Product Information
Name:Tuspetinib dihydrochloride
Synonyms:
- HM43239 dihydrochloride
Brand:Targetmol
Description:Tuspetinib (HM43239) dihydrochloride is a selective FLT3 inhibitor with oral bioactivity, exhibiting IC50 values of 1.1 nM for FLT3 wild type, 1.8 nM for FLT3ITD mutant type, and 1.0 nM for FLT3D835Y mutant type. As a reversible type I inhibitor, it directly suppresses FLT3 kinase activity and modulates p-STAT5, p-ERK, SYK, JAK1/2, and TAK1. Tuspetinib dihydrochloride inhibits the proliferation of leukemia cells and induces apoptosis (apoptosis).
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Chemical properties
Molecular weight:573.99
Formula:C29H35Cl3N6
Color/Form:Solid
Technical inquiry about: Tuspetinib dihydrochloride
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