
Inibitori
Gli inibitori sono molecole che si legano a enzimi, recettori o altre proteine per ridurre o bloccare la loro attività biologica. Questi composti sono ampiamente utilizzati nella ricerca per studiare le vie biologiche, comprendere i meccanismi delle malattie e sviluppare farmaci terapeutici. Gli inibitori svolgono un ruolo cruciale nel trattamento di varie malattie, tra cui il cancro, le malattie cardiovascolari e le infezioni. Presso CymitQuimica, offriamo una vasta gamma di inibitori di alta qualità per supportare le tue ricerche in biochimica, biologia cellulare e sviluppo farmaceutico.
Sottocategorie di "Inibitori"
- Angiogenesi(2.715 prodotti)
- Apoptosi(6.164 prodotti)
- Ciclo cellulare/Checkpoint(4.727 prodotti)
- Cromatina/Epigenetica(2.400 prodotti)
- Segnalazione citoscheletrica(1.492 prodotti)
- Danno al DNA/Riparazione del DNA(2.928 prodotti)
- Endocrinologia/Ormoni(3.653 prodotti)
- Enzima(3.661 prodotti)
- Proteina G/GPCR(8.861 prodotti)
- Immunologia e infiammazione(3.801 prodotti)
- Virus dell'influenza(299 prodotti)
- Segnalazione JAK/STAT(412 prodotti)
- Segnalazione MAPK(1.239 prodotti)
- Trasportatore di membrana/canale ionico(2.979 prodotti)
- Metabolismo(10.029 prodotti)
- Microbiologia/Virologia(7.445 prodotti)
- Neuroscienza(10.281 prodotti)
- Altri inibitori(36.478 prodotti)
- Ossidazione-riduzione(44 prodotti)
- Segnalazione PI3K/Akt/mTOR(1.443 prodotti)
- Proteasi/Proteasoma(1.695 prodotti)
- Cellule staminali e Derivati(829 prodotti)
- Adattatori Tirosin-chinasi(2.035 prodotti)
- Ubiquitinazione(1.693 prodotti)
Mostrare 16 più sottocategorie
Trovati 66676 prodotti di "Inibitori"
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ENMD-1068 hydrochloride
CAS:<p>ENMD-1068 hydrochloride: selective PAR2 antagonist, counters liver fibrosis, hinders endometrial cell growth, and induces apoptosis in studies.</p>Formula:C15H30ClN3O2Colore e forma:SolidPeso molecolare:319.87Olverembatinib dimesylate
CAS:Olverembatinib dimesylate (GZD824 Dimesylate) is a novel orally bioavailable Bcr-Abl inhibitor for Bcr-Abl(WT) and Bcr-Abl(T315I).Formula:C29H27F3N6O·2CH4O3SPurezza:97.66% - >99.99%Colore e forma:SolidPeso molecolare:724.774'-tert-Butylacetophenone
CAS:4'-tert-Butylacetophenone is used as medical intermediateFormula:C12H16OPurezza:99.39%Colore e forma:Clear Almost Colorless Liquid Mild OdorPeso molecolare:176.25ARV-771
CAS:<p>ARV-771 is an effective BET degrader based on PROTAC technology.Cost-effective and quality-assured.</p>Formula:C49H60ClN9O7S2Purezza:99.69%Colore e forma:SolidPeso molecolare:986.64Ethyl 4-amino-2-(methylthio)pyrimidine-5-carboxylate
CAS:ETHYL 4-AMINO-2-(METHYLTHIO)PYRIMIDINE-5-CARBOXYLATE used for preparation of pyrimidopyrimidines as protein kinase inhibitors.Formula:C8H11N3O2SPurezza:98.71%Colore e forma:SolidPeso molecolare:213.266-Phosphogluconic acid
CAS:6-Phosphogluconic acid competitively inhibits PGI with Ki: 0.048 mM for glucose 6-P, 0.042 mM for fructose 6-P.Formula:C6H13O10PPurezza:98%Colore e forma:SolidPeso molecolare:276.14XYLOBIOSE
CAS:XYLOBIOSE ia a natural product,and exhibited therapeutic potential for treating obesity which involved suppression of fat deposition and obesity-relatedFormula:C10H18O9Purezza:99.13% - 99.5%Colore e forma:SolidPeso molecolare:282.24Atractyloside potassium salt
CAS:<p>1.</p>Formula:C30H44K2O16S2Purezza:98.25% - 99.82%Colore e forma:SolidPeso molecolare:802.99Ioversol
CAS:Ioversol (MP-328) is a nonionic iodinated contrast agent.Formula:C18H24I3N3O9Purezza:99.11%Colore e forma:Odorless White PowderPeso molecolare:807.11VPC-80051 racemate
CAS:VPC-80051 is the first small molecule inhibitor of hnRNP A1 splicing activity by using a computer-aided drug discovery approach.Formula:C16H13F2N3OPurezza:97.36%Colore e forma:SolidPeso molecolare:301.29Isocurcumenol
CAS:1. Isocurcumenol inhibits 5α-reductase which converts testosterone to dihydrotestosterone (DHT).Formula:C15H22O2Purezza:99.29% - ≥95%Colore e forma:SolidPeso molecolare:234.33Desmethyl Erlotinib
CAS:Desmethyl Erlotinib (CP-473420) is the active metabolite of Erlotinib (EGFR inhibitor with IC50 of 2 nM).Formula:C21H21N3O4Purezza:97.92% - 98.62%Colore e forma:SolidPeso molecolare:379.41DSPS
CAS:<p>DSPS (Dioctadecanoylphosphatidylserine) is an important phospholipid membrane component, plays a key role in cell cycle signaling, specifically in apoptosis.</p>Formula:C42H82NO10PPurezza:mixture - mixtureColore e forma:SolidPeso molecolare:792.08Ilexgenin A
CAS:Ilexgenin A is a novel pentacyclic triterpenoid, is a compound extracted from leaves of Ilex hainanensis MerrFormula:C30H46O6Purezza:97.11% - 97.19%Colore e forma:SolidPeso molecolare:502.68Dansylglycine
CAS:Dansylglycine is a fluorescent probe for specific determination of halogenating activity of myeloperoxidase and eosinophil peroxidase[1].Formula:C14H16N2O4SPurezza:99.1%Colore e forma:SolidPeso molecolare:308.35Splitomicin
CAS:Splitomicin (1-Naphthalenepropanoic Acid) (IC50 of 60 μM), a specific inhibitor of NAD(+)-dependent histone deacetylase Sir2p, displays a high activity in aFormula:C13H10O2Purezza:97.09% - 99.11%Colore e forma:SolidPeso molecolare:198.22Potassium sorbate
CAS:<p>Potassium sorbate, an antifungal and corrosion inhibitor, is used with polyethylene films.</p>Formula:C6H7KO2Purezza:99.81%Colore e forma:White Solid CrystallinePeso molecolare:150.22Lobaplatin
CAS:Lobaplatin (D-19466) (D-19466) is a diastereometric mixture of platinum(II) complexe.Formula:C9H18N2O3PtPurezza:98.00%Colore e forma:SolidPeso molecolare:397.33IHR-1
CAS:IHR-1, a Smo inhibitor (IC50 7.6 nM), blocks Hedgehog pathway, not Wnt/Notch, and prevents Smo in primary cilium.Formula:C20H12Cl4N2O2Purezza:97.02%Colore e forma:SolidPeso molecolare:454.13Linoleic acid
CAS:<p>Linoleic acid (9,12-octadecadienoic acid) is a natural polyunsaturated fatty acid. Linoleic acid is an essential fatty acid. Cost-effective and quality-assured.</p>Formula:C18H32O2Purezza:97.71% - 99.61%Colore e forma:Less To Straw Colored Liquid A Polyunsaturated Fatty Acid Essential To Human DietPeso molecolare:280.45Trifloxystrobin
CAS:Trifloxystrobin is a fungicide against R. solani in sugar beets with EC50s: 23.0 μg/L for Daphnia neonates, 1.7 μg/L for embryos.Formula:C20H19F3N2O4Purezza:99.49%Colore e forma:SolidPeso molecolare:408.37HIV-1 Inhibitor 18A
CAS:HIV-1 Inhibitor 18A (HIV-1 Inhibitor-18A) specifically inhibits the entry of multiple HIV-1 isolates.Formula:C14H11N5O2SPurezza:99.79%Colore e forma:SolidPeso molecolare:313.33Ciprofibrate
CAS:Ciprofibrate (Win35833) is a fibrate derivative with antilipidemic activity.Formula:C13H14Cl2O3Purezza:99.63% - >99.99%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:289.15Decanedioic acid
CAS:Decanedioic acid (Sebacinsaure) is a saturated, straight-chain naturally occurring dicarboxylic acid.Formula:C10H18O4Purezza:99.73%Colore e forma:Reacts Violently With Bases And Oxidants Oxidants Solid PowderPeso molecolare:202.25N-Boc-O-tosyl hydroxylamine
CAS:<p>N-Boc-O-tosyl hydroxylamine is nitrogen source for the N-amination of aryl and alkyl amines.</p>Formula:C12H17NO5SPurezza:99.93%Colore e forma:SolidPeso molecolare:287.33Pristimerin
CAS:Pristimerin has anticancer properties, counters hypoxia-induced cancer spread, and reduces inflammation by inhibiting ROS/IKK/NF-κB pathways.Formula:C30H40O4Purezza:98.59% - 99.79%Colore e forma:SolidPeso molecolare:464.641,3,5-Trimethoxybenzene
CAS:1,3,5-Trimethoxybenzene, a flavonoid intake biomarker, has three methoxy groups.Formula:C9H12O3Purezza:99.57% - 99.85%Colore e forma:White To Off-White CrystalPeso molecolare:168.19Purpurogallin
CAS:Purpurogallin: natural phenol from Quercus spp., xanthine oxidase inhibitor (IC50: 0.2μM), antioxidant, anti-inflammatory.Formula:C11H8O5Purezza:96.44%Colore e forma:SolidPeso molecolare:220.18Secoxyloganin
CAS:Secoxyloganin possesses a hepato-protective effect.Formula:C17H24O11Purezza:99.45% - ≥95%Colore e forma:SolidPeso molecolare:404.37ADOS
CAS:ADOS (82692-96-4) is a biochemical reagent/chromogenic reagent.Formula:C12H18NNaO5SPurezza:99.84%Colore e forma:SolidPeso molecolare:311.33Motolimod
CAS:<p>Motolimod (VTX-378) (VTX-2337) is an effective and specific Toll-like receptor (TLR) 8 agonist (EC50: 100 nM), > 50-fold selectivity over TLR7.</p>Formula:C28H34N4O2Purezza:97.43% - 99.66%Colore e forma:SolidPeso molecolare:458.67,3',4'-Tri-O-methylluteolin
CAS:<p>7,3',4'-Tri-O-methylluteolin is anti-inflammatory, antibacterial, antifungal, and has moderate antitrypanosomal effects (MIC 19.0 ug/ml).</p>Formula:C18H16O6Purezza:98.66% - 99.79%Colore e forma:SolidPeso molecolare:328.32CK-636
CAS:CK-636 (CK-0944636), an Arp2/3 complex inhibitor, can inhibit actin polymerization induced by the human, fission yeast and bovine Arp2/3 complex.Formula:C16H16N2OSPurezza:98.1% - 98.88%Colore e forma:SolidPeso molecolare:284.38SB-590885
CAS:SB590885 is an effective B-Raf inhibitor (Ki: 0.16 nM, in a cell-free assay).Formula:C27H27N5O2Purezza:95.42% - 99.06%Colore e forma:SolidPeso molecolare:453.54Sodium taurocholate
CAS:Sodium taurocholate hydrate, a cholesterol breakdown product, cycles from bile to liver, changing forms via microbes and enzymes.Formula:C26H44NO7S·NaPurezza:95% - 99.64%Colore e forma:White PowderPeso molecolare:537.69Salvianolic acid B
CAS:Salvianolic acid B (Dan Shen Suan B) is an antioxidant. Salvianolic acid B has anticoagulant and antithrombotic effects. Cost-effective and quality-assured.Formula:C36H30O16Purezza:95% - 99.84%Colore e forma:SolidPeso molecolare:718.59KDU691
CAS:<p>KDU691 is a PI4K inhibitor.</p>Formula:C22H18ClN5O2Purezza:98.68%Colore e forma:SolidPeso molecolare:419.86Hydroxypropyl Cellulose
CAS:<p>Hydroxypropyl cellulose (HPC), soluble in water and organics, serves as a food additive and DNA separation aid.</p>Formula:C12H20N2Purezza:98%Colore e forma:SolidPeso molecolare:192.306Doxazosin
CAS:<p>Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.</p>Formula:C23H25N5O5Purezza:99.47% - 99.87%Colore e forma:SolidPeso molecolare:451.48Isosinensetin
CAS:1. Isosinensetin (6-Demethoxynobiletin) shows antioxidant and HIV-1 protease inhibiting activities.Formula:C20H20O7Purezza:99.98% - ≥95%Colore e forma:SolidPeso molecolare:372.37Almotriptan Malate
CAS:<p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>Formula:C17H25N3O2S·C4H6O5Purezza:99.95%Colore e forma:Pale Yellow SolidPeso molecolare:469.55N3-C5-NHS ester
CAS:N3-C5-NHS ester is a noncleavable ADC linker. N3-C5-NHS ester can be used in the synthesis of antibody-drug conjugates (ADCs).Formula:C10H14N4O4Purezza:99.76%Colore e forma:SolidPeso molecolare:254.24(+)-Nortrachelogenin
CAS:<p>(+)-Nortrachelogenin is a lignan isolated from Wikstroemia indica C.A. Meyer (Thymelaeaceae). (+)-Nortrachelogenin possesses antileukemic activity.</p>Formula:C20H22O7Purezza:99.88%Colore e forma:SolidPeso molecolare:374.38Batatasin III
CAS:Batatasin III inhibits cancer migration and invasion by suppressing epithelial to mesenchymal transition and FAK-AKT signals and possesses anti-cancerFormula:C15H16O3Purezza:99.16%Colore e forma:SolidPeso molecolare:244.29RO1138452
CAS:RO1138452 (CAY10441) blocks prostacyclin receptor; orally active, high affinity (Ki: 1.5 nM), analgesic in rats (2-20 mg/kg).Formula:C19H23N3OPurezza:97.01% - 99.34%Colore e forma:SolidPeso molecolare:309.41RKI1313
CAS:RKI1313 (RKI-1313) was a selective inhibitor for ROCK-dependent signaling, cytoskeletal changes, anchorage-independent colony formation, migration, and invasionFormula:C17H16N4O2SPurezza:99.53% - ≥95%Colore e forma:SolidPeso molecolare:340.4Siramesine hydrochloride
CAS:Siramesine hydrochloride (Lu 28-179 hydrochloride) is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of Y cells and to exhibitFormula:C30H32ClFN2OPurezza:99.72% - >99.99%Colore e forma:SolidPeso molecolare:491.045-FAM SE
CAS:5-FAM SE, a single-isomer green fluorophore, labels peptides, proteins, nucleotides.Formula:C25H15NO9Purezza:96.19% - 99.93%Colore e forma:Yellow To Orange SolidPeso molecolare:473.39TPTZ
CAS:<p>TPTZ is used exclusively as an analytical reagent.</p>Formula:C18H12N6Purezza:99.52% - 99.7%Colore e forma:Off-White PowderPeso molecolare:312.33Faropenem sodium
CAS:Faropenem sodium: Oral penem antibiotic for tuberculosis, pneumonia.Formula:C12H14NNaO5SPurezza:99.41%Colore e forma:Pale Yellow CrystalsPeso molecolare:307.3
