Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(939 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.945 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(148 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(407 prodotti)
- Recettore dell'endotelina(76 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(31 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(165 prodotti)
- Proteina Hedgehog/Smoothened(44 prodotti)
- Recettore dell'istamina(358 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(297 prodotti)
- PAFR(11 prodotti)
- PKA(48 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5352 prodotti di "Proteina G/GPCR"
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RE-640
CAS:<p>NSC-5844 (RE-640) (RE640) is a bisquinoline compound with C-C chemokine receptor type 1 (CCR1)-agonistic activities.</p>Formula:C20H16Cl2N4Purezza:99.60% - 99.87%Colore e forma:SolidPeso molecolare:383.27Siponimod hemifumarate
CAS:<p>Siponimod (BAF-312) is a potent S1P receptor modulator for multiple sclerosis research.</p>Formula:C62H74F6N4O10Colore e forma:SolidPeso molecolare:1149.282Cloprostenol sodium salt
CAS:<p>Cloprostenol sodium salt (ICI 80996 sodium salt) is a synthetic prostaglandin analogue, an agonist at the PGF2α receptor, with luteolytic properties.</p>Formula:C22H28ClNaO6Purezza:97.17% - 98.47%Colore e forma:White To Almost White Hygroscopic PowderPeso molecolare:446.9CB1-IN-1
CAS:<p>CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.</p>Formula:C33H31Cl2F3N6O3S2Purezza:99.08% - 99.76%Colore e forma:SolidPeso molecolare:751.67ACTH (1-39) human
CAS:<p>Adrenocorticotropic Hormone (ACTH) (1-39), human (ACTH (1-39), human) is an agonist of melanocortin receptor.</p>Formula:C207H308N56O58SPurezza:99.6%Colore e forma:White Lyophilised SolidPeso molecolare:4541.14RS 504393
CAS:RS 504393 is a highly selective CCR2 chemokine receptor antagonist (IC50s: 89 nM and > 100 μM for human recombinant CCR2 and CCR1).Formula:C25H27N3O3Purezza:98.64% - 99.62%Colore e forma:SolidPeso molecolare:417.5Bilastine
CAS:<p>Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of</p>Formula:C28H37N3O3Purezza:99.86% - >99.99%Colore e forma:SolidPeso molecolare:463.61ML 154
CAS:<p>ML 154 is a potent neuropeptide S receptor (NPSR) antagonist.</p>Formula:C29H26BrN2PSPurezza:99.53%Colore e forma:SolidPeso molecolare:545.47ARC-239
CAS:<p>ARC-239 is an agonist of α2-adrenergic receptor.</p>Formula:C24H29N3O3Colore e forma:SolidPeso molecolare:407.51Org 27569
CAS:<p>Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity and</p>Formula:C24H28ClN3OPurezza:>99.99% - ≥95%Colore e forma:SolidPeso molecolare:409.95MK 212 hydrochloride
CAS:<p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>Formula:C8H11ClN4·HClPurezza:99.88%Colore e forma:SolidPeso molecolare:235.12Neurokinin A(4-10) TFA(97559-35-8 free base)
<p>Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].</p>Formula:C36H55F3N8O12SPurezza:>99.99%Colore e forma:SolidPeso molecolare:880.932'-O-Methylisoliquiritigenin
CAS:<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Formula:C16H14O4Purezza:98.75%Colore e forma:SolidPeso molecolare:270.28REV 5901
CAS:<p>REV 5901: oral leukotriene receptor antagonist and 5-lipoxygenase inhibitor with Ki of 0.7 μM, researched for asthma.</p>Formula:C22H25NO2Colore e forma:SolidPeso molecolare:335.44Eltoprazine hydrochloride
CAS:<p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>Formula:C12H17ClN2O2Purezza:99.35%Colore e forma:SolidPeso molecolare:256.73Deslorelin acetate(57773-65-6 free base)
<p>Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)</p>Formula:C66H87N17O14Purezza:99.84%Colore e forma:SolidPeso molecolare:1342.5Ataciguat
CAS:<p>Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.</p>Formula:C21H19Cl2N3O6S3Purezza:99.09%Colore e forma:SolidPeso molecolare:576.49Etelcalcetide hydrochloride
CAS:<p>Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary hyperparathyroidism.</p>Formula:C38H73N21O10S2HClPurezza:>99.99%Colore e forma:SolidPeso molecolare:1353.33CYM-5541
CAS:<p>CYM-5541 (ML249) is a selective and allosteric S1P3 receptor agonist.</p>Formula:C19H28N2O2Purezza:99.74% - 99.76%Colore e forma:SolidPeso molecolare:316.44Phenelzine
CAS:Phenelzine is a MAOI antidepressant, boosting brain catecholamines, effective for endogenous depression.Formula:C8H12N2Purezza:98%Colore e forma:LiquidPeso molecolare:136.19Taladegib
CAS:<p>Taladegib (LY2940680), an oral Smo receptor antagonist, targets Hedgehog signaling for cancer treatment.</p>Formula:C26H24F4N6OPurezza:98.75% - >99.99%Colore e forma:SolidPeso molecolare:512.5Talnetant
CAS:<p>Talnetant (SB 223412) is a selective NK3 receptor antagonist that can penetrate the brain and modulate dopamine.</p>Formula:C25H22N2O2Purezza:97.88%Colore e forma:SolidPeso molecolare:382.45Pancreatic Polypeptide (human) acetate
<p>Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.</p>Purezza:97.26%Colore e forma:LiquidPeso molecolare:N/AAdipoRon hydrochloride
CAS:<p>AdipoRon hydrochloride is a specific, orally active AdipoR agonist, capable of binding AdipoR1 (Kd: 1.8 μM) and AdipoR2 (Kd: 3.1 μM).</p>Formula:C27H29ClN2O3Colore e forma:SolidPeso molecolare:464.99CAY10526
CAS:<p>CAY10526 (BTH) is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB signaling pathway.</p>Formula:C12H7BrO3SPurezza:98.75%Colore e forma:SolidPeso molecolare:311.15Clemizole
CAS:<p>Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.</p>Formula:C19H20ClN3Purezza:98% - 99.65%Colore e forma:SolidPeso molecolare:325.84PRX-08066
CAS:<p>PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.</p>Formula:C19H17ClFN5SPurezza:97.79% - 98.07%Colore e forma:SolidPeso molecolare:401.89ML-097
CAS:ML-097 (CID-2160985) is a pan activator of Ras-related GTPasesFormula:C14H11BrO3Purezza:99.12%Colore e forma:SolidPeso molecolare:307.139Neuropeptide Y (29-64), amide, human acetate
<p>Neuropeptide Y (29-64), amide, human acetate is involved in Alzheimer's disease (AD) and protects rat cortical neurons against β-Amyloid toxicity.</p>Purezza:98.42%Colore e forma:LiquidPeso molecolare:N/APiboserod
CAS:<p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>Formula:C22H31N3O2Purezza:97.21% - 99.49%Colore e forma:SolidPeso molecolare:369.5Laropiprant sodium
<p>Laropiprant sodium is a potent and selective DP receptor antagonist with Ki values of 0.57 nM for TP receptors and 2.95 nM for DP receptors.</p>Colore e forma:SolidAP1189 acetate
CAS:<p>AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.</p>Formula:C16H18N6O4Purezza:99.95%Colore e forma:SolidPeso molecolare:358.35[Lys8, Lys9]-Neurotensin (8-13) acetate
<p>[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2</p>Formula:C40H68N8O10Purezza:99.31%Colore e forma:SolidPeso molecolare:821.02R 396 acetate
<p>R 396 acetate is an NK-2 Tachykinin Receptor <br>Antagonist.</p>Formula:C41H55N9O12Purezza:99.52%Colore e forma:SolidPeso molecolare:865.93Betahistine EP Impurity C
CAS:<p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>Formula:C15H19N3Purezza:≥95%Colore e forma:SolidPeso molecolare:241.33HT-2157
CAS:<p>HT-2157 (SNAP-37889) is a selective, high-affinity competitive antagonist of the galanin-3 receptor (Gal3), demonstrating effective inhibition of this target.</p>Formula:C21H13F3N2OPurezza:98.33%Colore e forma:SolidPeso molecolare:366.34FSLLRY-NH2 TFA(245329-02-6 free base)
<p>FSLLRY-NH2 TFA inhibits PAR2, reverses taxol-induced pain, and reduces itch in mice; blocks ERK and collagen in fibroblasts.</p>Formula:C41H61F3N10O10Purezza:99.32%Colore e forma:SolidPeso molecolare:910.992-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)
<p>2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist.</p>Formula:C38H64F3N11O10Purezza:>99.99%Colore e forma:SolidPeso molecolare:891.98Ropinirole hydrochloride
CAS:<p>Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.</p>Formula:C16H24N2O·HClPurezza:99.87% - 99.98%Colore e forma:Off-White SolidPeso molecolare:296.84NIBR-0213
CAS:<p>NIBR-0213 is a potent and selective competitive S1P1 antagonist.Cost-effective and quality-assured.</p>Formula:C27H29ClN2O3Purezza:98.36% - 99.34%Colore e forma:SolidPeso molecolare:464.98LRGILS-NH2 acetate
<p>LRGILS-NH2 acetate is a PAR-2-inactive reversed peptide.</p>Formula:C29H56N10O7Purezza:96.65%Colore e forma:SolidPeso molecolare:656.82D3-βArr
CAS:<p>D3-βArr (NCGC00379308) is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by direct</p>Formula:C20H23N5Purezza:98.82%Colore e forma:SolidPeso molecolare:333.43BAY-545
CAS:<p>BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).</p>Formula:C18H22F3N3O4SPurezza:98.05%Colore e forma:SolidPeso molecolare:433.45SB-334867 free base
CAS:<p>SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.</p>Formula:C17H13N5O2Purezza:99.67% - >99.99%Colore e forma:SolidPeso molecolare:319.32Sitaxsentan sodium
CAS:<p>Sitaxsentan sodium (TBC11251 sodium salt) is a highly selective antagonist of endothelin A receptors.</p>Formula:C18H14ClN2O6S2·NaPurezza:98.39% - 99.01%Colore e forma:SolidPeso molecolare:476.89Calcitonin(salmon) Acetate(47931-85-1(free base))
<p>Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5</p>Formula:C145H240N44O48S2Purezza:99.29%Colore e forma:SolidPeso molecolare:3431.85Ibutamoren Mesylate
CAS:<p>Ibutamoren Mesylate (MK-0677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.</p>Formula:C28H40N4O8S2Purezza:97.98% - ≥98%Colore e forma:SolidPeso molecolare:624.77L-745870 hydrochloride
CAS:<p>L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptor</p>Formula:C18H20Cl2N4Purezza:97.36%Colore e forma:SolidPeso molecolare:363.28Gastrin I (human) acetate
<p>Gastrin I (human) acetate (Gastrin-17 acetate) is the endogenous peptide produced in the stomach, and increases gastric acid secretion via cholecystokinin 2 (</p>Formula:C99H128N20O33SPurezza:98.84%Colore e forma:SolidPeso molecolare:2158.25Aprepitant
CAS:<p>Aprepitant (Aprepitant`) is a Substance P/Neurokinin-1 Receptor Antagonist.</p>Formula:C23H21F7N4O3Purezza:98% - 99.68%Colore e forma:Off-White To Light Yellow Cyrstalline SolidPeso molecolare:534.43
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