PKC
PKC (Protein Kinase C) inhibitors target the PKC family of serine/threonine kinases, which are involved in a wide range of cellular processes, including cell cycle regulation, apoptosis, and differentiation. PKC plays a key role in signal transduction pathways that influence cell proliferation and survival. Inhibiting PKC can lead to changes in cell cycle progression, making these inhibitors valuable in research related to cancer, neurobiology, and cardiovascular diseases. At CymitQuimica, we provide a diverse selection of high-quality PKC inhibitors to support your research in signal transduction, cell cycle regulation, and therapeutic development.
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Y-33075
CAS:199433-58-4
Y-33075 is a selective inhibitor of ROCK derived from Y-27632, and is more potent than …
Formula:
C16H16N4O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
280.32
Ref: TM-T13384
| 2mg | 107.00 € | ||
| 25mg | 711.00 € | ||
| 50mg | 932.00 € | ||
| 100mg | 1,526.00 € | ||
| 1mL*10mM (DMSO) | 311.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
CGP60474
CAS:164658-13-3
CGP60474 is an inhibitor of VEGFR-2 (IC50 = 84 nM) and an inhibitor of ATP-competitive …
Formula:
C18H18ClN5O
Purity:
98.15%
Color and Shape:
Solid
Molecular weight:
355.82
Ref: TM-T14943
| 1mg | 35.00 € | ||
| 2mg | 47.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 324.00 € | ||
| 100mg | 537.00 € | ||
| 1mL*10mM (DMSO) | 82.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
DCPLA-ME
CAS:56687-67-3
DCPLA-ME (2-[(2-Pentylcyclopropyl)methyl]cyclopropaneoctanoic acid methyl ester) is the methyl ester form of DCPLA and can be …
Formula:
C21H38O2
Purity:
98.16%
Color and Shape:
Solid
Molecular weight:
322.53
Ref: TM-T10980
| 1mg | 85.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 254.00 € | ||
| 25mg | 419.00 € | ||
| 50mg | 591.00 € | ||
| 100mg | 797.00 € | ||
| 500mg | 1,588.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
VTX-27
CAS:1321924-70-2
VTX-27 is a selective inhibitor of protein kinase C θ (PKC θ) (Kis: 0.08 nM …
Formula:
C20H24ClFN6O
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
418.9
Ref: TM-T13314
| 1mg | 92.00 € | ||
| 2mg | 123.00 € | ||
| 5mg | 239.00 € | ||
| 10mg | 357.00 € | ||
| 25mg | 551.00 € | ||
| 50mg | 765.00 € | ||
| 100mg | 1,015.00 € | ||
| 1mL*10mM (DMSO) | 224.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
PKC-θ inhibitor 1
CAS:1160501-81-4
PKC-theta inhibitor 1 is an inhibitor of PKCθ (Ki of 6 nM)
Formula:
C17H15F3N4O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
348.32
Ref: TM-T12496
| 25mg | 1,688.00 € | ||
| 50mg | 2,225.00 € | ||
| 100mg | 2,897.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
TCS 21311
CAS:1260181-14-3
TCS 21311 (NIBR3049) selectively inhibits JAK3 (IC50: 8 nM) and PKCα/θ & GSK3β; >100x selective …
Formula:
C27H25F3N4O4
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
526.51
Ref: TM-T17019
| 1mg | 96.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
(-)-Indolactam V
CAS:90365-57-4
(-)-Indolactam V: PKC activator, antitumor, Ki 3.36 nM/1.03 μM for η/γ-CRD2, Kd 5.5-213 nM for …
Formula:
C17H23N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
301.38
Ref: TM-T17299
| 1mg | 710.00 € | ||
| 500µg | 375.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
PKC-IN-1
CAS:1046787-18-1
PKC-IN-1 is an ATP-competitive and reversible conventional PKC enzymes inhibitor (PKCα, PKCβI, PKCβII, PKCθ, PKCγ, …
Formula:
C25H37FN8O2
Purity:
98% - 98.79%
Color and Shape:
Solid
Molecular weight:
500.61
Ref: TM-T12494
| 2mg | 186.00 € | ||
| 5mg | 325.00 € | ||
| 25mg | 1,058.00 € | ||
| 50mg | 1,411.00 € | ||
| 100mg | 1,884.00 € | ||
| 1mL*10mM (DMSO) | 362.00 € |
Estimated delivery in United States, on Wednesday 19 Feb 2025
AS2521780
CAS:1214726-89-2
AS2521780 is an inhibitor of PKCθ (IC50: 0.48 nM).
Formula:
C30H41N7OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
547.76
Ref: TM-T14328
| 25mg | 2,662.00 € | ||
| 50mg | 3,522.00 € | ||
| 100mg | 4,844.00 € |
Estimated delivery in United States, on Wednesday 5 Mar 2025
Phorbol 12,13-dibutyrate
CAS:37558-16-0
Phorbol 12,13-dibutyrate (Phorbol dibutyrate) is a PKC activator that induces contraction of isolated rabbit vascular …
Formula:
C28H40O8
Purity:
100% - 99.32%
Color and Shape:
Solid
Molecular weight:
504.61
Ref: TM-T16526
| 1mg | 60.00 € | ||
| 5mg | 163.00 € | ||
| 10mg | 272.00 € | ||
| 25mg | 548.00 € | ||
| 50mg | 777.00 € | ||
| 100mg | 1,049.00 € | ||
| 1mL*10mM (DMSO) | 177.00 € |
Estimated delivery in United States, on Wednesday 5 Mar 2025
