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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

Mostrare 19 più sottocategorie

Trovati 6011 prodotti di "Proteina G/GPCR"

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  • 0990CL

    CAS:
    0990CL is an effective heterotrimer Gαi subunit specific inhibitor, which can interact with purified Go± in GDP-bound state, and can block α2AR mediated cAMP
    Formula:C21H21N5
    Purezza:98.99%
    Colore e forma:Solid
    Peso molecolare:343.42

    Ref: TM-T13983

    1mg
    192,00€
    5mg
    485,00€
    1mL*10mM (DMSO)
    507,00€
    10mg
    700,00€
    25mg
    1.063,00€
    50mg
    1.459,00€
    100mg
    1.963,00€
  • WAY-639889

    CAS:
    WAY-639889 is a small molecule compound with selective and potent inhibitory effects on neuropeptide Y-5 receptors.
    Formula:C25H27N5O
    Purezza:99.73%
    Colore e forma:Solid
    Peso molecolare:413.51

    Ref: TM-T77783

    1mg
    34,00€
    5mg
    82,00€
    10mg
    116,00€
    25mg
    225,00€
    50mg
    334,00€
    100mg
    477,00€
    200mg
    622,00€
  • Azelaprag

    CAS:
    Azelaprag (Example 263.0) is a candidate active molecule (EC50= 0.32 nM) for an apelin receptor agonist. treat nervous system diseases. High-Quality, Low-Cost!
    Formula:C25H29N7O4S
    Purezza:98.04% - >99.99%
    Colore e forma:Solid
    Peso molecolare:523.61

    Ref: TM-T14390

    1mg
    100,00€
    5mg
    236,00€
    1mL*10mM (DMSO)
    303,00€
    10mg
    371,00€
    25mg
    567,00€
  • SAG 21k

    CAS:
    SAG 21k is an orally bioactive and potent Hedgehog signaling activator that crosses the blood-brain barrier for the study of cartilage regeneration.
    Formula:C29H28ClF2N3O2S
    Purezza:99.51%
    Colore e forma:Solid
    Peso molecolare:556.07

    Ref: TM-T35559

    1mg
    109,00€
    5mg
    260,00€
    10mg
    389,00€
    25mg
    663,00€
    50mg
    888,00€
    100mg
    1.305,00€
  • GI 181771

    CAS:
    GI 181771 is an agonist of the cholecystokinin 1 receptor. GI 181771 can be used in studies about obesity.
    Formula:C34H31N5O6
    Purezza:95.02%
    Colore e forma:Solid
    Peso molecolare:605.64

    Ref: TM-T15382

    1mg
    175,00€
    5mg
    404,00€
    50mg
    1.243,00€
  • Osemozotan HCl

    CAS:
    Osemozotan is a 5-HT1A receptor agonist potentially for the treatment of generalized anxiety disorder.
    Formula:C19H22ClNO5
    Purezza:98.87% - 99.63%
    Colore e forma:Solid
    Peso molecolare:379.84

    Ref: TM-T28270

    1mg
    335,00€
    5mg
    803,00€
    10mg
    1.099,00€
    25mg
    1.639,00€
    50mg
    2.205,00€
    100mg
    2.952,00€
  • Calindol hydrochloride

    CAS:
    Calindol (hydrochloride) is a positive allosteric modulator (PAM) of calcimimetic calcium-sensing receptor (CaSR) with an EC50 of 132 nM.
    Formula:C21H21ClN2
    Purezza:99.47%
    Colore e forma:Solid
    Peso molecolare:336.86

    Ref: TM-T21758

    1mg
    52,00€
    5mg
    149,00€
    10mg
    246,00€
    25mg
    518,00€
    50mg
    825,00€
    100mg
    1.320,00€
    200mg
    1.776,00€
  • NMI 8739

    CAS:
    NMI 8739 (n-docosahexaenoyl dopamine) is an agonist of D2 autoreceptor.
    Formula:C30H41NO3
    Purezza:98.51%
    Colore e forma:Solid
    Peso molecolare:463.65

    Ref: TM-T11079

    1mg
    38,00€
    5mg
    80,00€
    1mL*10mM (DMSO)
    82,00€
    10mg
    114,00€
    25mg
    195,00€
    50mg
    286,00€
    100mg
    424,00€
    200mg
    617,00€
  • Selatogrel

    CAS:
    Selatogrel (ACT-246475) is a P2Y12 receptor antagonist with antithrombotic activity and inhibits platelet aggregation.
    Formula:C28H39N6O8P
    Purezza:98.43%
    Colore e forma:Solid
    Peso molecolare:618.62

    Ref: TM-T71364

    1mg
    99,00€
    5mg
    249,00€
    10mg
    409,00€
    25mg
    810,00€
    50mg
    1.305,00€
    100mg
    2.025,00€
    200mg
    2.740,00€
  • OPC-28326

    CAS:
    OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.
    Formula:C26H35N3O2
    Purezza:99.79%
    Colore e forma:Solid
    Peso molecolare:421.58

    Ref: TM-T13804

    1mg
    177,00€
    5mg
    432,00€
    1mL*10mM (DMSO)
    537,00€
    10mg
    587,00€
    25mg
    892,00€
    50mg
    1.198,00€
    100mg
    1.575,00€
    200mg
    2.133,00€
  • Adomeglivant

    CAS:
    Adomeglivant (LY2409021) is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus.
    Formula:C32H36F3NO4
    Purezza:99.91%
    Colore e forma:Solid
    Peso molecolare:555.63

    Ref: TM-T14130

    1mg
    35,00€
    5mg
    75,00€
    1mL*10mM (DMSO)
    93,00€
    10mg
    114,00€
    25mg
    178,00€
    50mg
    334,00€
    100mg
    557,00€
  • AS2717638

    CAS:
    AS2717638: oral LPA5 antagonist, IC50 38 nM, reduces PGF2α/PGE2/AMPA allodynia.
    Formula:C25H25N3O5
    Purezza:99.23%
    Colore e forma:Solid
    Peso molecolare:447.48

    Ref: TM-T10381

    1mg
    56,00€
    5mg
    118,00€
    1mL*10mM (DMSO)
    131,00€
    10mg
    190,00€
    25mg
    379,00€
    50mg
    612,00€
    100mg
    964,00€
    200mg
    1.305,00€
  • CGP-20712

    CAS:
    CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.
    Formula:C23H25F3N4O5
    Purezza:99.40% - 99.58%
    Colore e forma:Solid
    Peso molecolare:494.46

    Ref: TM-T30846

    1mg
    315,00€
    5mg
    745,00€
    10mg
    1.018,00€
    25mg
    1.431,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
    500mg
    4.410,00€
  • Selvigaltin

    CAS:
    Selvigaltin (GB1211) is a Gal-3 inhibitor with potential anticancer activity. Selvigaltin is used in the study of cirrhosis and cancer.
    Formula:C19H16BrF3N4O4S
    Purezza:99.49%
    Colore e forma:Solid
    Peso molecolare:533.32

    Ref: TM-T63751

    1mg
    250,00€
    5mg
    620,00€
    1mL*10mM (DMSO)
    743,00€
    10mg
    1.063,00€
    25mg
    2.142,00€
  • LGD-6972

    CAS:
    LGD-6972 is an antagonist of glucagon receptor.
    Formula:C43H46N2O5S
    Purezza:98.8% - 99.62%
    Colore e forma:Solid
    Peso molecolare:702.9

    Ref: TM-T11845

    1mg
    84,00€
    5mg
    177,00€
    10mg
    260,00€
    1mL*10mM (DMSO)
    268,00€
    25mg
    447,00€
    50mg
    655,00€
    100mg
    888,00€
  • ST-1006

    CAS:
    ST-1006: histamine H4 agonist, pKi 7.94, anti-inflammatory, anti-pruritic, promotes basophil migration.
    Formula:C16H20Cl2N6
    Purezza:99.96% - 99.98%
    Colore e forma:Solid
    Peso molecolare:367.28

    Ref: TM-T34709

    1mg
    86,00€
    1mL*10mM (DMSO)
    187,00€
    5mg
    188,00€
    10mg
    299,00€
    25mg
    487,00€
    50mg
    600,00€
    100mg
    743,00€
    200mg
    990,00€
  • AY 77

    CAS:

    AY 77: Potent, selective PAR2 agonist, favors Ca2+ (ec50=40nM) & ERK1/2 (ec50=2μM), boosts breast cancer cell migration.

    Formula:C21H32N4O4
    Purezza:99.7%
    Colore e forma:Solid
    Peso molecolare:404.5

    Ref: TM-T41190

    1mg
    391,00€
    5mg
    843,00€
    10mg
    1.130,00€
    25mg
    1.681,00€
    50mg
    2.270,00€
    100mg
    3.068,00€
  • Clazosentan

    CAS:
    Clazosentan (Ro 61-1790) is a selective ET_A receptor antagonist that inhibits ET-1 vasoconstriction and prevents cerebral vasospasm.
    Formula:C25H23N9O6S
    Purezza:95.39% - >99.99%
    Colore e forma:Solid
    Peso molecolare:577.57

    Ref: TM-T64084

    1mg
    71,00€
    5mg
    167,00€
    1mL*10mM (DMSO)
    205,00€
    10mg
    258,00€
    25mg
    565,00€
    50mg
    888,00€
    100mg
    1.161,00€
  • GV150013

    CAS:
    GV150013 is an antagonist of cholecystokinin-2 (CCK2) receptor.
    Formula:C33H34N4O3
    Purezza:99.93%
    Colore e forma:Solid
    Peso molecolare:534.65

    Ref: TM-T27503

    1mg
    177,00€
    5mg
    432,00€
    10mg
    587,00€
    1mL*10mM (DMSO)
    610,00€
    25mg
    892,00€
    50mg
    1.198,00€
    100mg
    1.575,00€
    200mg
    2.133,00€
  • α1 adrenoceptor-MO-1

    CAS:
    α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action.
    Formula:C20H24ClN5O
    Purezza:99.20% - 99.29%
    Colore e forma:Solid
    Peso molecolare:385.89

    Ref: TM-T10003

    1mg
    188,00€
    5mg
    371,00€
    1mL*10mM (DMSO)
    442,00€
    10mg
    513,00€
    25mg
    743,00€
    50mg
    1.018,00€
    100mg
    1.378,00€
    200mg
    1.863,00€