Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.687 produtos)
- Apoptose(6.097 produtos)
- Ciclo celular/Ponto de verificação(4.691 produtos)
- Cromatina/Epigenética(2.376 produtos)
- Sinalização Citoesquelética(1.472 produtos)
- Dano de DNA/Reparo de DNA(2.921 produtos)
- Endocrinologia/Hormónios(3.611 produtos)
- Enzima(3.655 produtos)
- GPCR/Proteína-G(8.755 produtos)
- Imunologia e Inflamação(3.765 produtos)
- Vírus da Influenza(298 produtos)
- Sinalização JAK/STAT(407 produtos)
- Sinalização MAPK(1.230 produtos)
- Transportador de Membranas/Canal Iónico(2.947 produtos)
- Metabolismo(9.940 produtos)
- Microbiologia/Virologia(7.347 produtos)
- Neurociência(10.240 produtos)
- Outros inibidores(36.533 produtos)
- Oxidação-Redução(43 produtos)
- Sinalização PI3K/Akt/mTOR(1.437 produtos)
- Proteases/Proteassoma(1.675 produtos)
- Células - tronco e Derivados(830 produtos)
- Tirosina Quinase/Adaptador(2.028 produtos)
- Ubiquitinação(1.682 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66582 produtos de "Inibidores"
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USP15-IN-1
CAS:<p>USP15-IN-1 is a potent USP15 inhibitor (IC50 is 3.76 μM).</p>Fórmula:C22H23N3O3Pureza:99.509% - 99.81%Cor e Forma:SolidPeso molecular:377.44Simmitecan hydrochloride
CAS:<p>Simmitecan hydrochloride is a camptothecin derivative, a topoisomerase I inhibitor with anticancer activity, which can be used to study is solid tumors.</p>Fórmula:C34H39ClN4O6Pureza:98.20% - 98.93%Cor e Forma:SolidPeso molecular:635.15JTK-109
CAS:JTK-109 is an inhibitor of hepatitis C virus NS5B RNA-dependent RNA polymerase inhibitor and inhibits G1b and G3a subgenomic replicons and recombinant enzymes.Fórmula:C37H33ClFN3O4Pureza:98.48% - 99.68%Cor e Forma:SolidPeso molecular:638.13Aleglitazar
CAS:<p>Aleglitazar (R1439) (R1439) is a potent dual PPARα/γ agonist, with IC50s of 38 nM and 19 nM for human PPARa and PPARγ, respectively.</p>Fórmula:C24H23NO5SPureza:99.03%Cor e Forma:SolidPeso molecular:437.51AKT Kinase Inhibitor
CAS:AKT Kinase Inhibitor is an Akt inhibitor with antitumor activity that selectively inhibits cell proliferation in a dose-dependent manner.Cost-effective and quality-assured.Fórmula:C16H19N7O3Pureza:97.83% - 99.13%Cor e Forma:SolidPeso molecular:357.37LY2979165
CAS:LY2979165 (mGlu2 agonist) is an orthosteric agonist of mGluR2 and can be used in studies about serving as an anti-depressant.Fórmula:C13H22N6O6SPureza:98.41%Cor e Forma:SolidPeso molecular:390.42Suzetrigine
CAS:Suzetrigine (VX-548) is an oral NaV1.8 inhibitor with analgesic properties for acute pain research.Fórmula:C21H20F5N3O4Pureza:98.08% - 99.27%Cor e Forma:SolidPeso molecular:473.39BDZ-g
CAS:BDZ-g: potent, selective AMPA receptor antagonist; useful for researching neurological disorders.Fórmula:C21H21N5O2SPureza:99.97%Cor e Forma:SolidPeso molecular:407.49NRX-252114
CAS:NRX-252114 promotes mutant β-catenin degradation, binding it to E3 ligase SCFβ-TrCP (EC50: 6.5 nM; Kd: 0.4 nM).Fórmula:C22H12Cl2F3N3O2SPureza:99.70%Cor e Forma:SolidPeso molecular:510.32BLU2864
CAS:BLU2864: oral PRKACA inhibitor, IC50=0.3 nM, potential in cancer/poly. kidney disease research.Fórmula:C24H19F3N4O2Pureza:97.58% - 99.92%Cor e Forma:SoildPeso molecular:452.43Picrotoxinin
CAS:<p>Picrotoxinin blocks chloride channels, antagonizes GABAA noncompetitively (IC50: 1.15 μM, α1β2γ2L), and induces convulsions.</p>Fórmula:C15H16O6Pureza:98.07%Cor e Forma:SolidPeso molecular:292.28CP-642931
CAS:CP-642931 (Sorbitol dehydrogenase-IN-1) is a sorbitol dehydrogenase inhibitor used in the study of diabetes mellitus and cardiovascular disease.Fórmula:C17H25N7OPureza:99.67% - >99.99%Cor e Forma:SolidPeso molecular:343.43SY-5609
CAS:SY-5609 (CDK7-IN-3) is a selective non-covalent CDK7 inhibitor, with weak inhibitory activity against CDK2, CDK9 and CDK12.Cost-effective and quality-assured.Fórmula:C23H26F3N6OPPureza:99.34% - >99.99%Cor e Forma:SolidPeso molecular:490.46GSK3368715 dihydrochloride
CAS:GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is a PRMTs inhibitor , with anticancer activity, for the study of advanced solid tumors.Fórmula:C20H40Cl2N4O2Pureza:99.66% - 99.66%Cor e Forma:SolidPeso molecular:439.46Zelasudil
CAS:<p>Zelasudil (RXC007) is a Rho-related (ROCK) kinase inhibitor for the study of idiopathic pulmonary fibrosis and inflammation.</p>Fórmula:C22H21F2N7OPureza:99.15%Cor e Forma:SolidPeso molecular:437.445Gepotidacin mesylate dihydrate
CAS:Gepotidacin mesylate dihydrate (GSK2140944 mesylate dihydrate) is an antibiotic and an inhibitor of bacterial type II topoisomerase.Fórmula:C25H36N6O8SPureza:99.85%Cor e Forma:SolidPeso molecular:580.65Cbl-b-IN-3
CAS:Cbl-b-IN-3 is a potent inhibitor of casitas b lineage lymphoma proto-oncogene-b (Cbl-b) (ic50 < 1 nM).Cost-effective and quality-assured.Fórmula:C30H34F3N5OPureza:97.63%Cor e Forma:SolidPeso molecular:537.62USP5-IN-1
<p>USP5-IN-1, a powerful USP5 deubiquitinase inhibitor, selectively binds with 2.8 μM affinity, blocking USP5's di-ubiquitin cleavage.</p>Fórmula:C19H20ClN3O5SPureza:99.76%Cor e Forma:SoildPeso molecular:437.9IDX184
CAS:IDX184 is a potent, orally active, targeted HCV polymerase inhibitor and nucleoside polymerase.IDX184 effectively inhibits HCV polymerase (IC50=0.31 μM, Ki=52.3Fórmula:C25H35N6O9PSPureza:97.15%Cor e Forma:SolidPeso molecular:626.62WAY-213613 hydrochloride
CAS:WAY-213613 hydrochloride: potent, selective GLT-1/EAAT2 inhibitor (IC50 85 nM); weaker for EAAT1/3; inactive at glutamate receptors; research tool for CNS.Fórmula:C16H13BrF2N2O4Pureza:99.14% - 99.37%Cor e Forma:SoildPeso molecular:415.19MAO-B-IN-17
CAS:MAO-B-IN-17 is a selective and potent monoamine oxidase B (MAO-B) inhibitor (IC50: 5.08 μM) for the study of central nervous system disorders like Parkinson's.Fórmula:C17H17F2NO2Pureza:99.41%Cor e Forma:SoildPeso molecular:305.32(+)-Tetrabenazine
CAS:(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-foldFórmula:C19H27NO3Pureza:98.69%Cor e Forma:SolidPeso molecular:317.42Vecabrutinib
CAS:<p>Vecabrutinib (SNS-062) is a potent and noncovalent BTK and ITK inhibitor (Kd: 0.3 nM and 2.2 nM, respectively). Vecabrutinib displays an IC50 of 24 nM for ITK.</p>Fórmula:C22H24ClF4N7O2Pureza:99.74%Cor e Forma:SolidPeso molecular:529.92AChE/BChE-IN-10
CAS:<p>AChE/BChE-IN-10 inhibits AChE/BChE (IC50: 0.176/0.47 μM), crosses the blood-brain barrier, and prevents Aβ-aggregation.</p>Fórmula:C26H30N2O2Pureza:99.55% - 99.88%Cor e Forma:SoildPeso molecular:402.53HRO761
CAS:HRO761 is a potent Werne r syndrome RecQ DNA deconjugase (WRN) inhibitor that can be used to study cancers such as colon and stomach cancer.Fórmula:C31H31ClF3N9O5Pureza:98.74% - 99.62%Cor e Forma:SolidPeso molecular:702.08HOIPIN-8 sodium
CAS:<p>HOIPIN-8 sodium is a LUBAC inhibitor for the study of inflammatory and immune diseases.</p>Fórmula:C23H15F2N4NaO3Pureza:97.34%Cor e Forma:SolidPeso molecular:456.38Obicetrapib
CAS:<p>Obicetrapib (AMG-899) is an inhibitor of cholesteryl ester transfer protein.</p>Fórmula:C32H31F9N4O5Pureza:99.26% - >99.99%Cor e Forma:SolidPeso molecular:722.6Treprostinil diethanolamine
CAS:<p>Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1,</p>Fórmula:C27H45NO7Pureza:99.86%Cor e Forma:SolidPeso molecular:495.65BCL6-IN-3
CAS:BCL6-IN-3: potent BCL6 inhibitor, 70 nM GI50 in SU-DHL4, affects cell functions, antitumor.Fórmula:C24H31ClF2N6O2Pureza:98.17%Cor e Forma:SolidPeso molecular:508.99NB-360
CAS:NB-360: potent, brain-penetrant BACE1/2 inhibitor; IC50s: 5-6 nM; high selectivity vs pepsin, cathepsin E/D.Fórmula:C21H19F4N5O2Pureza:99.72%Cor e Forma:SolidPeso molecular:449.4Iclepertin
CAS:Iclepertin (BI-425809) is a GlyT1 inhibitor.Iclepertin is used for the treatment of Alzheimer;s disease and other CNS disorders.Fórmula:C20H18F6N2O5SPureza:98.89% - 98.93%Cor e Forma:SolidPeso molecular:512.42Elacytarabine
CAS:<p>Elacytarabine (M7594 0037), a lipid-conjugated derivative of the nucleoside analog cytarabine, is an antineoplastic drug. It has cytotoxicity in solid tumors.</p>Fórmula:C27H45N3O6Pureza:97.69%Cor e Forma:SolidPeso molecular:507.66MIV-247
CAS:MIV-247 is a cathepsin S inhibitor that attenuates mechanically abnormal pain in preclinical neuropathic pain models and can be used to study myocardial injury.Fórmula:C17H24F3N3O4Pureza:99.27%Cor e Forma:SolidPeso molecular:391.39Zotizalkib
CAS:<p>TPX-0131: potent, selective, CNS-ready, oral ALK inhibitor (WT IC50: 1.4nM, G1202R/L1196M IC50: 0.3nM) with robust antitumor effects.</p>Fórmula:C21H20F3N5O3Pureza:98.7%Cor e Forma:SolidPeso molecular:447.41GLPG0974
CAS:<p>GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.</p>Fórmula:C25H25ClN2O4SPureza:99.8%Cor e Forma:SolidPeso molecular:484.99NDI-034858
CAS:NDI-034858 (TAK-279) is a tyrosine kinase 2 (TYK2) inhibitor (Kd<200 pM) that targets the JH2 structural domain of Tyk2 for the treatment of autoimmune diseasesFórmula:C23H24N8O3Pureza:>99.99%Cor e Forma:SolidPeso molecular:460.49BMS 299897
CAS:<p>BMS 299897, a sulfonamide γ-secretase inhibitor, inhibits Aβ production with an IC50 of 7 nM in HEK293 cells overexpressing APP.</p>Fórmula:C24H21ClF3NO4SPureza:99.82%Cor e Forma:SolidPeso molecular:511.94Dersimelagon
CAS:<p>Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist.Cost-effective and quality-assured.</p>Fórmula:C36H45F4N3O5Pureza:97.35% - 98.23%Cor e Forma:SolidPeso molecular:675.75KU-60019
CAS:<p>KU-60019 is a specific inhibitor of ATM kinase (IC50: 6.3 nM).</p>Fórmula:C30H33N3O5SPureza:98.05% - 98.50%Cor e Forma:SolidPeso molecular:547.67Cort108297
CAS:<p>Cort108297: selective GR modulator/antagonist, high GR affinity (Ki: 0.45nM), no other steroid receptor affinity.</p>Fórmula:C26H25F4N3O3SPureza:98.36% - 99.94%Cor e Forma:SolidPeso molecular:535.55Aldometanib
CAS:<p>Aldometanib (LXY-05-029) is an oral aldolase inhibitor that maintains metabolic balance by blocking FBP and activating lysosomal AMPK.</p>Fórmula:C27H43Cl2IN2Pureza:99.32% - 99.55%Cor e Forma:SolidPeso molecular:593.46Etamicastat hydrochloride
CAS:<p>Etamicastat hydrochloride (BIA 5-453 hydrochloride) is a peripherally selective dopamine beta-hydroxylase inhibitor that reduces hypertension.</p>Fórmula:C14H16ClF2N3OSPureza:98.54%Cor e Forma:SolidPeso molecular:347.81LLY-283
CAS:LLY-283, PRMT5 inhibitor, IC50 22 nM, Kd 6 nM, oral, selective, with antitumor effects.Fórmula:C17H18N4O4Pureza:99.49%Cor e Forma:SolidPeso molecular:342.35Vofopitant
CAS:Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for the study of post-traumatic stress disorder (PTSD).Fórmula:C21H23F3N6OPureza:97.86%Cor e Forma:SolidPeso molecular:432.44Rupintrivir
CAS:Rupintrivirvr (AG7088) is a mimetic peptide inhibitor of rhinovirus (HRV) 3C cysteine protease with antiviral activity for the study of viral infections.Fórmula:C31H39FN4O7Pureza:97.72% - 99.35%Cor e Forma:SolidPeso molecular:598.66DN02
<p>DN02: a potent, selective BRD8(1) bromodomain probe; Ki=32 nM; 30x more affine than BRD8(2).</p>Fórmula:C22H24FN3O3Pureza:98.22% - 99.74%Cor e Forma:SolidPeso molecular:397.44Eravacycline dihydrochloride
CAS:<p>Eravacycline dihydrochloride (TP-434-046) is a potent and broad-spectrum antibacterial agent against six E. coli (MICs: 0.125-0.25 mg/L).</p>Fórmula:C27H33Cl2FN4O8Pureza:94.59% - 95%Cor e Forma:SolidPeso molecular:631.48Pocenbrodib
CAS:<p>Pocenbrodib (FT-7051) is a potent inhibitor of the bromodomain of the CBP/p300 family with potential antitumour activity and is palatable for cancer research.</p>Fórmula:C28H32FN3O6Pureza:98.48% - 99.54%Cor e Forma:SolidPeso molecular:525.57STK-15
CAS:STK-15 is a candidate for use as a fatty acid binding protein 5 (FABP5) inhibitor.Fórmula:C34H29NO5Pureza:98.05%Cor e Forma:SolidPeso molecular:531.6AZD5462
CAS:<p>AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart failure and cancer.</p>Fórmula:C30H41FN2O6Pureza:98.32% - 99.63%Cor e Forma:SolidPeso molecular:544.65Vofopitant dihydrochloride
CAS:Vofopitant dihydrochloride (GR 205171A) is a tachykinin NK1 receptor antagonist and a potential compound for the treatment of pathologic vomiting.Fórmula:C21H25Cl2F3N6OPureza:98.99%Cor e Forma:SolidPeso molecular:505.36BQ-788
CAS:<p>BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation of coronary perfusion pressure.</p>Fórmula:C34H51N5O7Pureza:98.81%Cor e Forma:SolidPeso molecular:641.8Umibecestat
CAS:<p>Umibecestat inhibits human and mouse BACE-1 (IC50: 11 nM & 10 nM), potentially for Alzheimer's research.</p>Fórmula:C19H15ClF7N5O2Pureza:99.88%Cor e Forma:SolidPeso molecular:513.8ELOVL1-IN-2
CAS:ELOVL1-IN-2 weakly inhibits ELOVL1 enzyme (IC50: 21 μM) and shows moderate potency in HEK293 cells (IC50: 6.7 μM).Fórmula:C18H15FN2OPureza:99.94%Cor e Forma:SolidPeso molecular:294.32Milademetan
CAS:Milademetan (DS-3032), an MDM2 inhibitor, exhibits antitumor activity, induces G1 cell cycle arrest and apoptosis, and can be used to study solid tumors.Fórmula:C30H34Cl2FN5O4Pureza:>99.99%Cor e Forma:SolidPeso molecular:618.53JNJ-6204
CAS:JNJ-6204 is a deuterated compound that efficiently inhibits CSNK1D and CSNK1E.Fórmula:C19H11D6FN6OPureza:97.42% - 99.87%Cor e Forma:SolidPeso molecular:370.41VX-984
CAS:VX-984 (M9831) is an oral DNA-PK inhibitor, crossing the blood-brain barrier, targeting GBM and NSC-LC.Fórmula:C23H21D2N7OPureza:97.65% - 99.98%Cor e Forma:SolidPeso molecular:415.49AZ12601011
CAS:<p>AZ12601011 is a TGFBR1 kinase inhibitor that inhibits the growth of breast tumors.</p>Fórmula:C19H15N5Pureza:98.81%Cor e Forma:SolidPeso molecular:313.36Evixapodlin
CAS:Evixapodlin (PD-1/PD-L1-IN 7) is a human PD-1/PD-L1 protein/protein interaction inhibitor (IC50: 0.213).Evixapodlin has anticancer and antiviral activities.Fórmula:C34H36Cl2N8O4Pureza:99.07%Cor e Forma:SolidPeso molecular:691.61Enbezotinib
CAS:Enbezotinib is an inhibitor of RET autophosphorylation and can be used in cancer research.Fórmula:C21H21FN6O3Pureza:99.84%Cor e Forma:SolidPeso molecular:424.43SYM2206
CAS:<p>SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 μM.SYM2206 exhibits anticancer activity by blocking Nav1.6-mediated</p>Fórmula:C20H22N4O3Pureza:99.88%Cor e Forma:SolidPeso molecular:366.41ZD 7155 hydrochloride
CAS:ZD 7155 hydrochloride is an angiotensin II receptor type 1 (AT1 receptor) antagonist.Fórmula:C26H27ClN6OPureza:99.8%Cor e Forma:SolidPeso molecular:474.98Moiramide B
CAS:Moiramide B is an acetyl coenzyme A carboxylase inhibitor with antimicrobial activity, strongly inhibiting Gram-positive bacteria.Fórmula:C25H31N3O5Pureza:98.53% - 99.90%Cor e Forma:SolidPeso molecular:453.53NRX-1532
NRX-1532 is a small molecule β-catenin:β-TrCP interaction enhancer.Fórmula:C16H11F3N4O2Pureza:98.95% - 99.94%Cor e Forma:SolidPeso molecular:348.28SDZ 220-040
CAS:<p>SDZ 220-040 是一种选择性哺乳动物 NMDA 受体拮抗剂，可诱导根系生长的部分无重力模式 。</p>Fórmula:C16H16Cl2NO6PPureza:98.13%Cor e Forma:SolidPeso molecular:420.18SB-224289 hydrochloride
CAS:<p>SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.</p>Fórmula:C32H33ClN4O3Pureza:97.82% - 98.99%Cor e Forma:SolidPeso molecular:557.08PF-07258669
CAS:<p>PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.</p>Fórmula:C25H27FN6O2Pureza:99.9%Cor e Forma:SolidPeso molecular:462.52BODIPY FL prazosin
CAS:<p>BODIPY FL prazosin is an α1-adrenergic antagonist that inhibits α1a-AR and α1b-AR.</p>Fórmula:C28H32BF2N7O3Pureza:97.27%Cor e Forma:SolidPeso molecular:563.41CCF0058981
CAS:<p>CCF0058981: noncovalent inhibitor for SARS-CoV-2 & -1 proteases; IC50s: 68 nM (SC2) & 19 nM (SC1). Potential COVID-19 research use.</p>Fórmula:C24H19ClN6OPureza:98.94%Cor e Forma:SoildPeso molecular:442.9LSN3318839
CAS:<p>LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can</p>Fórmula:C26H23Cl2N3O2Pureza:99.21%Cor e Forma:SolidPeso molecular:480.39Odevixibat
CAS:Odevixibat (A4250) is a selective oral inhibitor for ileal bile acid transport, potentially treating primary biliary cirrhosis.Fórmula:C37H48N4O8S2Pureza:99.53% - 99.83%Cor e Forma:SolidPeso molecular:740.93Cap-dependent endonuclease-IN-1
CAS:Cap-dependent endonuclease-IN-1: potent, oral inhibitor with antiviral properties against influenza.Fórmula:C27H22F2N2O6SPureza:99.53% - 99.61%Cor e Forma:SolidPeso molecular:540.54BE1218
CAS:<p>BE1218 is a liver X receptor (LXR) inverse agonist active on LXRα and LXRβ with an IC50 of 9 nM and 7 nM, respectively.</p>Fórmula:C30H30FNO4S2Pureza:99.7%Cor e Forma:SoildPeso molecular:551.69NRX-103095
CAS:<p>NRX-103095 increases β-catenin binding to SCFβ-TrCP E3 ligase; EC50 is 163 nM for pSer33/Ser37 affinity boost.</p>Fórmula:C22H16Cl2F3N3O3SPureza:99.58% - 99.95%Cor e Forma:SolidPeso molecular:530.35FABPs ligand 6
CAS:FABPs ligand 6 (MF6) is an inhibitor of FABP5 and FABP7.Fórmula:C28H27FN2O3Pureza:97.45%Cor e Forma:SolidPeso molecular:458.52O-Propargyl-Puromycin
CAS:O-Propargyl-Puromycin (OP-puro) is a potent protein synthesis inhibitor, a puromycin acetylene analog.Fórmula:C24H29N7O5Pureza:97.83% - 99.29%Cor e Forma:SolidPeso molecular:495.53Tuvusertib
CAS:Tuvusertib (M1774), an oral ATR inhibitor (Ki<1µM), selectively blocks CHK1 phosphorylation, disrupts DNA repair, and induces tumor cell apoptosis.Fórmula:C16H12F2N8OPureza:98.44% - 99.66%Cor e Forma:SolidPeso molecular:370.32SB-423562
CAS:SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.Fórmula:C26H32N2O4Pureza:99.22%Cor e Forma:SolidPeso molecular:436.54INCB054329
CAS:INCB054329 is a BET inhibitor targeting BRD2/3/4 and BRDT with IC50s ranging from 1-119 nM.Fórmula:C19H16N4O3Pureza:99.52%Cor e Forma:SolidPeso molecular:348.36D75-4590
CAS:<p>D75-4590, a β-1,6-Glucan synthetase inhibitor, combats fungal infections by targeting cell walls.</p>Fórmula:C21H27N5Pureza:98.56% - 98.85%Cor e Forma:SolidPeso molecular:349.47SJ6986
CAS:SJ6986 is a potent, selective and orally active GSPT1/2 degrader. SJ6986 degrades GSPT1 with a DC 50 of 2.1 nM (D max 99%) [1].Fórmula:C20H14F3N3O7SPureza:99.73%Cor e Forma:SolidPeso molecular:497.4BMS453
CAS:BMS453 (BMS-189453), a synthetic retinoid, is a potent and selective agonist of RARβ and a potent testicular toxin.Fórmula:C27H24O2Pureza:99.93%Cor e Forma:SolidPeso molecular:380.48DRF-1042
CAS:DRF-1042 is a camptothecin analog with anticancer and insecticidal activity and is used to study solid tumors such as prostate and colon cancer.Fórmula:C22H20N2O6Pureza:98.34%Cor e Forma:SolidPeso molecular:408.4DRB18
CAS:DRB18 inhibits GLUT proteins, altering glucose metabolism and inducing cancer cell death by G1/S arrest and oxidative stress.Fórmula:C22H23ClN2O2Pureza:99.54%Cor e Forma:SolidPeso molecular:382.88Emprumapimod
CAS:Emprumapimod, an oral p38α MAPK inhibitor, targets RPMI-8226 cells, curbs LPS-induced IL-6; IC50: 100 pM; for cardiomyopathy, acute pain.Fórmula:C24H29F2N5O3Pureza:99.21% - >99.99%Cor e Forma:SolidPeso molecular:473.52ALOX15-IN-2
CAS:ALOX15-IN-2: Potent ALOX15 inhibitor. IC50: 1.55 μM for LA; 2.79 μM for AA. Stops linoleic/arachidonic acid oxidation.Fórmula:C23H29N3O4SPureza:99.98%Cor e Forma:SolidPeso molecular:443.56L-371,257
CAS:L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.Fórmula:C28H33N3O6Pureza:99.79%Cor e Forma:SolidPeso molecular:507.58AZD 3147
CAS:<p>AZD 3147 inhibits mTORC1 (40.7 nM), mTORC2 (5.75 nM), and PI3Kα/β/δ/γ (912/5495/9333/6310 nM IC50s).</p>Fórmula:C24H31N5O4S2Pureza:99.99%Cor e Forma:SolidPeso molecular:517.66Glycosyltransferase-IN-1
<p>Glycosyltransferase-IN-1 is a glycosyltransferase inhibitor with bacteriostatic activity, inhibiting MSSA, MRSA, Bacillus subtilis, and Enterobacteriaceae.</p>Fórmula:C19H21N5OPureza:99.76%Cor e Forma:SolidPeso molecular:335.4KI696
CAS:KI696 is a high-affinity probe that potently inhibits the interaction of Keap1 and NRF2.Fórmula:C28H30N4O6SPureza:99.74%Cor e Forma:SolidPeso molecular:550.63BMS-986141
CAS:<p>BMS-986141(UDM-003183) is a selective and potent protease-activated receptor-4 (PAR-4) antagonist with oral activity and an IC50 value of 0.4 nM.BMS-98614</p>Fórmula:C27H23N5O5S2Pureza:98.43% - 99.26%Cor e Forma:SolidPeso molecular:561.63Tigemonam
CAS:<p>Tigemonam is a monobactam, a novel orally administered monobactam that protects against gram-negative aerobic bacterial pathogens. Cost-effective and quality-assured.</p>Fórmula:C12H15N5O9S2Pureza:99.03% - >99.99%Cor e Forma:SolidPeso molecular:437.41EZM0414
CAS:EZM0414 is a potent, selective, orally bioavailable inhibitor of SETD2 with IC50 of 18 nM in SETD2 biochemical assay and IC50 of 34 nM in a cellular assay.Fórmula:C22H29FN4O2Pureza:99.58%Cor e Forma:SolidPeso molecular:400.49Dazostinag disodium
CAS:<p>Dazostinag disodium (TAK-676) is a synthetic novel interferon gene (STING) agonist.Cost-effective and quality-assured.</p>Fórmula:C21H20F2N8Na2O10P2S2Pureza:98.84% - 99.96%Cor e Forma:SolidPeso molecular:754.48Lometrexol
CAS:<p>Lometrexol (LY 264618) is an antifolate that inhibits GARFT, blocks purine synthesis, induces apoptosis, and has anticancer properties.</p>Fórmula:C21H25N5O6Pureza:97.76% - 99.56%Cor e Forma:SolidPeso molecular:443.45AM103
CAS:AM103 is an effective and selective inhibitor of FLAP (IC50 = 4.2 nM).Fórmula:C36H38N3NaO4SPureza:99.75%Cor e Forma:SolidPeso molecular:631.76NRX-103094
CAS:NRX-103094 boosts β-catenin binding to SCFβ-TrCP ligase with EC50 62 nM and Kd 0.6 nM.Fórmula:C20H11Cl2F3N2O4SPureza:99.13%Cor e Forma:SolidPeso molecular:503.28AZD-5672
CAS:<p>AZD-5672 is an antagonist of CCR5 with an IC50 of 0.32 nM.</p>Fórmula:C32H38F2N2O5S2Pureza:98.1%Cor e Forma:SolidPeso molecular:632.78BAY-3827
CAS:BAY-3827 is an AMPK inhibitor with antiproliferative activity and antitumor activity. BAY-3827 inhibits the phosphorylation of acetyl CoA carboxylase 1.Fórmula:C27H25FN6OPureza:99.90%Cor e Forma:SolidPeso molecular:468.53Darizmetinib
CAS:Darizmetinib (HRX215) is an MKK4 inhibitor.Fórmula:C21H17F2N5O3SPureza:98.03% - 99.57%Cor e Forma:SolidPeso molecular:457.45Dual FAAH/sEH-IN-1
CAS:<p>Dual FAAH/sEH-IN-1 inhibits both sEH (IC50: 9.6 nM) and FAAH (IC50: 7 nM), offering potent anti-inflammatory effects.</p>Fórmula:C25H22ClN3O3S2Pureza:99.89%Cor e Forma:SolidPeso molecular:512.04AChE-IN-26
CAS:<p>AChE-IN-26 (compound 4a) is an AChE (acetylcholinesterase) inhibitor (IC50: 0.42 μM).</p>Fórmula:C21H21BrN2O3Pureza:99.24% - 99.85%Cor e Forma:SoildPeso molecular:429.31PREP inhibitor-1
CAS:PREP inhibitor-1 is a prolyl oligopeptidase (PREP) inhibitor for the study of Alzheimer's disease.Fórmula:C22H28N4O2Pureza:98.78%Cor e Forma:SoildPeso molecular:380.48Sinefungin
CAS:Sinefungin (Adenosyl-Ornithine) is an effective inhibitor of virion mRNA(guanine-7-)-methyltransferase, mRNA(nucleoside-2'-)-methyltransferase, and viralFórmula:C15H23N7O5Pureza:98.12%Cor e Forma:SolidPeso molecular:381.3910-Methoxycamptothecin
CAS:10-Methoxycamptothecin is a natural bioactive derivative of camptothecin (CPT) isolated from Camptotheca acuminata and possesses high anti-cancer properties.Fórmula:C21H18N2O5Pureza:98.36%Cor e Forma:SolidPeso molecular:378.38TGFβRI-IN-3
CAS:<p>TGFβRI-IN-3 inhibits TGFβR1 with an IC 50 of 0.79 nM with 2000-fold selectivity against MAP4K4.</p>Fórmula:C28H23N3O2SPureza:99.85%Cor e Forma:SoildPeso molecular:465.57LY3143921 hydrate
CAS:<p>LY3143921 ((S)-Example 2) hydrate is an orally active CDC7 kinase inhibitor with broad in vitro anticancer activity [1].</p>Fórmula:C16H14FN5O2Pureza:98.43%Cor e Forma:SolidPeso molecular:327.31XMD-17-51 Trifluoroacetate
CAS:<p>XMD-17-51 Trifluoroacetate is a pyrimido-diazepinone compound that regulates protein kinases.</p>Fórmula:C23H25F3N8O3Pureza:99.65%Cor e Forma:SolidPeso molecular:518.49Durlobactam sodium salt
CAS:Durlobactam sodium salt (ETX2514) have an IC50 values of 4, 14 and 190 nM against class A KPC-2, class C AmpC and class D OXA-24.Cost-effective and quality-assured.Fórmula:C8H10N3NaO6SPureza:97.01% - 99.03%Cor e Forma:SolidPeso molecular:299.23BAY-8400
<p>BAY-8400 is an orally active, potent and selective DNA-dependent protein kinase ( DNA-PK ) inhibitor ( IC 50 =81 nM) which shows synergistic efficacy in</p>Fórmula:C21H17F2N5OPureza:99.53%Cor e Forma:SolidPeso molecular:393.39BRD0639
CAS:BRD0639 is a first-in-class PRMT5-substrate interaction inhibitor for PBM-dependent PRMT5 activity studies.Fórmula:C21H22ClN5O4SPureza:99.85%Cor e Forma:SolidPeso molecular:475.95PD 151746
CAS:<p>PD151746: calpain inhibitor, Ki μ-calpain=0.26μM, Ki m-calpain=5.33μM; reduces oxLDL cytotoxicity.</p>Fórmula:C11H8FNO2SPureza:98.63% - ≥95%Cor e Forma:SolidPeso molecular:237.25(E/Z)-GSK5182
CAS:<p>GSK5182 is a racemic mix of (E/Z) isomers, a selective ERRγ inverse agonist (IC50: 79 nM), and induces ROS in liver cancer.</p>Fórmula:C27H31NO3Pureza:97.58%Cor e Forma:SolidPeso molecular:417.54Rineterkib
CAS:Rineterkib (ERK-IN-1) is an inhibitor of RAF and ERK1/2 activating mutations in the MAPK pathway.Fórmula:C26H27BrF3N5O2Pureza:99.73%Cor e Forma:SolidPeso molecular:578.42ARN19702
CAS:ARN19702: orally active, brain-penetrant, selective NAAA inhibitor, IC50 230 nM, broad analgesic profile.Fórmula:C21H22FN3O3S2Pureza:99.86%Cor e Forma:SolidPeso molecular:447.55SR 11302
CAS:SR 11302 is an inhibitor of activator protein-1 (AP-1).Fórmula:C26H32O2Pureza:98.65%Cor e Forma:SolidPeso molecular:376.53CK2 inhibitor 2
CAS:CK2 Inhibitor 2, characterized as a potent, selective, and orally active inhibitor of CK2, demonstrates an impressive IC50 value of 0.66 nM.Fórmula:C21H17ClN4O2Pureza:99.02%Cor e Forma:SolidPeso molecular:392.84FGI-106 tetrahydrochloride
CAS:FGI-106 tetrahydrochloride demonstrates potent inhibitory activity across a broad spectrum of viruses, including those causing hemorrhagic fevers such as EbolaFórmula:C28H42Cl4N6Pureza:99.68%Cor e Forma:SolidPeso molecular:604.48JAK2-IN-7
CAS:JAK2-IN-7 selectively inhibits JAK2 (IC50: 3 nM), shows 14-fold selectivity over JAK1/3, FLT3, induces G0/G1 arrest, apoptosis, and has antitumor effects.Fórmula:C26H33N7OPureza:99.54%Cor e Forma:SolidPeso molecular:459.59Gemcitabine elaidate hydrochloride
CAS:<p>CP-4126, a lipophilic pro-drug of Gemcitabine, converts to active form by esterases, allowing oral administration with dose-dependent effects.</p>Fórmula:C27H44ClF2N3O5Pureza:98.50% - 99.6%Cor e Forma:SolidPeso molecular:564.11Rolapitant hydrochloride
CAS:Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki of 0.66 nM.Fórmula:C25H27ClF6N2O2Pureza:98.35% - 99.79%Cor e Forma:SolidPeso molecular:536.94LSZ-102
CAS:LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.Fórmula:C25H17F3O4SPureza:98.56%Cor e Forma:SolidPeso molecular:470.46INCB086550
CAS:<p>INCB086550 (PD-1/PD-L1-IN-8) (example 24) is a PD-1/PD-L1 inhibitor, with an IC50 <= 10 nM.</p>Fórmula:C41H39N7O4Pureza:98.49%Cor e Forma:SolidPeso molecular:693.79Sebetralstat
CAS:<p>Sebetralstat (KVD900) is an inhibitor of plasma kallikrein and can be used in studies about metabolic diseases.</p>Fórmula:C26H26FN5O4Pureza:99.85%Cor e Forma:SolidPeso molecular:491.51FX-11
CAS:<p>FX-11: potent LDHA inhibitor (Ki 8 μM), activates PKM2, reduces ATP, induces oxidative stress/ROS, cell death, shows antitumor effects.</p>Fórmula:C22H22O4Pureza:98.95%Cor e Forma:SolidPeso molecular:350.41Clorophene
CAS:Clorophene (Clorofene) is an antimicrobial agent and can be used in personal care products.Fórmula:C13H11ClOPureza:99.87%Cor e Forma:White To Light Tan Or Pink Flakes Phenolic Odor (Ntp 1992)Peso molecular:218.68GAS6 Protein, Human, Recombinant (His)
<p>GAS6 (Growth arrest-specific protein 6) is also known as AXL receptor tyrosine kinase ligand, AXLLG, is a multimodular protein that is up-regulated by a wide variety of cell types in response to growth arrest. Gas6 binds and induces signaling through the receptor tyrosine kinases Axl, Dtk, and Mer whose signaling is implicated in cell growth and survival, cell adhesion and cell migration. GAS6/AXL signaling plays a role in various processes such as endothelial cell survival during acidification by preventing apoptosis, optimal cytokine signaling during human natural killer cell development, hepatic regeneration, gonadotropin-releasing hormone neuron survival and migration, platelet activation, or regulation of thrombotic responses. GAS6 Protein, Human, Recombinant (His) is expressed in HEK293 cells.</p>Pureza:＞99.90%Cor e Forma:SoildPeso molecular:72.7 KDa (Predicted), 80-90 KDa (Reducing conditions)sodium 4-pentynoate
CAS:<p>sodium 4-pentynoate is a alkynylacetate analogue.</p>Fórmula:C5H5NaO2Pureza:98%Cor e Forma:SolidPeso molecular:120.08N-Octylmaleimide
CAS:<p>N-Octylmaleimide is an alkylmaleimide, which can inhibit rat liver glucose 6-phosphatase.</p>Fórmula:C12H19NO2Cor e Forma:SolidPeso molecular:209.28TEM1/CD248 Protein, Mouse, Recombinant (His)
<p>TEM1/CD248 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 73.6 kDa and the accession number is Q91V98.</p>Cor e Forma:SolidPeso molecular:73.6 kDa (predicted). Due to glycosylation, the protein migrates to 75-140 kDa based on Tris-Bis PAGE result.TCblR Protein, Human, Recombinant (His)
<p>TCblR Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with C-6xHis tag. The predicted molecular weight is 32-58 KDa and the accession number is Q9NPF0.</p>Cor e Forma:SolidPeso molecular:32-58 KDa (reducing condition)Ref: TM-TMPJ
Produto descontinuado4-Ethoxycoumarin
CAS:<p>4-Ethoxycoumarin has antimicrobial activity.</p>Fórmula:C11H10O3Pureza:99.64%Cor e Forma:SolidPeso molecular:190.2Relacorilant
CAS:<p>Relacorilant is an oral glucocorticoid receptor antagonist with Ki of 7.2 nM, potential for treating Cushing's syndrome.</p>Fórmula:C27H22F4N6O3SPureza:98.53% - 99%Cor e Forma:SolidPeso molecular:586.56PRGL493
CAS:<p>PRGL493 blocks ACSL4, halts PC3/MDA-MB-231 cancer cell spread, and inhibits MA-10 tumor progesterone. Effective in mouse PC3 tumor model at 0.25 mg/kg.</p>Fórmula:C25H21N7O2Pureza:98.80% - 99.11%Cor e Forma:SolidPeso molecular:451.483-Methoxyphenylacetic acid
CAS:<p>3-Methoxyphenylacetic acid belongs to the class of organic compounds known as anisoles. 3-Methoxyphenylacetic acid is slightly soluble (in water) and a weakly acidic compound (based on its pKa).3-Methoxyphenylacetic acid (m-Methoxyphenylacetic acid), a m-hydroxyphenylacetic acid (m-OHPAA) derivative, is a phytotoxin in Rhizoctonia solani. 3-Methoxyphenylacetic acid is used to develop a toxin-mediated bioassay for resistance to rhizoctonia root rot</p>Fórmula:C9H10O3Pureza:98.61%Cor e Forma:White SolidPeso molecular:166.17(-)-Isopulegol
CAS:<p>Isopulegol has antioxidant, and neuroactive properties. It also has gastroprotective effects induced by isopulegol appear to be mediated, at least in part, by endogenous prostaglandins, K+ATP channel opening and antioxidant proprieties related to GSH increased.</p>Fórmula:C10H18OPureza:99.89%Cor e Forma:LiquidPeso molecular:154.25EGFR-IN-7
CAS:<p>EGFR-IN-7 (TQB3804) is a selective and potent EGFR kinase inhibitor.</p>Fórmula:C32H41BrN9O2PPureza:95.32% - 99.64%Cor e Forma:SolidPeso molecular:694.62'-Hydroxy-4'-methylacetophenone
CAS:<p>2'-Hydroxy-4'-methylacetophenone, a phenolic compound isolated from Angelicae koreana roots possesses acaricidal property. 2'-Hydroxy-4'-methylacetophenone has acaricidal activity, it could be used in the preparation of 4'-methyl-2'-[(p-tolylsulfonyl) oxy] acetophenone.</p>Fórmula:C9H10O2Pureza:99.88%Cor e Forma:Black LiquidPeso molecular:150.17Anisylacetone
CAS:<p>Anisylacetone (Anisylacetone) is an effective lure for the male melon fly.</p>Fórmula:C11H14O2Pureza:99.74%Cor e Forma:LiquidPeso molecular:178.23α-Terpineol
CAS:<p>Terpineol possesses antifungal activity against Trichophyton mentagrophytes, it also exhibits strong antimicrobial activity against periodontopathic and cariogenic bacteria. α-Terpineol (Terpineol) shows anticonvulsant, and anti-inflammatory activities, it inhibits the gene expression of the IL-6 receptor.</p>Fórmula:C10H18OPureza:97.55%Cor e Forma:Colorless LiquidPeso molecular:154.253-Acetylcoumarin
CAS:<p>3-Acetylcoumarin as a practical ligand for copper-catalyzed CN coupling reactions at room temperature. It has neuroprotective and acaricidal properties.</p>Fórmula:C11H8O3Pureza:99.41%Cor e Forma:Yellow Crystalline PowderPeso molecular:188.18(5R)-Platyphyllone
CAS:<p>(5R)-Platyphyllone has a wide range of applications in life science related research.</p>Fórmula:C19H22O4Pureza:98%Cor e Forma:SolidPeso molecular:314.381Antibacterial agent 83
CAS:<p>Compound 17h is a potent antibacterial against VRE and MRSA, reduces MRSA biofilms, and is stable in liver microsomes.</p>Fórmula:C11H5Cl2N3O2Cor e Forma:SolidPeso molecular:282.08Dabigatran Acyl-β-D-Glucuronide
CAS:<p>Dabigatran acyl-β-D-glucuronide is a major active metabolite of the thrombin inhibitor dabigatran .</p>Fórmula:C31H33N7O9Cor e Forma:SolidPeso molecular:647.645Gd-NMC-3
CAS:<p>Gd-NMC-3, a bimodal imaging probe, exhibits high resolution and sensitivity for tumor imaging with favorable biocompatibility, demonstrating significant</p>Fórmula:C77H114Gd2N14O24S2Cor e Forma:SolidPeso molecular:1998.449-Azido-Neu5DAz
CAS:<p>9-Azido-Neu5DAz is a non-natural bifunctional carbohydrates as imaging agent.</p>Fórmula:C14H22N6O8Pureza:98%Cor e Forma:SolidPeso molecular:402.36Ref: TM-T19168
Produto descontinuadoThalidomide-NH-PEG4-Ms
CAS:<p>Thalidomide-NH-PEG4-Ms: cereblon ligand + linker, for PROTAC BCL-XL degrader XZ739.</p>Fórmula:C22H29N3O10SCor e Forma:SolidPeso molecular:527.55Leishman's stain
CAS:Leishman's stain is a vital dye for staining peripheral blood and bone marrow smears, which appear pale bluish-grey to deep blue when viewed under an oil-Cor e Forma:SolidAnticancer agent 11
CAS:<p>Anticancer agent 11 suppresses angiogenesis and induces DNA cross-links for broad-spectrum efficacy.</p>Fórmula:C20H21N3O2Cor e Forma:SolidPeso molecular:335.40Cgp 11130
CAS:<p>Cgp 11130 is a bio-active chemical.</p>Fórmula:C10H12FNO2Cor e Forma:SolidPeso molecular:197.21BPH-629
CAS:<p>BPH-629 is a bioactive chemical.</p>Fórmula:C20H18O8P2Cor e Forma:SolidPeso molecular:448.3Zanamivir-Cholesterol Conjugate
CAS:<p>Zanamivir-cholesterol conjugate is an extended-duration neuraminidase inhibitor highly effective against drug-resistant influenza strains.</p>Fórmula:C61H104N8O15Cor e Forma:SolidPeso molecular:1189.5442',3'-cGAMP-C2-SH
CAS:<p>2', 3'-cGAMP-C2-SH is a ADC cytotoxin.</p>Fórmula:C22H28N10O12P2SCor e Forma:SolidPeso molecular:718.53SIAIS117
CAS:<p>SIAIS117: A Brigatinib-VHL-1 ALK PROTAC; degrades ALK G1202R, inhibits SR/H2228 cells, may fight small cell lung cancer.</p>Fórmula:C57H76ClN10O7PSCor e Forma:SolidPeso molecular:1111.77Nutlin carboxylic acid
CAS:<p>Nutlin carboxylic acid is a Nutlin 3-based MDM2 ligand; used with a linker to create PROTACs.</p>Fórmula:C32H32Cl2N4O6Pureza:98%Cor e Forma:SolidPeso molecular:639.53Ref: TM-T17874
Produto descontinuadoERK1/2 inhibitor 4
CAS:<p>ERK1/2 inhibitor 5 targets MAPK pathway, potentially aiding cancer and inflammation research.</p>Fórmula:C28H31ClFN5O5SCor e Forma:SolidPeso molecular:604.09m-PEG11-Tos
<p>m-PEG11-Tos is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs[1].</p>Fórmula:C28H50O13SPureza:98%Cor e Forma:SolidPeso molecular:626.75MCA17-1
CAS:<p>MCA17-1 exhibits superior bioactivity compared to the positive control, obeticholic acid (OCA), in the treatment of liver fibrosis.</p>Fórmula:C14H15NO5Cor e Forma:SolidPeso molecular:277.276Questiomycin A derivatives 14
<p>Questiomycin A derivatives 14 is a Questiomycin A derivative.</p>Fórmula:C18H18N2O3Pureza:99.73%Cor e Forma:SoildPeso molecular:310.351-(2,3-Dichlorphenyl)-piperazine
CAS:<p>1-(2,3-Dichlorphenyl)-piperazine (DCPP) is a potent DHCR7 inhibitor. DHCR7 is the last enzyme in cholesterol biosynthesis.</p>Fórmula:C10H12Cl2N2Pureza:98%Cor e Forma:Brown OilPeso molecular:231.12Cap-dependent endonuclease-IN-15
CAS:<p>Cap-dependent endonuclease-IN-15: potent CEN inhibitor, halts influenza virus replication, aids viral research.</p>Fórmula:C27H23F2N3O7SeCor e Forma:SolidPeso molecular:618.44DFHBI-2T
CAS:<p>DFHBI-2T, a membrane-permeable fluorescence probe activated by RNA aptamers (ex/em=500 nm/523 nm), is utilized for imaging RNA within live cells.</p>Fórmula:C12H7F5N2O2Cor e Forma:SolidPeso molecular:306.192SKF 89748
CAS:SKF 89748 is an agonists of alpha 1-adrenoceptor.Fórmula:C12H17NOSPureza:98%Cor e Forma:SolidPeso molecular:223.33PEG2-bis(phosphonic acid)
CAS:<p>PEG2-bis(phosphonic acid) is a PEG Linker.</p>Fórmula:C6H16O8P2Cor e Forma:SolidPeso molecular:278.13TAK-683
CAS:TAK-683: a full KISS1R agonist, IC50=170 pM; a nonapeptide metastin analog with human EC50=0.96 nM, rat EC50=1.6 nM.Fórmula:C64H83N17O13Pureza:98%Cor e Forma:SolidPeso molecular:1298.45Contezolid acefosamil
CAS:<p>Contezolid acefosamil (MRX-4), oral prodrug of Contezolid (MRX-I), treats multidrug-resistant Gram-positive bacteria, including MRSA.</p>Fórmula:C20H18F3N4O8PCor e Forma:SolidPeso molecular:530.353Taragarestrant meglumine
CAS:<p>Taragarestrant (D-0502) is an oral SERD with potent activity against ER+ breast cancer.</p>Fórmula:C32H42Cl2FN3O7Cor e Forma:SolidPeso molecular:670.60ER degrader 2
CAS:<p>ER degrader 2: Potent estrogen receptor disruptor; key for cancer research.</p>Fórmula:C34H42F3N5O3Cor e Forma:SolidPeso molecular:625.72MCAAD-3
CAS:<p>MCAAD-3, a near-infrared Aβ imaging probe, exhibits blood-brain barrier permeability and strong affinity for Aβ polymers (Ki >106 nM).</p>Fórmula:C17H18N2O2Cor e Forma:SolidPeso molecular:282.34Elamipretide TFA
CAS:<p>Elamipretide TFA (RX-31 TFA) is a cardiolipin peroxidase inhibitor and mitochondria-targeting peptide[1].</p>Fórmula:C34H50F3N9O7Pureza:98%Cor e Forma:SolidPeso molecular:753.81Ref: TM-TP1096
Produto descontinuadogp91ds-tat
<p>gp91ds-tat is a useful organic compound for research related to life sciences and the catalog number is T35393.</p>Pureza:98%Cor e Forma:SolidZ-(L-Arg)-AMC (hydrochloride)
CAS:<p>Z-(L-Arg)-AMC releases fluorescent AMC upon cleavage by trypsin, cathepsins B & H, used to measure their activity (Ex/Em: 340-360/440-460 nm).</p>Fórmula:C24H28ClN5O5Cor e Forma:SolidPeso molecular:501.97(3,4-Dihydroxy-5-methoxybenzoyl)taraxerol
CAS:<p>(3,4-Dihydroxy-5-methoxybenzoyl)taraxerol is a natural products from plants</p>Fórmula:C38H56O5Pureza:98%Cor e Forma:SolidPeso molecular:592.85Ref: TM-TN2397
Produto descontinuadoPD-1/PD-L1-IN 5 TFA
CAS:<p>PD-1/PD-L1-IN 5 is an inhibitor of PD-1/PD-L1 protein/protein interaction (IC50 of ≤100 nM).</p>Fórmula:C22H18N4O3S·xC2HF3O2Pureza:98%Cor e Forma:SolidPhototherapeutic agent-1
CAS:<p>Phototherapeutic agent-1: a light-activated, ROS-generating cancer cell killer with aggregation-induced emission.</p>Fórmula:C39H33F6N2O2PS3Cor e Forma:SolidPeso molecular:802.853'-O-Angeloylhamaudol
<p>3'-O-Angeloylhamaudol is a useful organic compound for research related to life sciences and the catalog number is T124112.</p>Fórmula:C20H22O6Cor e Forma:SolidPeso molecular:358.39PROTAC eEF2K degrader-1
CAS:<p>PROTAC eEF2K degrader-1 (11l) targets eEF2K, induces apoptosis in MDA-MB-231 cells, and degrades eEF2K.</p>Fórmula:C31H33N9O11Cor e Forma:SolidPeso molecular:707.65Fungicide5
CAS:<p>Fungicide5 is a fungicide candidate targeting succinate dehydrogenase ( K i = 0.095 μM).</p>Fórmula:C20H13F8N3O2Cor e Forma:SolidPeso molecular:479.33Sel-green
CAS:<p>Sel-green: a probe for quantifying Sec in thioredoxin reductase and imaging Sec in live HepG2 cells.</p>Fórmula:C19H18N4O8SCor e Forma:SolidPeso molecular:462.433-Hydroxyephedrine
CAS:3-Hydroxyephedrine is a bioactive chemical.Fórmula:C10H15NO2Cor e Forma:SolidPeso molecular:181.232-(7-Hydroxy-2-oxo-2H-chromen-4-yl)acetic acid
CAS:2-(7-Hydroxy-2-oxo-2H-chromen-4-yl)acetic acid is a useful organic compound for research related to life sciences.Fórmula:C11H8O5Cor e Forma:SolidPeso molecular:220.1782BKM1740
CAS:BKM1740 induced apoptosis in prostate cancer (PCa) cells by repressing survivin at both the mRNA and protein levels in vitro.Fórmula:C39H46Cl2F5N3O9P2Pureza:98%Cor e Forma:SolidPeso molecular:928.65Mca-Ala-Pro-Lys(Dnp)-OH
CAS:<p>Mca-Ala-Pro-Lys(Dnp)-OH, a specific quenched fluorogenic substrate for ACE2, enables the detection of ACE2 activity in various tissues including urinary, heart</p>Fórmula:C32H36N6O12Cor e Forma:SolidPeso molecular:696.67Stephalonine L
CAS:<p>Stephalonine L is a natural product for research related to life sciences. The catalog number is TN6290 and the CAS number is 2379277-60-6.</p>Fórmula:C30H35NO10Pureza:98%Cor e Forma:SolidPeso molecular:569.6Ref: TM-TN6290
Produto descontinuado1,2-Diaminoanthraquinone
CAS:<p>1,2-Diaminoanthraquinone serves as a sensitive, specific, and nontoxic fluorescent probe for nitric oxide (NO), facilitating the detection of NO production in</p>Fórmula:C14H10N2O2Cor e Forma:SolidPeso molecular:238.24BPH-252
CAS:<p>BPH-252 is a bioactive chemical.</p>Fórmula:C10H24O7P2Cor e Forma:SolidPeso molecular:318.24H-L-Photo-lysine hydrochloride
<p>H-L-Photo-lysine HCl is a diazirine lysine for site-specific protein incorporation and in vivo cross-linking.</p>Fórmula:C11H21ClN4O4Pureza:98%Cor e Forma:SolidPeso molecular:308.76Spirolingzhine D
CAS:<p>Spirolingzhine D is a useful organic compound for research related to life sciences. The catalog number is T125689 and the CAS number is 1612239-54-9.</p>Fórmula:C16H16O6Cor e Forma:SolidPeso molecular:304.298Xibornol
CAS:Xibornol (Nanbacine) 具有广谱的抗菌和抗病毒活性，可用于研究革兰氏阳性菌感染和人呼吸道合胞病毒与人冠状病毒229E感染。Fórmula:C18H26OCor e Forma:SolidPeso molecular:258.4Deutetrabenazine metabolite M4
CAS:Deutetrabenazine's metabolite M4 depletes monoamines by reversibly inhibiting VMAT2, affecting nerve terminals.Fórmula:C19H21D6NO4Pureza:98%Cor e Forma:SolidPeso molecular:339.46Glabralide A
CAS:<p>Glabralide A is a natural product from plants</p>Fórmula:C27H32O5Pureza:98%Cor e Forma:SolidPeso molecular:436.54Ref: TM-TN2407
Produto descontinuadoTL4830031
CAS:<p>TL4830031 (8i), quinolone derivative, Axl inhibitor, IC50: 26 nM, blocks Axl phosphorylation, cell invasion & migration; for cancer research.</p>Fórmula:C35H33F2N5O6Cor e Forma:SolidPeso molecular:657.66Aflatoxin M1
CAS:<p>Aflatoxin M1, a toxic metabolite of Aflatoxin B1, is produced by Aspergillus fungi, with a toxicity order: B1 > M1 > G1 > B2 > M2 > G2.</p>Fórmula:C17H12O7Cor e Forma:SolidPeso molecular:328.276LY 280748
CAS:LY 280748 is a bio-active chemical.Fórmula:C23H29N4NaO2Cor e Forma:SolidPeso molecular:416.49rel-(11S,31S)-16,36,37,54-Tetramethoxy-12,32-dimethyl-11,12,13,14,31,32,33,34-octahydro-2,6-dioxa-1(7,1),3(8,1)-diisoquinolina-5(1,3),7(1,4)-dibenzenacyclooctaphane
<p>rel-(11S,31S)-16,36,37,54-Tetramethoxy-12,32-dimethyl-11,12,13,14,31,32,33,34-octahydro-2,6-dioxa-1(7,1),3(8,1)-diisoquinolina-5(1,3),7(1,4)-dibenzenacyclooctaphane is a useful organic compound for research related to life sciences and the catalog number is T64548.</p>Pureza:98%GEM-5
CAS:<p>GEM-5, a gemcitabine conjugate with HIF-1α inhibitor YC-1 (IC50=30 nM), down-regulates HIF-1α, up-regulates p53, and induces A2780 cell apoptosis.</p>Fórmula:C32H29F2N5O8Cor e Forma:SolidPeso molecular:649.60Cap-dependent endonuclease-IN-22
CAS:<p>Cap-dependent endonuclease-IN-22 is a powerful inhibitor of cap-dependent endonuclease (CEN) [1].</p>Fórmula:C37H37ClF2N6O7S2Cor e Forma:SolidPeso molecular:815.31FGFR-IN-1
CAS:<p>FGFR-IN-1 targets FGFR1-3 with IC50 <100 nM. (US20130338134A1, ex 219)</p>Fórmula:C26H24F2N4O6SCor e Forma:SolidPeso molecular:558.55Coumarin 314
CAS:<p>Coumarin 314 is a useful organic compound for research related to life sciences. The catalog number is T66908 and the CAS number is 55804-66-5.</p>Fórmula:C18H19NO4Cor e Forma:SolidPeso molecular:313.353
