
Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.524 produtos)
- Apoptose(5.793 produtos)
- Ciclo celular/Ponto de verificação(4.452 produtos)
- Cromatina/Epigenética(2.242 produtos)
- Sinalização Citoesquelética(1.382 produtos)
- Dano de DNA/Reparo de DNA(2.826 produtos)
- Endocrinologia/Hormónios(3.507 produtos)
- Enzima(3.640 produtos)
- GPCR/Proteína-G(8.333 produtos)
- Imunologia e Inflamação(3.527 produtos)
- Vírus da Influenza(296 produtos)
- Sinalização JAK/STAT(404 produtos)
- Sinalização MAPK(1.203 produtos)
- Transportador de Membranas/Canal Iónico(2.792 produtos)
- Metabolismo(9.449 produtos)
- Microbiologia/Virologia(6.981 produtos)
- Neurociência(9.926 produtos)
- Outros inibidores(37.921 produtos)
- Oxidação-Redução(41 produtos)
- Sinalização PI3K/Akt/mTOR(1.400 produtos)
- Proteases/Proteassoma(1.597 produtos)
- Células - tronco e Derivados(830 produtos)
- Tirosina Quinase/Adaptador(2.015 produtos)
- Ubiquitinação(1.650 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66639 produtos de "Inibidores"
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Ilaprazole sodium
CAS:<p>Ilaprazole sodium (IY-81149 sodium) , a substituted benzimidazole prodrug, is a selective and irreversible proton pump inhibitor.</p>Fórmula:C19H17N4NaO2SPureza:99.06%Cor e Forma:SolidPeso molecular:388.42Vps34-IN-4
CAS:<p>VPS34 inhibitor 1 (Compound 19, PIK-III analogue) (PIK-III analogue) is a potent and selective inhibitor of VPS34( IC50 : 15 nM)</p>Fórmula:C21H25N7OPureza:98.6%Cor e Forma:SolidPeso molecular:391.47Pseudolaric acid A-O-β-D-glucopyranoside
CAS:<p>Pseudolaric acid A-O-β-D-glucopyranoside (Pseudolaric acid A-O-beta-D-glucopyranoside) is a natural product with antibacterial, anticancer</p>Fórmula:C28H38O11Pureza:99.5% - 99.7%Cor e Forma:SolidPeso molecular:550.60MSDC 0160
CAS:<p>MSDC 0160 (CAY10415) is a prototype mTOT-modulating insulin sensitizer being used in trials studying the treatment of Type 2 Diabetes and Alzheimer's Disease.</p>Fórmula:C19H18N2O4SPureza:98.11% - 99.53%Cor e Forma:SolidPeso molecular:370.42BIIB021
CAS:<p>BIIB021 (CNF2024) is an orally-available, fully synthetic inhibitor of HSP90(Ki=1.7 nM, EC50=38 nM).</p>Fórmula:C14H15ClN6OPureza:98% - 99.82%Cor e Forma:SolidPeso molecular:318.76PSA1 141-150 acetate
<p>PSA1 141-150 acetate is used in the immunotherapy of cancer experiments that is a prostate specific antigen 1 peptide.</p>Fórmula:C57H97N13O15SPureza:96.41%Cor e Forma:SolidPeso molecular:1236.52Genz-644282
CAS:<p>Genz-644282, a novel non-camptothecin topoisomerase I inhibitor for cancer treatment.</p>Fórmula:C22H21N3O5Pureza:97.49%Cor e Forma:SolidPeso molecular:407.42Tolimidone
CAS:<p>Tolimidone (NSC 314335) is a chemical compound which inhibits acid secretion in animal models and also acts as a bronchodilator in histamine-challenged animals.</p>Fórmula:C11H10N2O2Pureza:99.85% - 99.85%Cor e Forma:SolidPeso molecular:202.21Tipifarnib (S enantiomer)
CAS:<p>Tipifarnib S enantiomer ((S)-(-)-R-115777) is the S-enantiomer of Tipifarnib. Tipifarnib is a potent and specific farnesyltransferase inhibitor (IC50: 0.6 nM).</p>Fórmula:C27H22Cl2N4OPureza:99.05%Cor e Forma:SolidPeso molecular:489.4ABT-724
CAS:<p>ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)</p>Fórmula:C17H19N5Pureza:99.73%Cor e Forma:SolidPeso molecular:293.37Zofenopril calcium
CAS:<p>Zofenopril calcium (SQ26991) is an antioxidant that acts as an angiotensin-converting enzyme inhibitor.</p>Fórmula:C44H44CaN2O8S4Pureza:98.37%Cor e Forma:White Or Whitish Crystalline PowderPeso molecular:897.17Ondansetron hydrochloride
CAS:<p>Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation</p>Fórmula:C18H19N3O·HClPureza:99.78%Cor e Forma:White PowderPeso molecular:329.82Silmitasertib
CAS:<p>Silmitasertib (CX-4945) is a potent, orally bioavailable inhibitor of casein kinase 2 (CK2; Ki: 0.38 nM).</p>Fórmula:C19H12ClN3O2Pureza:98% - 99.90%Cor e Forma:SolidPeso molecular:349.77Tecalcet Free Base
CAS:<p>Tecalcet Free Base is an oral calcium receptor agonist</p>Fórmula:C18H22ClNOCor e Forma:SolidPeso molecular:303.83bis(p-methoxyphenyl)iodonium bromide
CAS:<p>Di(p-anisyl)iodonium bromide used in polymer synthesis, nanoparticle prep, and dye creation.</p>Fórmula:C14H14BrIO2Pureza:99.56%Cor e Forma:SolidPeso molecular:421.07D-Galacturonic acid hydrate
CAS:<p>D-Galacturonic acid hydrate is used in the synthesis of N-(D-galacturonoyl) amino acids and dipeptides.</p>Fórmula:C6H12O8Pureza:97% - 99.97%Cor e Forma:White To Light Beige Fine PowderPeso molecular:212.15β-Sitosterol
CAS:<p>Beta-Sitosterol induces G2/M arrest, endoreduplication, and apoptosis, possibly affecting cancer therapy, cholesterol metabolism, and inflammation.</p>Fórmula:C29H50OPureza:98.54% - 99.95%Cor e Forma:White SolidPeso molecular:414.71Dehydropachymic acid
CAS:<p>Dehydropachymic acid shows antiinflammatory activity.</p>Fórmula:C33H50O5Pureza:99.61% - 99.78%Cor e Forma:SolidPeso molecular:526.75Midostaurin
CAS:<p>PKC412(Midostaurin (PKC412); CGP41231; CGP41251) is a broad spectrum protein kinase inhibitor.</p>Fórmula:C35H30N4O4Pureza:97.61% - >99.99%Cor e Forma:SolidPeso molecular:570.643-Hydroxybutyric acid
CAS:<p>Butanoic acid is an endogenous histone deacetylase (HDAC) inhibitor,IC50 for HDAC3, HDAC4, and HDAC1 is 2.4 mM, 4.5 mM, and 5.3 mM. High-Quality, Low-Cost!</p>Fórmula:C4H8O3Pureza:97.31% - 99.77%Cor e Forma:SolidPeso molecular:104.1trans-4-Hydroxycyclohexanecarboxylic Acid
CAS:<p>trans-4-Hydroxycyclohexanecarboxylic Acid is an organic intermediate.</p>Fórmula:C7H12O3Pureza:96.24%Cor e Forma:SolidPeso molecular:144.17Neoandrographolide
CAS:<p>Neoandrographolide has hypolipidemic, cardio-protective, anti-inflammatory effects, and enhances chemo-sensitivity without major liver harm.</p>Fórmula:C26H40O8Pureza:98.52% - 99.00%Cor e Forma:Less Columnar Crystal Colorless Columnar CrystalPeso molecular:480.59TP-2857
CAS:<p>TP-2857 (TAP2857) is a potent antimicrobial agent.</p>Fórmula:C28H38N2O5SiPureza:98.43%Cor e Forma:SolidPeso molecular:510.7Maoecrystal B
CAS:<p>Maoecrystal B is a diterpenoid isolated from the leaves of Isodon eriocalyx var.</p>Fórmula:C22H28O6Pureza:97.00%Cor e Forma:SolidPeso molecular:388.45Olanexidine
CAS:<p>Olanexidine: broad-spectrum antibacterial/antiseptic, targets gram-positive/negative bacteria, used in infection/inflammation research.</p>Fórmula:C17H27Cl2N5Cor e Forma:SolidPeso molecular:372.34Lucanthone hydrochloride
CAS:<p>Lucanthone hydrochloride is a novel acridine derivative which supresses autophagic degradation and triggers apoptosis in colon cancer cells.</p>Fórmula:C20H25ClN2OSCor e Forma:SolidPeso molecular:376.94Piperacetazine
CAS:<p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>Fórmula:C24H30N2O2SPureza:99.9% - 99.92%Cor e Forma:SolidPeso molecular:410.57SCH772984
CAS:<p>SCH772984 is an ERK inhibitor and is highly selective and ATP-competitive. SCH772984 exhibits antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C33H33N9O2Pureza:97.565% - 98.75%Cor e Forma:SolidPeso molecular:587.67ELOVL6-IN-1
CAS:<p>ELOVL6-IN-1: selective, oral ELOVL6 inhibitor; IC50 of 0.35 μM; noncompetitive with Ki of 994 nM.</p>Fórmula:C27H24F3N3O3Pureza:99.54%Cor e Forma:SolidPeso molecular:495.49iMDK
CAS:<p>iMDK quarterhydrate, a PI3K inhibitor, blocks MDK growth factor and enhances NSCLC treatment with MEK inhibitors, sparing normal cells.</p>Fórmula:C21H13FN2O2SPureza:99.99%Cor e Forma:SolidPeso molecular:376.44-Cyclohexylphenol
CAS:<p>4-Cyclohexylphenol (p-Cyclohexylphenol) is a biochemical compound for proteomics research.</p>Fórmula:C12H16OPureza:99.72%Cor e Forma:Brown Crystalline Solid With A Weak Characteristic OdorPeso molecular:176.25VU 0238429
CAS:<p>VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).</p>Fórmula:C17H12F3NO4Pureza:>99.99%Cor e Forma:SolidPeso molecular:351.28HhAntag
CAS:<p>HhAntag is a small molecule inhibitor of GLI1-mediated transcription, an essential down-stream element of the Hedgehog (Hh) pathway with the anti-tumor activity</p>Fórmula:C24H23ClN4O3Pureza:95.73%Cor e Forma:SolidPeso molecular:450.92SM-7368
CAS:<p>The NF-κB Activation Inhibitor III, controls the biological activity of NF-κB. It is primarily used for Inflammation/Immunology applications.</p>Fórmula:C10H5ClN4O5SPureza:99.64%Cor e Forma:SolidPeso molecular:328.69Cinnarizine clofibrate
CAS:<p>Cinnarizine clofibrate: a piperazine derivative, calcium channel inhibitor, antihistamine, prevents motion sickness-induced vomiting.</p>Fórmula:C36H39ClN2O3Cor e Forma:SolidPeso molecular:583.17paulownin
CAS:<p>Paulownin, a furofuran lignan from Paulownia tomentosa,has the action of anti-inflammation,analgesia,immunity,hypoglycemia and has little toxicity.</p>Fórmula:C20H18O7Pureza:99.95% - ≥95%Cor e Forma:SolidPeso molecular:370.35BMS-582949 hydrochloride
CAS:<p>The BMS-582949 hydrochloride (BMS-582949 HCl) is a highly specific p38α MAPK inhibitor (IC50: 13 nM).</p>Fórmula:C22H27ClN6O2Pureza:97.57% - 98.75%Cor e Forma:SolidPeso molecular:442.955'-N-Ethylcarboxamidoadenosine
CAS:<p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>Fórmula:C12H16N6O4Pureza:98.95% - ≥95%Cor e Forma:PowderPeso molecular:308.29Chelerythrine chloride
CAS:<p>Chelerythrine Chloride is a cell-permeable inhibitor of protein kinase C, competitive with respect to the phosphate acceptor and non-competitive with respect to</p>Fórmula:C21H18ClNO4Pureza:95% - 99.19%Cor e Forma:Yellow To Orange SolidPeso molecular:383.83OF-1
CAS:<p>OF-1 is a potent inhibitor of BRPF1B and BRPF2 bromodomain.</p>Fórmula:C17H18BrN3O4SPureza:98.55% - ≥95%Cor e Forma:SolidPeso molecular:440.31Linzagolix
CAS:<p>Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei</p>Fórmula:C22H15F3N2O7SPureza:99.33%Cor e Forma:SolidPeso molecular:508.42RGX-202
CAS:<p>RGX-202 (β-GPA) is an orally active inhibitor of the SLC6A8 transport protein. RGX-202 is a creatine analog that alters skeletal muscle energy expenditure.</p>Fórmula:C4H9N3O2Pureza:99.67% - 99.8%Cor e Forma:SolidPeso molecular:131.13GJ103
CAS:<p>GJ103 sodium salt, an active GJ072 analog, shows read-through activity similar to RTC13/14 with better A-T cell tolerance.</p>Fórmula:C16H14N4O3SPureza:95.78% - 99.04%Cor e Forma:SolidPeso molecular:342.372-Undecanone
CAS:<p>2-Undecanone (Methylnonylketone) is a volatile organic compound that inhibits DnaKJE-ClpB dione-dependent refolding of heat-inactivated bacterial fluorokinase.</p>Fórmula:C11H22OPureza:98.84%Cor e Forma:Colorless To Pale Yellow LiquidPeso molecular:170.29Dimebolin
CAS:<p>Dimebolin (Latrepirdine) is a 5-HT6 antagonist.</p>Fórmula:C21H25N3Pureza:99.69%Cor e Forma:White PowderPeso molecular:319.44RNAIII-inhibiting peptide TFA
<p>RNAIII-inhibiting peptide TFA (RNAIII-inhibiting peptide(TFA))(228544-21-6 free base) inhibits S.</p>Fórmula:C47H57F3N10O13Pureza:98.68%Cor e Forma:SolidPeso molecular:1027.01Ginsenoside Rg4
CAS:<p>Ginsenoside Rg4 is isolated from the leaves of Panax ginseng C.</p>Fórmula:C42H70O12Pureza:99.17%Cor e Forma:SolidPeso molecular:767Picaridin
CAS:<p>Picaridin (Lcaridin) is a topical insect repellent.</p>Fórmula:C12H23NO3Pureza:99.8% - 99.93%Cor e Forma:Less Liquid Colourless LiquidPeso molecular:229.32Transcrocetinate disodium
CAS:<p>Transcrocetinate disodium (Disodium trans-crocetinate), extracted from saffron (Crocus sativus L.), is a high-affinity antagonist of NMDA receptor.</p>Fórmula:C20H22Na2O4Pureza:98.27% - 99.22%Cor e Forma:SolidPeso molecular:372.37Gadolinium chloride
CAS:<p>Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist</p>Fórmula:Cl3GdPureza:98%Cor e Forma:White Crystalline SolidPeso molecular:263.61
