Enzima
Os inibidores de enzimas são moléculas que se ligam a enzimas e diminuem sua atividade. Esses inibidores são amplamente utilizados em pesquisas para estudar a cinética enzimática, regulação e o papel de enzimas específicas nas vias metabólicas. Os inibidores de enzimas também são cruciais no desenvolvimento de medicamentos, pois muitos agentes terapêuticos funcionam inibindo enzimas envolvidas em processos patológicos. Ao direcionar enzimas, esses inibidores podem modular vias bioquímicas e oferecer tratamentos potenciais para várias doenças. Na CymitQuimica, oferecemos uma ampla seleção de inibidores de enzimas de alta qualidade para apoiar sua pesquisa em bioquímica, farmacologia e descoberta de medicamentos.
Subcategorias de "Enzima"
- Anidrase carbónica(177 produtos)
- Hidroxilase(30 produtos)
- MPO(2 produtos)
- Redutase(52 produtos)
- Tirosinase(67 produtos)
Foram encontrados 3586 produtos de "Enzima"
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Acipimox
CAS:<p>Acipimox (K-9321), a niacin derivative, treats hyperlipidemia in type 2 diabetics.</p>Fórmula:C6H6N2O3Pureza:98.98%Cor e Forma:Low Yellow Liquid Or CrystallinePeso molecular:154.12Arbutin
CAS:<p>Arbutin, a bearberry extract, blocks melanin by inhibiting tyrosinase.</p>Fórmula:C12H16O7Pureza:99.58% - 99.93%Cor e Forma:Colorless Elongated Prisms From Moist Ethyl Acetate White PowderPeso molecular:272.255-Feruloylquinic acid
CAS:<p>5-Feruloylquinic acid, a potent Sirt1 activator, may aid in developing anti-aging drugs.</p>Fórmula:C17H20O9Pureza:99.03%Cor e Forma:SolidPeso molecular:368.34KW-2450 Formate
<p>KW-2450 Formate is an IGF-1R/IR tyrosine kinase inhibitor with antitumor effects that acts through inhibition of Aurora A and B kinases.KW-2450 Formate inhibits the growth of TNBC xenografts and induces tetraploid accumulation.</p>Fórmula:C29H31N5O5SPureza:99.28%Cor e Forma:SolidPeso molecular:561.654-Chlorosalicylic acid
CAS:<p>4-Chlorosalicylic acid (4-Chloro-2-hydroxybenzoic acid, 4-chloro salicylic acid) is antimicrobial compositions comprising a metal salt and a benzoic acid analog</p>Fórmula:C7H5ClO3Pureza:98.59%Cor e Forma:Off-White To Light Beige PowderPeso molecular:172.57Telotristat ethyl
CAS:<p>Telotristat ethyl (LX1606) is a orally-delivered inhibitor of tryptophan hydroxylase that reduces serotonin production.</p>Fórmula:C27H26ClF3N6O3Pureza:98% - 99.89%Cor e Forma:White SolidPeso molecular:574.98Topiramate
CAS:<p>Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.</p>Fórmula:C12H21NO8SPureza:99.79% - 99.92%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:339.36Methocarbamol
CAS:<p>Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.</p>Fórmula:C11H15NO5Pureza:99.96%Cor e Forma:Crystals From Benzene SolidPeso molecular:241.24ACT-678689
CAS:<p>ACT-678689 (Compound Example 1.53.4) (Compound Example 1.53.4) is a tryptophan hydroxylase (TPH) inhibitor with an IC50 of 8 nM[1].</p>Fórmula:C23H22ClFN6O4S2Pureza:99.46%Cor e Forma:SolidPeso molecular:565.04Benzthiazide
CAS:<p>Benzthiazide treats edema and hypertension by promoting diuresis and inhibiting kidney Na+/Cl- reuptake, but may reduce potassium and raise uric acid.</p>Fórmula:C15H14ClN3O4S3Pureza:99.34% - 99.79%Cor e Forma:Crystals From Acetone SolidPeso molecular:431.94Methazolamide
CAS:<p>Methazolamide (CL 8490) is a carbonic anhydrase inhibitor that is used as a diuretic and in the treatment of glaucoma.</p>Fórmula:C5H8N4O3S2Pureza:99.31% - 99.77%Cor e Forma:Crystals From Water SolidPeso molecular:236.27Tioxolone
CAS:<p>Tioxolone is a metalloenzyme carbonic anhydrase I inhibitor.</p>Fórmula:C7H4O3SPureza:97.79%Cor e Forma:Light Yellow To Beige PowderPeso molecular:168.17Flanvotumab
CAS:<p>Flanvotumab (IMC-20D7S) is a humanized antibody targeting TYRP1 with strong antitumor effects via NK cells and ADCC.</p>Pureza:> 95%Cor e Forma:LiquidPeso molecular:145.42 kDap-Ethynylphenylalanine hydrochloride
CAS:<p>p-Ethynylphenylalanine hydrochloride (4-Ethynyl-L-phenylalanine HCL) is a novel, potent and specific inhibitor of TPH[1].</p>Fórmula:C11H12ClNO2Pureza:99.03%Cor e Forma:SolidPeso molecular:225.67Fenclonine
CAS:<p>Fenclonine (CP-10188) is a selective and irreversible inhibitor of tryptophan hydroxylase, a rate-limiting enzyme in the biosynthesis of serotonin.</p>Fórmula:C9H10ClNO2Pureza:98.81% - >99.99%Cor e Forma:Crystals From Methanol White SolidPeso molecular:199.63Zonisamide
CAS:<p>Zonisamide (AD 810), a sulfonamide anticonvulsant, is approved for use as an adjunctive treatment in adults with partial-onset seizures.</p>Fórmula:C8H8N2O3SPureza:99.05% - 99.9%Cor e Forma:Off-White PowderPeso molecular:212.23Actarit
CAS:<p>Actarit (4-acetylaminophenylacetic acid) is an anti-inflammatory drug.</p>Fórmula:C10H11NO3Pureza:99.64% - 99.74%Cor e Forma:White Or Off-White Crystal Or Crystalline SolidPeso molecular:193.2Brinzolamide
CAS:<p>Brinzolamide (AL-4862) is a Carbonic Anhydrase Inhibitor. The mechanism of action of brinzolamide is as a Carbonic Anhydrase Inhibitor.</p>Fórmula:C12H21N3O5S3Pureza:99.84% - >99.99%Cor e Forma:Crystalline SolidPeso molecular:383.51pNNP
CAS:<p>pNNP is a substrate for PP2C assays and inhibits β-carbonic anhydrase, α-carbonate dehydrogenase, and H. pylori.</p>Fórmula:C6H6NO6PPureza:99.73%Cor e Forma:SolidPeso molecular:219.09Tyrosinase-IN-38
<p>Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.</p>Cor e Forma:Odour SolidPotassium iodide
CAS:<p>Potassium iodide 用于治疗过度活跃的甲状腺，并保护甲状腺免受吞咽或吸入放射性碘的辐射影响。可在意外接触放射性碘后或服用含放射性碘的药物前后使用。</p>Fórmula:IKCor e Forma:White Solid CrystallinePeso molecular:166.01TPH1-IN-1
<p>TPH1-IN-1 (compound 40) is a xanthine derivative that serves as an inhibitor of tryptophan hydroxylase TPH1, with an IC50 of 110.1 nM.</p>Fórmula:C21H18N6O4SCor e Forma:SolidPeso molecular:450.47CA inhibitor 2
<p>Compound 4H is a potent carbonic anhydrase inhibitor with an IC50 value of 0.033 μM [1].</p>Fórmula:C7H9N7O3S3Pureza:98%Cor e Forma:SolidPeso molecular:335.392-Methoxy-4-propylphenol
CAS:<p>2-Methoxy-4-propylphenol is an inhibitor of human carbonic anhydrase isoenzymes 1/2/9/12 and has antifungal activity.</p>Fórmula:C10H14O2Cor e Forma:SolidPeso molecular:166.22CAIX/CAXII-IN-3
<p>CAIX/CAXII-IN-3 (compound 11) serves as an inhibitor for CAIX/CAXII, exhibiting an IC50 value of less than 65 nM. Additionally, this compound effectively inhibits the proliferation of human melanoma cells.</p>Cor e Forma:Odour SolidCalmodulin-dependent Protein Kinase II fragment 290-309
CAS:Fórmula:C103H185N31O24SPeso molecular:2273.83hCA/VEGFR-2-IN-1
<p>hCA/VEGFR-2-IN-1 (compound 13a) is a potent dual inhibitor targeting both Carbonic Anhydrase (CA) IX/XII and Vascular Endothelial Growth Factor Receptor 2 (</p>Fórmula:C21H17FN6O3SPureza:98%Cor e Forma:SolidPeso molecular:452.46Tyrosinase-IN-13
<p>Tyrosinase-IN-13 (compound 3c), stemming from Flurbiprofen, acts as a potent non-competitive inhibitor of tyrosinase, exhibiting IC50 and Ki values of 68 μM and</p>Fórmula:C23H18ClFN4OSPureza:98%Cor e Forma:SolidPeso molecular:452.935,6-Dihydro-2H-pyran-2-one
CAS:<p>5,6-Dihydro-2H-pyran-2-one is a carbonic anhydrase 1/9 inhibitor that inhibits KB cell viability.</p>Fórmula:C5H6O2Cor e Forma:SolidPeso molecular:98.1hCAI/II/IV-IN-28
CAS:<p>hCAI/II/IV-IN-28(WAY-638358) is a potent carbonic anhydrase inhibitor with potential anticonvulsant activity.</p>Fórmula:C14H15N3O3SPureza:96.48%Cor e Forma:SolidPeso molecular:305.35L-Lactate Dehydrogenase from bovine heart, powder, approx. 300 U/mg
CAS:Cor e Forma:Lyophilised powderhCAIX/VII-IN-1
<p>hCAIX/VII-IN-1 is a selective inhibitor of human carbonic anhydrase isoforms VII and IX.</p>Fórmula:C16H13BFN3O3Pureza:98%Cor e Forma:SolidPeso molecular:325.12,3-Dihydroisoginkgetin
CAS:<p>2,3-Dihydroisoginkgetin is a Tyrosinase inhibitor with 36.84% inhibition at 0.1 mM.</p>Fórmula:C32H24O10Pureza:98%Cor e Forma:SolidPeso molecular:568.53Bendroflumethiazide
CAS:<p>Bendroflumethiazide (Naturetin) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE. It has been used in the treatment of familial hyperkalemia, hypertension, edema, and urinary tract disorders. (From Martindale, The Extra Pharmacopoeia, 30th ed, p810)</p>Fórmula:C15H14F3N3O4S2Pureza:98% - >99.99%Cor e Forma:Crystals From Dioxane SolidPeso molecular:421.41(Z)-SU14813
CAS:<p>(Z)-SU14813 is a tyrosine kinase inhibitor with anticardiogenic and antitumor activity.</p>Fórmula:C23H27FN4O4Pureza:98.18%Cor e Forma:SolidPeso molecular:442.48SH7s
<p>SH7s is an effective carbonic anhydrase inhibitor, exhibiting Ki values of 15.9 nM for hCA IX and 55.2 nM for hCA XII. Additionally, SH7s acts as a hypoxia-mediated chemosensitizer in colorectal cancer cells.</p>Fórmula:C24H19ClF3N5O4SCor e Forma:SolidPeso molecular:565.95hTYR/AbTYR-IN-1
CAS:<p>hTYR/AbTYR-IN-1 is a dual hTYR/AbTYR inhibitor with inhibitory effects on hTYR and AbTYR, with IC50s of 5.4 μM and 3.52 μM, respectively.</p>Fórmula:C18H20N2O3Pureza:99.59%Cor e Forma:SoildPeso molecular:312.36hCAIX-IN-19
<p>hCAIX-IN-19 is a sulfonamide inhibitor with an inhibition constant (KI) of 6.2 nM for hCAIX, exhibiting significant selectivity towards hCAIX over hCAI (hCA I/</p>Cor e Forma:Odour SolidCarbonic anhydrase inhibitor 15
<p>Carbonic Anhydrase Inhibitor 15 (Compound 8), with an inhibitory constant (K_i) of 8.5 nM for hCA II, exhibits analgesic effects [1].</p>Fórmula:C27H33N5O2S2Pureza:98%Cor e Forma:SolidPeso molecular:523.71GZ22-4
<p>GZ22-4 is a near-infrared (NIR) fluorescent probe with a high affinity for carbonic anhydrase IX (CAIX), exhibiting a dissociation constant (Kd) of 0.2 nM. It is applicable in studies for visualizing CAIX-positive tumors.</p>Fórmula:C88H126F3N6NaO24S4Peso molecular:1858.75561Tyrosinase-IN-19
<p>Tyrosinase-IN-19 (compound 9), a competitive tyrosinase inhibitor, exhibits potent antioxidant activities by neutralizing ROS, ABTS+, and DPPH radicals and</p>Pureza:98%Cor e Forma:Odour SolidATP2A2 Protein, Human, Recombinant (C-His)
<p>ATP2A2 Protein, Human, Recombinant (C-His) is expressed in E.</p>Pureza:95%Cor e Forma:SoildPeso molecular:55.2 kDa (Predicted)KRAS Protein, Human, Recombinant (G12C, His)
<p>KRAS Protein, Human, Recombinant (G12C, His) is expressed in E.</p>Pureza:> 99.9% - Greater than 95% as determined by reducing SDS-PAGE.Cor e Forma:Lyophilized PowderPeso molecular:26 KDa (reducing condition)Tyrosinase
CAS:<p>Tyrosinase (Polyphenol oxidase) is a key rate-limiting enzyme encoded by the TYR gene that controls melanin production and catalyzes tyrosine oxidation.</p>Cor e Forma:SolidDOTA-XYIMSR-01
CAS:<p>DOTA-XYIMSR-01 is a molecular probe targeting CAIX, capable of being labeled with 177Lu for the treatment and localization of malignant gliomas. The uptake of [177Lu]Lu-XYIMSR-01 in U87MG tumors is 6.19% injected dose per gram (% ID/g), with a tumor-to-muscle uptake ratio of 20.14. In an orthotopic glioma model, co-administration with temozolomide significantly enhances survival rates and inhibits tumor growth in mice. DOTA-XYIMSR-01 shows potential for research in the field of cancer treatment.</p>Fórmula:C61H88N16O22S2Cor e Forma:SolidPeso molecular:1461.57Dorzolamide
CAS:<p>Dorzolamide is an anti-glaucoma agent and is a carbonic anhydrase inhibitor.</p>Fórmula:C10H16N2O4S3Pureza:98%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:324.44Anhydrotetracycline hydrochloride
CAS:<p>Anhydrotetracycline (hydrochloride) is a potent competitive inhibitor of broad-spectrum tetracycline destructase enzymes.</p>Fórmula:C22H23ClN2O7Pureza:98.90%Cor e Forma:SolidPeso molecular:462.88VM4-037
CAS:<p>VM4-037 is a PET imaging agent used for carbonic anhydrase IX.</p>Fórmula:C26H29FN6O7S2Cor e Forma:SolidPeso molecular:620.67hCAIX/XII-IN-7
<p>Compound 3e (hCAIX/XII-IN-7) is a potent inhibitor of human carbonic anhydrase (hCA) isozymes IX and XII, displaying inhibitory constants (Kis) of 503.7 nM for</p>Fórmula:C17H14N6O3SPureza:98%Cor e Forma:SolidPeso molecular:382.4CA Ⅱ-IN-1
<p>CAⅡ-IN-1 (compound 2i) is an inhibitor of the CA Ⅱ isozyme, exhibiting an IC50 of 0.44 µM. This compound is utilized in metabolic research.</p>Fórmula:C18H19NO6SCor e Forma:SolidPeso molecular:377.41AV22-149
<p>AV22-149 (compound 22) is an inhibitor of Carbonic Anhydrase .</p>Fórmula:C23H28F3N3O6S2Cor e Forma:SolidPeso molecular:563.61hCAI/II-IN-10
<p>hCAI/II-IN-10 (Compound 5d) is an inhibitor of human carbonic anhydrase I and II (hCA I and hCA II), with IC50 values of 4.32 nM and 3.89 nM, respectively.</p>Fórmula:C24H17Cl2N3O3S2Cor e Forma:SolidPeso molecular:530.446Chlorothiazide
CAS:<p>Chlorothiazide (Diuril) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE.</p>Fórmula:C7H6ClN3O4S2Pureza:98.46% - 98.91%Cor e Forma:Crystals Physical Description Crystals; White Powder (Ntp 1992)Peso molecular:295.72hCAII-IN-7
<p>hCAII-IN-7 (R-13) inhibits human CA I, II, IV, IX with K i of 60.7, 320.7, 2298, 35.2 nM respectively.</p>Fórmula:C20H25N3O4SCor e Forma:SolidPeso molecular:403.5Carbonic anhydrase inhibitor 26
<p>Compound 6T, designated as Carbonic anhydrase inhibitor26, acts as an inhibitor of Carbonic Anhydrase II (Carbonic AnhydraseII), exhibiting an IC50 value of 9.10 ± 0.26 μM.</p>Fórmula:C17H14N6O4Cor e Forma:SolidPeso molecular:366.33Pyrocatechol
CAS:<p>Pyrocatechol, often known as catechol or benzene-1,2-diol, is a benzenediol, Pyrocatechol was produced at a large scale industrially, mainly as precursors to pesticides, flavors, and fragrances. Its sulfonic acid is often present in the urine of many mammals.</p>Fórmula:C6H6O2Cor e Forma:SolidPeso molecular:110.11hCAII-IN-6
<p>"hCAII-IN-6 (S-13) inhibits hCA II (4.4 nM) and isoforms I, IV, IX (9.2, 480.2, 14.7 nM). For glaucoma research."</p>Fórmula:C20H25N3O4SCor e Forma:SolidPeso molecular:403.5Swertiajaponin
CAS:<p>Swertiajaponin possesses antimicrobial activity.</p>Fórmula:C22H22O11Pureza:99.85%Cor e Forma:SolidPeso molecular:462.4Acesulfame
CAS:<p>Acesulfame inhibits CA9/12 and can be used to study inflammation-related diseases.</p>Fórmula:C4H5NO4SCor e Forma:SolidPeso molecular:163.15Carbonic anhydrase inhibitor 18
<p>Carbonic anhydrase inhibitor18 (Compound 9) is an inhibitor of human carbonic anhydrase (hCA) isozymes, with Ki values of 604.8 nM for hCA I, 333.6 nM for hCA II, 1.9 nM for hCA IX, and 6.7 nM for hCA XII. Carbonic anhydrase inhibitor18 is applicable in cancer research.</p>Fórmula:C26H28N4O6S2Peso molecular:556.14503β-Glucosidase, from almonds
CAS:Pureza:approx. 90% (biuret)Cor e Forma:White to pale yellow or beige powderPeso molecular:-Thrombopoietin Protein, Mouse, Recombinant
<p>Expression system: E. coli<br>Length: 22-195, Partial<br>Activity: Cell Activity</p>Cor e Forma:Lyophilized PowderPeso molecular:18.7 kDa (Predicted)(E)-Dehydrodiconiferyl alcohol
CAS:<p>(E)-Dehydrodiconiferyl alcohol inhibits hCA IX/XII enzymes and blocks NF-κB nuclear translocation in healing tissues.</p>Fórmula:C20H22O6Cor e Forma:SolidPeso molecular:358.39Tyrosinase-IN-15
<p>Tyrosinase-IN-15 (Compound 39), with an IC50 of 7.12 μM and a Ki of 11.8 μM, functions as a tyrosinase inhibitor [1].</p>Pureza:98%Cor e Forma:Odour SolidhCA XII-IN-6
<p>Compound 4d, known as hCA XII-IN-6, is a potent inhibitor of human carbonic anhydrase XII (hCA XII) with a Ki value of 84.2 nM and exhibits anti-proliferative</p>Fórmula:C11H9N5O3S2Pureza:98%Cor e Forma:SolidPeso molecular:323.35Carbonic anhydrase inhibitor 30
<p>Carbonic anhydrase inhibitor30 (compound 17) is an inhibitor of carbonic anhydrase with Ki values of 2.13 μM for hCA I and 0.161 μM for hCA II[1].</p>Fórmula:C23H22FN3O5SCor e Forma:SolidPeso molecular:471.12642hCAXII-IN-7
<p>hCAXII-IN-7 (compound 6e) functions as an inhibitor of human carbonic anhydrase XII (hCA XII) and possesses blood-brain barrier (BBB) permeability.</p>Fórmula:C26H25N5O6S2Pureza:98%Cor e Forma:SolidPeso molecular:567.64hCA/VEGFR-2-IN-2
<p>Compound 8g (hCA/VEGFR-2-IN-2) is an indolinonylbenzenesulfonamide identified as a potential dual inhibitor targeting cancer-associated isozymes hCA IX/XII and</p>Fórmula:C23H26N6O5SPureza:98%Cor e Forma:SolidPeso molecular:498.55hCA/VEGFR-2-IN-4
<p>hCA/VEGFR-2-IN-4 (compound 15b), an indolinylbenzenesulfonamide, serves as a potential dual inhibitor targeting cancer-related human carbonic anhydrases hCA IX/</p>Fórmula:C22H23FN6O5SPureza:98%Cor e Forma:SolidPeso molecular:502.52hCAIX/XII-IN-14
<p>hCAIX/XII-IN-14 (Compound 1i) is an inhibitor of hCAIX and hCAXII, with Ki values of 9.4 nM for hCAII, 5.6 nM for hCAIX, and 6.3 nM for hCAXII.</p>Fórmula:C16H14F3N3O4SCor e Forma:SolidPeso molecular:401.36α-Pyrone
CAS:<p>Alpha-Pyrone exhibits inhibitory activity against tyrosinase, carbonic anhydrase 1, and carbonic anhydrase 9</p>Fórmula:C5H4O2Cor e Forma:SolidPeso molecular:96.08Carbonic anhydrase
CAS:<p>Carbonic anhydrase, a zinc enzyme in all life forms, converts CO2 to bicarbonate; studied for cancer, glaucoma, obesity, epilepsy.</p>Cor e Forma:SolidCAIX/CAXII-IN-4
<p>CAIX/CAXII-IN-4 (Compound 7h) is an inhibitor of carbonic anhydrase (CA) that binds to CAIX, CA XII, and CAII with Ki values of 1.324 μM, 0.435 μM, and 3.035 μM, respectively. This compound exhibits broad-spectrum anti-tumor activity and inhibits the proliferation of central nervous system tumor cells U251, with a GI50 of 0.361 μM.</p>Fórmula:C23H21N5O3SCor e Forma:SolidPeso molecular:447.51TSPO/Carbonic Anhydrase Modulator 1
<p>TSPO/Carbonic Anhydrase Modulator 1 (Compound 3) acts as a dual modulator of mitochondrial translocator protein and carbonic anhydrase, with a TSPOKi of 1.340 μM and a CAVII KA of 10.7 μM. It enhances neurosteroid production, increases BDNF gene expression, and demonstrates neuroprotective activity.</p>Fórmula:C35H51N3O3Cor e Forma:SolidPeso molecular:561.798Tyrosinase-IN-36
<p>Tyrosinase-IN-36 is a moderately potent inhibitor of tyrosine, exhibiting an inhibition percentage of 42.75% compared to kojic acid at a concentration of 100 μM and possesses antioxidant activity.</p>Cor e Forma:Odour SolidGirentuximab
CAS:<p>Girentuximab (G250) is an anti-carbonic anhydrase IX (CAIX) monoclonal antibody with anti-cancer activity for the study of uroepithelial carcinoma PET (ZiPUP).</p>Cor e Forma:LiquidPeso molecular:145.55 kDaTyrosinase-IN-40
<p>Tyrosinase-IN-40 (Compound 9r) is a competitive inhibitor of tyrosinase, boasting an IC50 value of 17.02 µM and a Ki value of 14.87 µM. This compound also exhibits antioxidant activity and can be utilized in studies related to melanin.</p>Fórmula:C34H29N9O10Cor e Forma:SolidPeso molecular:723.648CAIX Inhibitor S4
CAS:<p>CAIX Inhibitor S4 (S4) is an effective inhibitor of carbonic anhydrase IX/XII with a Ki of 7 nM and 2 nM, respectively.</p>Fórmula:C15H17N3O4SPureza:99.07%Cor e Forma:SolidPeso molecular:335.38hCAII-IN-8
CAS:<p>Compound CDy9 is a highly selective inhibitor of carbonic anhydrase (CA) with an IC50 value of 0.18 μM for hCA II.</p>Fórmula:C15H16N2O5SPureza:99.73%Cor e Forma:SoildPeso molecular:336.36Carbonic anhydrase inhibitor 32
<p>Carbonic anhydrase inhibitor32 (compound 5B) is an orally active, selective inhibitor of hCA (carbonic anhydrase) II/VII, with Ki values of 6.3 nM for hCA II, 10.1 nM for hCA VII, and 681 nM for hCA I. It shows potential for neuroprotection and anticonvulsant effects by reducing mTOR activation and increasing hippocampal KCC2 levels.</p>Fórmula:C17H16N6O3SCor e Forma:SolidPeso molecular:384.41Carbonic anhydrase inhibitor 31
<p>Carbonic anhydrase inhibitor31 is an mtCA2 inhibitor (Ki: 5.2 nM) that can be used in antituberculosis research.</p>Fórmula:C24H20N6O5SCor e Forma:SolidPeso molecular:504.12159hCAIX-IN-17
<p>hCA IX-IN-1 inhibits hCA I/II/IX/XII with Ki of 331.4/28.4/9.4/17.8 nM, has anticancer properties.</p>Fórmula:C19H18N2O3SCor e Forma:SolidPeso molecular:354.42hCAII/XII-IN-1
<p>hCAII/XII-IN-1 (compound 4l) is a potent inhibitor of hCAXII and hCAII, with Ki values of 8.4 nM and 9.4 nM, respectively. It plays a significant role in cancer research.</p>Fórmula:C22H20N4O6S2Cor e Forma:SolidPeso molecular:500.547CA IX/VEGFR-2-IN-3
<p>CAIX/VEGFR-2-IN-3 (Compound 6i) is an inhibitor of Carbonic Anhydrase IX and VEGFR-2, with IC50 values of 41 and 48 nM, respectively. It exhibits anticancer activity by inhibiting the growth of MCF-7 breast cancer cells (IC50 of 22.33 μM) and mouse fibroblast cell line 3T3, where cell viability is reduced to below 40% at a concentration of 100 μM. This compound is applicable for research in the field of cancer treatment.</p>Fórmula:C19H16ClN3O5S2Cor e Forma:SolidPeso molecular:465.93hCA/VEGFR-2-IN-3
<p>hCA/VEGFR-2-IN-3 (compound 8j) is an indolinonylbenzenesulfonamide with potential as a dual inhibitor of cancer-associated hCA IX/XII and VEGFR-2.</p>Fórmula:C24H28N6O6SPureza:98%Cor e Forma:SolidPeso molecular:528.58Peroxidase
CAS:Pureza:≥ 85units/mg (dry basis)Cor e Forma:Beige to light-brown, reddish brown or dark brown lyophilised powderPeso molecular:-hCAII/IX-IN-1
<p>hCAII/IX-IN-1 (compound 4o) is a potent inhibitor of hCAII and hCAIX, with Ki values of 7.4 nM and 7.0 nM, respectively. It plays a significant role in cancer research.</p>Fórmula:C23H22N4O7S2Cor e Forma:SolidPeso molecular:530.573hCA/Wnt/β-catenin-IN-1
<p>hCA/Wnt/β-catenin-IN-1 (Compd 15) serves as an inhibitor with selective affinity for hCA isoforms II, IX, and XII, exhibiting K i values of 33.6, 24.1, and 6.8</p>Cor e Forma:Odour SolidCarbonic anhydrase inhibitor 29
<p>Carbonic anhydrase inhibitor29 (Compound 5d) is an inhibitor targeting carbonic anhydrase IX and XII, with an inhibition constant (Ki) of 26.6 nM for carbonic anhydrase IX and a Ki of 10.9 nM for carbonic anhydrase XII. Carbonic anhydrase inhibitor29 can be used in cancer research.</p>Cor e Forma:Odour SolidPyridine-2-aldoxime methochloride
CAS:Fórmula:C7H9N2O·ClPureza:≥ 98.0%Cor e Forma:White to off-white or light yellow crystalline powderPeso molecular:172.61CAXII-IN-2
<p>CAXII-IN-2 (compound 3j) is a highly effective inhibitor of CAXII. It demonstrates inhibitory activity against CA IX and CAXII, with Ki values of 27.4 nM and 4.0 nM, respectively.</p>Fórmula:C16H13FNO4PCor e Forma:SolidPeso molecular:333.05662IOX2-NH2-1
CAS:<p>IOX2-NH2-1 inhibits E. coli EGLN-3 (prolyl hydroxylase) with an IC50 of 0.02–1 μM.</p>Fórmula:C19H17N3O5Pureza:98.77% - 99.91%Cor e Forma:SoildPeso molecular:367.36α-Glycosidase-IN-2
<p>α-Glycosidase-IN-2 (compound 8b) is an inhibitor of α-glycosidase, displaying Ki values of 74.16 nM and 6.09 nM for aldose reductase and α-glycosidase, respectively. This compound is utilized in research related to diabetes.</p>Fórmula:C25H22N6OS2Cor e Forma:SolidPeso molecular:486.61DPP IV/hCA II-IN-1
CAS:<p>DPP IV/hCA II-IN-1: strong DPP IV & CA inhibitor, IC50=0.049μM (DPP IV), Ki=0.0361-3.034μM (CA II-IV).</p>Fórmula:C17H20N2O5SCor e Forma:SolidPeso molecular:364.42Trypsin, bovine origin
CAS:Pureza:≥ 2000units/mg (USP)Cor e Forma:White or almost white crystalline powderPeso molecular:-Phenylsulfamide
CAS:<p>Phenylsulfamide (Compound 10), acting as an inhibitor of human carbonic anhydrase-II (hCA-II), exhibits a dissociation constant (Kd) of 45.50 μM and an</p>Fórmula:C6H8N2O2SCor e Forma:SolidPeso molecular:172.2hCAIX/XII-IN-11
<p>hCAIX/XII-IN-11 (Compound 6c) is an inhibitor of hCA IX and hCA XII, exhibiting Ki values of 0.7 μM for both isoforms. This compound is applicable in cancer research.</p>Fórmula:C13H10FN3O4Peso molecular:291.06553TPT-004
<p>TPT-004, a TPH inhibitor, exhibits superior pharmacokinetic and pharmacodynamic properties, and demonstrates efficacy in preclinical models for attenuating</p>Cor e Forma:Odour SolidAc-[Nle4,D-Phe7]-α-MSH (4-10)-NH2
CAS:<p>Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2, a melanotropin derivative and melanocyte-stimulating hormone, activates tyrosinase and demonstrates a thermoregulatory effect</p>Fórmula:C47H64N14O10Cor e Forma:SolidPeso molecular:985.1Tyrosinase-IN-14
<p>Tyrosinase-IN-14 (compound 7m), a tyrosinase inhibitor, modulates the enzyme's secondary structure to diminish its catalytic function, exhibits low cytotoxicity</p>Fórmula:C21H13Br2N3O3SPureza:98%Cor e Forma:SolidPeso molecular:547.22Peroxidase, from horseradish, approx. 200 U/mg
CAS:Pureza:≥ 150U/mgCor e Forma:Beige to light-brown, reddish brown or dark brown lyophilised powderPeso molecular:-Proteinase K
CAS:Pureza:≥ 30units/mg (pH 7.5, 37°C, dried basis)Cor e Forma:White or almost white lyophilized powderPeso molecular:-Tyrosinase-IN-34
<p>Tyrosinase-IN-34 (compound 5a), a human tyrosinase inhibitor (IC 50: 3.5 μM), shows promise in regulating melanogenesis and pigmentation.</p>Fórmula:C19H14BrClN4OCor e Forma:SolidPeso molecular:429.7Tyrosinase-IN-32
<p>Tyrosinase-IN-32 (compound 11), a hydroxamate-based alkaloid extracted from black pepper (Piper nigrum L.), functions as an inhibitor of mushroom tyrosinase. In addition to its inhibitory properties, it exhibits antioxidant activity.</p>Fórmula:C15H19NO3Cor e Forma:SolidPeso molecular:261.32Lysozyme, from chicken egg white
CAS:Pureza:≥ 20,000U/mgCor e Forma:White to off-white powderPeso molecular:-TrkA Protein, Rabbit, Recombinant (His)
<p>TrkA Protein, Rabbit, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.</p>Cor e Forma:Lyophilized PowderPeso molecular:43.4 kDa (predicted)TrkB Protein, Canine, Recombinant (hFc)
<p>TrkB Protein, Canine, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag.</p>Cor e Forma:Lyophilized PowderPeso molecular:71.2 kDa (predicted)TrkA Protein, Rat, Recombinant (hFc)
<p>TrkA Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag.</p>Cor e Forma:Lyophilized PowderPeso molecular:69.2 kDa (predicted); 92-102 kDa (reducing conditions)Cuprizone
CAS:<p>Cuprizone is a copper chelator.Cuprizone is used to induce schizophrenia in mice.Cuprizone induces oligodendrocyte death and induces a demyelination response.</p>Fórmula:C14H22N4O2Pureza:≥98%Cor e Forma:SolidPeso molecular:278.35TrkA Protein, Human, Recombinant (His)
<p>TrkA Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.</p>Pureza:98.7%Cor e Forma:Lyophilized PowderPeso molecular:39.5 kDa (predicted); 60-65 kDa (reducing condition, due to glycosylation)HER3/ERBB3 Protein, Cynomolgus/Rhesus macaque, Recombinant (His)
<p>Her3, also called ErbB3, is a type I membrane glycoprotein that is a member of the ErbB family of tyrosine kinase receptors.Her3 is expressed in keratinocytes,</p>Cor e Forma:Lyophilized PowderPeso molecular:69.54 kDa (predicted). Due to glycosylation, the protein migrates to 85-105 kDa based on Tris-Bis PAGE result.p38 γ/MAPK12 Protein, Human, Recombinant
<p>p38 gamma/MAPK12 Protein, Human, Recombinant is expressed in Baculovirus insect cells.</p>Cor e Forma:Lyophilized PowderPeso molecular:42.1 kDa (predicted); 43 kDa (reducing conditions)Thrombopoietin Protein, Mouse, Recombinant (C-His)
<p>Expression System: HEK293 Cells<br>Length: 22-356, Full Length of Mature Protein<br>Activity: Cell Activity</p>Peso molecular:37.20 kDa (Predicted); 75-95 kDa (Due to glycosylation)Carbonic Anhydrase 12 Protein, Human, Recombinant (His) V2
<p>Expression System: HEK293 Cells<br>Length: 25-301, Extracellular Domain<br>Activity: Enzyme Activity</p>Peso molecular:32.22 kDa (Predicted); 40-50 kDa (Due to glycosylation)ErbB4 Protein, Rat, Recombinant (His)
<p>ErbB4 Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.</p>Cor e Forma:Lyophilized PowderPeso molecular:71.3 kDa (predicted); 75-95 kDa (reducing condition, due to glycosylation)TrkB Protein, Human, Recombinant (His), Biotinylated
<p>Expression system: HEK293 Cells<br>Length: 1-430, Partial<br>Activity: ELISA</p>Cor e Forma:Lyophilized PowderPeso molecular:45.66 kDa (predicted); 65.4 kDa (reducing contition, due to glycosylation)DDR2 Protein, Human, Recombinant (His & Avi), Biotinylated
<p>Expression system: HEK293 Cells<br>Length: 1-399, Partial<br>Activity: BLI</p>Cor e Forma:Lyophilized PowderPeso molecular:45.84 kDa (predicted); 60.4 kDa (reducing contition)Anti-Tyrosinase/TYR Antibody (7Z445)
<p>Anti-Tyrosinase/TYR Antibody (7Z445) is an antibody targeting Tyrosinase/TYR. Anti-Tyrosinase/TYR Antibody (7Z445) can be used in ELISA, IF.</p>Cor e Forma:Odour LiquidTrkA Protein, Human, Recombinant
<p>TrkA Protein, Human, Recombinant is expressed in HEK293 Cells. The accession number is P04629.</p>Pureza:> 95% as analyzed by SDS-PAGE - > 95% as analyzed by SDS-PAGECor e Forma:Lyophilized PowderPeso molecular:65~85 kDa (Reducing conditions)HER3/ERBB3 Protein, Mouse, Recombinant (His)
<p>HER3/ERBB3 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.</p>Pureza:97.1%Cor e Forma:Lyophilized PowderPeso molecular:70 kDa (predicted); 95 kDa (reducing condition, due to glycosylation)TrkA Protein, Cynomolgus, Recombinant (His)
<p>TrkA Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.</p>Cor e Forma:Lyophilized PowderPeso molecular:43.95 kDa (predicted); 86 kDa (reducing conditions)HER3/ERBB3 Protein, Mouse, Recombinant (hFc)
<p>HER3/ERBB3 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag.</p>Cor e Forma:Lyophilized PowderPeso molecular:95.23 kDa (predicted); 117.08 kDa (reducing conditions)p38 γ/MAPK12 Protein, Human, Recombinant (His & GST)
<p>p38 gamma/MAPK12 Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag.</p>Cor e Forma:Lyophilized PowderPeso molecular:69.8 kDa (predicted); 65 kDa (reducing conditions)TrkB Protein, Human, Recombinant (His) V2
<p>Expression System: HEK293 Cells<br>Length: 32-430, Extracellular Domain<br>Activity: ELISA</p>Peso molecular:45.2 kDa (Predicted); 65-80 kDa (Due to glycosylation)HER3/ERBB3 Protein, Human, Recombinant (His & Avi), FITC-Labeled
<p>Her3, also called ErbB3, is a type I membrane glycoprotein that is a member of the ErbB family of tyrosine kinase receptors.Her3 is expressed in keratinocytes,</p>Cor e Forma:Lyophilized PowderPeso molecular:71.6 kDa (predicted). Due to glycosylation, the protein migrates to 72-75 kDa based on Tris-Bis PAGE result.PTP α/PTPRA Protein, Human, Recombinant (aa 174-793, His & GST)
<p>PTPRA is reported to be involved in cancer development and progression through activating the Src family kinase (SFK) signaling pathways.</p>Cor e Forma:Lyophilized PowderPeso molecular:99 kDa (predicted); 90 kDa (reducing conditions)Mer Protein, Mouse, Recombinant (hFc)
<p>Mer Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag.</p>Cor e Forma:Lyophilized PowderPeso molecular:79.3 kDa (predicted); 130 kDa (reducing condition, due to glycosylation)HER3/ERBB3 Protein, Rhesus, Recombinant
<p>HER3/ERBB3 Protein, Rhesus, Recombinant is expressed in HEK293 mammalian cells.</p>Pureza:92.6%Cor e Forma:Lyophilized PowderPeso molecular:69.5 kDa (predicted)HER3/ERBB3 Protein, Human, Recombinant (hFc), Biotinylated
<p>HER3/ERBB3 Protein, Human, Recombinant (hFc), Biotinylated is expressed in HEK293 mammalian cells with hFc tag.</p>Cor e Forma:Lyophilized PowderPeso molecular:95.4 kDa (predicted)
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