
Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.523 produtos)
- Apoptose(5.792 produtos)
- Ciclo celular/Ponto de verificação(4.449 produtos)
- Cromatina/Epigenética(2.238 produtos)
- Sinalização Citoesquelética(1.383 produtos)
- Dano de DNA/Reparo de DNA(2.825 produtos)
- Endocrinologia/Hormónios(3.507 produtos)
- Enzima(3.640 produtos)
- GPCR/Proteína-G(8.333 produtos)
- Imunologia e Inflamação(3.526 produtos)
- Vírus da Influenza(296 produtos)
- Sinalização JAK/STAT(404 produtos)
- Sinalização MAPK(1.202 produtos)
- Transportador de Membranas/Canal Iónico(2.790 produtos)
- Metabolismo(9.448 produtos)
- Microbiologia/Virologia(6.981 produtos)
- Neurociência(9.926 produtos)
- Outros inibidores(37.926 produtos)
- Oxidação-Redução(41 produtos)
- Sinalização PI3K/Akt/mTOR(1.400 produtos)
- Proteases/Proteassoma(1.597 produtos)
- Células - tronco e Derivados(831 produtos)
- Tirosina Quinase/Adaptador(2.016 produtos)
- Ubiquitinação(1.650 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66641 produtos de "Inibidores"
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TCN 201
CAS:<p>TCN 201 is a selective antagonist of NMDA receptors containing the NR2A subunit.</p>Fórmula:C21H17ClFN3O4SPureza:98.5%Cor e Forma:SolidPeso molecular:461.89Mildronate
CAS:<p>Mildronate (Meldonium) is an inhibitor of biosynthesis of L-carnitine by gamma-butyrobetaine (GBB) hydroxylase and as a competitive inhibitor of renal carnitine</p>Fórmula:C6H14N2O2Pureza:99.94%Cor e Forma:White Crystalline PowderPeso molecular:146.19Gypenoside XLVI
CAS:<p>Gypenoside XLVI shows strong cytotoxic activity against A549 cells, with the IC50 values of 52.63±8.31 ug/ml.</p>Fórmula:C48H82O19Pureza:98.59%Cor e Forma:SolidPeso molecular:963.15JNJ-5207852 dihydrochloride
CAS:<p>JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor</p>Fórmula:C20H34Cl2N2OPureza:99.51%Cor e Forma:SolidPeso molecular:389.4Emapunil
CAS:<p>Emapunil (XBD-173) is an anxiolytic and selective TSPO agonist, targeting peripheral benzodiazepine receptors.</p>Fórmula:C23H23N5O2Pureza:98% - 99.9%Cor e Forma:SolidPeso molecular:401.46Sofosbuvir
CAS:<p>Sofosbuvir (GS 7977) is a uridine monophosphate analog inhibitor of hepatitis C virus (HCV) polymerase NS5B that is used as an antiviral agent in the treatment</p>Fórmula:C22H29FN3O9PPureza:99.77% - 99.82%Cor e Forma:SolidPeso molecular:529.45Brigatinib
CAS:<p>Brigatinib (AP-26113) is a highly potent and selective ALK inhibitor.</p>Fórmula:C29H39ClN7O2PPureza:97.18% - >99.99%Cor e Forma:SolidPeso molecular:584.09Indirubin
CAS:<p>Indirubin (Couroupitine B) is a potent cyclin-dependent kinases and GSK-3β inhibitor with IC50 of about 5 uM and 0.6 uM.</p>Fórmula:C16H10N2O2Pureza:97.21% - 99.74%Cor e Forma:Reddish-Violet PowderPeso molecular:262.26Coretinphencone
CAS:<p>Coretinphencone is a natural product that is isolated from the buds of Coreopsis tinctoria Nutt.</p>Fórmula:C14H18O9Pureza:99.95%Cor e Forma:SolidPeso molecular:330.29Lauryl benzalkonium chloride
CAS:<p>Lauryl benzalkonium chloride (Benzododecinium chloride) is a quaternary ammonium compound.Benzododecinium chloride is an irritant for eye.</p>Fórmula:C21H38ClNPureza:99.88%Cor e Forma:LiquidPeso molecular:339.99Hemokinin 1 (mouse) acetate(208041-90-1 free base)
<p>Mouse Hemokinin-1 acetate: NK1 receptor agonist, Ki=0.175 nM; NK2 Ki=560 nM.</p>Fórmula:C63H104N22O17SPureza:98.33%Cor e Forma:SolidPeso molecular:1473.72N2-methylguanine
CAS:<p>N2-methylguanine (N2-methylguanine) is an endogenous methylated nucleoside found in human fluids and a modified nucleoside.</p>Fórmula:C6H7N5OPureza:99.86%Cor e Forma:SolidPeso molecular:165.15Ginkgolic Acid
CAS:<p>Ginkgolic Acid (Romanicardic acid) C15:1 represses curli genes and prophage genes in EHEC.</p>Fórmula:C22H34O3Pureza:98.69% - 99.9%Cor e Forma:White PowderPeso molecular:346.5Semagacestat
CAS:<p>Semagacestat (LY450139) (LY450139) is a γ-secretase blocker for Aβ42/Aβ40/Aβ38 (IC50: 10.9/12.1/12.0 nM) and also inhibits Notch signaling (IC50: 14.1 nM).</p>Fórmula:C19H27N3O4Pureza:97.1% - 99.9%Cor e Forma:SolidPeso molecular:361.44Deltamethrin
CAS:<p>Deltamethrin, a pyrethroid insecticide, causes reversible hind limb rigidity in rats and is used for crop protection and disease control.</p>Fórmula:C22H19Br2NO3Pureza:99.25% - 99.85%Cor e Forma:White To Off-White Crystals Or PowderPeso molecular:505.20Tyrphostin A9
CAS:<p>Tyrphostin A9 (SF 6847) is an Agricultural acaricide, now superseded. Tyrphostin A9 is firstly designed as an EGFR inhibitor</p>Fórmula:C18H22N2OPureza:98.21% - 99.87%Cor e Forma:Yellow SolidPeso molecular:282.38Fmoc-N-Me-Leu-OH
CAS:<p>Fmoc-N-Me-Leu-OH is available for the peptide-coupling reaction.</p>Fórmula:C22H25NO4Pureza:99.51%Cor e Forma:White PowderPeso molecular:367.44Aloe-emodin-8-O-β-D-glucopyranoside
CAS:<p>Aloe-emodin-8-O-β-D-glucopyranoside (Aloe-emodin-8-O-beta-D-glucopyranoside) shows moderate bioactivity against human Protein Tyrosine Phosphatase 1B (hPTP1B)</p>Fórmula:C21H20O10Pureza:99.21% - 99.91%Cor e Forma:SolidPeso molecular:432.38Sonidegib
CAS:<p>Sonidegib (Erismodegib), a Smoothened (Smo) antagonist, inhibits Hedgehog (Hh) signaling with IC50 of 1.3 nM (mouse) and 2.5 nM (human), respectively.</p>Fórmula:C26H26F3N3O3Pureza:98% - 99.97%Cor e Forma:SolidPeso molecular:485.5GDC-0214
CAS:<p>GDC-0214 is an inhaled small-molecule JAK1 inhibitor and reduces fractional exhaled nitric oxide (Feno).</p>Fórmula:C28H28ClF2N9O3Pureza:99.75%Cor e Forma:SolidPeso molecular:612.03[11C]MP 10
CAS:<p>[11C]MP 10 (PF-2545920), a specific and effective PDE10A inhibitor (IC50=0.37 nM), is with more than1000-fold specificity activity over the PDE.</p>Fórmula:C25H20N4OPureza:99.5%Cor e Forma:SolidPeso molecular:391.45WIN 18446
CAS:<p>inhibitor of aldehyde dehydrogenase 1a2 (ALDH1a2)</p>Fórmula:C12H20Cl4N2O2Pureza:99.69%Cor e Forma:SolidPeso molecular:366.11H-PRO-HIS-CYS-LYS-ARG-MET-OH acetate
CAS:<p>H-PRO-HIS-CYS-LYS-ARG-MET-OH acetate acts as antioxidant by reacting with active oxygen species such as superoxide and hydroxyl radicals.</p>Fórmula:C33H58N12O9S2Pureza:98.74% - 99.4%Cor e Forma:SolidPeso molecular:831.02Mdivi-1
CAS:<p>Mdivi-1 (Mitochondrial division inhibitor 1) is a mitochondrial division inhibitor that inhibits DRP1 and Dynamin I (IC50=1-10 μM).</p>Fórmula:C15H10Cl2N2O2SPureza:96.57% - 99.23%Cor e Forma:SolidPeso molecular:353.22N-Methylsarcosine
CAS:<p>N-Methylsarcosine improves athletic performance, boosts immunity, treats autism/epilepsy, tracks COPD, and aids in ionic liquid development.</p>Fórmula:C4H9NO2Pureza:98.17%Cor e Forma:SolidPeso molecular:103.12cim0216
CAS:<p>CIM0216 is a synthetic TRPM3 activator whose potency and apparent affinity greatly exceeds that of the canonical TRPM3 agonist.</p>Fórmula:C21H21N3O2Pureza:99.87%Cor e Forma:SolidPeso molecular:347.41Toloxatone
CAS:<p>Toloxatone (MD 69276) is a reversible monoamine oxidase A (MAOA) inhibitor.</p>Fórmula:C11H13NO3Pureza:98.58%Cor e Forma:SolidPeso molecular:207.232-Amino-4'-fluorobenzophenone
CAS:2-Amino-4'-fluorobenzophenone, a benzophenone derivative, synthesizes p-fluorobenzoyl chloride and probes DNA/RNA.Fórmula:C13H10FNOPureza:99.52%Cor e Forma:SolidPeso molecular:215.22CAY10603
CAS:<p>CAY10603 (BML-281) is a potent and selective inhibitor of HDAC6.</p>Fórmula:C22H30N4O6Pureza:95.75% - 98.1%Cor e Forma:SolidPeso molecular:446.5Phenylethyl isothiocyanate
CAS:<p>Phenylethyl isothiocyanate (JC5411) is an HDAC inhibitor. It potentially for the treatment of benign prostatic hypertrophy.</p>Fórmula:C9H9NSPureza:98.14% - 99.78%Cor e Forma:Less To Pale Yellow Liquid Colourless To Pale Yellow LiquidPeso molecular:163.24N-Methylpyrrolidone
CAS:<p>N-Methylpyrrolidone, a cyclic amide, is a polar solvent for adhesives, paints, fuels, and drugs.</p>Fórmula:C5H9NOPureza:98.28%Cor e Forma:Clear Colorless LiquidPeso molecular:99.13Benzyldodecyldimethylammonium Chloride Dihydrate
CAS:<p>Benzyldodecyldimethylammonium chloride dihydrate: a QAC biocide against MRSA, MDR P. aeruginosa.</p>Fórmula:C21H42ClNO2Pureza:99.36%Cor e Forma:SolidPeso molecular:376.02HOMOPLANTAGININ
CAS:<p>Homoplantaginin is a flavonoid from a traditional Chinese medicine Salvia plebeia,it has a protective and therapeutic effect on hepatocyte injury and shows</p>Fórmula:C22H22O11Pureza:97.63% - 99.66%Cor e Forma:SolidPeso molecular:462.4PHA-767491 hydrochloride
CAS:<p>PHA-767491 (CAY-10572) is a potent Cdc7/CDK9 inhibitor (IC50: 10/34 nM), selective against GSK3-β, CDK1/2, CDK5, MK2, CHK2, PLK1.</p>Fórmula:C12H12ClN3OPureza:99.56% - 99.92%Cor e Forma:SolidPeso molecular:249.69Isoxaflutole
CAS:<p>Isoxaflutole (RP-201772) is a low toxic herbicide and has been marketed as a substitute for atrazine.</p>Fórmula:C15H12F3NO4SPureza:98.49%Cor e Forma:SolidPeso molecular:359.32Cyclopiazonic acid
CAS:<p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>Fórmula:C20H20N2O3Pureza:99.27% - 99.80%Cor e Forma:SolidPeso molecular:336.38Dihydrolapachenole
CAS:<p>Dihydrolapachenole (6-methoxy-2,2-dimethyl-3,4-dihydro-2H-benzo[h]chromene) can be isolated from T. chrysantha.</p>Fórmula:C16H18O2Pureza:99.75%Cor e Forma:SolidPeso molecular:242.31Zearalenone
CAS:<p>Zearalenone (F2 toxin) is a mycotoxin produced mainly by fungi belonging to the genus Fusarium in foods and feeds.</p>Fórmula:C18H22O5Pureza:98.39% - 99.11%Cor e Forma:This Chemical May Be Sensitive To Prolonged Exposure To Air Insoluble In Water Physical Description White Micr°Crystals Or White Powder (Ntp 1992)Peso molecular:318.36PXS-4728A
CAS:<p>BI-1467335 HCl(BI 1467335) is a selective, orally active inhibitor of semicarbazide-sensitive amine oxidase (SSAO) that helps improve chronic obstructive</p>Fórmula:C15H22ClFN2O2Pureza:98.61%Cor e Forma:SolidPeso molecular:316.8ODM-203
CAS:<p>ODM-203, a Selective Inhibitor of FGFR and VEGFR, Shows Strong Antitumor Activity, and Induces Antitumor Immunity</p>Fórmula:C26H21F2N5O2SPureza:99.85%Cor e Forma:SolidPeso molecular:505.54Sarpogrelate hydrochloride
CAS:<p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>Fórmula:C24H32ClNO6Pureza:99.73%Cor e Forma:Colorless LiquidPeso molecular:465.97[D-Ala2]leucine-enkephalin
CAS:<p>[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.</p>Fórmula:C29H39N5O7Pureza:98.06%Cor e Forma:SolidPeso molecular:569.65Mertansine
CAS:<p>Mertansine is a tubulin inhibitor and an antibody-conjugable maytansinoid alkaloid. The IC50 of Mertansine against HCT-15 and A431 cells is 0.750 and 0.04nM.Cost-effective and quality-assured.</p>Fórmula:C35H48ClN3O10SPureza:98% - >99.99%Cor e Forma:SolidPeso molecular:738.29Vitexin-4''-O-glucoside
CAS:<p>Vitexin-4''-O-glucoside (Vitexin -4''-O-glucoside) could effectively protect ECV-304 cells against cytotoxicity induced by TBHP through resuming mitochondrial</p>Fórmula:C27H30O15Pureza:98.58% - 99.64%Cor e Forma:SolidPeso molecular:594.52Substance P
CAS:<p>Substance P (Neurokinin P) (SP) is an undecapeptide (a peptide composed of a chain of 11 amino acid residues) member of the tachykinin neuropeptide family.</p>Fórmula:C63H98N18O13SPureza:98% - 99.51%Cor e Forma:White PowderPeso molecular:1347.63Gypenoside XVII
CAS:<p>Gypenoside XVII (Gynosaponin S) confers protection against Aβ25-35-induced neurotoxicity through estrogen receptor-dependent activation of PI3K/Akt pathways,</p>Fórmula:C48H82O18Pureza:98% - 99.89%Cor e Forma:SolidPeso molecular:947.155-(2-furyl)-N-propylisoxazole-3-carboxamide
CAS:<p>5-(2-furyl)-isoxazole combats glutamate toxicity, oxidative stress, and inflammation; potential in Alzheimer's and Parkinson's therapy.</p>Fórmula:C11H12N2O3Pureza:99.64%Cor e Forma:SolidPeso molecular:220.22Dihydroactinidiolide
CAS:<p>Dihydroactinidiolide (R-(-)Dihydro actinidiolide)is avolatileterpene. It has a sweet,tea-likeodorand is used as a fragrance.</p>Fórmula:C11H16O2Pureza:99.94%Cor e Forma:Less Crystal Colorless CrystalPeso molecular:180.24Tazarotene
CAS:<p>Tazarotene (Zorac), a synthetic topical retinoid, treats psoriasis by normalizing keratinocytes and reducing growth.</p>Fórmula:C21H21NO2SPureza:97.01% - 99.14%Cor e Forma:White SolidPeso molecular:351.462,5-Dihydroxybenzaldehyde
CAS:<p>2,5-Dihydroxybenzaldehyde (Gentisaldehyde) has antioxidant activity against Mycobacterium avium subsp.</p>Fórmula:C7H6O3Pureza:99.55% - 99.75%Cor e Forma:SolidPeso molecular:138.12
