Asenapine Maleate

CAS: 85650-56-2

Ref. TR-A788025

Product Information

• Name: Asenapine Maleate
• Synonyms: 1H-Dibenz[2,3:6,7]oxepino[4,5-c]pyrrole, 5-chloro-2,3,3a,12b-tetrahydro-2-methyl-, (3aR,12bR)-rel-, (2Z)-2-butenedioate (1:1), 1H-Dibenz[2,3:6,7]oxepino[4,5-c]pyrrole, 5-chloro-2,3,3a,12b-tetrahydro-2-methyl-, trans-, (Z)-2-butenedioate (1:1), Org 5222, (3aR,12bR)-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1H-dibenzo[2,3:6,7]oxepino[4,5-c]pyrrole (2Z)-but-2-enedioate, (3aS,12bS)-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1H-dibenzo[2,3:6,7]oxepino[4,5-c]pyrrole (2Z)-but-2-enedioate, 1H-Dibenz[2,3:6,7]oxepino[4,5-c]pyrrole, 5-chloro-2,3,3a,12b-tetrahydro-2-methyl-, (3aR,12bR)-rel-, (2Z)-2-butenedioate (1:1), 1H-Dibenz[2,3:6,7]oxepino[4,5-c]pyrrole, 5-chloro-2,3,3a,12b-tetrahydro-2-methyl-, trans-, (Z)-2-butenedioate (1:1)

Description

Applications Asenapine Maleate, is a 5-HT receptor antagonist developed for the treatment of acute schizophrenia and bipolar mania. Antagonist of serotonin, norepinephrine, dopamine and histamine receptors.
Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package
References Tarazi. F.I., et al.: Drugs. Today., 45, 865 (2009); Boboaca, S.D., et al.: Int. J. Molec. Sci., 12, 4348 (2011); Audinot, V., et al.: Neuropsycopharmacol., 25, 410 (2001);

• Brand: TRC

Chemical properties

• Molecular weight: 401.84
• Formula: C₁₇H₁₆ClNO·C₄H₄O₄
• Color/Form: Neat
• InChI: 5-3(6)1-2-4(7)8/h2-8,14-15H,9-10H2,1H3, 1-2H,(H,5,6)(H,7,8)/b, 2-1-/t14-,15-, /m1./s1, InChI=1S/C17H16ClNO.C4H4O4/c1-19-9-14-12-4-2-3-5-16(12)20-17-7-6-11(18)8-13(17)15(14)10-19
• InChI key: InChIKey=GMDCDXMAFMEDAG-BTJKTKAUSA-N
• SMILES: CN1C[C@@H]2c3ccccc3Oc3ccc(Cl)cc3[C@H]2C1.O=C(O)/C=C\C(=O)O