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VR23
CAS:<p>VR23: Potent proteasome inhibitor; IC50: 1 nM trypsin, 50-100 nM chymotrypsin, 3 μM caspase-like.</p>Formula:C19H16ClN5O6SPurity:98.99% - 99.22%Color and Shape:SolidMolecular weight:477.88PF-06427878
CAS:<p>PF-06427878 is an orally active, potent and selective diacylglycerol acyltransferase 2 inhibitor.</p>Formula:C26H28N4O5Color and Shape:SolidMolecular weight:476.52Berotralstat HCl
CAS:Berotralstat HCl is a selective plasma kallikrein inhibitor, reducing pain and swelling in HAE by blocking bradykinin release.Formula:C30H28Cl2F4N6OColor and Shape:SolidMolecular weight:635.4886GPA512
CAS:<p>GPA512 is a prodrug of aliellalactone, inhibiting STAT3 and preventing the transcription of STAT3 regulated genes.</p>Formula:C17H25NO6SColor and Shape:SolidMolecular weight:371.45Bizine dihydrochloride
CAS:Bizine dihydrochloride is a potent LSD1 inhibitor in vitro, being selective versus monoamine oxidases A/B and the LSD1 homologue, LSD2.Formula:C18H25Cl2N3OColor and Shape:SolidMolecular weight:370.32LASSBio-1829 HCl
CAS:LASSBio-1829 HCl is an orally active IKK2 inhibitor.Formula:C25H19ClN4OColor and Shape:SolidMolecular weight:426.9V-125
CAS:V-125 is an agonist of retinoid X receptors.Formula:C23H30N2O2Color and Shape:SolidMolecular weight:366.5Indinavir monohydrate
CAS:Indinavir monohydrate is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability.Formula:C36H49N5O5Color and Shape:SolidMolecular weight:631.82BP-5-087
CAS:BP-5-087 is a STAT3 inhibitor, combining with BCR-ABL1 inhibition to overcome kinase-independent resistance in chronic myeloid leukemia.Formula:C36H30F8N2O6SColor and Shape:SolidMolecular weight:770.69Tofacitinib HCl
CAS:Tofacitinib (tasocitinib, CP-690550) is a JAK inhibitor impacting phosphorylation/activation of STATs with varied IC50 values.Formula:C16H21ClN6OColor and Shape:SolidMolecular weight:348.835UAWJ-247
CAS:UAWJ-247 is a SARS-CoV-2 Main Protease inhibitor (IC50 = 45 nM).Formula:C24H28N3NaO8SColor and Shape:SolidMolecular weight:541.55WNK463
CAS:WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all four WNK family members (WNK1/2/3/4).Formula:C21H24F3N7O2Purity:>99.99% - ≥95%Color and Shape:SolidMolecular weight:463.46Milvexian TFA
CAS:Milvexian (BMS-986177/JNJ-70033093) is a factor XIa inhibitor with Ki=44 nM for kallikrein, Ki=35 nM for chymotrypsin, 32% bioavailability.Formula:C30H26Cl2F5N9O4Color and Shape:SolidMolecular weight:742.49GSK1379767A
CAS:GSK1379767A is a dual inhibitor of BPTF and Brd4.Formula:C26H30N6O6Color and Shape:SolidMolecular weight:522.55NY0173
CAS:<p>NY0173 is a potent exchange protein activated by cAMP antagonists.</p>Formula:C18H15Cl3N4O2Color and Shape:SolidMolecular weight:425.7NY0123
CAS:NY0123 is an active EPAC antagonist with low micromolar inhibitory activity.Formula:C16H13Cl3N4O2Color and Shape:SolidMolecular weight:399.66Fadaltran
CAS:Fadaltran is an α2-adrenoreceptor antagonist.Formula:C24H29N5O2Color and Shape:SolidMolecular weight:419.52P7170
CAS:<p>P7170 is an anti-cancer agent active as an mTORC1/C2 and activin receptor-like kinase 1 (ALK1) inhibitor.</p>Formula:C21H16F3N9Color and Shape:SolidMolecular weight:451.42OAT-177
CAS:OAT-177 is a potent, selective, orally active acidic mammalian chitinase (AMCase) inhibitor.Formula:C19H29ClN6Color and Shape:SolidMolecular weight:376.93Sonidegib metabolite M25
CAS:Sonidegib metabolite M25 is a smoothened (SMO) antagonist.Formula:C26H26F3N3O4Color and Shape:SolidMolecular weight:501.5THIQ-40
CAS:THIQ-40: potent ERα antagonist, oral SERD with antitumor effects.Formula:C28H29NO3Color and Shape:SolidMolecular weight:427.53WZB117
CAS:WZB117 inhibits GLUT1; IC50 ~10μM slows A549 lung & MCF7 breast cancer cell growth.Formula:C20H13FO6Purity:99.03% - 99.18%Color and Shape:SolidMolecular weight:368.31LFS-829
CAS:LFS-829: small molecule, inhibits exportin-1, low nanomolar activity, orally reverses colitis in mice, low toxicity, promising for clinical trials.Formula:C13H9F6NOS2Color and Shape:SolidMolecular weight:373.34FFA3-Antagonist-6
CAS:FFA3-Antagonist-6 is a PAM-antagonist of the function of C3 at FFA3.Formula:C30H28N2O3Color and Shape:SolidMolecular weight:464.55NVP-BHS345
CAS:<p>NVP-BHS345 is a dual inhibitor of TORC1 and TORC2.</p>Formula:C25H20N6OColor and Shape:SolidMolecular weight:420.47Eptapirone fumarate
CAS:Eptapirone (F11440) is a strong 5HT1A agonist with high anxiolytic and antidepressant effects, more potent than buspirone and flesinoxan.Formula:C20H27N7O6Color and Shape:SolidMolecular weight:461.479YM-60828 dihydrochloride
CAS:YM-60828 dihydrochloride is a Factor Xa (FXa) inhibitor and anticoagulant used in the treatment of venous thromboembolic disease.Formula:C27H33Cl2N5O5SColor and Shape:SolidMolecular weight:610.55Desmethyl atenolol
CAS:Desmethyl atenolol is an impurity of Atenolol -- a selective β1 receptor antagonist.Formula:C13H20N2O3Color and Shape:SolidMolecular weight:252.31Methazolamide-d6
CAS:<p>Methazolamide-d6 is a GC/LC-MS standard for measuring methazolamide, a glaucoma drug that lowers eye pressure and fluid, reduces seizures, and combats ROS.</p>Formula:C5H2D6N4O3S2Color and Shape:SolidMolecular weight:242.31NPC-18915
CAS:NPC-18915 is a benzofuran compound, inhibitor of neutophil activation.Formula:C23H16O3Color and Shape:SolidMolecular weight:340.37ER-34122
CAS:<p>ER-34122, a novel orally available dual 5-lipoxygenase/cyclooxygenase inhibitor with potent anti-inflammatory activity.</p>Formula:C27H26ClN3O5Purity:>99.99%Color and Shape:SolidMolecular weight:507.96Navoximod phosphate
CAS:<p>Navoximod phosphate is an indoleamine 2,3-dioxygenase (IDO) inhibitor, immunomodulator and antineoplastic.</p>Formula:C18H24FN2O6PColor and Shape:SolidMolecular weight:414.37Z-IETD-FMK
CAS:<p>Z-IETD-FMK (Z-IE(OMe)TD(OMe)-FMK) is a selective caspase 8 inhibitor, which has cell permeable.</p>Formula:C30H43FN4O11Purity:95% - 99.81%Color and Shape:SolidMolecular weight:654.68Tinostamustine HCl
CAS:Tinostamustine (EDO-S101) is an alkylating HDACi fusion molecule, enhancing potency and overcoming drug resistance.Formula:C19H29Cl3N4O2Color and Shape:SolidMolecular weight:451.82GI261520A
CAS:GI261520A is a potent egfr/erbb2 dual inhibitorFormula:C22H19N3O2Color and Shape:SolidMolecular weight:357.41NC-2100
CAS:<p>NC-2100 is an aperoxisome proliferator-activated receptor-gamma (PPARgamma) activator.</p>Formula:C20H16N2O3SColor and Shape:SolidMolecular weight:364.42APC-366 HCl
CAS:APC-366 is a selective inhibitor of the mast cell tryptase that inhibits tryptase-induced histamine release from human tonsil and lung cells.Formula:C22H29ClN6O4Color and Shape:SolidMolecular weight:476.96AM92016
CAS:AM92016 is a specific blocker of the time dependent delayed rectifier potassium current. AM92016 does not show any β-adrenoceptor blocking activity.Formula:C26H30Cl2N2O6SColor and Shape:SolidMolecular weight:569.49NL-103
CAS:NL-103, a dual-targeting compound, inhibits HDACs & Hh pathway, countering vismodegib-resistant Smo mutations.Formula:C26H27Cl2N5O4Color and Shape:SolidMolecular weight:544.43AZD1446 HCl
CAS:AZD1446 (TC-6683) is a selective α4β2 receptor agonist, showing promise in treating cognitive deficits and Alzheimer's.Formula:C11H14Cl2N2O2Color and Shape:SolidMolecular weight:277.15AQ 148
CAS:<p>AQ 148 is a potent competitive inhibitor of HIV-1 PR.</p>Formula:C30H37N3O4Color and Shape:SolidMolecular weight:503.63Atrasentan sodium
CAS:Atrasentan (ABT-627) is an oral ETA receptor blocker with potential cancer-fighting properties, inhibiting angiogenesis and tumor growth.Formula:C29H37N2NaO6Color and Shape:SolidMolecular weight:532.61Enecadin HCl
CAS:<p>Enecadin HCl is a voltage-dependent sodium and calcium channel blocker.</p>Formula:C21H29ClFN3OColor and Shape:SolidMolecular weight:393.93Z-VAD-FMK
CAS:<p>Z-VAD-FMK (Caspase Inhibitor VI) is a broad-spectrum inhibitor of caspases.Z-VAD-FMK binds to activated caspases and inhibits apoptosis.Z-VAD-FMK does not</p>Formula:C21H28FN3O7Purity:98.24% - 99.79%Color and Shape:SolidMolecular weight:453.46VU590 HCl
CAS:VU590 is a small molecule inhibitor of KCNJ1 (IC50 = 294 nM).Formula:C24H34Cl2N4O7Color and Shape:SolidMolecular weight:561.457S 16020-2
CAS:<p>S 16020-2 is an olivacine derivative, and DNA topoisomerase II inhibitor endowed with a remarkable antitumor activity against various experimental tumors.</p>Formula:C22H26Cl2N4O2Color and Shape:SolidMolecular weight:449.376DDR1-IN-1 dihydrochloride
CAS:DDR1-IN-1 dihydrochloride: potent DDR1 kinase inhibitor; IC50=105 nM; 4x less effective on DDR2 (IC50=413 nM).Formula:C30H33Cl2F3N4O3Color and Shape:SolidMolecular weight:625.51Galloflavin Potassium
CAS:<p>Galloflavin Potassium is an inhibitor of lactate dehydrogenase.</p>Formula:C12H5KO8Color and Shape:SolidMolecular weight:316.26XM 412
CAS:XM 412, also known as DMP 450, is an HIV protease inhibitor.Formula:C35H44N4O9S2Color and Shape:SolidMolecular weight:728.876IND8
CAS:IND8 is a selective and potent α7-nAChR agonist.Formula:C17H19N5Color and Shape:SolidMolecular weight:293.37Clorgyline
CAS:Clorgyline,M&B 9302, an irreversible and selective MAO-A inhibitor with the advantages of oral activity and blood-brain barrier permeability, antidepressant.Formula:C13H15Cl2NOPurity:98.39%Color and Shape:SolidMolecular weight:272.17Pimodivir tosylate
CAS:Pimodivir (VX-787/JNJ-872) inhibits influenza by targeting PB2, with KD 24 nM and EC50 1.6 nM, effective against various strains, including NAI-resistant ones.Formula:C27H27F2N5O5SColor and Shape:SolidMolecular weight:571.6SB1-B-57
CAS:SB1-B-57 is an USP14 inhibitor.Formula:C22H22N4O2Color and Shape:SolidMolecular weight:374.44Nepicastat hydrochloride monohydrate
CAS:<p>Nepicastat hydrochloride monohydrate is an inhibitor of dopamine beta-hydroxylase, an enzyme that catalyzes the conversion of dopamine to norepinephrine.</p>Formula:C14H18ClF2N3OSColor and Shape:SolidMolecular weight:349.82ZM241385
CAS:<p>ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.</p>Formula:C16H15N7O2Purity:97.02% - 99.69%Color and Shape:SolidMolecular weight:337.34FT-1101 free base
CAS:FT-1101 is a potent, selective oral BET inhibitor disrupting gene expression to inhibit tumor growth.Formula:C26H34N4O2Color and Shape:SolidMolecular weight:434.57U 95133
CAS:<p>U 95133 is a potent, broad-spectrum nonnucleoside reverse transcriptase inhibitor of drug-resistant isolates of human immunodeficiency virus type 1.</p>Formula:C25H34N6O3SColor and Shape:SolidMolecular weight:498.64BRD7929
CAS:BRD7929 is a multistage antimalarial inhibitor for single-dose treatment of malaria in mouse models.Formula:C33H38N4O2Color and Shape:SolidMolecular weight:522.68Clonazoline
CAS:Clonazoline: imidazoline-derived alpha-agonist for coronary dilation, nasal decongestion, and vasoconstriction.Formula:C14H13ClN2Color and Shape:SolidMolecular weight:244.72Omiloxetine
CAS:Omiloxetine, an SSRI developed by Ferrer Internacional, was shelved in 2005 after preclinical trials.Formula:C27H25F2NO4Color and Shape:SolidMolecular weight:465.49IMB-YH-8
CAS:<p>IMB-YH-8 is an inhibitor of protein kinase B (PknB), inhibiting PknB auto-phosphorylation and the phosphorylation of GarA by PknB in a dose-dependent manner.</p>Formula:C12H12O4Color and Shape:SolidMolecular weight:220.22ISP-VT
CAS:<p>ISP-VT is a Novel inhibitor of COX and neutrophil migration.</p>Formula:C11H14O4Color and Shape:SolidMolecular weight:210.23PEG300
CAS:PEG300 (Polyethylene glycol 300) is a polymer formed from repeating units of ethylene glycol that is water soluble, low immunogenicity, and biocompatible.Formula:C5H15NO2Purity:FW~300 - mw~300Color and Shape:Transparent Liquid ViscousMolecular weight:10000Tazomeline citrate
CAS:Tazomeline citrate is used for alzheimer's disease treatment (Cholinergic Agonist).Formula:C20H31N3O7S2Color and Shape:SolidMolecular weight:489.602Dibefurin
CAS:Dibefurin blocks calcineurin, a calcium-dependent enzyme, reducing T lymphocyte activation.Formula:C18H16O8Color and Shape:SolidMolecular weight:360.31Ethonafide
CAS:Ethonafide, a non-cardiotoxic anthracene derivative, potently fights multidrug-resistant cancers and halts prostate cancer growth at nanomolar levels.Formula:C22H22N2O3Color and Shape:SolidMolecular weight:362.42UA8967
CAS:UA8967, a non-selective, membrane-active anti-tumor compound, exhibits IC50s of 12-61 μM across various cancer cells.Formula:C20H23N3Color and Shape:SolidMolecular weight:305.42Bupivacaine tartrate
CAS:<p>Bupivacaine blocks various K channels and Na channels, acting as an anesthetic; high doses may cause neurotoxicity.</p>Formula:C22H34N2O7Color and Shape:SolidMolecular weight:438.521L-159884
CAS:L-159884 is a radiolabelled, nonpeptide angiotensin II antagonist that is useful for angiotensin II, AT1 receptor imagingFormula:C31H30N4O4SColor and Shape:SolidMolecular weight:554.66Amentoflavone hexaacetate
CAS:<p>Amentoflavone hexaacetate is a 3,5-cyclic nucleotide phosphodiesterase inhibitor. It has anti-angiogenic and anti-metastatic effects.</p>Formula:C42H30O16Color and Shape:SolidMolecular weight:790.68BPIQ-I
CAS:<p>BPIQ-I (PD 159121), an ATP-competitive EGFR tyrosine kinase inhibitor, exhibits potent anti-proliferative activity.</p>Formula:C16H12BrN5Color and Shape:SolidMolecular weight:354.2AT-1015 free base
CAS:AT-1015 free base is a serotonin (5-HT)2 receptor antagonist that blocks vascular and platelet 5-HT2A receptors.Formula:C29H33N3O2Color and Shape:SolidMolecular weight:455.59Laromustine
CAS:<p>Laromustine (VNP40101M) is a sulfonyl hydrolysis alkylation prodrug for cancer treatment with significant anticancer activity, inhibiting thioredoxin reductase.</p>Formula:C6H14ClN3O5S2Purity:≥98%Color and Shape:SolidMolecular weight:307.78FPTI
CAS:FPTI is an inhibitor against SYT-SSX1 fusion protein in synovial sarcoma which down-regulates SYT-SSX1 and modulates its downstream target genes.Formula:C15H10FN5Color and Shape:SolidMolecular weight:279.27Osanetant HCl
CAS:Osanetant HCl is the (R)-enantiomer; neurokinin-3 receptor antagonistFormula:C35H42Cl3N3O2Color and Shape:SolidMolecular weight:643.093,4-Dephostatin
CAS:3,4-Dephostatin is an inhibitor of the interactions of CFTR-associated ligand (CAL) and PSD-95/Dlg1/ZO-1 (PDZ) domain.Formula:C7H8N2O3Color and Shape:SolidMolecular weight:168.15Efegatran HCl
CAS:Efegatran (GYKI-14166, RGH-2958, LY294468) is a thrombin inhibitor in development by IVAX for thromboembolic disorders.Formula:C21H34Cl2N6O3Color and Shape:SolidMolecular weight:489.442Cacospongionolide B
CAS:<p>Cacospongionolide B from Fasciospongia cavernosa inhibits secretory phospholipase A2, curbing inflammation.</p>Formula:C25H36O4Color and Shape:SolidMolecular weight:400.55Cemadotin hydrochloride
CAS:Cemadotin hydrochloride (LU103793) is a synthetic mitosis inhibitor derived from Dolastatin 15 for treating solid tumors.Formula:C35H57ClN6O5Color and Shape:SolidMolecular weight:677.33Isonitrosoacetone
CAS:<p>Isonitrosoacetone is an acetylcholinesterase reactivator.</p>Formula:C3H5NO2Color and Shape:SolidMolecular weight:87.08HX-600
CAS:HX-600 is a synthetic agonist for the RXR-Nurr1 heterodimer complex. HX-600 prevents ischemia-induced neuronal damage.Formula:C29H30N2O2Color and Shape:SolidMolecular weight:438.56FPL-64170XX
CAS:FPL-64170XX is a selective inhibitor of the enzyme 5-lipoxygenase.Formula:C19H19N3O2Color and Shape:SolidMolecular weight:321.37CP-64434 hydrate
CAS:CP-64434 hydrate is an antibiotic; anti-proliferative HDAC inhibitor.Formula:C37H70N2O12Color and Shape:SolidMolecular weight:734.96Qingyangshengenin
CAS:Qingyangshengenin (Cynanchagenin) is a steroid used in the preparation of antiepileptic agents.Formula:C28H36O8Purity:99.62% - 99.89%Color and Shape:SolidMolecular weight:500.58Caparratriene
CAS:<p>Caparratriene: a new sesquiterpene from Ocotea caparrapi, may inhibit CEM leukemia cell growth.</p>Formula:C15H26Color and Shape:SolidMolecular weight:206.37KY 234
CAS:<p>KY 234 is a thromboxane synthetase antagonist.</p>Formula:C33H35N5O2Color and Shape:SolidMolecular weight:533.676SC 8109
CAS:<p>SC 8109 is an aldosterone antagonist.</p>Formula:C21H28O3Color and Shape:SolidMolecular weight:328.45TAC 363
CAS:TAC 363 is a tachykinin NK-2-receptor antagonist.Formula:C38H48N8O6Color and Shape:SolidMolecular weight:712.84JRN73958
CAS:JRN73958, a precursor to scytonemin (a cyanobacteria pigment), inhibits cell growth in multiple myeloma, acting as a Plk1 inhibitor.Formula:C36H24N2O4Color and Shape:SolidMolecular weight:548.59PD159206
CAS:<p>PD-159206 is a nucleocapsid inhibitor. It exhibits good antiviral activity against HIV.</p>Formula:C26H32N2O6S2Color and Shape:SolidMolecular weight:532.674991W93
CAS:4991W93 is a 5HT(1B/1D) agonist that blocks neurogenic inflammation and inhibits CGRP release.Formula:C18H23N3O2Color and Shape:SolidMolecular weight:313.39Desmethylene Tadalafil
CAS:Desmethylene Tadalafil is a phosphodiesterase 5 inhibitor.Formula:C21H19N3O4Color and Shape:SolidMolecular weight:377.39Rehmannioside D
CAS:Rehmannioside D is a carotenoid glycoside that existed in the roots of Rehmannia glutinosa.Formula:C27H42O20Purity:99.91% - 99.96%Color and Shape:SolidMolecular weight:686.61Demeclocycline calcium
CAS:<p>Demeclocycline, a semisynthetic antibiotic from S. aureofaciens, blocks protein synthesis and vasopressin, causing diuresis.</p>Formula:C42H40CaCl2N4O16Color and Shape:SolidMolecular weight:967.77Hexestrol diphosphate tetrasodium
CAS:Hexestrol diphosphate tetrasodium: synthetic ER agonist, may cause cancer, inhibits microtubule assembly, leads to mitotic arrest and DNA adducts.Formula:C18H24O8P2·xNaColor and Shape:SolidMolecular weight:518.26RU1968 bis-TFA salt
CAS:<p>RU1968 bis-TFA salt is an inhibitor of the sperm-specific Ca2+ channel CatSper, thereby inhibiting human Slo3 with about 15-fold lower potency than CatSper.</p>Formula:C24H38N2OColor and Shape:SolidMolecular weight:370.57R 1714
CAS:<p>R 1714 is an orally available cholesterol-lowering compound.</p>Formula:C24H38N2OPurity:99.61%Color and Shape:SoildMolecular weight:370.57R 1714 dihydrochloride
CAS:R 1714 dihydrochloride is an orally available cholesterol-lowering compound.Formula:C24H40Cl2N2OPurity:97.76%Color and Shape:SoildMolecular weight:443.49Nordimaprit
CAS:Nordimaprit is effective agonist in the inhibition of lymphocyte activation.Formula:C5H13N3SColor and Shape:SolidMolecular weight:147.24FE-999011
CAS:FE-999011 is a dipeptidyl peptidase IV inhibitor.Formula:C11H19N3OColor and Shape:SolidMolecular weight:209.29
