
Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.524 produtos)
- Apoptose(5.793 produtos)
- Ciclo celular/Ponto de verificação(4.452 produtos)
- Cromatina/Epigenética(2.242 produtos)
- Sinalização Citoesquelética(1.382 produtos)
- Dano de DNA/Reparo de DNA(2.826 produtos)
- Endocrinologia/Hormónios(3.507 produtos)
- Enzima(3.640 produtos)
- GPCR/Proteína-G(8.333 produtos)
- Imunologia e Inflamação(3.527 produtos)
- Vírus da Influenza(296 produtos)
- Sinalização JAK/STAT(404 produtos)
- Sinalização MAPK(1.203 produtos)
- Transportador de Membranas/Canal Iónico(2.792 produtos)
- Metabolismo(9.449 produtos)
- Microbiologia/Virologia(6.981 produtos)
- Neurociência(9.926 produtos)
- Outros inibidores(37.921 produtos)
- Oxidação-Redução(41 produtos)
- Sinalização PI3K/Akt/mTOR(1.400 produtos)
- Proteases/Proteassoma(1.597 produtos)
- Células - tronco e Derivados(830 produtos)
- Tirosina Quinase/Adaptador(2.015 produtos)
- Ubiquitinação(1.650 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66639 produtos de "Inibidores"
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Alizarin
CAS:Alizarin, red dye from madder roots, inhibits CYP1A1 (IC50=6.2μM), CYP1A2 (IC50=10μM), CYP1B1 (IC50=2.7μM).Fórmula:C14H8O4Pureza:98.62%Cor e Forma:Orange-Red Crystals Or PowderPeso molecular:240.21Meglumine
CAS:<p>Meglumine (Meglumin), a derivative of sorbitol, is used in conjunction with iodinated organic compounds as contrast medium.</p>Fórmula:C7H17NO5Pureza:99.98%Cor e Forma:DrypowderPeso molecular:195.211-Methylxanthine
CAS:1-Methylxanthine: caffeine derivative, human urinary metabolite, increases tumor cell radiosensitivity.Fórmula:C6H6N4O2Pureza:99.11%Cor e Forma:SolidPeso molecular:166.14Letrozole
CAS:<p>Letrozole (CGS 20267) is an Aromatase Inhibitor. The mechanism of action of letrozole is as an Aromatase Inhibitor.</p>Fórmula:C17H11N5Pureza:98.67% - 99.84%Cor e Forma:White To Off-Whitecrystalline PowderPeso molecular:285.3Zolmitriptan
CAS:<p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>Fórmula:C16H21N3O2Pureza:99.69% - 99.91%Cor e Forma:White Or Kind Of White PowderPeso molecular:287.36Orlistat
CAS:<p>Orlistat (Tetrahydrolipstatin) is a lipase inhibitor and a FASN inhibitor. Orlistat has been shown to promote weight loss. Cost effective and quality assured.</p>Fórmula:C29H53NO5Pureza:99.58% - >99.99%Cor e Forma:White Crystalline PowderPeso molecular:495.73Icopezil
CAS:<p>Icopezil: small molecule, AChE inhibitor, treats neurological disorders, used in Alzheimer's research.</p>Fórmula:C23H25N3O2Pureza:99.35%Cor e Forma:SolidPeso molecular:375.46L-Ascorbic acid
CAS:<p>L-Ascorbic acid (Vitamin C) is a natural product that is a potent reducing agent and antioxidant.</p>Fórmula:C6H8O6Pureza:99.85% - 99.89%Cor e Forma:Crystals (Usually Plates Sometimes Needles Mon°Clinic System) Taste Almost Odorless (Ntp 1992)Peso molecular:176.12WAY-640509
CAS:<p>WAY-640509 is a glucocerebrosidase inhibitor.</p>Fórmula:C25H23N5O4SPureza:99.36%Cor e Forma:SolidPeso molecular:489.55Risperidone
CAS:<p>Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.</p>Fórmula:C23H27FN4O2Pureza:99.73%Cor e Forma:Crystalline SolidPeso molecular:410.48Mucic Acid
CAS:<p>Mucic Acid (Tetrahydroxyadipic acid) is an aldaric acid obtained by nitric acid oxidation of galactose or galactose-containing compounds.</p>Fórmula:C6H10O8Pureza:99.31%Cor e Forma:Crystalline Powder SolidPeso molecular:210.14pNNP
CAS:<p>pNNP is a substrate for PP2C assays and inhibits β-carbonic anhydrase, α-carbonate dehydrogenase, and H. pylori.</p>Fórmula:C6H6NO6PPureza:99.73%Cor e Forma:SolidPeso molecular:219.09Docusate sodium
CAS:<p>Docusate sodium (Aerosol OT) is an orally available, over-the-counter laxative and stool softener used to treat or prevent constipation.</p>Fórmula:C20H37NaO7SPureza:99.34%Cor e Forma:White Wax-Like Solid With Water (Uscg 1999)Peso molecular:444.56Fendiline hydrochloride
CAS:<p>Fendiline hydrochloride (Fendiline HCl) is a non-selective blocker of calcium channel.</p>Fórmula:C23H26ClNPureza:98.76% - 99.75%Cor e Forma:SolidPeso molecular:351.91ZT 52656A hydrochloride
CAS:<p>ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.</p>Fórmula:C19H26ClF3N2OPureza:98.78%Cor e Forma:SolidPeso molecular:390.87Itepekimab
CAS:<p>Itepekimab (REGN-3500), a potent IL-33 monoclonal antibody, may help study asthma by reducing airway inflammation.</p>Pureza:92.8%Cor e Forma:LiquidPeso molecular:144.63kDaMK-0533
CAS:<p>MK-0533 is a novel PPARγ partial agonist for the prevention of vascular endothelial dysfunction (VED) and VED-related cardiovascular disease.</p>Fórmula:C28H24F3NO6Pureza:99.03%Cor e Forma:SoildPeso molecular:527.49Methylsyringol
CAS:<p>Methylsyringol is a natural product from Pinus yunnanensis.</p>Fórmula:C9H12O3Pureza:99.47%Cor e Forma:SolidPeso molecular:168.19Pazopanib
CAS:<p>Pazopanib (GW786034) is an inhibitor of protein tyrosine kinases that inhibits VEGFR1/2/3. Pazopanib has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C21H23N7O2SPureza:98.78% - 99.85%Cor e Forma:White PowderPeso molecular:437.52MK-0812 Succinate
CAS:<p>MK-0812 Succinate is an effective and selective CCR2 antagonist.</p>Fórmula:C28H40F3N3O7Pureza:98.62% - 99.93%Cor e Forma:SolidPeso molecular:587.63YQ128
CAS:<p>YQ128 is a potent and selective inhibitor of second-generation NLRP3 (NOD-like receptor P3) inflammasome(IC50 of 0.30 µM), with anti-inflammatory activity.</p>Fórmula:C27H29ClN2O4S2Pureza:99.89%Cor e Forma:SolidPeso molecular:545.11Ciliobrevin D
CAS:<p>Ciliobrevin D is a AAA+ ATPase motor cytoplasmic dynein inhibitor.</p>Fórmula:C17H8Cl3N3O2Pureza:98.09%Cor e Forma:SolidPeso molecular:392.62Bendamustine hydrochloride
CAS:<p>Bendamustine hydrochloride (EP-3101) (IC50 of 50 μM) is an alkylating agent associated with DNA damage.</p>Fórmula:C16H21Cl2N3O2·HClPureza:97.71%Cor e Forma:SolidPeso molecular:394.72Quinestrol
CAS:<p>Quinestrol (Ethinylestradiol 3-cyclopentyl ether) is a synthetic estrogen, applied in hormone replacement therapy, and occasionally to use in cancer and</p>Fórmula:C25H32O2Pureza:99.36% - 99.72%Cor e Forma:SolidPeso molecular:364.525-hydroxytryptophan
CAS:<p>5-hydroxytryptophan (NSC-92523) is the immediate precursor in the biosynthesis of SEROTONIN from tryptophan. It is used as an antiepileptic and antidepressant.</p>Fórmula:C11H12N2O3Pureza:99.52%Cor e Forma:Minute Rods Or Needles From Ethanol White SolidPeso molecular:220.22Amiselimod hydrochloride
CAS:<p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>Fórmula:C19H31ClF3NO3Pureza:99.55%Cor e Forma:SolidPeso molecular:413.9CDK4/6-IN-2
CAS:<p>CDK4/6-IN-2 是一种CDK4和CDK6抑制剂,IC50分别为 2.7 和 16 nM。</p>Fórmula:C27H32F2N8Pureza:99.47%Cor e Forma:SolidPeso molecular:506.59Glipizide
CAS:<p>Glipizide (CP 28720) is a short-acting, second-generation sulfonylurea with hypoglycemic activity.</p>Fórmula:C21H27N5O4SPureza:99.67% - 99.75%Cor e Forma:SolidPeso molecular:445.54Ac-FLTD-CMK
CAS:<p>Ac-FLTD-CMK, an abscisicin D derivative, selectively inhibits inflammatory caspases-1, -4, and -11 (IC50: 46.7 nM, 1.49 μM, 329 nM) but not caspase-3.</p>Fórmula:C26H37ClN4O8Pureza:95.17%Cor e Forma:SolidPeso molecular:569.05Mizoribine
CAS:<p>Mizoribine (NSC-289637) belongs to the family of 1-Ribosyl-imidazolecarboxamides. Mizoribine has been investigated for the treatment of Rheumatoid Arthritis.</p>Fórmula:C9H13N3O6Pureza:98.38% - 99.95%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:259.22Linaclotide
CAS:<p>Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.</p>Fórmula:C59H79N15O21S6Pureza:97.93% - 98.71%Cor e Forma:SolidPeso molecular:1526.74L-Ornithine
CAS:<p>L-Ornithine ((S)-2, 5-diaminopentanoic acid) is a non-protein amino acid. in the urea cycle to remove excess nitrogen from the body. High-Quality, Low-Cost!</p>Fórmula:C5H12N2O2Pureza:99.73% - 99.91%Cor e Forma:SolidPeso molecular:132.16Pulrodemstat benzenesulfonate
CAS:<p>Pulrodemstat benzenesulfonate (CC-90011 benzenesulfonate) is a potent and orally inhibitor of lysine specific demethylase-1 (LSD1) with anticancer effect.</p>Fórmula:C30H29F2N5O5SPureza:97.67%Cor e Forma:SolidPeso molecular:609.64Elacestrant
CAS:<p>Elacestrant (RAD1901) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant is an orally available selective estrogen receptor degrader .</p>Fórmula:C30H38N2O2Pureza:98.31%Cor e Forma:SolidPeso molecular:458.63CDKI-73
CAS:<p>CDKI-73: strong CDK9 blocker, Ki 4 nM, kills CLL cells selectively, aids cisplatin.</p>Fórmula:C15H15FN6O2S2Pureza:98.11%Cor e Forma:SolidPeso molecular:394.45MOG peptide (35-55), mouse, rat acetate
<p>Mouse, rat MOG peptide (35-55) acetate, part of myelin glycoprotein, for immune disease research.</p>Pureza:97.88%Cor e Forma:SoildDeoxycholic acid
CAS:<p>Deoxycholic acid (Cholanoic Acid) is a bile acid formed by bacterial action from cholate.</p>Fórmula:C24H40O4Pureza:99.91% - 99.91%Cor e Forma:Crystals From Alc SolidPeso molecular:392.57PIT
CAS:<p>PIT (2,2'-Pyridylisatogen tosylate) is a specific and non-competitive antagonist of the Purinergic receptor P2Y1 with an IC50 of 0.14 μM for human P2Y1.</p>Fórmula:C20H16N2O5SPureza:98.63%Cor e Forma:SolidPeso molecular:396.42CXCR7 antagonist-1
CAS:<p>CXCR7 antagonist-1 is a specific antagonist of the binding of the SDF-1 chemokine or I-TAC to the chemokine receptor CXCR7.</p>Fórmula:C21H19FN6OPureza:99.93%Cor e Forma:SolidPeso molecular:390.41Chloramphenicol
CAS:<p>Chloramphenicol (Chloromycetin) is a broad-spectrum antibiotic that inhibits the biosynthesis of bacterial proteins. Cost-effective and quality-assured.</p>Fórmula:C11H12Cl2N2O5Pureza:99.6% - 99.84%Cor e Forma:Needles Or Elongated Plates From Water Or Ethylene Dichloride SolidPeso molecular:323.13Apidaecin IB acetate
<p>Apidaecin IB acetate: insect antibacterial peptide, minimum 8 μM effective against E. coli strains.</p>Fórmula:C97H154N32O25Pureza:99.91%Cor e Forma:SolidPeso molecular:2168.46SNDX-5613
CAS:<p>Revumenib (SNDX-5613) is a potent and selective oral inhibitor of menin-KMT2A interaction.Cost-effective and quality-assured.</p>Fórmula:C32H47FN6O4SPureza:99.12% - 99.74%Cor e Forma:SolidPeso molecular:630.82Zonisamide
CAS:<p>Zonisamide (AD 810), a sulfonamide anticonvulsant, is approved for use as an adjunctive treatment in adults with partial-onset seizures.</p>Fórmula:C8H8N2O3SPureza:99.05% - 99.9%Cor e Forma:Off-White PowderPeso molecular:212.23Maltitol
CAS:<p>Maltitol (4-O-α-glucopyranosyl-D-sorbitol) is a sugar alcohol (polyol) used as a sugar substitute.</p>Fórmula:C12H24O11Pureza:99.72% - 99.82%Cor e Forma:White Powder LiquidPeso molecular:344.31Pseudobaptigenin
CAS:<p>Pseudobaptigenin (Psi-baptigenin) is an isoflavone, a flavonoid lipid molecule that is a natural product found in Pterocarpus marsupium, Dalbergia spruceana.</p>Fórmula:C16H10O5Pureza:98.61%Cor e Forma:SolidPeso molecular:282.25Florfenicol
CAS:<p>Florfenicol treats BRD in cattle, effective against Mannheimia, Pasteurella, Haemophilus, Fusobacterium, and Bacteroides.</p>Fórmula:C12H14Cl2FNO4SPureza:98.93%Cor e Forma:SolidPeso molecular:358.21Oxytetracycline
CAS:<p>Oxytetracycline (Terramycin) is a TETRACYCLINE analog isolated from the actinomycete STREPTOMYCES rimosus and used in a wide variety of clinical conditions.</p>Fórmula:C22H24N2O9Pureza:99.11%Cor e Forma:Light-Yellow Crystals Or Needles From Aqueous Meoh Physical Description Odorless Fluffy Yellow Solid Or Yellow Powder Bitter Taste (Ntp 1992)Peso molecular:460.43PF-3450074
CAS:<p>PF-3450074 (PF-74) is a specific HIV-1 inhibitor, blocking viral replication and uncoating at submicromolar EC50=8-640 nM.</p>Fórmula:C27H27N3O2Pureza:99.92%Cor e Forma:SolidPeso molecular:425.52Inobrodib
CAS:<p>Inobrodib (CBP-IN-1) is a potent inhibitor of p300/CBP bromodomain.</p>Fórmula:C30H32F2N4O3Pureza:98.91% - 99.18%Cor e Forma:SolidPeso molecular:534.6DiI
CAS:<p>DiI (DiIC18(3)) is a lipophilic membrane dye commonly used as a long-term tracer for neurons and other cells (λex/em=549/565 nm). Cost-effective and quality-assured.</p>Fórmula:C59H97ClN2O4Pureza:99.19% - 99.95%Cor e Forma:SolidPeso molecular:933.87
