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Receptor opioide

Receptor opioide

Os receptores opioides são um grupo de receptores acoplados à proteína G que mediam os efeitos dos opioides endógenos e exógenos. Estes receptores desempenham um papel central na modulação da dor, regulação do humor e comportamentos aditivos. Agonistas e antagonistas dos receptores opioides são amplamente utilizados no manejo da dor e tratamento de dependências, bem como em pesquisas sobre distúrbios neurológicos e psiquiátricos. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores opioides de alta qualidade para apoiar sua pesquisa em neurobiologia, manejo da dor e terapia de dependência.

Foram encontrados 326 produtos de "Receptor opioide"

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  • Trimebutine maleate

    CAS:
    <p>Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.</p>
    Fórmula:C26H33NO9
    Pureza:99.76% - 99.98%
    Cor e Forma:White Solid
    Peso molecular:503.55

    Ref: TM-T1197

    1g
    34,00€
  • ZT 52656A hydrochloride

    CAS:
    ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.
    Fórmula:C19H26ClF3N2O
    Pureza:98.78%
    Cor e Forma:Solid
    Peso molecular:390.87

    Ref: TM-T13414

    1mg
    540,00€
    5mg
    1.198,00€
    10mg
    1.786,00€
    25mg
    3.030,00€
    50mg
    3.924,00€
    1mL*10mM (DMSO)
    1.026,00€
  • Matrine

    CAS:
    Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.
    Fórmula:C15H24N2O
    Pureza:99.77% - >99.99%
    Cor e Forma:Solid
    Peso molecular:248.36

    Ref: TM-T2870

    25mg
    43,00€
    50mg
    58,00€
    100mg
    81,00€
    200mg
    117,00€
    500mg
    250,00€
    1mL*10mM (DMSO)
    49,00€
  • CP 866087

    CAS:
    CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.
    Fórmula:C24H30N2O3S
    Pureza:99.22% - 99.74%
    Cor e Forma:Solid
    Peso molecular:426.57

    Ref: TM-T31081L

    1mg
    185,00€
    5mg
    459,00€
    10mg
    657,00€
    25mg
    1.026,00€
    50mg
    1.415,00€
  • Naltrexone hydrochloride

    CAS:
    <p>Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.</p>
    Fórmula:C20H24ClNO4
    Pureza:98.72% - 99.65%
    Cor e Forma:White Crystalline Powder
    Peso molecular:377.862

    Ref: TM-T0963

    1g
    163,00€
    25mg
    35,00€
    50mg
    44,00€
    100mg
    55,00€
    500mg
    111,00€
  • Apitegromab

    CAS:
    Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases including
    Pureza:97.59% (SDS-PAGE); 99.78% (SEC-HPLC) - >95.0% (SDS-PAGE); 99.62% (SEC-HPLC)
    Cor e Forma:Liquid
    Peso molecular:145.06 kDa

    Ref: TM-T77445

    1mg
    160,00€
    5mg
    472,00€
    10mg
    755,00€
    25mg
    1.121,00€
    50mg
    1.501,00€
  • Moguisteine

    CAS:
    Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.
    Fórmula:C16H21NO5S
    Pureza:99.98%
    Cor e Forma:Solid
    Peso molecular:339.41

    Ref: TM-T1169

    50mg
    34,00€
    1mL*10mM (DMSO)
    34,00€
  • BTRX-335140

    CAS:
    <p>BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.</p>
    Fórmula:C25H32FN5O2
    Pureza:98% - 99.89%
    Cor e Forma:Solid
    Peso molecular:453.55

    Ref: TM-T14835

    1mg
    105,00€
    2mg
    155,00€
    5mg
    250,00€
    10mg
    406,00€
    25mg
    840,00€
    50mg
    1.378,00€
    100mg
    1.882,00€
    200mg
    2.632,00€
  • Meptazinol hydrochloride

    CAS:
    Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.
    Fórmula:C15H23NO·HCl
    Pureza:99.75%
    Cor e Forma:White Solid
    Peso molecular:269.81

    Ref: TM-T0201

    5mg
    48,00€
    10mg
    55,00€
    25mg
    87,00€
    50mg
    116,00€
    100mg
    168,00€
    200mg
    227,00€
    1mL*10mM (DMSO)
    55,00€
  • Alvimopan

    CAS:
    <p>Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.</p>
    Fórmula:C25H32N2O4
    Pureza:99.47% - 99.78%
    Cor e Forma:Solid
    Peso molecular:424.53

    Ref: TM-T1242

    1mg
    48,00€
    5mg
    88,00€
    10mg
    135,00€
    25mg
    245,00€
    50mg
    378,00€
    100mg
    560,00€
    200mg
    797,00€
  • Loperamide hydrochloride

    CAS:
    Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.
    Fórmula:C29H34Cl2N2O2
    Pureza:99.91% - >99.99%
    Cor e Forma:Crystals Practically Insoluble In Water
    Peso molecular:513.50

    Ref: TM-T0209

    1g
    107,00€
    50mg
    44,00€
    100mg
    55,00€
    500mg
    85,00€
    1mL*10mM (DMSO)
    55,00€
  • Sinomenine hydrochloride

    CAS:
    Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.
    Fórmula:C19H24ClNO4
    Pureza:99.43%
    Cor e Forma:Solid
    Peso molecular:365.85

    Ref: TM-T2921

    1g
    70,00€
    200mg
    34,00€
    500mg
    52,00€
  • Samidorphan HCl

    CAS:
    <p>Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.</p>
    Fórmula:C21H27ClN2O4
    Pureza:96.79% - 97.85%
    Cor e Forma:Soild
    Peso molecular:406.9

    Ref: TM-T67888L

    1mg
    164,00€
    5mg
    393,00€
    10mg
    582,00€
    25mg
    930,00€
    50mg
    1.254,00€
    100mg
    1.691,00€
  • LY2940094

    CAS:
    LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.
    Fórmula:C22H23ClF2N4O2S
    Pureza:99.4%
    Cor e Forma:Solid
    Peso molecular:480.96

    Ref: TM-T15799

    1mg
    81,00€
    2mg
    106,00€
    5mg
    163,00€
    10mg
    274,00€
    25mg
    542,00€
    50mg
    778,00€
    100mg
    1.074,00€
    1mL*10mM (DMSO)
    180,00€
  • DPDPE

    CAS:
    DPDPE is selective δ-opioid receptor agonist peptide.
    Fórmula:C30H39N5O7S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:645.79

    Ref: TM-TP2036

    1mg
    545,00€
  • ICI 174,864

    CAS:
    Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.
    Fórmula:C38H53N5O7
    Pureza:98%
    Cor e Forma:White Solid
    Peso molecular:691.87

    Ref: TM-TP2013

    1mg
    677,00€
  • Neurotransmitter Receptor Compound Library


    <p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>
    Cor e Forma:Odour Solid

    Ref: TM-L2610

    1mg
    A consultar
  • Biphalin TFA

    CAS:
    Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.
    Fórmula:C46H56N10O10·xC2HF3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:909.00 (free base)

    Ref: TM-T80074

    5mg
    A consultar
    50mg
    A consultar
  • [DPro10] Dynorphin A (1-11)acetate,porcine


    [DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.
    Fórmula:C65H107N21O15
    Pureza:99.59%
    Cor e Forma:Soild
    Peso molecular:1422.7

    Ref: TM-T76341L

    2mg
    38,00€
    5mg
    59,00€
    10mg
    87,00€
    25mg
    131,00€
    50mg
    190,00€
    100mg
    279,00€
    200mg
    394,00€
  • β-Endorphin, equine TFA


    β-Endorphin, equine TFA, an endogenous opioid peptide, demonstrates high affinity binding to μ/δ opioid receptors and possesses analgesic properties [1] [2] [3
    Fórmula:C156H249F3N42O46S
    Cor e Forma:Solid
    Peso molecular:3537.96

    Ref: TM-T76027

    5mg
    A consultar
    50mg
    A consultar