
Receptor opioide
Os receptores opioides são um grupo de receptores acoplados à proteína G que mediam os efeitos dos opioides endógenos e exógenos. Estes receptores desempenham um papel central na modulação da dor, regulação do humor e comportamentos aditivos. Agonistas e antagonistas dos receptores opioides são amplamente utilizados no manejo da dor e tratamento de dependências, bem como em pesquisas sobre distúrbios neurológicos e psiquiátricos. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores opioides de alta qualidade para apoiar sua pesquisa em neurobiologia, manejo da dor e terapia de dependência.
Foram encontrados 326 produtos de "Receptor opioide"
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Trimebutine maleate
CAS:<p>Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.</p>Fórmula:C26H33NO9Pureza:99.76% - 99.98%Cor e Forma:White SolidPeso molecular:503.55ZT 52656A hydrochloride
CAS:ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.Fórmula:C19H26ClF3N2OPureza:98.78%Cor e Forma:SolidPeso molecular:390.87Matrine
CAS:Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.Fórmula:C15H24N2OPureza:99.77% - >99.99%Cor e Forma:SolidPeso molecular:248.36CP 866087
CAS:CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.Fórmula:C24H30N2O3SPureza:99.22% - 99.74%Cor e Forma:SolidPeso molecular:426.57Naltrexone hydrochloride
CAS:<p>Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.</p>Fórmula:C20H24ClNO4Pureza:98.72% - 99.65%Cor e Forma:White Crystalline PowderPeso molecular:377.862Apitegromab
CAS:Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases includingPureza:97.59% (SDS-PAGE); 99.78% (SEC-HPLC) - >95.0% (SDS-PAGE); 99.62% (SEC-HPLC)Cor e Forma:LiquidPeso molecular:145.06 kDaMoguisteine
CAS:Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.Fórmula:C16H21NO5SPureza:99.98%Cor e Forma:SolidPeso molecular:339.41BTRX-335140
CAS:<p>BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.</p>Fórmula:C25H32FN5O2Pureza:98% - 99.89%Cor e Forma:SolidPeso molecular:453.55Ref: TM-T14835
1mg105,00€2mg155,00€5mg250,00€10mg406,00€25mg840,00€50mg1.378,00€100mg1.882,00€200mg2.632,00€Meptazinol hydrochloride
CAS:Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.Fórmula:C15H23NO·HClPureza:99.75%Cor e Forma:White SolidPeso molecular:269.81Alvimopan
CAS:<p>Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.</p>Fórmula:C25H32N2O4Pureza:99.47% - 99.78%Cor e Forma:SolidPeso molecular:424.53Loperamide hydrochloride
CAS:Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.Fórmula:C29H34Cl2N2O2Pureza:99.91% - >99.99%Cor e Forma:Crystals Practically Insoluble In WaterPeso molecular:513.50Sinomenine hydrochloride
CAS:Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.Fórmula:C19H24ClNO4Pureza:99.43%Cor e Forma:SolidPeso molecular:365.85Samidorphan HCl
CAS:<p>Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.</p>Fórmula:C21H27ClN2O4Pureza:96.79% - 97.85%Cor e Forma:SoildPeso molecular:406.9LY2940094
CAS:LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.Fórmula:C22H23ClF2N4O2SPureza:99.4%Cor e Forma:SolidPeso molecular:480.96Ref: TM-T15799
1mg81,00€2mg106,00€5mg163,00€10mg274,00€25mg542,00€50mg778,00€100mg1.074,00€1mL*10mM (DMSO)180,00€DPDPE
CAS:DPDPE is selective δ-opioid receptor agonist peptide.Fórmula:C30H39N5O7S2Pureza:98%Cor e Forma:SolidPeso molecular:645.79ICI 174,864
CAS:Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.Fórmula:C38H53N5O7Pureza:98%Cor e Forma:White SolidPeso molecular:691.87Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>Cor e Forma:Odour SolidBiphalin TFA
CAS:Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.Fórmula:C46H56N10O10·xC2HF3O2Pureza:98%Cor e Forma:SolidPeso molecular:909.00 (free base)[DPro10] Dynorphin A (1-11)acetate,porcine
[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.Fórmula:C65H107N21O15Pureza:99.59%Cor e Forma:SoildPeso molecular:1422.7β-Endorphin, equine TFA
β-Endorphin, equine TFA, an endogenous opioid peptide, demonstrates high affinity binding to μ/δ opioid receptors and possesses analgesic properties [1] [2] [3Fórmula:C156H249F3N42O46SCor e Forma:SolidPeso molecular:3537.96

