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Opioid Receptor

Opioid Receptor

Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.

Found 350 products for "Opioid Receptor".

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  • Matrine

    CAS:
    Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.
    Formula:C15H24N2O
    Purity:99.77% - >99.99%
    Color and Shape:White Solid
    Molecular weight:248.3639
  • Naltrexone hydrochloride

    CAS:
    Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.
    Formula:C20H24ClNO4
    Purity:98.72% - 99.65%
    Color and Shape:Solid
    Molecular weight:377.862
  • Alvimopan

    CAS:
    Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.
    Formula:C25H32N2O4
    Purity:99.47% - 99.78%
    Color and Shape:Solid
    Molecular weight:424.5326
  • Apitegromab

    CAS:
    Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases including
    Purity:97.59% (SDS-PAGE); 99.78% (SEC-HPLC) - >95.0% (SDS-PAGE); 99.62% (SEC-HPLC)
    Color and Shape:Liquid
    Molecular weight:145.06 kDa (Predicted)
  • Loperamide hydrochloride

    CAS:
    Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.
    Formula:C29H34Cl2N2O2
    Purity:99.91% - >99.99%
    Color and Shape:White Solid
    Molecular weight:513.498
  • LY2940094

    CAS:
    LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.
    Formula:C22H23ClF2N4O2S
    Purity:99.4%
    Color and Shape:White Solid
    Molecular weight:480.958
  • Samidorphan HCl

    CAS:
    Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.
    Formula:C21H27ClN2O4
    Purity:96.79% - 97.85%
    Color and Shape:Solid
    Molecular weight:406.9
  • ZT 52656A hydrochloride

    CAS:
    ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.
    Formula:C19H26ClF3N2O
    Purity:98.78%
    Color and Shape:Solid
    Molecular weight:390.871
  • Moguisteine

    CAS:
    Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.
    Formula:C16H21NO5S
    Purity:99.98%
    Color and Shape:White Solid
    Molecular weight:339.41
  • BTRX-335140

    CAS:
    BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.
    Formula:C25H32FN5O2
    Purity:98% - 99.89%
    Color and Shape:White Solid
    Molecular weight:453.5523
  • Meptazinol hydrochloride

    CAS:
    Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.
    Formula:C15H23NO·HCl
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:269.81
  • CP 866087

    CAS:
    CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.
    Formula:C24H30N2O3S
    Purity:99.22% - 99.74%
    Color and Shape:Solid
    Molecular weight:426.57
  • Trimebutine maleate

    CAS:
    Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.
    Formula:C26H33NO9
    Purity:99.89% - 99.98%
    Color and Shape:White Solid
    Molecular weight:503.55
  • Sinomenine hydrochloride

    CAS:
    Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.
    Formula:C19H24ClNO4
    Purity:99.43%
    Color and Shape:White Solid
    Molecular weight:365.85
  • SNC 80

    CAS:
    SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 nM), with analgesic and antidepressant potential.
    Formula:C28H39N3O2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:449.63
  • Dermorphin

    CAS:
    Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
    Formula:C40H50N8O10
    Purity:98.82%
    Color and Shape:White Solid
    Molecular weight:802.8726
  • KOR agonist 6


    KOR agonist 6 is a KOR agonist with a Ki value of 0.25 pM. In CHO cells, it exhibits agonistic activity on MOR and DOR and inhibits forskolin-stimulated cAMP accumulation. The compound stimulates KOR-mediated [35S]GTPγS binding in HEK293 cells expressing KOR and effectively suppresses cAMP accumulation as a potent agonist, showing lower β-arrestin recruitment efficacy. Additionally, KOR agonist 6 demonstrates analgesic effects in mice and can be employed in the study of analgesics with reduced central nervous system (CNS) side effects.
    Color and Shape:Odour Solid
  • Dynorphin (2-17), amide, porcine


    Dynorphin (2-17), amide, porcine is a C-terminally amidated KOR agonist with enhanced protease resistance.
    Formula:C90H147N31O20
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1983.33
  • μ/κ/δ opioid receptor agonist 1


    μ/κ/δopioid receptor agonist1 is an agonist for the μ opioid receptor (MOR), κ opioid receptor (KOR), and δ opioid receptor (DOR). It produces potent and long-lasting analgesic effects in the tail flick test through peripheral MOR and KOR activation.
    Formula:C35H45FN8O8
    Color and Shape:Solid
    Molecular weight:724.33444
  • Dynorphin (2-17), porcine acetate


    Dynorphin (2-17), porcine acetate is a porcine dynorphin fragment that acts as a potent KOR agonist.
    Formula:C92H150N30O23
    Purity:98.19%
    Molecular weight:2044.40