EGFR
EGFR (epidermal growth factor receptor) inhibitors are compounds that block the signaling of EGFR, a receptor that is often overexpressed in various cancers and plays a critical role in angiogenesis. EGFR inhibitors are used to prevent tumor growth and metastasis by disrupting the pathways that promote blood vessel formation in tumors. These inhibitors are widely used in cancer research and therapy. At CymitQuimica, we offer a diverse selection of high-quality EGFR inhibitors to support your research in oncology and angiogenesis.
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(E)-AG 99
CAS:122520-85-8
(E)-AG 99 ((E)-Tyrphostin AG 99) is an inhibitor of EGFR kinase (IC50: 10 μM in …
Formula:
C10H8N2O3
Purity:
99.23%
Color and Shape:
Solid
Molecular weight:
204.18
Ref: TM-T5155
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 157.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
JCN037
CAS:2305154-31-6
JCN037 is potent, non-covalent and brain-penetrant inhibitor of EGFR(EGFR, p-wtEGFR and pEGFRvⅢ with IC50 of …
Formula:
C16H11BrFN3O2
Purity:
99.50%
Color and Shape:
Solid
Molecular weight:
376.18
Ref: TM-T8431
| 2mg | 39.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 263.00 € | ||
| 100mg | 377.00 € | ||
| 200mg | 537.00 € | ||
| 1mL*10mM (DMSO) | 81.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Biochanin A
CAS:491-80-5
Biochanin A: an isoflavone from red clover with anticancer properties and inhibits FAAH.
Formula:
C16H12O5
Purity:
97.1% - 97.69%
Color and Shape:
Solid
Molecular weight:
284.26
Ref: TM-T2859
| 100mg | 40.00 € | ||
| 200mg | 55.00 € | ||
| 500mg | 94.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
EGFR/ErbB-2/ErbB-4 inhibitor-2
CAS:179248-61-4
EGFR/ErbB-2/ErbB-4 inhibitor-2 (EGFR/ErbB2 Inhibitor) is a cell-permeable inhibitor of EGFR and c-ErbB2 (IC50s = 20 …
Formula:
C23H21N3O3
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
387.43
Ref: TM-T21954
| 1mg | 73.00 € | ||
| 2mg | 90.00 € | ||
| 5mg | 136.00 € | ||
| 10mg | 197.00 € | ||
| 25mg | 359.00 € | ||
| 50mg | 538.00 € | ||
| 100mg | 781.00 € | ||
| 200mg | 1,035.00 € | ||
| 1mL*10mM (DMSO) | 151.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Olmutinib
CAS:1802181-20-9
Olmutinib (BI1482694) is a Novel Epidermal Growth Factor Receptor Tyrosine Kinase Inhibitor
Formula:
C26H26N6O2S
Purity:
97.46%
Color and Shape:
Solid
Molecular weight:
486.59
Ref: TM-T8460
| 2mg | 36.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 129.00 € | ||
| 50mg | 181.00 € | ||
| 100mg | 277.00 € | ||
| 200mg | 454.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
AEE788
CAS:497839-62-0
AEE788 (NVP-AEE 788) has been used in trials studying the treatment of Cancer, Glioblastoma Multiforme, …
Formula:
C27H32N6
Purity:
100% - 98.94%
Color and Shape:
Solid
Molecular weight:
440.58
Ref: TM-T2116
| 2mg | 46.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 319.00 € | ||
| 100mg | 481.00 € | ||
| 500mg | 1,078.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
WHI-P180
CAS:211555-08-7
WHI-P180 (Janex 3) is a potent EGFR and Cdk2 inhibitors with IC50 of 4.0 and …
Formula:
C16H15N3O3
Purity:
97.74%
Color and Shape:
Solid
Molecular weight:
297.31
Ref: TM-T2032
| 1mg | 46.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 215.00 € | ||
| 50mg | 321.00 € | ||
| 100mg | 463.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Trastuzumab
CAS:180288-69-1
Trastuzumab is a humanized monoclonal antibody for patients with invasive breast cancers that overexpress HER2.
Purity:
98% - 99.50%
Color and Shape:
Liquid
Molecular weight:
Approximately 145.53 kDa
Ref: TM-T9912
| 1mg | 152.00 € | ||
| 5mg | 511.00 € | ||
| 10mg | 640.00 € | ||
| 25mg | 1,009.00 € | ||
| 50mg | 1,364.00 € | ||
| 100mg | 1,831.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Sulforaphene
CAS:592-95-0
Sulforaphene, from radish seeds, aids cancer cell apoptosis and inhibits migration; has an ED50 for …
Formula:
C6H9NOS2
Purity:
98.01% - 99.19%
Color and Shape:
Slightly Yellowish Liquid
Molecular weight:
175.27
Ref: TM-TL0016
| 1mg | 36.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 222.00 € | ||
| 50mg | 331.00 € | ||
| 100mg | 489.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
SU5204
CAS:186611-11-0
SU5204 (3-[(2-Ethoxyphenyl)methylidene]-1H-indol-2-one), an analogue of SU5025, pharmacologically inhibits VEGFR2(IC50s of 4 and 51.5 μM for …
Formula:
C17H15NO2
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
265.31
Ref: TM-T22431
| 5mg | 34.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 84.00 € | ||
| 50mg | 112.00 € | ||
| 100mg | 174.00 € | ||
| 200mg | 256.00 € | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PP2
CAS:172889-27-9
PP2 (AG 1879,AGL 1879) is a effective inhibitor of Lck/Fyn (IC50:4/5 nM) , ~100-fold less …
Formula:
C15H16ClN5
Purity:
95.65%
Color and Shape:
White Solid
Molecular weight:
301.77
Ref: TM-T6266
| 2mg | 46.00 € | ||
| 5mg | 68.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 314.00 € | ||
| 100mg | 498.00 € | ||
| 200mg | 709.00 € | ||
| 1mL*10mM (DMSO) | 75.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Tyrphostin AG30
CAS:122520-79-0
Tyrphostin AG30 (AG30) (AG30) is a potent protein tyrosine kinases (PTK) inhibitor.
Formula:
C10H7NO4
Purity:
99.02%
Color and Shape:
Solid
Molecular weight:
205.17
Ref: TM-T7101
| 2mg | 46.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 301.00 € | ||
| 100mg | 500.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PD-161570
CAS:192705-80-9
PD-161570 is a potent and ATP-competitive human FGF-1 receptor inhibitor with an IC50 of 39.9 …
Formula:
C26H35Cl2N7O
Purity:
99.23%
Color and Shape:
Solid
Molecular weight:
532.51
Ref: TM-T23127
| 1mg | 36.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 295.00 € | ||
| 50mg | 473.00 € | ||
| 100mg | 673.00 € | ||
| 200mg | 926.00 € | ||
| 1mL*10mM (DMSO) | 121.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Lazertinib
CAS:1903008-80-9
Lazertinib (GNS-1480) is a potent, selective, irreversible EGFR-TKI; IC50: 1.7-76 nM for various EGFR mutations.
Formula:
C30H34N8O3
Purity:
98.7% - 99.53%
Color and Shape:
Solid
Molecular weight:
554.64
Ref: TM-T4485
| 1mg | 48.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 147.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 319.00 € | ||
| 100mg | 462.00 € | ||
| 500mg | 1,072.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Tyrphostin A1
CAS:2826-26-8
Tyrphostin A1 (Tyrphostin 1) is an inhibitor of EGFR tyrosine kinase .
Formula:
C11H8N2O
Purity:
99.13%
Color and Shape:
Solid
Molecular weight:
184.19
Ref: TM-T7649
| 10mg | 35.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 81.00 € | ||
| 100mg | 93.00 € | ||
| 200mg | 136.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
WZ4002
CAS:1213269-23-8
WZ4002 is a mutant-selective EGFR inhibitor for EGFR(L858R) and EGFR(T790M) with IC50 of 2 nM/8 …
Formula:
C25H27ClN6O3
Purity:
98.12%
Color and Shape:
Solid
Molecular weight:
494.97
Ref: TM-T6238
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 115.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 325.00 € | ||
| 200mg | 478.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Brigatinib
CAS:1197953-54-0
Brigatinib (AP-26113) is a highly potent and selective ALK inhibitor.
Formula:
C29H39ClN7O2P
Purity:
100% - 99.93%
Color and Shape:
Solid
Molecular weight:
584.09
Ref: TM-T3621
| 2mg | 36.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 112.00 € | ||
| 100mg | 163.00 € | ||
| 200mg | 235.00 € | ||
| 500mg | 400.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MAZ51
CAS:163655-37-6
MAZ51 is a VEGFR-3 (Flt-4) tyrosine kinase inhibitor.
Formula:
C21H18N2O
Purity:
98.53%
Color and Shape:
Solid
Molecular weight:
314.38
Ref: TM-T8496
| 1mg | 40.00 € | ||
| 2mg | 56.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 242.00 € | ||
| 50mg | 403.00 € | ||
| 100mg | 599.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Gefitinib-based PROTAC 3
CAS:2230821-27-7
Gefitinib-PROTAC 3 degrades EGFR in cancer cells; DC50s: 11.7 nM (HCC827) and 22.3 nM (H3255).
Formula:
C47H57ClFN7O8S
Purity:
97.29% - 98.25%
Color and Shape:
Solid
Molecular weight:
934.51
Ref: TM-T5437
| 2mg | 44.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 248.00 € | ||
| 100mg | 358.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Dacomitinib hydrate
CAS:1042385-75-0
Dacomitinib hydrate (PF 299804) is a highly selective and second-generation small-molecule inhibitor of the pan-epidermal …
Formula:
C24H27ClFN5O3
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
487.96
Ref: TM-T19965
| 5mg | 50.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 136.00 € | ||
| 100mg | 204.00 € | ||
| 200mg | 301.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
