A 922500

CAS: 959122-11-3

Ref. 3D-FA64929

Product Information

• Name: A 922500
• Brand: Biosynth
• Description: Inhibits human and mouse diacylglycerol O-acyltransferase 1 (DGAT-1) with IC50 values of 9 and 22 nM, respectively. Selective for DGAT-1 over DGAT-2 (IC50 = 53 µM), acyl coenzyme A transferase (IC50 = 296 µM) and other acyltransferases. Reduces plasma and liver triglycerides, FFA, chylomicron secretion and increases HDL cholesterol in vivo.

Chemical properties

• Molecular weight: 428.48 g/mol
• Formula: C₂₆H₂₄N₂O₄
• Purity: Min. 95%