Product Information
Name:PROTAC CBP/p300/BRD4 Degrader-1
Brand:Targetmol
Description:PROTAC CBP/p300/BRD4 Degrader-1 is a dual-targeting PROTAC degrader with DC50 values of 8.8 pM for BRD4, 6.55 nM for CBP, and 1.05 nM for p300. It facilitates CRBN and proteasome-dependent degradation of BRD4 and CBP/p300, leading to the downregulation of c-Myc and acetyl-H3K27, and triggers apoptosis. As an antiproliferative and antitumor agent, PROTAC CBP/p300/BRD4 Degrader-1 demonstrates tumor growth inhibition in xenograft models. It is applicable in research on prostate and colorectal cancers.
Notice:Our products are intended for lab use only. For any other use, please contact us.
Chemical properties
Molecular weight:801.81
Formula:C41H42F3N7O7
Technical inquiry about: PROTAC CBP/p300/BRD4 Degrader-1
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