
Microtúbulo associado
Os inibidores de proteínas associadas aos microtúbulos têm como alvo as proteínas que interagem com os microtúbulos, os componentes estruturais do citoesqueleto da célula que são essenciais para a divisão celular. Essas proteínas regulam a estabilidade e a dinâmica dos microtúbulos durante a mitose. A inibição de proteínas associadas aos microtúbulos pode interromper a função dos microtúbulos, levando à parada do ciclo celular e à apoptose, especialmente em células cancerígenas de rápida divisão. Esses inibidores são amplamente utilizados na pesquisa do câncer e no desenvolvimento de medicamentos. Na CymitQuimica, oferecemos uma ampla gama de inibidores de proteínas associadas aos microtúbulos de alta qualidade para apoiar sua pesquisa em divisão celular, dinâmica do citoesqueleto e terapia do câncer.
Foram encontrados 273 produtos de "Microtúbulo associado"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Tubulin polymerization-IN-30
CAS:Compound 6e inhibits tubulin polymerization, disrupts microtubules, halts G2/M phase, and targets HeLa, SGC-7901, A549 with low IC50.Fórmula:C22H25N5O3Cor e Forma:SolidPeso molecular:407.47Tubulin polymerization-IN-15
CAS:Tubulin polymerization-IN-15 (compound 4) is a highly effective inhibitor of tubulin polymerization, with significant potential in cancer research [1].Fórmula:C18H17N3O4Cor e Forma:SolidPeso molecular:339.35Tubulin polymerization-IN-20
CAS:Tubulin aggregation-IN-20, a potent inhibitor, may be studied for breast and drug-resistant colon cancers.Fórmula:C25H24FNO5Cor e Forma:SolidPeso molecular:437.46Tubulin inhibitor 18
CAS:"Tubulin inhibitor 18 (5j), a potent chalcone, uniquely structured for cancer research."Fórmula:C22H26O5Cor e Forma:SolidPeso molecular:370.44Tubulin/MMP-IN-1
Tubulin/MMP-IN-1 inhibits tubulin, MMP, and cancer cell growth; disrupts cell cycles and induces apoptosis.Fórmula:C38H44NO9PCor e Forma:SolidPeso molecular:689.73Synstab A
CAS:Synstab A is a microtubule stabilizer.Fórmula:C15H13BrCl3N3O3SCor e Forma:SolidPeso molecular:501.61Tubulin inhibitor 12
CAS:New tubulin inhibitor 12 (Hit 9); potent anti-cancer agent; IC50=25.3 μM; strong anti-tumor effect.Fórmula:C24H20N2OCor e Forma:SolidPeso molecular:352.43Tau tracer 1
CAS:Tau tracer 1 is a radiopharmaceutical for imaging Tau aggregates linked to neurodegenerative disease diagnosis.Fórmula:C34H23N5O2Cor e Forma:SolidPeso molecular:533.591SB-216
CAS:SB-216, a potent anti-cancer compound, inhibits tubulin polymerization and curbs growth in various cancer cells.
Fórmula:C17H18N4O2Pureza:99.70%Cor e Forma:SolidPeso molecular:310.35CID-663143
CAS:CID-663143 inhibits cancer cell growth and shows microtubule-binding activity.Fórmula:C19H18N4O2SPureza:99.68% - 99.77%Cor e Forma:SolidPeso molecular:366.44Ref: TM-T23889
1mg50,00€5mg105,00€1mL*10mM (DMSO)109,00€10mg155,00€25mg224,00€50mg315,00€100mg424,00€200mg560,00€Erbulozole
CAS:Erbulozole (R 55104) is a synthetic microtubule inhibitor with anti-invasive activity that induces Wernicke's encephalopathy-like neurotoxicity.Fórmula:C24H27N3O5SPureza:99.88%Cor e Forma:SolidPeso molecular:469.55LY3372689
CAS:LY3372689 (Formulaic Ia) is an orally active O-GlcNAcase (OGA) enzyme inhibitor for tau protein-based disorders including Alzheimer's disease.
Fórmula:C16H22FN5O3SPureza:99.43% - 99.53%Cor e Forma:SolidPeso molecular:383.44TCS 2210
CAS:TCS 2210 promotes neuronal differentiation in stem cells, boosting β-III tubulin and enolase markers.Fórmula:C18H17N3O3Pureza:98.62%Cor e Forma:SolidPeso molecular:323.35Ref: TM-T23446
1mg86,00€2mg116,00€5mg172,00€1mL*10mM (DMSO)177,00€10mg259,00€25mg444,00€50mg610,00€100mg867,00€500mg1.738,00€Tubulin inhibitor 8
CAS:Tubulin inhibitor 8 blocks tubulin polymerization, stunts K562 cancer cell growth; IC50: 0.73 μM, 14 nM.
Fórmula:C21H14N2O3Pureza:98.51% - 99.87%Cor e Forma:SolidPeso molecular:342.35Rosabulin
CAS:v Rosabulin (STA 5312) is an orally active microtubule inhibitor with potency.Fórmula:C22H16N4O2SPureza:98.86%Cor e Forma:SolidPeso molecular:400.45Ref: TM-T16788
1mg92,00€5mg230,00€1mL*10mM (DMSO)251,00€10mg344,00€25mg623,00€50mg888,00€100mg1.341,00€Tubulin polymerization-IN-52
CAS:Tubulin polymerization-IN-52 (compound SC23) effectively inhibits tubulin polymerization, exhibiting an IC50 value of 2.9 μM [1].Fórmula:C21H18F3N5O3Cor e Forma:SolidPeso molecular:445.39JG-23
CAS:JG-23, a 4-chloro-modified analog, effectively induces t-tau degradation and demonstrates robust metabolic stability, exhibiting an extended half-life (T1/2) ofFórmula:C19H16ClN3OS2Cor e Forma:SolidPeso molecular:401.93Valecobulin hydrochloride
CAS:Valecobulin hydrochloride (CKD-516 hydrochloride) is the valine prodrug and vasoblocker of S516.Cost-effective and quality-assured.Fórmula:C26H29ClN6O5SPureza:99.52%Cor e Forma:SolidPeso molecular:573.06Ref: TM-T13278
1mg84,00€5mg161,00€1mL*10mM (DMSO)197,00€10mg245,00€25mg406,00€50mg572,00€100mg772,00€200mg1.035,00€Anticancer agent 40
CAS:Anticancer agent 3e targets SKBR-3, SKOV-3, PC-3, U-87 (IC50 ~0.95 nM) and HDF cells (IC50: 2.13 nM).Fórmula:C25H29NO6Cor e Forma:SolidPeso molecular:439.5Tubulin inhibitor 25
CAS:Potent Tubulin inhibitor 25: IC50 0.98 μM, blocks HT29 cell growth, hinders cell migration & microtubule formation, anti-angiogenic.Fórmula:C26H22O8Cor e Forma:SolidPeso molecular:462.45
