Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(942 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.949 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(149 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(410 prodotti)
- Recettore dell'endotelina(75 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(32 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(166 prodotti)
- Proteina Hedgehog/Smoothened(45 prodotti)
- Recettore dell'istamina(359 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(298 prodotti)
- PAFR(11 prodotti)
- PKA(49 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5378 prodotti di "Proteina G/GPCR"
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15-keto Prostaglandin F2α
CAS:<p>15-keto Prostaglandin F2α is a metabolite of Prostaglandin F2α that lowers intraocular pressure in rabbits.</p>Formula:C20H32O5Purezza:98%Colore e forma:SolidPeso molecolare:352.47Cinnarizine D8
CAS:<p>Cinnarizine D8 is a deuterium-labeled Cinnarizine which is an antihistamine and a calcium channel blocker.</p>Formula:C26H28N2Purezza:98%Colore e forma:SolidPeso molecolare:376.573Ticlopidine
CAS:<p>Ticlopidine (PCR 5332) is an antiplatelet drug in the thienopyridine family which is an adenosine diphosphate (ADP) receptor inhibitor.</p>Formula:C14H14ClNSPurezza:99.67%Colore e forma:SolidPeso molecolare:263.79(RS)-ICI-118551 Hydrochloride
CAS:ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3Formula:C17H27NO2·HClPurezza:98.02%Colore e forma:SolidPeso molecolare:313.865-Methyltryptamine hydrochloride
CAS:<p>5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.</p>Formula:C11H15ClN2Purezza:99.45%Colore e forma:SolidPeso molecolare:210.703Vanoxerine
CAS:<p>Vanoxerine is an antagonist of dopamine transporter (Ki: 16.9nM).</p>Formula:C28H32F2N2OPurezza:98%Colore e forma:SolidPeso molecolare:450.56R-138727
CAS:<p>R-138727 is a novel P2Y12 receptor inhibitor.</p>Formula:C18H20FNO3SPurezza:98%Colore e forma:SolidPeso molecolare:349.42Isoproterenol sulfate anhydrous
CAS:<p>Isoproterenol sulfate anhydrous is a useful alkaloid. It is used for biological research.</p>Formula:C22H36N2O10SPurezza:98%Colore e forma:CoaPeso molecolare:520.59Ridazolol HCl
CAS:<p>Ridazolol HCl (CAS 413) is a novel β-adrenoceptor (β-AR) blocker with α-adrenerolytic activity.</p>Formula:C15H19Cl3N4O3Purezza:99.48%Colore e forma:SoildPeso molecolare:409.7Itopride free base
CAS:<p>Itopride HCl combats dyspepsia and GERD, inhibiting AChE and blocking D2 receptors.</p>Formula:C20H26N2O4Colore e forma:WhitePeso molecolare:358.43SB 271046 hydrochloride
CAS:<p>SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is > 200-fold selective over 55 other receptors, enzymes and ion channels.</p>Formula:C20H22ClN3O3S2·HClPurezza:99.77%Colore e forma:SolidPeso molecolare:488.457-Desmethyl-3-hydroxyagomelatine
CAS:<p>7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.</p>Formula:C14H15NO3Purezza:98%Colore e forma:SolidPeso molecolare:245.27Atenolol Hydrochloride
CAS:<p>Atenolol Hydrochloride is a selective antagonist of ß1 receptor.</p>Formula:C14H23ClN2O3Purezza:98%Colore e forma:SolidPeso molecolare:302.807-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene
CAS:<p>7-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene is a liver receptor homolog-1 (LRH-1) antagonist (IC50: 3.1 μM).</p>Formula:C42H44N2O6SPurezza:98%Colore e forma:SolidPeso molecolare:704.87Hydroxy ziprasidone
CAS:<p>Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.</p>Formula:C21H21ClN4O2SPurezza:98%Colore e forma:SolidPeso molecolare:428.94Dehydroabiethylamine
CAS:<p>Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs & cholesterol transport, and has anti-tumor effects.</p>Formula:C20H31NPurezza:98.79%Colore e forma:Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber LiquidPeso molecolare:285.47MK-447
CAS:<p>MK-447 is a nonsteroidal antiinflammatory agent.</p>Formula:C11H16INOPurezza:98%Colore e forma:SolidPeso molecolare:305.16Amidephrine
CAS:<p>Amidephrine is an adrenergic agent.</p>Formula:C10H16N2O3SColore e forma:SolidPeso molecolare:244.31Ketanserinol
CAS:<p>Ketanserinol is a metabolite of the antihypertensive drug ketanserin, which blocks 5-HT2 receptors to treat protamine-induced pulmonary hypertension.</p>Formula:C22H24FN3O3Colore e forma:SolidPeso molecolare:397.44Diclofensine
CAS:<p>Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.</p>Formula:C17H17Cl2NOPurezza:97.01% - 98.13%Colore e forma:SolidPeso molecolare:322.23Amidephrine hydrochloride
CAS:<p>Amidephrine hydrochloride is a biochemical.</p>Formula:C10H17ClN2O3SColore e forma:SolidPeso molecolare:280.77Caerulein, desulfated
CAS:Caerulein, desulfated (FI-6934, desulfated) is a desulfated compound formed after caerulein hydrolysis, a neuropeptide with lower smooth muscle activity.Formula:C58H73N13O18SPurezza:99.46%Colore e forma:SolidPeso molecolare:1272.34Amthamine
CAS:<p>Compound AMTHAMINE DIHYDROBROMIDE is a useful organic compound for research related to life sciences.</p>Formula:C6H11N3SColore e forma:SoildPeso molecolare:157.24Pardoprunox
CAS:<p>Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.</p>Formula:C12H15N3O2Purezza:98%Colore e forma:SolidPeso molecolare:233.27Tivumecirnon
CAS:<p>Tivumecirnon (FLX475) is a selective and oral CCR4 antagonist inhibits the infiltration and migration of Treg into the tumour microenvironment, antitumour</p>Formula:C24H27Cl2F3N6OPurezza:99.88%Colore e forma:SolidPeso molecolare:543.41Penbutolol sulfate
CAS:<p>Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.</p>Formula:C18H29NO2H2O4SPurezza:98.55%Colore e forma:SolidPeso molecolare:340.47Norreticuline
CAS:<p>Norreticuline is a potential adrenoceptor-α/β agonist and CYP2D6 and D2 receptor inhibitor for the study of neurodegenerative diseases.</p>Formula:C18H21NO4Colore e forma:SolidPeso molecolare:315.36S 25585
CAS:<p>S 25585 is a neuropeptide Y (NPY) Y5 receptor antagonist.</p>Formula:C22H23F3N4O6SPurezza:98%Colore e forma:SolidPeso molecolare:528.5Litorin
CAS:<p>Litorin suppresses appetite and stimulates smooth muscle, gastrin, gastric acid, and pancreatic secretion.</p>Formula:C51H68N14O11SColore e forma:White PowderPeso molecolare:1085.24Roxatidine acetate
CAS:<p>Roxatidine acetate: anti-ulcer, blocks histamine, reduces acid. Safer at lower doses.</p>Formula:C19H28N2O4Purezza:98%Colore e forma:White Or Off-White PowderPeso molecolare:348.44Ciproxifan
CAS:<p>Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).</p>Formula:C16H18N2O2Purezza:98.00%Colore e forma:SolidPeso molecolare:270.33Guacetisal
CAS:<p>Guacetisal, from acetylsalicylic acid and guaiacol, may treat chronic bronchitis.</p>Formula:C16H14O5Purezza:99.18%Colore e forma:SolidPeso molecolare:286.28LY 344864
CAS:<p>LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.</p>Formula:C21H22FN3OPurezza:98%Colore e forma:SolidPeso molecolare:351.42Lodoxamide tromethamine
CAS:<p>Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergic</p>Formula:C19H28ClN5O12Purezza:98.8%Colore e forma:SolidPeso molecolare:553.91MK-5046
CAS:MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).Formula:C20H18F6N4OPurezza:98.56%Colore e forma:SolidPeso molecolare:444.37Dolasetron Mesylate
CAS:<p>Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea following</p>Formula:C20H24N2O6SPurezza:99.05%Colore e forma:White PowderPeso molecolare:420.48Paroxetine hydrochloride hemihydrate
CAS:<p>Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).</p>Formula:C38H44Cl2F2N2O7Purezza:99.949%Colore e forma:SolidPeso molecolare:749.67CH 141
CAS:<p>CH 141 is a new type of peripheral vasodilator.</p>Formula:C19H21N3OColore e forma:SolidPeso molecolare:307.39OPC-14523 free base
CAS:OPC-14523, a 5-HT1A receptor agonist, is used potentially for the treatment of depression and neuropathic pain.Formula:C23H28ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:413.94Ranitidine bismuth citrate
CAS:<p>Ranitidine bismuth citrate, oral H2 blocker, IC50 3.3 µM, targets SARS-CoV-2 cells, treats H. pylori; MIC90 16 ng/L.</p>Formula:C19H27BiN4O10SColore e forma:SolidPeso molecolare:712.48Fulimetibant
CAS:<p>Fulimetibant is a bradykinin receptor antagonist.</p>Formula:C25H21F4N3O3Colore e forma:SolidPeso molecolare:487.45SB 258719 hydrochloride
CAS:<p>Selective 5-HT7 receptor antagonist</p>Formula:C18H31ClN2O2SPurezza:98%Colore e forma:SolidPeso molecolare:374.97E-3620
CAS:E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study dyskinesia and gastrointestinal dysfunction.Formula:C20H27Cl2N3O2Purezza:98.88% - 98.88%Colore e forma:SolidPeso molecolare:412.35OMDM-6
CAS:<p>OMDM-6 is a dual agonist of TRPV1(EC50 = 75 nM) and CB1 (Ki = 3.2 μM). OMDM-6 inhibits anandamide cellular uptake with a Ki of 7.0 μM.</p>Formula:C28H42N2O3Purezza:99.66%Colore e forma:SolidPeso molecolare:454.64(R)-Viloxazine Hydrochloride
CAS:<p>(R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.</p>Formula:C13H20ClNO3Purezza:99.88% - 99.94%Colore e forma:SolidPeso molecolare:273.76VPC 23019
CAS:<p>VPC 23019 is a competitive antagonist at the S1P1 and S1P3 receptors (pKi= 7.86 and 5.93, respectively).</p>Formula:C17H29N2O5PPurezza:98%Colore e forma:SolidPeso molecolare:372.4ABT-239
CAS:<p>ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.</p>Formula:C22H22N2OPurezza:>99.99%Colore e forma:SolidPeso molecolare:330.42Zolantidine dimaleate
CAS:<p>H2 receptor antagonist</p>Formula:C26H31N3O5SPurezza:98%Colore e forma:SolidPeso molecolare:497.61GSK-894490A
CAS:<p>GSK-894490A is an agonist of ghrelin receptor. GSK-894490A crosses the blood/brain barrier and elicit pro-cognitive effects.</p>Formula:C24H30ClN3O4SColore e forma:SolidPeso molecolare:492.03JNJ-10191584
CAS:<p>JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammation</p>Formula:C13H15ClN4OColore e forma:SolidPeso molecolare:278.74
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