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Inibidores

Inibidores

Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.

Subcategorias de "Inibidores"

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Foram encontrados 66639 produtos de "Inibidores"

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  • Agmatine sulfate

    CAS:
    <p>Agmatine sulfate (Agmatine sulfate salt) is a bioactive metabolite of the arginine amino acid.</p>
    Fórmula:C5H16N4O4S
    Pureza:99.56% - 99.86%
    Cor e Forma:White To Off-White Powder
    Peso molecular:228.27
  • Nirogacestat

    CAS:
    <p>Nirogacestat (PF 03084014) is a specific γ-secretase inhibitor (IC50: 6.2 nM, in a cell-free assay).</p>
    Fórmula:C27H41F2N5O
    Pureza:97.98% - 99.63%
    Cor e Forma:Solid
    Peso molecular:489.64
  • BMS-833923

    CAS:
    <p>BMS-833923 (XL-139), an orally bioavailable Smoothened antagonist, inhibits BODIPY cyclopamine binding to SMO in a dose-dependent manner (IC50: 21 nM).</p>
    Fórmula:C30H27N5O
    Pureza:99.47% - 99.76%
    Cor e Forma:Solid
    Peso molecular:473.57
  • lufenuron

    CAS:
    <p>Lufenuron (Fluphenacur) is a chitin-synthesis inhibitor.</p>
    Fórmula:C17H8Cl2F8N2O3
    Pureza:99.87%
    Cor e Forma:Coa
    Peso molecular:511.15
  • Tyrphostin AG1296

    CAS:
    <p>Tyrphostin AG1296 (Tyrphostin AG 1296) is an inhibitor of PDGFR with IC50 of 0.3-0.5 μM, no activity to EGFR.</p>
    Fórmula:C16H14N2O2
    Pureza:99.94% - >99.99%
    Cor e Forma:Solid
    Peso molecular:266.29
  • ALSTERPAULLONE

    CAS:
    <p>Alsterpaullone is a Cyclin-Dependent Kinase Inhibitor, Mediated Toxicity in HeLa Cells Through Apoptosis-Inducing Effec</p>
    Fórmula:C16H11N3O3
    Pureza:99.8%
    Cor e Forma:Solid
    Peso molecular:293.28
  • PF-3758309

    CAS:
    <p>PF-3758309 (PF-03758309) (IC50=1.3 nM), a pyrrolopyrazole inhibitor of PAK4, has effective ATP-competition.</p>
    Fórmula:C25H30N8OS
    Pureza:97.70%
    Cor e Forma:Solid
    Peso molecular:490.62
  • ELR510444

    CAS:
    <p>ELR510444 (LR510444) is a novel microtubule disruptor; inhibits MDA-MB-231 cell proliferation with IC50 of 30.9 nM.</p>
    Fórmula:C19H16N2O2S2
    Pureza:97.67% - 98.69%
    Cor e Forma:Solid
    Peso molecular:368.47
  • Methyl N-methylanthranilate

    CAS:
    <p>Methyl N-methylanthranilate (Methyl2-(methylamino)benzoate) is anatural product.</p>
    Fórmula:C9H11NO2
    Pureza:98.44%
    Cor e Forma:Pale-Yellow Liq With Slight Bluish Fluorescence Liquid
    Peso molecular:165.19
  • SN-011

    CAS:
    <p>SN-011 (GUN35901) is a STING inhibitor, which inhibited the activation of the STING signal pathway and to prevent or treat a STING- mediated disease.</p>
    Fórmula:C25H19FN2O4S
    Pureza:97.99% - 98.03%
    Cor e Forma:Solid
    Peso molecular:462.49
  • ACEPROMAZINE MALEATE

    CAS:
    <p>ACEPROMAZINE MALEATE is a dopamine receptor antagonist</p>
    Fórmula:C23H26N2O5S
    Pureza:98.87% - 99.51%
    Cor e Forma:Off White Or Yellow Crystalline Powder
    Peso molecular:442.53
  • Acetophenone

    CAS:
    <p>Acetophenone (Phenylethanone) is used in chemical synthesis and as a fragrance.</p>
    Fórmula:C8H8O
    Pureza:99.53%
    Cor e Forma:Acetophenone Is A Colorless Liquid Liquid
    Peso molecular:120.15
  • CZ415

    CAS:
    <p>CZ415 is a potent and highly selective mTOR inhibitor.</p>
    Fórmula:C22H29N5O4S
    Pureza:97.54% - 98.36%
    Cor e Forma:Solid
    Peso molecular:459.56
  • 7-Ethoxyresorufin

    CAS:
    <p>7-Ethoxyresorufin (Resorufin ethyl ether) (7-ER) is a fluorometric substrate for and competitive inhibitor of cytochrome P450, especially CYP1A1.</p>
    Fórmula:C14H11NO3
    Pureza:99.09% - 99.62%
    Cor e Forma:Red Solid
    Peso molecular:241.24
  • SMCC-DM1

    CAS:
    <p>SMCC-DM1 is a drug-coupler coupler consisting of a potent microtubule disrupter, DM1, and a coupler, SMCC, for the preparation of antibody-drug couplers.Cost-effective and quality-assured.</p>
    Fórmula:C51H66ClN5O16S
    Pureza:97.07% - 99.25%
    Cor e Forma:Solid
    Peso molecular:1072.61
  • Lapachol

    CAS:
    <p>Lapachol (CI75490): antimicrobial, anti-inflammatory, analgesic, antibiotic, inhibits epithelial tumors in Drosophila.</p>
    Fórmula:C15H14O3
    Pureza:99.01% - 99.38%
    Cor e Forma:White To Yellow Powder
    Peso molecular:242.27
  • Centhaquin

    CAS:
    <p>Centhaquin (Centhaquine)e is an adrenergic receptor potentially for the treatment of postoperative pain and for the resuscitation of hypovolemic shock</p>
    Fórmula:C22H25N3
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:331.45
  • Linderane

    CAS:
    <p>1. Linderane was characterized as a mechanism-based inactivator of CYP2C9.</p>
    Fórmula:C15H16O4
    Pureza:98.25%
    Cor e Forma:Solid
    Peso molecular:260.29
  • Desmethylanethol trithione

    CAS:
    <p>Desmethylanethol trithione (ADT-OH), a synthetic H2S donor, modulates tPA effects, reduces stroke damage, and improves recovery in mice.</p>
    Fórmula:C9H6OS3
    Pureza:98.05% - 98.41%
    Cor e Forma:Solid
    Peso molecular:226.34
  • 2-Hydroxydecanoic acid

    CAS:
    <p>2-Hydroxydecanoic acid ((±)-α-hydroxy Decanoic Acid) is a fatty acid found in the lipophilic portion of the lipopolysaccharide fraction of the aerobic bacterium</p>
    Fórmula:C10H20O3
    Pureza:99.1%
    Cor e Forma:White Solid
    Peso molecular:188.26
  • Purpurogallin

    CAS:
    <p>Purpurogallin: natural phenol from Quercus spp., xanthine oxidase inhibitor (IC50: 0.2μM), antioxidant, anti-inflammatory.</p>
    Fórmula:C11H8O5
    Pureza:96.44%
    Cor e Forma:Solid
    Peso molecular:220.18
  • tris(dibenzylideneacetone)dipalladium

    CAS:
    <p>tris(dibenzylideneacetone)dipalladium (Tris DBA) is a N-myristoyltransferase-1 (NMT-1) inhibitor</p>
    Fórmula:C51H42O3Pd2
    Pureza:98%
    Cor e Forma:Purple Crystals
    Peso molecular:915.71
  • Banoxantrone

    CAS:
    <p>Banoxantrone (AQ4N), a hypoxia-targeting drug, turns into AQ4 to inhibit topoisomerase II and selectively kills hypoxic cells, potentiated by radiation.</p>
    Fórmula:C22H28N4O6
    Cor e Forma:Solid
    Peso molecular:444.48
  • Cinacalcet metabolite M4

    CAS:
    <p>Cinacalcet metabolite M4 (Rarechem AL BW 1078) is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.</p>
    Fórmula:C10H12F3N
    Pureza:97.13%
    Cor e Forma:Solid
    Peso molecular:203.2
  • 3-(2,6-dichlorophenyl)-1-methyl-7-(methylsulfanyl)-1H,2H,3H,4H-pyrimido[4,5-d][1,3]diazin-4-one

    CAS:
    <p>Compound treats tumors, Alzheimer's, Parkinson's, inflammation, and pain; has chlorophenyl, methyl, and methylsulfanyl groups.</p>
    Fórmula:C14H12Cl2N4OS
    Pureza:98.95%
    Cor e Forma:Solid
    Peso molecular:355.24
  • o-Phenanthroline monohydrate

    CAS:
    <p>o-Phenanthroline monohydrate (1, 10-Phenanthroline monohydrate) is an inhibitor of metallopeptidases, inhibits zinc-dependent hydrolysis of Fa-Gly-Leu-NH2.</p>
    Fórmula:C12H10N2O
    Pureza:98.73%
    Cor e Forma:White Crystals Or Powder
    Peso molecular:198.22
  • L-Histidine

    CAS:
    <p>L-Histidine (L-(-)-Histidine) is a semi-essential amino acid (children should obtain it from food) needed in humans for growth and tissue repair, L-Histidine is</p>
    Fórmula:C6H9N3O2
    Pureza:99.62% - 99.92%
    Cor e Forma:Needles Or Plates Solid
    Peso molecular:155.15
  • Raltegravir sodium

    CAS:
    <p>Raltegravir (MK 0518) sodium is a potent, orally active HIV integrase (IN) inhibitor.</p>
    Fórmula:C20H20FN6NaO5
    Cor e Forma:Solid
    Peso molecular:466.405
  • Procyanidin B1

    CAS:
    <p>Procyanidin B1, isolated from commonly eaten fruits, binds to the TLR4/MD-2 complex and has anti-inflammatory activity.</p>
    Fórmula:C30H26O12
    Pureza:98.00% - 99.91%
    Cor e Forma:Red-Brown Powder
    Peso molecular:578.52
  • 1-Oleoyl-sn-glycero-3-phosphocholine

    CAS:
    <p>1-Oleoyl-sn-glycero-3-phosphocholine is a reference for the analysis of lysolecithins</p>
    Fórmula:C26H52NO7P
    Pureza:99.19%
    Cor e Forma:Solid
    Peso molecular:521.67
  • TAK-715

    CAS:
    <p>TAK-715 is a p38 MAPK inhibitor for p38α.</p>
    Fórmula:C24H21N3OS
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:399.51
  • Ethoxysanguinarine

    CAS:
    <p>Ethoxysanguinarine inhibits HuAChE and HuBuChE with IC50s of 0.83 and 4.20 μM, respectively.</p>
    Fórmula:C22H19NO5
    Pureza:99.24% - 99.48%
    Cor e Forma:Solid
    Peso molecular:377.39
  • Telaprevir

    CAS:
    <p>Telaprevir (Incivek) (VX-950) is an effective inhibitor of HCV NS3-4A serine protease (IC50: 0.35 μM).</p>
    Fórmula:C36H53N7O6
    Pureza:96.9% - 98.89%
    Cor e Forma:Solid
    Peso molecular:679.85
  • NS9283

    CAS:
    <p>NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.</p>
    Fórmula:C14H8N4O
    Pureza:99.12%
    Cor e Forma:Solid
    Peso molecular:248.24
  • CID 16020046

    CAS:
    <p>CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.</p>
    Fórmula:C25H19N3O4
    Pureza:99.03%
    Cor e Forma:Solid
    Peso molecular:425.44
  • Ethyl gallate

    CAS:
    <p>Ethyl gallate reduces breast cancer cell growth, invasion, and shows cytotoxicity via PI3K/Akt and MMPs pathway modulation; potential in cancer therapy.</p>
    Fórmula:C9H10O5
    Pureza:99.96%
    Cor e Forma:White Granular
    Peso molecular:198.17
  • DS-1971a

    CAS:
    <p>DS-1971a is a highly potent and selective NaV1.7 inhibitor. DS-1971a exhibits a favorable toxicological profile and analgesic effects.</p>
    Fórmula:C20H21ClFN5O3S
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:465.93
  • Omadacycline HCl

    CAS:
    <p>Omadacycline, a first-class aminomethylcycline, treats pneumonia and skin infections including MRSA, and overcomes tetracycline resistance.</p>
    Fórmula:C29H41ClN4O7
    Cor e Forma:Solid
    Peso molecular:593.118
  • Tiaprofenic acid

    CAS:
    <p>Tiaprofenic acid (Acido tiaprofenico) is a non-steroidal anti-inflammatory drug used to treat pain, especially arthritic pain.</p>
    Fórmula:C14H12O3S
    Pureza:99.51%
    Cor e Forma:Solid
    Peso molecular:260.31
  • Seletalisib

    CAS:
    <p>Seletalisib (UCB5857) (UCB5857) is a potent and specific PI3Kδ inhibitor (IC50: 12 nM).</p>
    Fórmula:C23H14ClF3N6O
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:482.85
  • PHYTOL

    CAS:
    <p>Phytol is a diterpene alcohol with antinociceptive, antioxidant, anti-inflammatory, and antiallergic properties, activating PPARα.</p>
    Fórmula:C20H40O
    Pureza:97.71 - 99.62%
    Cor e Forma:Liquid
    Peso molecular:296.53
  • D-Tagatose

    CAS:
    <p>D-Tagatose, a rare hexoketose and isomer of d-galactose, is naturally found in Sterculia setigera gum and various dairy products.</p>
    Fórmula:C6H12O6
    Pureza:99.78% - 99.96%
    Cor e Forma:White Crystalline Powder
    Peso molecular:180.16
  • BAR 501 impurity

    CAS:
    <p>BAR 501 impurity 在 BAR501 制剂中发现的一种杂质,可作为 G 蛋白偶联胆汁酸激活受体 (GP-BAR1) 的激动剂。 BAR501 杂质 (10 µM) 在 GP-BAR1 报告基因检测中诱导荧光素酶活性增加 150%。</p>
    Fórmula:C26H46O3
    Pureza:98.78%
    Cor e Forma:Solid
    Peso molecular:406.64
  • LIXIVAPTAN

    CAS:
    <p>Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)</p>
    Fórmula:C27H21ClFN3O2
    Pureza:98.36%
    Cor e Forma:Solid
    Peso molecular:473.93
  • LF3

    CAS:
    <p>LF3 is a specific inhibitor of canonical Wnt signaling by disrupting the interaction between β-catenin and TCF4 (IC50 &lt; 2 μM)</p>
    Fórmula:C20H24N4O2S2
    Pureza:99.63%
    Cor e Forma:Solid
    Peso molecular:416.56
  • Adenine hydrochloride

    CAS:
    <p>Adenine hydrochloride (6-Aminopurine hydrochloride) is a hydrochloride salt form of adenine which is a nucleobase with a variety of roles in biochemistry.</p>
    Fórmula:C5H5N5·HCl
    Pureza:98.86%
    Cor e Forma:White To Light Yellow Crystal Powder
    Peso molecular:171.59
  • BX-795 hydrochloride

    CAS:
    <p>BX-795 hydrochloride is a TBK1 and IKKε inhibitor. BX-795 is a potential maternal embryonic leucine zipper kinase inhibitor.</p>
    Fórmula:C23H27ClIN7O2S
    Cor e Forma:Solid
    Peso molecular:627.93
  • ABT-639 hydrochloride

    CAS:
    <p>ABT-639 hydrochloride is a selective, novel T-type Ca2+ channel blocker.</p>
    Fórmula:C20H21Cl2F2N3O3S
    Cor e Forma:Solid
    Peso molecular:492.36
  • Levolansoprazole

    CAS:
    <p>Levolansoprazole ((S)-Lansoprazole), a proton pump inhibitor, irreversibly inhibits H+/K+-stimulated ATPase pumps in parietal cells (IC50: 5.2 μM).</p>
    Fórmula:C16H14F3N3O2S
    Pureza:98.629%
    Cor e Forma:Solid
    Peso molecular:369.36
  • Thalidomide 4-fluoride

    CAS:
    <p>Thalidomide 4-fluoride (E3 ligase Ligand 4) (Cereblon ligand 4) is the Thalidomide-based Cereblon ligand.</p>
    Fórmula:C13H9FN2O4
    Pureza:99.12%
    Cor e Forma:Solid
    Peso molecular:276.22