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Inibidores

Inibidores

Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.

Subcategorias de "Inibidores"

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Foram encontrados 66618 produtos de "Inibidores"

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  • NS3623

    CAS:
    <p>NS3623 is an activator of human ether-a-go-go-related gene potassium channels.</p>
    Fórmula:C15H10BrF3N6O
    Pureza:97.06%
    Cor e Forma:Solid
    Peso molecular:427.18
  • Pranoprofen

    CAS:
    <p>Pranoprofen (Pyranoprofen) (INN) is a non-steroidal anti-inflammatory drug used in ophthalmology.</p>
    Fórmula:C15H13NO3
    Pureza:97.98% - 99.85%
    Cor e Forma:Solid
    Peso molecular:255.27
  • Bromperidol

    CAS:
    <p>Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.</p>
    Fórmula:C21H23BrFNO2
    Pureza:99.89%
    Cor e Forma:Tan Solid
    Peso molecular:420.32
  • Retinyl palmitate

    CAS:
    <p>Retinyl palmitate (Vitamin A palmitate) is a naturally-occurring phenyl analogue of retinol, with potential antineoplastic and chemopreventive activities.</p>
    Fórmula:C36H60O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:524.86
  • Tramiprosate

    CAS:
    <p>Tramiprosate (Alzhemed) is an orally active, BBB-crossing, naturally occurring amino acid that binds soluble Aβ and maintains it in a non-protofibrillar form.</p>
    Fórmula:C3H9NO3S
    Pureza:99%
    Cor e Forma:White Crystals Or Crystalline Power
    Peso molecular:139.17
  • MYCMI-6

    CAS:
    <p>MYCMI-6 inhibits MYC:MAX, reduces tumor growth, triggers apoptosis, minimal side effects.</p>
    Fórmula:C20H19N7O
    Pureza:99.23%
    Cor e Forma:Solid
    Peso molecular:373.41
  • Ifenprodil Tartrate

    CAS:
    <p>Ifenprodil is a selective NMDA receptor (glutamate) antagonist.</p>
    Fórmula:C21H27NO2C4H6O6
    Pureza:99.02% - 99.55%
    Cor e Forma:Solid
    Peso molecular:400.49
  • Pefloxacin Mesylate

    CAS:
    Pefloxacin Mesylate (Pefloxacinium mesylate) is a synthetic broad-spectrum fluoroquinolone antibacterial agent active against most gram-negative and gram-
    Fórmula:C18H24FN3O6S
    Pureza:99.86%
    Cor e Forma:Solid
    Peso molecular:429.46
  • D-AP5

    CAS:
    <p>D-AP5 (D-APV) is a NMDA receptor antagonist.</p>
    Fórmula:C5H12NO5P
    Pureza:98.77% - >99.99%
    Cor e Forma:White Fine Crystalline Powder
    Peso molecular:197.13
  • CMP8

    CAS:
    <p>CMP8, an estrogen receptor ligand, selectively binds to ERLBD with IC50: 29 nM (MGERα), 41 nM (MGRERα), 1100 nM (hERα), 2200 nM (hERβ).</p>
    Fórmula:C33H34ClNO3
    Pureza:99.36%
    Cor e Forma:Solid
    Peso molecular:528.08
  • Promethazine

    CAS:
    <p>Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .</p>
    Fórmula:C17H20N2S
    Pureza:99.76%
    Cor e Forma:Crystals
    Peso molecular:284.42
  • Enarodustat

    CAS:
    <p>Enarodustat (JTZ-951) is an orally active factor inhibitor of prolyl hydroxylase (EC50: 0.22 μM) and has the potential for renal anemia treatment.</p>
    Fórmula:C17H16N4O4
    Pureza:99.73% - 99.75%
    Cor e Forma:Solid
    Peso molecular:340.33
  • Shikimic Acid

    CAS:
    Shikimic Acid (Shikimate) is a tri-hydroxy cyclohexene carboxylic acid important in the biosynthesis that the shikimate pathway is named after it.
    Fórmula:C7H10O5
    Pureza:98.85% - 98.86%
    Cor e Forma:Off-White Solid Crystalline
    Peso molecular:174.15
  • RA190

    CAS:
    <p>RA190 inhibits proteasome function by covalently binding to cysteine 88 of ubiquitin receptor RPN13.</p>
    Fórmula:C28H23Cl5N2O2
    Pureza:97.7%
    Cor e Forma:Solid
    Peso molecular:596.76
  • Labetalol hydrochloride

    CAS:
    <p>Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.</p>
    Fórmula:C19H25ClN2O3
    Pureza:99.54% - 99.85%
    Cor e Forma:Solid
    Peso molecular:364.87
  • Sulfamethoxazole

    CAS:
    <p>Sulfamethoxazole (STX 608), a sulfonamide antimicrobial, inhibits Cytochrome P450 2C9.</p>
    Fórmula:C10H11N3O3S
    Pureza:99.71% - 99.92%
    Cor e Forma:Crystals Or White Powder
    Peso molecular:253.28
  • D-Mannitol

    CAS:
    <p>D-Mannitol (Mannitol) is a diuretic and renal diagnostic aid related to sorbitol.</p>
    Fórmula:C6H14O6
    Pureza:99.66% - 99.68%
    Cor e Forma:Orthorhombic Needles From Alc (Ntp 1992)
    Peso molecular:182.17
  • DCZ0415

    CAS:
    <p>DCZ0415: Potent TRIP13 inhibitor; combats myeloma in vitro, in vivo, and in drug-resistant patients; hinders DNA repair and NF-κB activity.</p>
    Fórmula:C23H20N2O2
    Pureza:99.34% - 99.95%
    Cor e Forma:Solid
    Peso molecular:356.42
  • 2-Phenylbutanoic acid

    CAS:
    <p>2-Phenylbutanoic acid (2-Phenylbutyric acid) is used as an industrial intermediate.</p>
    Fórmula:C10H12O2
    Pureza:98.25%
    Cor e Forma:Solid
    Peso molecular:164.2
  • 2',5'-Dideoxyadenosine

    CAS:
    <p>2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).</p>
    Fórmula:C10H13N5O2
    Pureza:99.55%
    Cor e Forma:White Solid
    Peso molecular:235.24
  • STAT3-IN-1

    CAS:
    <p>STAT3-IN-1 selective and orally active inhibitor of STAT3(in HT29 and MDA-MB 231 cells, with IC50 values of 1.82 μM and 2.14 μM , respectively), induces tumor</p>
    Fórmula:C28H29NO6
    Pureza:95.89% - 95.89%
    Cor e Forma:Solid
    Peso molecular:475.53
  • Zagotenemab

    CAS:
    <p>Zagotenemab: humanized antibody targeting tau protein to study neurological disorders, including Alzheimer's.</p>
    Pureza:95% - > 95%
    Cor e Forma:Liquid
    Peso molecular:145.3 kDa
  • Gabexate mesylate

    CAS:
    Gabexate mesylate (FOY) inhibits thrombin, plasmin, kallikrein; used for pancreatitis, DIC, hemodialysis anticoagulant.
    Fórmula:C17H27N3O7S
    Pureza:99.2% - 99.64%
    Cor e Forma:White Crystal
    Peso molecular:417.48
  • Florfenicol

    CAS:
    <p>Florfenicol treats BRD in cattle, effective against Mannheimia, Pasteurella, Haemophilus, Fusobacterium, and Bacteroides.</p>
    Fórmula:C12H14Cl2FNO4S
    Pureza:98.93%
    Cor e Forma:Solid
    Peso molecular:358.21
  • DSP Crosslinker

    CAS:
    DSP Crosslinker is a cleavable ADC linker, used in antibody-drug conjugates (ADCs) synthesis[1].
    Fórmula:C14H16N2O8S2
    Pureza:97.89% - 99.94%
    Cor e Forma:Powder
    Peso molecular:404.42
  • GPX-100

    CAS:
    <p>GPX-100 (13-deoxydoxorubicin) is an anthracycline antitumour antibiotic that inhibits DNA replication by interacting with topoisomerase II.</p>
    Fórmula:C27H31NO10
    Pureza:95.91%
    Cor e Forma:Solid
    Peso molecular:529.54
  • Nevanimibe hydrochloride

    CAS:
    <p>Nevanimibe hydrochloride (PD-132301 hydrochloride) is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50</p>
    Fórmula:C27H40ClN3O
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:458.08
  • Gusacitinib

    CAS:
    <p>Gusacitinib (ASN-002) (ASN-002) is spleen tyrosine kinase (SYK) and janus kinase (JAK) inhibitor (IC50: 5-46 nM).</p>
    Fórmula:C24H28N8O2
    Pureza:98.06% - 99.94%
    Cor e Forma:Solid
    Peso molecular:460.53
  • hGPR91 antagonist 1

    CAS:
    <p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>
    Fórmula:C31H23F4N3O
    Pureza:98.89%
    Cor e Forma:Solid
    Peso molecular:529.53
  • Ethylenediaminetetraacetic acid trisodium salt

    CAS:
    <p>Ethylenediaminetetraacetic acid trisodium salt (EDTA Trisodium) used to bind metal ions in the chelation therapy.</p>
    Fórmula:C10H13N2Na3O8
    Pureza:99.92% - 99.96%
    Cor e Forma:White Crystals
    Peso molecular:358.19
  • Ciproquazone

    CAS:
    <p>Ciproquazone has analgesic activity and is used to treat spondylitis.</p>
    Fórmula:C19H18N2O2
    Pureza:99.30%
    Cor e Forma:Solid
    Peso molecular:306.36
  • Tigecycline

    CAS:
    <p>Tigecycline (GAR-936), a broad-spectrum glycylcycline, disrupts protein synthesis by binding the 30S ribosomal subunit.</p>
    Fórmula:C29H39N5O8
    Pureza:98.81% - >99.99%
    Cor e Forma:Powder
    Peso molecular:585.65
  • L-Ascorbic acid 2-phosphate trisodium

    CAS:
    <p>L-Ascorbic acid 2-phosphate trisodium (Sodium ascorbyl phosphate) is a long-acting vitamin C derivative that stimulates collagen expression and formation.</p>
    Fórmula:C6H6Na3O9P
    Pureza:99.81% - >99.99%
    Cor e Forma:Solid
    Peso molecular:322.05
  • Centrinone

    CAS:
    <p>Centrinone (LCR-263) (LCR-263) is a reversible inhibitor of polo-like kinase 4 (PLK4; Ki:0.16 nM).</p>
    Fórmula:C26H25F2N7O6S2
    Pureza:98.76%
    Cor e Forma:Solid
    Peso molecular:633.65
  • Tiragolumab

    CAS:
    <p>Tiragolumab, a monoclonal antibody, targets TIGIT and is used with Atezolizumab to treat solid tumors like lung cancer.</p>
    Pureza:SDS-PAGE:95.3%;SEC-HPLC:98.8%
    Cor e Forma:Liquid
    Peso molecular:148.3 kDa
  • Inobrodib

    CAS:
    <p>Inobrodib (CBP-IN-1) is a potent inhibitor of p300/CBP bromodomain.</p>
    Fórmula:C30H32F2N4O3
    Pureza:98.91% - 99.18%
    Cor e Forma:Solid
    Peso molecular:534.6
  • Rapamycin

    CAS:
    <p>Rapamycin, a macrolide from Streptomyces hygroscopicus, inhibits mTOR (IC50: 0.1 nM) and promotes autophagy with immunosuppressive effects.</p>
    Fórmula:C51H79NO13
    Pureza:97.08% - 99.80%
    Cor e Forma:Yellow Solid
    Peso molecular:914.17
  • ATG7-IN-1

    CAS:
    <p>ATG7-IN-1 is a selective ATG7 inhibitor with an IC50 of 62 nM.</p>
    Fórmula:C17H19FN6O5S2
    Pureza:99.85% - >99.99%
    Cor e Forma:Solid
    Peso molecular:470.5
  • Oxolinic acid

    CAS:
    <p>Oxolinic acid (Nidantin) is a synthetic antimicrobial related to NALIDIXIC ACID and used in URINARY TRACT INFECTIONS.</p>
    Fórmula:C13H11NO5
    Pureza:98.39% - 99.72%
    Cor e Forma:Crystals From Dimethylformamide White Crystalline Powder
    Peso molecular:261.23
  • Articaine hydrochloride

    CAS:
    <p>Articaine hydrochloride (Hoe-045) is a thiophene-containing local anesthetic pharmacologically similar to MEPIVACAINE.</p>
    Fórmula:C13H21ClN2O3S
    Pureza:99.76%
    Cor e Forma:White Crystalline Powder
    Peso molecular:320.84
  • Devapamil

    CAS:
    <p>Devapamil (Devapamilo) is a phenylalkylamine that blocks L-type calcium currents from the inner side of membrane cells in a use-dependent manner.</p>
    Fórmula:C26H36N2O3
    Pureza:99.63%
    Cor e Forma:Solid
    Peso molecular:424.58
  • EC23

    CAS:
    <p>EC23 (AGN 190205) is a stable synthetic retinoid analogue. It is also induces neuronal differentiation.</p>
    Fórmula:C23H24O2
    Pureza:99.64%
    Cor e Forma:Solid
    Peso molecular:332.44
  • Nidanilimab

    CAS:
    <p>Nidanilimab (CAN04) is an IL1RAP antibody with 1.10 pM affinity and antitumor effects on NSCLC and PDAC.</p>
    Pureza:> 95%
    Cor e Forma:Soild
    Peso molecular:150 kDa
  • HBX 19818

    CAS:
    <p>HBX 19818 is a specific ubiquitin-specific protease 7 (USP7) inhibitor (IC50: 28.1 μM).</p>
    Fórmula:C25H28ClN3O
    Pureza:97.71%
    Cor e Forma:Solid
    Peso molecular:421.96
  • AP20187

    CAS:
    <p>AP20187: Cell-permeable ligand dimerizing FKBP fusion proteins for signaling and gene expression control.</p>
    Fórmula:C82H107N5O20
    Pureza:99.05% - 99.80%
    Cor e Forma:Solid
    Peso molecular:1482.75
  • Muraglitazar

    CAS:
    Muraglitazar (BMS-298585) is a PPAR α/γ dual agonist for the treatment of type 2 diabetes and associated dyslipidemia.
    Fórmula:C29H28N2O7
    Pureza:99.17%
    Cor e Forma:Solid
    Peso molecular:516.54
  • GSK3145095

    CAS:
    GSK3145095 is an orally active inhibitor of RIPK1 with IC50 of 5 nM, with potential immunomodulatory activities and antineoplastic.
    Fórmula:C20H17F2N5O2
    Pureza:99.50%
    Cor e Forma:Solid
    Peso molecular:397.38
  • Col003

    CAS:
    <p>Col003 is a selective and potent inhibitor of Hsp47 and competitively binds to the collagen-binding site on Hsp47 (IC50: 1.8 μM).</p>
    Fórmula:C14H11NO4
    Pureza:98.67% - 99.03%
    Cor e Forma:Solid
    Peso molecular:257.24
  • Doxepin hydrochloride

    CAS:
    <p>Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.</p>
    Fórmula:C19H22ClNO
    Pureza:99.65% - 99.91%
    Cor e Forma:White To Off-White Powder
    Peso molecular:315.84
  • DUPA(OtBu)-OH

    CAS:
    <p>DUPA(OtBu)-OH, a DUPA precursor, targets PSMA with high affinity (Ki=8nM) to deliver Docetaxel for prostate cancer therapy.</p>
    Fórmula:C23H40N2O9
    Pureza:97.29%
    Cor e Forma:Solid
    Peso molecular:488.57
  • Oxeladin citrate

    CAS:
    <p>Oxeladin citrate: potent, non-addictive cough suppressant safe for all ages and heart patients; no common antitussive side effects.</p>
    Fórmula:C26H41NO10
    Pureza:97.23%
    Cor e Forma:Solid
    Peso molecular:527.6
  • Pralidoxime Chloride

    CAS:
    <p>Pralidoxime Chloride (2-PAM chloride) is a agent in the treatment of organophosphate poisoning, which binds to organophosphate-inactivated acetylcholinesterase.</p>
    Fórmula:C7H9ClN2O
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:172.61
  • (R)-ADX-47273

    CAS:
    <p>(R)-ADX-47273 is a potent mGluR5 positive allosteric modulator(EC50 of 168 nM for potentiation ).</p>
    Fórmula:C20H17F2N3O2
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:369.36
  • trans-C75

    CAS:
    <p>trans-C75 ((±)-C75) is an enantiomer of C75. C75 is an inhibitor of fatty-acid synthase (FASN).</p>
    Fórmula:C14H22O4
    Pureza:98.88% - 99.57%
    Cor e Forma:White To Off-White Solid
    Peso molecular:254.32
  • Aminophylline

    CAS:
    <p>Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.</p>
    Fórmula:C7H8O2·C2H8N2
    Pureza:99.31%
    Cor e Forma:White Or Slightly Yellowish Granules Or Powder Solid
    Peso molecular:420.43
  • Enoxacin

    CAS:
    <p>Enoxacin (NSC-629661) is a broad-spectrum 6-fluoronaphthyridinone antibacterial agent (fluoroquinolones) structurally related to nalidixic acid.</p>
    Fórmula:C15H17FN4O3
    Pureza:98.68% - 99.89%
    Cor e Forma:Off-White To Yellow Crystals
    Peso molecular:320.32
  • BI-1935

    CAS:
    <p>BI-1935 is an inhibitor of soluble epoxide hydrolase (sEH). For diseases related to cardiovascular disease.</p>
    Fórmula:C24H21F3N6O3
    Pureza:97.55%
    Cor e Forma:Solid
    Peso molecular:498.46
  • Lonidamine

    CAS:
    <p>Lonidamine (Diclondazolic Acid) is an indazole carboxylic acid derivative, principally inhibiting aerobic glycolytic activity, by its effect on mitochondrially-</p>
    Fórmula:C15H10Cl2N2O2
    Pureza:97.90%
    Cor e Forma:White To Light Yellow Crystal
    Peso molecular:321.16
  • Maltose monohydrate

    CAS:
    <p>D-(+)-Maltose monohydrate (D-(+)-Maltose monohydrate), a dextrodisaccharide from starch and malt, is used as a fermentable intermediate and sweetening agent in</p>
    Fórmula:C12H2201·H2O
    Pureza:98.41%
    Cor e Forma:Powder
    Peso molecular:360.31
  • Sulfamethoxypyridazine

    CAS:
    <p>Sulfamethoxypyridazine (CL 13494) is a sulfanilamide antibacterial agent.</p>
    Fórmula:C11H12N4O3S
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:280.3
  • SLU-PP-332

    CAS:
    <p>SLU-PP-332 is a pan-estrogen receptor-related receptor (ERR) agonist with high affinity for ERRα, ERRβ, and ERRγ with EC50 values of 98, 230, and 430 nM,</p>
    Fórmula:C18H14N2O2
    Pureza:98.3% - 98.60%
    Cor e Forma:Soild
    Peso molecular:290.32
  • Isotretinoin

    CAS:
    <p>Isotretinoin (13-cis-Retinoic acid) binds to and activates nuclear retinoic acid receptors (RARs); activated RARs serve as transcription factors that promote</p>
    Fórmula:C20H28O2
    Pureza:97.01% - 98.06%
    Cor e Forma:Reddish-Orange Plates From Isopropyl Alcohol (Ntp 1992)
    Peso molecular:300.44
  • Cyclamic acid

    CAS:
    <p>Cyclamic acid, a synthetic sweetener (NSC-220327), often used as Na/Ca cyclamate. Banned in USA over disputed cancer risk.</p>
    Fórmula:C6H13NO3S
    Pureza:98.42%
    Cor e Forma:White Crystals
    Peso molecular:179.24
  • Vitamin D2

    CAS:
    <p>Ergocaliferol (Vitamin D2), derived from ergosterol by UV, inhibits bladder tumor promotion and leukemia, and blocks DNA Polymerase.</p>
    Fórmula:C28H44O
    Pureza:98.73% - 99.89%
    Cor e Forma:Prisms From Acetone 1998)
    Peso molecular:396.65
  • Clopidogrel

    CAS:
    <p>Clopidogrel (SR-25990C), a P2Y12 receptor antagonist, decreases platelet aggregation.</p>
    Fórmula:C16H16ClNO2S
    Pureza:98.23% - 98.83%
    Cor e Forma:White Powder
    Peso molecular:321.82
  • Retagliptin Phosphate

    CAS:
    <p>Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.</p>
    Fórmula:C19H21F6N4O7P
    Pureza:98.70%
    Cor e Forma:Solid
    Peso molecular:562.36
  • Metyrapone

    CAS:
    <p>Metyrapone (NSC-25265) blocks steroid 11β-monooxygenase, used to diagnose Cushing's syndrome.</p>
    Fórmula:C14H14N2O
    Pureza:99.03% - ≥95%
    Cor e Forma:Crystals From Ether & Pentane Solid
    Peso molecular:226.27
  • Acemetacin

    CAS:
    <p>Acemetacin (TVX 1322) is a carboxymethyl ester of indometacin.</p>
    Fórmula:C21H18ClNO6
    Pureza:99.26%
    Cor e Forma:Light Yellow Solid
    Peso molecular:415.82
  • Diminazene Aceturate

    CAS:
    <p>Diminazene is a trypanocidal agent.</p>
    Fórmula:C22H29N9O6
    Pureza:96.86% - 99.58%
    Cor e Forma:Solid
    Peso molecular:515.52
  • MIM1

    CAS:
    <p>MIM1 (Inhibitor of Mcl-1) is an myeloid cell factor 1 (Mcl-1) inhibitor.</p>
    Fórmula:C17H21N3O3S
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:347.43
  • Sulfalene

    CAS:
    <p>Sulfalene (SMP2), a long-acting sulfonamide antibiotic, is used for the therapy of chronic bronchitis, urinary tract infections, and malaria.</p>
    Fórmula:C11H12N4O3S
    Pureza:99.24% - 99.52%
    Cor e Forma:White Or Slightly Yellow Crystal Powder
    Peso molecular:280.3
  • p-MPPI hydrochloride

    CAS:
    <p>p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.</p>
    Fórmula:C25H28ClIN4O2
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:578.87
  • Benazepril hydrochloride

    CAS:
    <p>Benazepril hydrochloride (CGS 14824A HCl) is an angiotensin-converting enzyme (ACE) inhibitor widely used in the therapy of hypertension.</p>
    Fórmula:C24H29ClN2O5
    Pureza:99.68% - ≥95%
    Cor e Forma:Crystalline Solid
    Peso molecular:460.95
  • ZX-29

    CAS:
    <p>ZX-29: Strong ALK inhibitor; IC50 - ALK 2.1 nM, L1196M 1.3 nM, G1202R 3.9 nM; triggers autophagy; anti-cancer.</p>
    Fórmula:C23H28ClN7O3S
    Pureza:98.32%
    Cor e Forma:Solid
    Peso molecular:518.03
  • Omeprazole metabolite Omeprazole sulfone

    CAS:
    <p>Omeprazole metabolite Omeprazole sulfone can inhibit proton pump.</p>
    Fórmula:C17H19N3O4S
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:361.42
  • Hydralazine hydrochloride

    CAS:
    <p>Hydralazine hydrochloride, an antihypertensive phthalazine, induces vasodilation and may inhibit tumor DNA methylation.</p>
    Fórmula:C8H9ClN4
    Pureza:99.85% - 99.86%
    Cor e Forma:Yellow Crystals White Crystalline Solid
    Peso molecular:196.64
  • Regorafénib N-oxyde (M2)

    CAS:
    <p>Regorafénib N-oxyde M2 is an active metabolite of Regorafenib.</p>
    Fórmula:C21H15ClF4N4O4
    Pureza:98.03% - 98.26%
    Cor e Forma:Solid
    Peso molecular:498.81
  • Medrysone

    CAS:
    <p>Medrysone is a synthetic glucocorticoid for topical use with anti-inflammatory and anti-allergic effects, altering gene expression to reduce inflammation.</p>
    Fórmula:C22H32O3
    Pureza:97.72% - 99.91%
    Cor e Forma:Solid
    Peso molecular:344.49
  • Zidebactam

    CAS:
    <p>Zidebactam (WCK-5107) is an effective β-lactamase inhibitor. Zidebactam also is a penicillin-binding protein2 inhibitor (IC50: 0.26 μg/mL).</p>
    Fórmula:C13H21N5O7S
    Pureza:96.85% - 99.69%
    Cor e Forma:Solid
    Peso molecular:391.4
  • 4-Nonylphenol polyethoxylate

    CAS:
    <p>4-Nonylphenol polyethoxylate (Nonoxinol-9) is a typical surfactant used as a vaginal spermicide. Spermicides are locally acting non-hormonal contraceptives.</p>
    Fórmula:(C2H4O)nC15H24O
    Pureza:98%
    Cor e Forma:Compounds With N20 Are Pale-Yellow To Off-White Pastes Or Waxes Liquid Liquid
    Peso molecular:514.69
  • AZ7550 hydrochloride

    CAS:
    <p>AZ7550 hydrochloride (AZ7550 hydrochloride ), an active metabolite of AZD9291, inhibits the activity of IGF1R (IC50: 1.6 μM).</p>
    Fórmula:C27H32ClN7O2
    Pureza:99.65%
    Cor e Forma:Solid
    Peso molecular:522.04
  • Teneliximab

    CAS:
    <p>Teneliximab (BMS 224819) is a chimeric monoclonal antibody that blocks CD40-CD40L interactions.Cost-effective and quality-assured.</p>
    Pureza:95.00% - 99.19% (SEC-HPLC)
    Cor e Forma:Liquid
    Peso molecular:146.06 kDa
  • K-604 dihydrochloride

    CAS:
    <p>K-604 dihydrochloride is a potent and selective acyl-CoA:cholesterol acyltransferase 1 inhibitor with an IC50 of 0.45±0.06 μM.</p>
    Fórmula:C23H32Cl2N6OS3
    Pureza:99.10% - 99.74%
    Cor e Forma:Solid
    Peso molecular:575.64
  • Bispyrazolone

    CAS:
    <p>Bispyrazolone (NSC-37393) is light yellow or white crystalline powder.</p>
    Fórmula:C20H18N4O2
    Pureza:99.40%
    Cor e Forma:Cream To Yellow Crystalline Powder
    Peso molecular:346.38
  • Allylestrenol

    CAS:
    Allylestrenol (Gestanin) is a synthetic steroid with progestational activity.
    Fórmula:C21H32O
    Pureza:>99.99%
    Cor e Forma:White Crystalline Powder
    Peso molecular:300.48
  • Tetracaine hydrochloride

    CAS:
    <p>Tetracaine HCl (Pontocaine), a potent local anesthetic and antipruritic, is used in eye care and for surface/spinal anesthesia.</p>
    Fórmula:C15H25ClN2O2
    Pureza:99.72% - 99.94%
    Cor e Forma:White Or Off White Crystalline Powder
    Peso molecular:300.82
  • (-)-Syringaresinol

    CAS:
    <p>(-)-Syringaresinol from Annona Montana stems inhibits HL-60 cell growth, induces G1 arrest, apoptosis, and has anti-cancer properties.</p>
    Fórmula:C22H26O8
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:418.44
  • (+)-Camphor

    CAS:
    <p>(+)-Camphor (D-Camphor) is the oil extracted from the wood of the Camphor tree Cinnamomum Camphora with anti-inflammatory and analgesic properties.</p>
    Fórmula:C10H16O
    Pureza:98.82%
    Cor e Forma:Less Or White Crystals Sublimes Flash Point 149°F Burns Readily With A Bright Smoky Flame Penetrating Aromatic Odor Pungent Aromatic Taste Followed By A Sensation Of
    Peso molecular:152.23
  • Trifluridine

    CAS:
    <p>Trifluridine is a fluorinated thymidine analog with antineoplastic and antiviral properties, disrupting DNA and protein synthesis, leading to apoptosis.</p>
    Fórmula:C10H11F3N2O5
    Pureza:99.39% - 99.82%
    Cor e Forma:White Crystalline Powder
    Peso molecular:296.2
  • Onvatilimab

    CAS:
    <p>Onvatilimab (JNJ-61610588) is a human IgG1 κ monoclonal antibody with antitumor effects for advanced head and neck cancers.</p>
    Pureza:98.11% (SEC-HPLC) - > 95%
    Cor e Forma:Liquid
    Peso molecular:144.52 kDa
  • Glipizide

    CAS:
    <p>Glipizide (CP 28720) is a short-acting, second-generation sulfonylurea with hypoglycemic activity.</p>
    Fórmula:C21H27N5O4S
    Pureza:99.67% - 99.75%
    Cor e Forma:Solid
    Peso molecular:445.54
  • Boc-Gln-Ala-Arg-AMC hydrochloride

    CAS:
    <p>Boc-Gln-Ala-Arg-AMC HCl: A fluorescent tracer for trypsin and TMPRSS2 protein hydrolysis.</p>
    Fórmula:C29H43ClN8O8
    Pureza:99.59%
    Cor e Forma:Solid
    Peso molecular:667.15
  • Orlistat

    CAS:
    Orlistat (Tetrahydrolipstatin) is a lipase inhibitor and a FASN inhibitor. Orlistat has been shown to promote weight loss. Cost effective and quality assured.
    Fórmula:C29H53NO5
    Pureza:99.58% - >99.99%
    Cor e Forma:White Crystalline Powder
    Peso molecular:495.73
  • Nimodipine

    CAS:
    <p>Nimodipine (BAY-e 9736), a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle cells.</p>
    Fórmula:C21H26N2O7
    Pureza:99.64% - 99.79%
    Cor e Forma:Solid
    Peso molecular:418.44
  • Monoelaidin

    CAS:
    <p>Monoelaidin is a poorly water-soluble drug enhancer of solubility and oral bioavailability.</p>
    Fórmula:C21H40O4
    Pureza:99.05%
    Cor e Forma:Solid
    Peso molecular:356.54
  • Thioctamide

    CAS:
    <p>Thioctamide is 6,8-dithiooctanoic amide; carboxyl changes to amide linking to proteins/amines.</p>
    Fórmula:C8H15NOS2
    Pureza:99.47%
    Cor e Forma:Solid
    Peso molecular:205.34
  • Pepstatin

    CAS:
    <p>Pepstatin (Pepsin Inhibitor S 735A) is a specific and orally aspartate protease inhibitor that also inhibits HIV protease activity. Cost effective and quality assured.</p>
    Fórmula:C34H63N5O9
    Pureza:96.74% - 99.94%
    Cor e Forma:Solid
    Peso molecular:685.89
  • Amoxapine

    CAS:
    <p>Amoxapine (CL-67772) exerts its antidepressant effect by inhibiting the re-uptake of norepinephrine and, to a lesser degree, of serotonin, at adrenergic nerve</p>
    Fórmula:C17H16ClN3O
    Pureza:98.25% - 98.80%
    Cor e Forma:Solid
    Peso molecular:313.78
  • Amatuximab

    CAS:
    <p>Amatuximab is a chimeric humanized IgG1/k antibody targeting MSLN with antitumor effects for solid tumors.</p>
    Pureza:SDS-PAGE:95.2%;SEC-HPLC:98.4%
    Cor e Forma:Liquid
    Peso molecular:144.31 kDa
  • Nithiamide

    CAS:
    <p>Nithiamide (CL-5279) is an orally available antiprotozoan agent used in the treatment of vaginal trichomoniasis.</p>
    Fórmula:C5H5N3O3S
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:187.18