Product Information
Name:DBPR116
Brand:Targetmol
Description:DBPR116 is a prodrug of BPRMU191 that can penetrate the blood-brain barrier. It significantly enhances the delivery efficiency of drugs targeting the central nervous system. When combined with the antagonist Naltrexone, DBPR116 demonstrates superior safety and analgesic effects compared to morphine in various in vivo pharmacological studies, including thermal pain models, cancer pain models, constipation, sedation, psychological dependence, heart rate, and respiratory frequency. As a strategy for peripheral administration, DBPR116 effectively alleviates pain while reducing adverse effects, showing promise as a safer opioid analgesic.
Notice:Our products are intended for lab use only. For any other use, please contact us.
Chemical properties
Molecular weight:359.42
Formula:C19H18FNO3S
Color/Form:Solid
Technical inquiry about: DBPR116
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