forma:SolidPeso molecolare:382.5419-deoxy-9-methylene Prostaglandin E2
CAS:<p>9-deoxy-9-methylene PGE2: stable PGE2 analog with similar effects, less side effects, equal potency in rats, gerbils, primates.</p>Formula:C21H34O4Colore e forma:SolidPeso molecolare:350.499(+)-Oxypeucedanin methanolate
CAS:<p>(+)-Oxypeucedanin methanolate (compound 9) is a natural compound that inhibits prostaglandin E2 production [1].</p>Formula:C17H18O6Colore e forma:SolidPeso molecolare:318.32PAR 4 (1-6)
CAS:<p>PAR 4 (1-6) can be used for relevant research in the life sciences. Its product number is T36293 and CAS number is 225779-44-2.</p>Formula:C28H41N7O9Colore e forma:SolidPeso molecolare:619.676EP4 receptor antagonist 3
CAS:<p>EP4 receptor antagonist 3 from patent WO2010019796 A1 targets EP4 for research on pain, arthritis, and cancer.</p>Formula:C26H21F3N2O3SColore e forma:SolidPeso molecolare:498.52GLP-1 receptor agonist 4
CAS:<p>GLP-1 receptor agonist 4 targets GLP-1R, EC50 64.5 nM, potential diabetes treatment research.</p>Formula:C51H44Cl2N4O6Purezza:98%Colore e forma:SolidPeso molecolare:879.824-fluoro MBZP
CAS:<p>4-fluoro MBZP is a novel psychoactive substance in the phenylpiperazine class, utilized for studies on the 5-HT2 receptors in the central nervous system.</p>Formula:C12H17FN2Colore e forma:SolidPeso molecolare:208.28LUF6096
CAS:<p>LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically while</p>Formula:C22H21Cl2N3OPurezza:99.5%Colore e forma:SolidPeso molecolare:414.33Firazorexton
CAS:<p>Firazorexton is a potent orexin type 2 receptor (OX2R) agonist.</p>Formula:C22H25F3N2O4SColore e forma:SolidPeso molecolare:470.51DOTA-LM3 TFA
<p>DOTA-LM3 TFA is a somatostatin receptor (SSTR) antagonist with the molecular structure p-Cl-Phe-cyclo(D-Cys-Tyr-D-4-amino-Phe(carbamoyl)-Lys-Thr-Cys)D-Tyr-NH2.</p>Formula:C71H94ClF3N16O21S2Colore e forma:SolidPeso molecolare:1664.18SB-408124
CAS:SB408124: Non-peptide, OX1 receptor antagonist, Ki 57 nM (whole cell) and 27 nM (membrane), 50x more selective than OX2.Formula:C19H18F2N4OPurezza:99.81%Colore e forma:SolidPeso molecolare:356.37LY 344864 racemate
CAS:<p>LY 344864 racemate is a 5-HT1F receptor agonist.</p>Formula:C21H22FN3OPurezza:99.75%Colore e forma:SoildPeso molecolare:351.42PAR-4 Agonist Peptide, amide acetate
<p>PAR-4 Agonist Peptide, amide acetate is an agonist of proteinase-activated receptor-4 (PAR-4).</p>Formula:C36H52N8O9Purezza:98%Colore e forma:SolidPeso molecolare:740.865-Bromoimidazo[1,2-A]Pyrazine
CAS:<p>5-Bromoimidazo[1,2-a]pyrazine inhibits phosphodiesterase and beta-adrenergic receptors.5-Bromoimidazo[1,2-a]pyrazine shows antibronchospastic activity in vitro.</p>Formula:C6H4BrN3Purezza:97.04%Colore e forma:SolidPeso molecolare:198.02Ro60-0175
CAS:<p>Ro60-0175 is a selective 5-HT2B and 5-HT2C serotonin receptor agonist, often used as fumarate.</p>Formula:C11H12ClFN2Purezza:97.09%Colore e forma:SolidPeso molecolare:226.68PF-232798
CAS:<p>PF-232798 is a second generation oral CCR5 antagonist with potent broad-spectrum anti-HIV-1 activity.</p>Formula:C29H40FN5O2Colore e forma:SolidPeso molecolare:509.66GLI1-IN-3
<p>GLI1-IN-3 (Compound 11a) is a triterpenoid-like compound that inhibits Hedgehog signaling in cancer cells with GLI1 overexpression. It suppresses the proliferation of non-small cell lung cancer and prostate cancer cell lines with excessive Hh signaling activation. Additionally, GLI1-IN-3 reduces the expression of GLI1 protein and its target genes associated with tumor progression and proliferation in A549 and DU-145 cancer cells.</p>Colore e forma:Odour SolidBombinakinin M acetate
<p>Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and is</p>Formula:C102H163N31O26Purezza:99.80%Colore e forma:SolidPeso molecolare:2239.58PACAP-Related Peptide (PRP), human
<p>PRP, human: 29-amino-acid PACAP precursor segment, synthesized for biological/structural research.</p>Formula:C139H229N41O42Purezza:98%Colore e forma:SolidPeso molecolare:3146.574-Chloromethamphetamine hydrochloride
CAS:<p>4-Chloromethamphetamine hydrochloride is a novel psychoactive substance belonging to the amphetamine class.</p>Formula:C10H15Cl2NColore e forma:SolidPeso molecolare:220.14Tamuzimod
CAS:<p>Tamuzimod, an effective immunomodulator, exhibits modulatory activity on S1P Receptors with EC50 values below 1 μM [1] [2].</p>Formula:C21H13Cl3F3N5O3Colore e forma:SolidPeso molecolare:546.71HPP-9
<p>HPP-9, a Proteolysis-Targeting Chimera (PROTAC) derived from Hedgehog Pathway Inhibitor-1 (HPI-1) with a pIC50 value of 6.71, is designed to degrade BET</p>Formula:C49H52N6O11Colore e forma:SolidPeso molecolare:900.97ACT-1016-0707
CAS:<p>ACT-1016-0707 is a selective, insurmountable LPA1 antagonist with antifibrotic and anti-inflammatory activity in lung fibrosis models</p>Formula:C19H23ClN4O4SPurezza:99.905%Colore e forma:SolidPeso molecolare:438.93L-770644 dihydrochloride
CAS:<p>L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.</p>Formula:C30H38ClN7O4SColore e forma:SolidPeso molecolare:628.19GLP-1R agonist 4
CAS:<p>GLP-1R agonist 4, potentially for diabetes research, is a potent GLP-1R stimulator linked to hypoglycemia.</p>Formula:C32H30ClF2N3O5Colore e forma:SolidPeso molecolare:610.05Histamine & Melatonin Receptor-Targeted Compound Library
<p>A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS</p>Colore e forma:Odour SolidUpacicalcet HCl
<p>Upacicalcet HCl, a calcium mimetic, reduces blood PTH by targeting parathyroid receptors; treats secondary hyperparathyroidism.</p>Formula:C11H15Cl2N3O6SPurezza:98.56%Colore e forma:SoildPeso molecolare:388.22Preclamol hydrochloride
CAS:<p>Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.</p>Formula:C14H22ClNOColore e forma:SolidPeso molecolare:255.78Zalospirone
CAS:<p>Zalospirone is a 5-HT1A receptor agonist that can be used to study anxiety disorders and major depressive disorder.</p>Formula:C24H29N5O2Purezza:98.41% - 99.82%Colore e forma:SolidPeso molecolare:419.52O-Desethyl Dapagliflozin
CAS:<p>O-Desethyl Dapagliflozin (Empagliflozin-4) is a SGLT2 inhibitor, IC50=33nM.</p>Formula:C19H21ClO6Purezza:98.33%Colore e forma:SolidPeso molecolare:380.82tBPC
CAS:<p>Enhances Y4R response to PP, NPY & PYY with EC50 of 0.03, 0.4, 0.5 nM; selective for Y4R over Y1R, Y2R, Y5R.</p>Formula:C16H24O2Colore e forma:SolidPeso molecolare:248.36(Iso)-RJW100
CAS:<p>Potent LRH-1/NR5A2 and SF-1/NR5A1 agonist; pEC50: 6.4 (LRH-1), 7.2 (SF-1).</p>Formula:C28H34OPurezza:99.79%Colore e forma:SoildPeso molecolare:386.57GPR55 agonist 4
<p>GPR55 agonist 4 (Compound 28), with an EC50 of 131 nM for hGPR55 and 1.41 nM for rGPR55, effectively induces β-arrestin recruitment to human GPR55 [1].</p>Formula:C19H16FN5O2Colore e forma:SolidPeso molecolare:365.36Xanthine amine congener trihydrochloride
CAS:<p>Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.</p>Formula:C21H29ClN6O4Purezza:98.81%Colore e forma:SolidPeso molecolare:464.95CAY10580
CAS:<p>CAY10580 is a potent and selective prostaglandin EP 4 receptor agonist ( K i =35 nM).</p>Formula:C19H35NO4Colore e forma:SolidPeso molecolare:341.49Sufotidine
CAS:<p>Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.</p>Formula:C20H31N5O3SPurezza:99.03% - 99.92%Colore e forma:SolidPeso molecolare:421.56Bradykinin (1-6)
CAS:<p>Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.</p>Formula:C30H45N9O8Purezza:98%Colore e forma:SolidPeso molecolare:659.73CAP-100
<p>CAP-100 is a monoclonal antibody targeting CCR7. It neutralizes the ligand binding site and signaling of CCR7. This compound effectively inhibits migration, extravasation, homing, and survival in chronic lymphocytic leukemia (CLL) samples induced by CCR7. CAP-100 can mediate potent tumor cell killing through host immune mechanisms and exhibits favorable toxicity profiles in related hematopoietic cell subsets. It is involved in research on antitumor activity and diseases like chronic lymphocytic leukemia (CLL).</p>Colore e forma:Odour LiquidSR-31747 free base
CAS:SR-31747: immunosuppressive anti-inflammatory agent, inhibits cell growth by blocking sterol isomerase.Formula:C23H34ClNColore e forma:SolidPeso molecolare:359.98Galanin Receptor Ligand M35
CAS:<p>M35, a galanin(1-13)-bradykinin(2-9) amide, acts as a galanin antagonist in rats and inhibits mouse pancreatic islets.</p>Formula:C107H153N27O26Purezza:98%Colore e forma:SolidPeso molecolare:2233.6PY-60
CAS:<p>PY-60 can effectively activate YAP transcriptional activity against annexin A2 (ANXA2).Cost-effective and quality-assured.</p>Formula:C16H15N3O2SPurezza:99.5% - 99.67%Colore e forma:SolidPeso molecolare:313.37ELA-32(human)
CAS:<p>Potent apelin receptor agonist with IC50 = 0.27 nM; does not bind GPR15/GPR25. Boosts hESC self-renewal and angiogenesis.</p>Formula:C170H289N63O39S4Purezza:98%Colore e forma:SolidPeso molecolare:3967.8DETQ
CAS:<p>DETQ enhances human D1 dopamine receptor signaling, EC50=5.8 nM, less effective in rats/mice, inactive on D5.</p>Formula:C22H25Cl2NO3Colore e forma:SolidPeso molecolare:422.34GLP-1 receptor agonist 13
<p>Compound (S)-9, a GLP-1 receptor agonist, exhibits an EC50 of 76 nM for the glucagon GLP-1 receptor [1].</p>Formula:C25H23ClF2N6OColore e forma:SolidPeso molecolare:496.94Fasitibant chloride hydrochloride
CAS:Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.Formula:C36H50Cl4N6O6SColore e forma:SolidPeso molecolare:836.7Bremelanotide
CAS:<p>Bremelanotide is a synthetic peptide analog of alpha-MSH and is an agonist at melanocortin receptors including the MC3R and MC4R.</p>Formula:C50H68N14O10Purezza:98%Colore e forma:White PowderPeso molecolare:1025.16DSP-1053
CAS:<p>Dsp-1053 is a powerful SERT (Ki=1.02 nM) inhibitor with partial 5-HT1A receptor (Ki=5.05 nM) agonizing activity.</p>Formula:C26H32BrNO4Purezza:98%Colore e forma:SolidPeso molecolare:502.44LU AA33810
CAS:<p>LU AA33810 is a neuropeptide Y (NPY) Y5 receptor antagonist.</p>Formula:C19H25N3O2S3Purezza:98%Colore e forma:SolidPeso molecolare:423.62Linaclotide acetate
CAS:<p>Linaclotide acetate, an oral guanylate cyclase C agonist with 14 amino acids, treats constipation-predominant IBS and chronic constipation.</p>Formula:C61H83N15O23S6Purezza:98%Colore e forma:SolidPeso molecolare:1586.79GLP-1R agonist 16
CAS:<p>Compound 115a, a GLP-1R agonist, effectively activates the GLP-1 receptor with an EC50 of 0.15 nM [1].</p>Formula:C50H58FN10O6PColore e forma:SolidPeso molecolare:945.03Prostaglandin D2 methyl ester
CAS:<p>PGD2: made in mast cells during allergic reactions, causes vasodilation and inhibits blood clots. PGD2 methyl ester is a similar, fat-soluble prodrug.</p>Formula:C21H34O5Colore e forma:SolidPeso molecolare:366.498GRL093-22
<p>GRL093-22 is an effective and selective inhibitor of G protein-coupled receptor kinases (GRK), with IC50 values of 60 nM for GRK5 and 40 nM for GRK6. It shows potential for research in heart failure and multiple myeloma.</p>Formula:C33H29FN6O3Colore e forma:SolidPeso molecolare:576.62Amylin (8-37), rat
CAS:<p>Amylin (8-37), rat, an analog of IAPP, blocks insulin's effects on muscle glucose uptake and glycogen storage.</p>Formula:C140H227N43O43Purezza:98%Colore e forma:SolidPeso molecolare:3200.61Albiglutide fragment TFA
<p>Albiglutide fragment (GLP-1 (7-36) analog) TFA represents a biologically active segment of Albiglutide, resistant to DPP-4 degradation due to its structure as a</p>Formula:C148H224N40O45·xC2HF3O2Colore e forma:SolidBIBP3226
CAS:<p>BIBP3226 is a potent and selective antagonist for the Neuropeptide Y receptor Y1 and the neuropeptide FF receptor.</p>Formula:C27H31N5O3Colore e forma:SolidPeso molecolare:473.57CCR4 antagonist 3 hydrochloride
CAS:<p>Orally active CCR4 antagonist 3 hydrochloride with potent selectivity, IC50s: 22/50 nM; has antitumor properties.</p>Formula:C24H27Cl2N7O·xHClColore e forma:SolidImnopitant dihydrochloride
CAS:<p>Imnopitant dihydrochloride is a neurokinin NK1 receptor antagonist [1] .</p>Formula:C28H30Cl2F6N4OColore e forma:SolidPeso molecolare:623.46Lys-γ3-MSH(human)
CAS:<p>Pro-opiomelanocortin (POMC) derived peptide that stimulates lipolysis</p>Formula:C128H193N45O39SPurezza:98%Colore e forma:SolidPeso molecolare:3018.25Neuropeptide Y 13-36 (porcine)
CAS:<p>Neuropeptide Y 13-36 (porcine) is a selective neuropeptide Y2 receptor agonist.</p>Formula:C135H209N41O36Colore e forma:SolidPeso molecolare:2982.408Khusimol
CAS:Khusimol is a vasopressin V1a receptors non-peptide ligand that acts by inhibiting the binding of vasopressin.Formula:C15H24OPurezza:98%Colore e forma:SolidPeso molecolare:220.35Ramelteon metabolite M-II
CAS:<p>Ramelteon M-II binds MT1/MT2 with IC50s: 208/1470 pM; it's the main metabolite and a melatonin receptor agonist.</p>Formula:C16H21NO3Purezza:98%Colore e forma:SolidPeso molecolare:275.34Alverine hydrochloride
CAS:<p>Alverine hydrochloride is a parasympatholytic.</p>Formula:C20H28ClNColore e forma:SolidPeso molecolare:317.9HTL22562
CAS:<p>HTL22562 is a calcitonin gene-related peptide (CGRP) receptor antagonist for acute treatment of migraine.</p>Formula:C40H49N11O5Colore e forma:SolidPeso molecolare:763.904(S)-V-0219 hydrochloride
<p>(S)-V-0219 hydrochloride, a GLP-1R PAM, triggers calcium in hGLP-1R HEK cells, lowers glucose in mice, and reduces fasting hunger.</p>Formula:C20H26ClF3N4O2Colore e forma:SolidPeso molecolare:446.89PACAP (6-38), human, ovine, rat
CAS:<p>PACAP (6-38) in humans, sheep, rats: a strong inhibitor of PACAP 38, outperforms PACAP (6-27) in blocking PACAP-27-induced adenylate cyclase.</p>Formula:C182H300N56O45SPurezza:98%Colore e forma:SolidPeso molecolare:4024.74Orexin B, rat, mouse
CAS:<p>Orexin B, rat, mouse is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.</p>Formula:C126H215N45O34SPurezza:98%Colore e forma:SolidPeso molecolare:2936.45Metaraminol
CAS:<p>Metaraminol is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.</p>Formula:C9H13NO2Colore e forma:SolidPeso molecolare:167.21Bodilisant
CAS:<p>Bodilisant: nanomolar-affinity hH3R ligand, derived from piperidine, with BODIPY fluorophore.</p>Formula:C27H34BF2N3OColore e forma:SolidPeso molecolare:465.4Hemokinin 1 (mouse)
CAS:<p>Hemokinin 1 (mouse) is a selective excitogen 1 receptor agonist with a Ki value of 0.175 nM for the human NK1 receptor and 560 nM for the human NK2 receptor.</p>Formula:C61H100N22O15SPurezza:98%Colore e forma:White PowderPeso molecolare:1413.65Neuropeptide FF
CAS:<p>Endogenous antiopioid peptide and agonist at NPFF1 and NPFF2 receptors (Ki values are 2.82 and 0.21 nM respectively).</p>Formula:C54H76N14O10Purezza:98%Colore e forma:SolidPeso molecolare:1081.27Prazobind
CAS:<p>Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.</p>Formula:C23H27N5O3Colore e forma:SolidPeso molecolare:421.501Methapyrilene hydrochloride
CAS:<p>Methapyrilene hydrochloride is a biochemical.</p>Formula:C14H20ClN3SColore e forma:Liquid Solution) 5 5 (Ntp 1992)Peso molecolare:297.85Plecanatide acetate
CAS:Plecanatide acetate: GC-C receptor agonist, EC50=190 nM (T84 cells), anti-inflammatory in murine colitis.Formula:C67H108N18O28S4Purezza:98%Colore e forma:SolidPeso molecolare:1741.94d[Leu4,Lys8]-VP
CAS:<p>Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.</p>Formula:C47H67N11O11S2Purezza:98%Colore e forma:SolidPeso molecolare:1026.2FXR/TGR5 agonist 1
CAS:<p>FXR/TGR5 agonist 1 acts as an agonist on both FXR and TGR5 receptors and is utilized for treating fatty liver disease.</p>Formula:C31H32ClN3O3Colore e forma:SolidPeso molecolare:530.07[D-Trp8]-γ-MSH
CAS:<p>[D-Trp8]-γ-MSH is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively).</p>Formula:C74H99N21O16SPurezza:98%Colore e forma:SolidPeso molecolare:1570.798-iso Prostaglandin E2
CAS:<p>"8-iso PGE2: Isoprostane from arachidonic acid, potent rat renal vasoconstrictor, reduces GFR and renal flow by 80%, no BP effect."</p>Formula:C20H32O5Colore e forma:SolidPeso molecolare:352.47Neuropeptide Y5 receptor ligand-1
CAS:<p>Neuropeptide Y5 receptor ligand-1 (Compound 54), a carbazole derivative, acts as a powerful antagonist to the neuropeptide Y5 (NPY-5) receptor [1].</p>Formula:C19H17N3O2Colore e forma:SolidPeso molecolare:319.36Neurokinin B
CAS:<p>NKB, a tachykinin peptide, impacts human functions like gonadotropin-releasing hormone secretion.</p>Formula:C55H79N13O14S2Purezza:98%Colore e forma:SolidPeso molecolare:1210.4217-phenyl trinor Prostaglandin F2α cyclopropyl methyl amide
CAS:<p>Prostaglandin F2α (PGF2α) activates the FP receptor, promoting smooth muscle contraction and luteolysis.</p>Formula:C27H39NO4Colore e forma:SolidPeso molecolare:441.612Bz-Dab(nbd)-awfpp-nle-NH2
CAS:<p>Bz-Dab(nbd)-ala-trp-phe-pro-pro-nle-NH2 is a fluorescent NK2 antagonist.</p>Formula:C56H65N13O11Colore e forma:SolidPeso molecolare:1096.2L-797,591
CAS:<p>L-797,591 is a selective agonist of somatostatin receptor subtype 1.</p>Formula:C38H49N5O2Colore e forma:SolidPeso molecolare:607.83dCNP
<p>dCNP binds to NPR-B/C receptors (NPR-B/C receptor), initiating the cGMP signaling pathway and regulating vascular function. It exhibits anti-hypoxic effects by downregulating hypoxia-related genes such as HIF1α and HIF2α. Additionally, dCNP inhibits tumor stroma induction, demonstrating antifibrotic properties. It also enhances immune response by upregulating CTL, NK cells, and conventional type 1 dendritic cells in tumors.</p>Formula:C141H248N38O36S3Colore e forma:SolidPeso molecolare:3147.91RGS2-Galpha-q interaction-IN-1
RGS2–Galpha-q interaction-IN-1 (Compound AJ-3) is an inhibitor of the RGS2-Galpha-q interaction. It inhibits the growth of cancer cell lines that express RGS2 and has anti-cell migration properties.Formula:C30H30ClN7O3Colore e forma:SolidPeso molecolare:572.06Apelin-12 acetate
<p>Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.</p>Formula:C66H107N21O16SPurezza:98.82%Colore e forma:SolidPeso molecolare:1482.7517-phenoxy trinor Prostaglandin F2α ethyl amide
CAS:<p>Prostaglandin F2α (PGF2α), acting through the FP receptor, causes smooth muscle contraction and exhibits potent luteolytic activity.</p>Formula:C25H37NO5Colore e forma:SolidPeso molecolare:431.573Avorelin
CAS:<p>Avorelin, a luteinizing hormone releasing hormone (LH-RH) agonist, is used potentially for the treatment of prostate.</p>Formula:C65H85N17O12Purezza:98%Colore e forma:SolidPeso molecolare:1296.48NI-0701
<p>NI-0701 is a humanized antibody targeting CCL5/RANTES.</p>Purezza:95.4% (SDS-PAGE); 99.4% (SEC-HPLC) - 95.4% (SDS-PAGE); 99.4% (SEC-HPLC)Colore e forma:LiquidPeso molecolare:145.5kDaM40
CAS:<p>Potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in rat</p>Formula:C94H145N23O24Purezza:98%Colore e forma:SolidPeso molecolare:1981.33[Nle11]-Substance P
CAS:<p>'[Nle11]-Substance P is a gut and brain peptide, resisting methionine oxidation and causing excitatory neural effects.'</p>Formula:C64H100N18O13Purezza:98%Colore e forma:SolidPeso molecolare:1329.59Calcitonin Gene Related Peptide (CGRP) II, rat
CAS:<p>CGRP II is a potent vasodilator that boosts pancreatic enzyme levels by activating β-cell receptors.</p>Formula:C163H267N51O50S2Purezza:98%Colore e forma:SolidPeso molecolare:3805.31Antisauvagine-30
CAS:<p>CRF2 receptor antagonist; Kd 1.4 nM (mCRF2β), 153.6 nM (rCRF1). Blocks sauvagine-induced cAMP in cells & stress-related responses in mice.</p>Formula:C161H274N48O46SPurezza:98%Colore e forma:SolidPeso molecolare:3650.29Cloprostenol isopropyl ester
CAS:<p>(+)-Chloprostol is a PGF2α agonist, mimics prostaglandin F2α, induces luteal dissolution in mares without side effects or stress.</p>Formula:C25H35ClO6Colore e forma:SolidPeso molecolare:466.99Bertilimumab
CAS:<p>Bertilimumab (CAT 213; iCo-008), a human monoclonal antibody that targets eotaxin-1 (CCL11), shows promise in the research of allergic disorders [1].</p>Colore e forma:LiquidGalanin (1-16), mouse, porcine, rat TFA
<p>Galanin (1-16) agonizes hippocampal receptors; Kd 3 nM. Active on locus coeruleus neurons in mice, pigs, rats.</p>Formula:C80H117F3N20O23Purezza:98%Colore e forma:SolidPeso molecolare:1783.917-phenyl trinor Prostaglandin F2α cyclopropyl amide
CAS:<p>17-phenyl trinor Prostaglandin F2α cyclopropyl amide (17-phenyl trinor PGF2α cyclopropyl amide) is a novel analog of 17-phenyl trinor PGF2α ethyl amide.</p>Formula:C26H37NO4Colore e forma:SolidPeso molecolare:427.585Dehydro Aripiprazole (hydrochloride)
CAS:<p>Dehydro aripiprazole, an active atypical antipsychotic metabolite of aripiprazole, is formed by CYP3A4 and CYP2D6.</p>Formula:C23H26Cl3N3O2Colore e forma:SolidPeso molecolare:482.83[D-Phe12]-Bombesin
CAS:<p>Bombesin receptor antagonist</p>Formula:C74H112N22O18SPurezza:98%Colore e forma:SolidPeso molecolare:1629.88GLP-1R Antagonist 1
CAS:<p>GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).</p>Formula:C16H11ClF6N4O2Purezza:99.84%Colore e forma:SolidPeso molecolare:440.73Adenosine receptor antagonist 1
CAS:<p>A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.</p>Formula:C22H15ClFN7OColore e forma:SolidPeso molecolare:447.86Adenosine 2',5'-diphosphate sodium
CAS:<p>Adenosine 2',5'-diphosphate sodium is a competitive P2Y1 antagonist with non-selective antagonism at recombinant and human platelet P2X1 receptors.</p>Formula:C10H15N5NaO10P2Colore e forma:SolidPeso molecolare:450.192Antipsychotic agent-2
<p>Compound 11: potent antipsychotic, binds 5-HT1A/2A/2C, D2, H1 receptors; K is 56.6-1140 nM, BBB permeable.</p>Formula:C22H26FN5OColore e forma:SolidPeso molecolare:395.47Glucagon receptor antagonists-1
CAS:<p>Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.</p>Formula:C29H34FNO2Purezza:98%Colore e forma:SolidPeso molecolare:447.58Somatostatin-28 (1-14)
CAS:<p>Somatostatin-28 (1-14) is a truncated neuropeptide from prosomatostatin cleavage.</p>Formula:C61H105N23O21SPurezza:98%Colore e forma:SolidPeso molecolare:1528.71[Ala1,3,11,15]-Endothelin
CAS:<p>Selective ETB endothelin receptor agonist (IC50 values are 0.33 and 2200 nM for displacing [125I]-ET-1 from ETB and ETA receptors respectively).</p>Formula:C109H163N25O32SPurezza:98%Colore e forma:SolidPeso molecolare:2368Nebentan
CAS:<p>Nebentan (YM598) is an oral, selective ETA antagonist; Ki: 0.697 nM (ETA), 569 nM (ETB); may slow cor pulmonale, myocardial infarction.</p>Formula:C24H21N5O5SColore e forma:SolidPeso molecolare:491.52Bim 21009
CAS:Bim 21009 is an inhibitor of gonadorelin.Formula:C74H92ClN17O13Purezza:98%Colore e forma:SolidPeso molecolare:1463.08IRL-1620
CAS:<p>IRL-1620 is an effective and selective agonist of endothelin receptor type B (ETB) (Ki: 16 pM).</p>Formula:C86H117N17O27Purezza:98%Colore e forma:SolidPeso molecolare:1820.974Dipentylone hydrochloride
CAS:<p>Dipentylone hydrochloride (Bk-dmbdp HCl) is a psychoactive synthetic cathinone and sympathomimetic stimulant. Its inhibitory activity towards the dopamine transporter (IC50=0.233µM) is tenfold higher than that towards NET and SERT, inhibiting dopamine uptake and stimulating locomotor activity in mice.</p>Formula:C14H20ClNO3Purezza:99.94%Colore e forma:SolidPeso molecolare:285.77α-CGRP, rat
CAS:Endogenous neuropeptide, potent vasodilatorFormula:C162H262N50O52S2Purezza:98%Colore e forma:SolidPeso molecolare:3806.25Vapiprost hydrochloride
CAS:<p>Vapiprost hydrochloride is a biochemicla.</p>Formula:C30H40ClNO4Colore e forma:SolidPeso molecolare:514.117-phenyl trinor Prostaglandin E2 ethyl amide
CAS:<p>17-phenyl trinor PGE2 ethyl amide, an EP1/EP3 agonist (Ki: 14-54 nM), enhances lipid solubility and tissue uptake, is a potent antifertility agent.</p>Formula:C25H35NO4Colore e forma:SolidPeso molecolare:413.5516-phenoxy tetranor Prostaglandin F2α methyl ester
CAS:<p>Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor.</p>Formula:C23H32O6Colore e forma:SolidPeso molecolare:404.503GB-110 hydrochloride
<p>GB-110 HCl: potent, nonpeptidic oral PAR2 agonist; triggers Ca2+ release in HT29 cells; EC50 0.28 μM.</p>Formula:C33H49ClN6O5Colore e forma:SolidPeso molecolare:645.23Rubraxanthone
CAS:<p>Rubraxanthone is a PAF inhibitor isolated from Garcinia parvifolia Miq.</p>Formula:C24H26O6Colore e forma:SolidPeso molecolare:410.466β-CGRP, human
CAS:<p>β-CGRP, human ,a 37-amino acid peptide,is the beta form of Calcitonin-gene-related peptide (β-CGRP), involved extensively in regulation of the cardiovascular</p>Formula:C162H267N51O48S3Purezza:98%Colore e forma:SolidPeso molecolare:3793.41Gulgafafusp alfa
CAS:<p>Gulgafafusp alfa is a human IgG2κ monoclonal antibody that selectively binds to the glucagon-like peptide 1 receptor (GLP1R) [1].</p>Colore e forma:LiquidApelin-36(rat, mouse)
CAS:Endogenous APJ agonist from adipocytes; binds APJ tightly, inhibits cAMP, regulates heart function and fluid balance, blocks some HIV strains.Formula:C185H304N68O43SPurezza:98%Colore e forma:SolidPeso molecolare:4200.93S(-)-Bisoprolol fumarate
CAS:<p>S(-)-Bisoprolol fumarate is a selective β1-blocker for hypertension and heart research.</p>Formula:C18H31NO4·xC4H4O4Colore e forma:SolidPeso molecolare:441.521Eletriptan
CAS:<p>Eletriptan, second-generation triptans used to treat migraines, is used as an abortion drug.</p>Formula:C22H26N2O2SColore e forma:SolidPeso molecolare:382.52Cetirizine D8 dihydrochloride
CAS:<p>Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.</p>Formula:C21H26Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:433.4Vicasinabin
CAS:<p>Vicasinabin: potent CB2 agonist; researches chronic pain, atherosclerosis, bone mass, neuroinflammation.</p>Formula:C15H22N10OColore e forma:SolidPeso molecolare:358.4115-keto Latanoprost
CAS:<p>Latanoprost, a PG analog for ocular pressure, metabolizes into 15-keto latanoprost, a less potent variant reducing intraocular pressure and pupil size.</p>Formula:C26H38O5Colore e forma:SolidPeso molecolare:430.58Substance P (1-9)
CAS:<p>Substance P (1-9), a nonapeptide, slows its own inactivation and stimulates neurons.</p>Formula:C52H77N15O12Purezza:98%Colore e forma:SolidPeso molecolare:1104.26(S, R)-LSN 3318839
CAS:<p>(S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.</p>Formula:C26H23Cl2N3O2Purezza:99.57%Colore e forma:SoildPeso molecolare:480.39Besipirdine hydrochloride
CAS:<p>Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with cardiovascular activity that inhibits the uptake of biogenic amines.</p>Formula:C16H18ClN3Purezza:98.45%Colore e forma:SoildPeso molecolare:287.79THX-B
CAS:<p>THX-B, a potent non-peptidic p75 NTR antagonist, aids in researching diabetic kidney disease and neurodegenerative and inflammatory disorders.</p>Formula:C16H24N6O4Colore e forma:SolidPeso molecolare:364.4Spantide II
CAS:<p>Spantide II is an antagonist of tachykinin.</p>Formula:C86H104Cl2N18O13Purezza:98%Colore e forma:SolidPeso molecolare:1668.77LHRH, Ala(6)-
CAS:<p>LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.</p>Formula:C56H77N17O13Colore e forma:SolidPeso molecolare:1196.32Losulazine
CAS:<p>Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.</p>Formula:C27H22F4N4O3SPurezza:98.83%Colore e forma:SolidPeso molecolare:558.55PACAP (1-27), human, ovine, rat
CAS:PACAP (1-27) (the N-terminal fragment of PACAP-38) is a novel neuropeptides originally isolated from bovine hypothalamus, also found in humans and rats.Formula:C142H224N40O39SPurezza:98%Colore e forma:SolidPeso molecolare:3147.66{Val1}-Exendin-3/4
{Val1}- exendin-3/4 is the first n-terminal 1-28 residue of exendin-4 peptide.Formula:NAPurezza:98%Colore e forma:SolidPeso molecolare:3241.7Apelin-36(human)
CAS:Endogenous APJ agonist, EC50=20nM, regulates cardiovascular function, fluid balance, and feeding; blocks certain HIV strains.Formula:C184H297N69O43SPurezza:98%Colore e forma:SolidPeso molecolare:4195.87PF-03382792
CAS:<p>PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.</p>Formula:C23H32FN3O4Purezza:99.64%Colore e forma:SolidPeso molecolare:433.52A71378
CAS:<p>A71378 is a high potency, selectivity CCK-A receptors agonist.</p>Formula:C48H62N8O13SPurezza:98%Colore e forma:SolidPeso molecolare:991.12(R)-CJ 11974
CAS:<p>(R)-CJ 11974: non-peptide NK1 receptor antagonist, may relieve pain and prevent chemo-induced vomiting.</p>Formula:C31H38N2OPurezza:97.15%Colore e forma:SoildPeso molecolare:454.65RWJ 676070
CAS:<p>RWJ 676070 is an antagonist of vasopressin V1A/V2 receptor.</p>Formula:C30H26ClFN2O5Colore e forma:SolidPeso molecolare:548.99Chemerin-9 (149-157) TFA
<p>Chemerin-9 (149-157) TFA is a peptide located at positions 149-157 of chemerin-9, acting as a ChemR23/CMKLR1 agonist.</p>Formula:C56H67F3N10O15Purezza:99.77%Colore e forma:SolidPeso molecolare:1177.18FR190997
CAS:<p>FR190997 is an agonist of bradykinin B2 receptor.</p>Formula:C37H33Cl2N5O5Colore e forma:SolidPeso molecolare:698.59Ecraprost
CAS:<p>Ecraprost is used as a prodrug of prostaglandin E1.</p>Formula:C28H48O6Colore e forma:SolidPeso molecolare:480.68Enuvaptan
CAS:<p>Enuvaptan is a vasopressin receptor antagonist and has the potential for research into renal and cardiovascular diseases.</p>Formula:C21H15ClF6N8O3Colore e forma:SolidPeso molecolare:576.84I-BOP
CAS:<p>I-BOP is an agonist (KD=0.61 nM) at the thromboxane A2 receptor (TP).</p>Formula:C23H29IO5Colore e forma:SolidPeso molecolare:512.384CRL-42872 free base
CAS:<p>CRL-42872 free base is a bioactive chemical.</p>Formula:C22H26N6O6SColore e forma:SolidPeso molecolare:502.54AB21 HCl
<p>AB21 HCl: σ1 receptor antagonist, Ki 13 nM; less potent at σ2 (102 nM). Reduces mechanical hypersensitivity.</p>Formula:C23H29ClN2OPurezza:99.91%Colore e forma:SolidPeso molecolare:384.2NF157
CAS:<p>NF157, a selective P2Y11 antagonist with pKi 7.35, lowers MMP-3/MMP-13, aiding OA treatment; IC50s: P2Y11 463 nM, P2Y1 1811 μM, P2Y2 170 μM.</p>Formula:C49H28F2N6Na6O23S6Purezza:98%Colore e forma:SolidPeso molecolare:1437.1(R)-V-0219 hydrochloride
<p>(R)-V-0219 hydrochloride: Oral GLP-1R PAM, enantiomer of V-0219, triggers Ca2+ flux in hGLP-1R HEK cells.</p>Formula:C20H26ClF3N4O2Colore e forma:SolidPeso molecolare:446.89Leukotriene B4 Ethanolamide
CAS:<p>LTB4 binds to BLT1 (high affinity) and BLT2. LTB4-EA, a metabolite, is a stronger BLT1 antagonist, suggesting anti-inflammatory properties.</p>Formula:C22H37NO4Colore e forma:SolidPeso molecolare:379.541GLP-1R agonist 27
<p>GLP-1R agonist 27 (compound 21) is a potent and orally active GLP-1R agonist. It enhances the accumulation of cyclic adenosine monophosphate (cAMP), reduces blood glucose levels, and decreases food intake. GLP-1R agonist 27 shows potential for research in obesity and type 2 diabetes mellitus (T2DM).</p>Formula:C32H33N5O4SeColore e forma:SolidPeso molecolare:630.6
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