CAS 95093-99-5

(2R)-1-(9H-carbazol-4-yloxy)-3-{[2-(2-methoxyphenoxy)ethyl]amino}propan-2-ol

Description:

The chemical substance known as (2R)-1-(9H-carbazol-4-yloxy)-3-{[2-(2-methoxyphenoxy)ethyl]amino}propan-2-ol, with the CAS number 95093-99-5, is a complex organic compound characterized by its unique structural features. It contains a carbazole moiety, which is a fused ring system known for its aromatic properties and potential applications in organic electronics and pharmaceuticals. The presence of a propanol group suggests that it may exhibit alcohol-like properties, potentially influencing its solubility and reactivity. Additionally, the compound features ether and amine functional groups, which can enhance its biological activity and interaction with various biological targets. The methoxyphenoxy group may contribute to its lipophilicity, affecting its pharmacokinetics. Overall, this compound's intricate structure indicates potential utility in medicinal chemistry, particularly in the development of therapeutic agents, although specific biological activities and applications would require further investigation through empirical studies.

Formula: C₂₄H₂₆N₂O₄

InChI: InChI=1/C24H26N2O4/c1-28-21-10-4-5-11-22(21)29-14-13-25-15-17(27)16-30-23-12-6-9-20-24(23)18-7-2-3-8-19(18)26-20/h2-12,17,25-27H,13-16H2,1H3/t17-/m1/s1

SMILES: COc1ccccc1OCCNC[C@H](COc1cccc2c1c1ccccc1[nH]2)O

(2R)-1-(9H-Carbazol-4-yloxy)-3-[[2-(2-methoxyphenoxy)ethyl]amino]-2-propanol

CAS: 95093-99-5

Formula: C₂₄H₂₆N₂O₄

Purity: 98%

Color and Shape: Solid

Molecular weight: 406.4742

Ref: IN-DA01CCHP

(R)-Carvedilol

CAS: 95093-99-5

Formula: C₂₄H₂₆N₂O₄

Molecular weight: 406.48

Ref: 4Z-C-026

(S)-(+)-4’-Hydroxyphenyl Carvedilol-d4

CAS: 95093-99-5

Formula: C₂₄H₂₂D₄N₂O₅

Molecular weight: 426.51

Ref: 4Z-C-0266

(R)-(+)-Carvedilol

Controlled Product

CAS: 95093-99-5

Stability Hygroscopic
Applications The optically active isomer of Carvedilol (C184625), a nonselective ß-adrenergic blocker with a1-blocking activity. An antihypertensive used in the treatment of congestive heart failure.
Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package
References Hirohashi, M., et al.: Arzneim.-Forsch., 40, 735 (1990),

Formula: C₂₄H₂₆N₂O₄

Color and Shape: Off White Solid

Molecular weight: 406.47

Ref: TR-C184630

(R)-(+)-Carvedilol

Controlled Product

CAS: 95093-99-5

Carvedilol is a racemic mixture of the enantiomers (-) and (+) that are mirror images of each other. It is used in the treatment of congestive heart failure and ventricular dysfunction by acting as a vasodilator and reducing cardiac workload. Carvedilol has been shown to reduce blood pressure, decrease plasma levels of α1-acid glycoprotein, increase the excretion of teicoplanin, and inhibit cytosolic calcium release. Carvedilol also binds stereoselectively to the ryanodine receptor in rat hearts and inhibits on-line cytosolic calcium release. The (+) enantiomer has been shown to have greater potency than (-) at binding to the ryanodine receptor.

Formula: C₂₄H₂₆N₂O₄

Purity: Min. 95%

Color and Shape: White Powder

Molecular weight: 406.47 g/mol

Ref: 3D-FC19827

Carvedilol (R)-Isomer

CAS: 95093-99-5

Formula: C₂₄H₂₆N₂O₄

Molecular weight: 406.48

Ref: ST-EA-CP-C10040

(R)-Carvedilol

CAS: 95093-99-5

(R)-Carvedilol is a non-selective blocker of β/α-1. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).

Formula: C₂₄H₂₆N₂O₄

Purity: 98%

Color and Shape: Solid

Molecular weight: 406.47

Ref: TM-T12615