Receptor de Bradicinina
Os receptores de bradicinina são GPCRs que mediam os efeitos da bradicinina, um peptídeo envolvido em respostas inflamatórias, sensação de dor e regulação da pressão arterial. Existem dois principais tipos de receptores de bradicinina, B1 e B2, cada um desempenhando papéis distintos em processos fisiopatológicos. Antagonistas dos receptores de bradicinina são usados no tratamento de condições como angioedema hereditário, dor crônica e hipertensão. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores de bradicinina de alta qualidade para apoiar sua pesquisa em inflamação, manejo da dor e biologia cardiovascular.
Foram encontrados 61 produtos de "Receptor de Bradicinina"
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Anatibant 2HCl
CAS:Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.
Fórmula:C34H36Cl2N6O5S·2ClHPureza:99.17% - 99.58%Cor e Forma:SoildPeso molecular:784.58Bradykinin (1-7)
CAS:Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.Fórmula:C35H52N10O9Pureza:98%Cor e Forma:White Lyophilized PowderPeso molecular:756.85FR167344 free base
CAS:FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.Fórmula:C30H28BrCl2N5O4Pureza:98%Cor e Forma:SolidPeso molecular:673.38Bradykinin (1-6)
CAS:Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.Fórmula:C30H45N9O8Pureza:98%Cor e Forma:SolidPeso molecular:659.73Labradimil
CAS:Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.Fórmula:C49H75N15O12SPureza:98%Cor e Forma:SolidPeso molecular:1098.29MEN 11270
CAS:B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.Fórmula:C60H90N20O11SPureza:98%Cor e Forma:SolidPeso molecular:1299.56Bradykinin (1-3)
CAS:Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.
Fórmula:C16H28N6O4Pureza:98%Cor e Forma:SolidPeso molecular:368.43[Des-Arg9]-Bradykinin
CAS:[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.
Fórmula:C44H61N11O10Pureza:98%Cor e Forma:SolidPeso molecular:904.02Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS:Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.Fórmula:C47H66N12O11Pureza:98%Cor e Forma:SolidPeso molecular:975.11Icatibant
CAS:Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).Fórmula:C59H89N19O13SPureza:98%Cor e Forma:White SolidPeso molecular:1304.52Lys-[Des-Arg9]Bradykinin
CAS:Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.Fórmula:C50H73N13O11Pureza:98%Cor e Forma:SolidPeso molecular:1032.21[Des-Arg10]-HOE I40 TFA
[Des-Arg10]-HOE I40 TFA is a potent antagonist of the bradykinin B1 receptor.
Fórmula:C53H77N15O12S·xC2HF3O2Cor e Forma:SolidBombinakinin M
CAS:Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.Fórmula:C100H159N31O24Pureza:98%Cor e Forma:SolidPeso molecular:2179.55[Phe8Ψ(CH-NH)-Arg9]-Bradykinin
CAS:Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage.Fórmula:C50H75N15O10Pureza:98%Cor e Forma:SolidPeso molecular:1046.23Fasitibant chloride
CAS:Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.
Fórmula:C36H49Cl3N6O6SCor e Forma:SolidPeso molecular:800.23NPC 567
CAS:NPC 567 is an antagonist of the bradykinin receptor.Fórmula:C60H87N19O13Pureza:98%Cor e Forma:SolidPeso molecular:1282.48Fasitibant chloride hydrochloride
CAS:Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.Fórmula:C36H50Cl4N6O6SCor e Forma:SolidPeso molecular:836.7Lys-Bradykinin
CAS:Endogenous bradykinin receptor agonistFórmula:C56H85N17O12Pureza:98%Cor e Forma:SolidPeso molecular:1188.38Zoliprofen
CAS:Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.Fórmula:C12H11NO3SPureza:99.62%Cor e Forma:SolidPeso molecular:249.29Ref: TM-T68025
1mg85,00€5mg170,00€10mg256,00€25mg480,00€50mg655,00€100mg933,00€500mg1.872,00€1mL*10mM (DMSO)168,00€Retrobradykinin
CAS:Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.Fórmula:C50H73N15O11Cor e Forma:SolidPeso molecular:1060.228
![[Des-Arg9]-Bradykinin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT7645.webp&w=3840&q=75)
![Sar-[D-Phe8]-des-Arg9-Bradykinin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1917.webp&w=3840&q=75)
![Lys-[Des-Arg9]Bradykinin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1918.webp&w=3840&q=75)
![[Phe8Ψ(CH-NH)-Arg9]-Bradykinin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP2076.webp&w=3840&q=75)
