PKC
PKC (Protein Kinase C) inhibitors target the PKC family of serine/threonine kinases, which are involved in a wide range of cellular processes, including cell cycle regulation, apoptosis, and differentiation. PKC plays a key role in signal transduction pathways that influence cell proliferation and survival. Inhibiting PKC can lead to changes in cell cycle progression, making these inhibitors valuable in research related to cancer, neurobiology, and cardiovascular diseases. At CymitQuimica, we provide a diverse selection of high-quality PKC inhibitors to support your research in signal transduction, cell cycle regulation, and therapeutic development.
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CMPD101
CAS:865608-11-3
CMPD101 is a membrane-permeable small-molecule inhibitor of GRK2/3 (IC50: 18 nM and 5.4 nM).
Formula:
C24H21F3N6O
Purity:
98.34% - 99.01%
Color and Shape:
Solid
Molecular weight:
466.46
Ref: TM-T14989
| 1mg | 65.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 193.00 € | ||
| 25mg | 389.00 € | ||
| 50mg | 582.00 € | ||
| 1mL*10mM (DMSO) | 130.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
N-Desmethyltamoxifen hydrochloride
CAS:15917-65-4
N-Desmethyltamoxifen hydrochloride is the major tamoxifen metabolite in humans.
Formula:
C25H28ClNO
Purity:
99.15%
Color and Shape:
Solid
Molecular weight:
393.95
Ref: TM-T12148
| 1mg | 41.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 220.00 € | ||
| 50mg | 332.00 € | ||
| 100mg | 498.00 € | ||
| 500mg | 1,049.00 € | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
A-3 hydrochloride
CAS:78957-85-4
A-3 hydrochloride: potent, reversible kinase antagonist; permeable; inhibits PKC, CKI, PKA, CKII, MLCK; Ki: 4.3-80 …
Formula:
C12H14Cl2N2O2S
Purity:
99.32%
Color and Shape:
Solid
Molecular weight:
321.22
Ref: TM-T14069
| 1mg | 35.00 € | ||
| 5mg | 68.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 278.00 € | ||
| 100mg | 445.00 € | ||
| 500mg | 920.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Delcasertib
CAS:949100-39-4
Delcasertib (KAI-9803) is a potent and selective inhibitor of δ-protein kinase C (δPKC).
Formula:
C120H199N45O34S2
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
2880.28
Ref: TM-T11740
| 1mg | 198.00 € | ||
| 5mg | 503.00 € | ||
| 10mg | 723.00 € | ||
| 25mg | 1,100.00 € | ||
| 50mg | 1,505.00 € | ||
| 100mg | 2,032.00 € | ||
| 1mL*10mM (DMSO) | 1,680.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Mitoxantrone dihydrochloride
CAS:70476-82-3
Mitoxantrone dihydrochloride (NSC-301739) is an anthracenedione antibiotic with antineoplastic activity. Mitoxantrone is a type II …
Formula:
C22H30Cl2N4O6
Purity:
100% - 99.85%
Color and Shape:
Blue-Black Solid From Water Ethanol Solid
Molecular weight:
517.4
Ref: TM-T0158
| 50mg | 54.00 € | ||
| 100mg | 78.00 € | ||
| 500mg | 170.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Bisindolylmaleimide VIII acetate
CAS:138516-31-1
Bisindolylmaleimide VIII acetate is a selective PKC inhibitor with an IC50 of 158 nM in …
Formula:
C26H26N4O4
Purity:
99.27%
Color and Shape:
Solid
Molecular weight:
458.51
Ref: TM-T10549
| 1mg | 46.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 292.00 € | ||
| 50mg | 424.00 € | ||
| 100mg | 592.00 € | ||
| 1mL*10mM (DMSO) | 133.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
K-252c
CAS:85753-43-1
K-252c is a staurosporine analog isolated from Nocardiopsis sp.
Formula:
C20H13N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
311.34
Ref: TM-T15638
| 5mg | 809.00 € | ||
| 10mg | 1,404.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
SAMβA TFA
SAMβA TFA, a selective antagonist of Mfn1-βIIPKC association conjugated to the cell permeable peptide TAT47-57, …
Formula:
C50H73N17O16·xC2HF3O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1168.22 (free acid)
Ref: TM-T78220
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Protein Kinase C (19-31)
CAS:121545-65-1
Protein Kinase C (19-31), a PKC inhibitor derived from PKCa, has a serine at position …
Formula:
C67H118N26O16
Purity:
98%
Color and Shape:
Lyophilized Powder
Molecular weight:
1543.82
Ref: TM-TP1053
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 7 Jan 2025
LY 379196
LY 379196, a potent PKC-β inhibitor (IC 50: 50 nM for PKC βI and 30 …
Formula:
C30H34N4O5S
Color and Shape:
Liquid
Molecular weight:
562.68
Ref: TM-T89929
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 7 Jan 2025
K-252b
CAS:99570-78-2
K-252b, an indolocarbazole derived from the actinomycete Nocardiopsis, functions as a protein kinase C (PKC) …
Formula:
C26H19N3O5
Purity:
98%
Color and Shape:
Ready-To-Use Solution
Molecular weight:
453.45
Ref: TM-T15637
| 1mg | 795.00 € | ||
| 500µg | 463.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Fasudil
CAS:103745-39-7
Fasudil (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.
Formula:
C14H17N3O2S
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
291.37
Ref: TM-T1606
| 50mg | 39.00 € | ||
| 100mg | 49.00 € | ||
| 200mg | 67.00 € | ||
| 500mg | 104.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
1-Oleoyl-2-acetyl-sn-glycerol
CAS:86390-77-4
1-Oleoyl-2-acetyl-sn-glycerol (1-oleoyl-2-acetyl-glycerol) is a PKC activator that induces superoxide production.
Formula:
C23H42O5
Color and Shape:
Liquid
Molecular weight:
398.58
Ref: TM-T40972
| 5mg | 140.00 € | ||
| 10mg | 188.00 € | ||
| 25mg | 367.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Bisindolylmaleimide III
CAS:137592-43-9
Bisindolylmaleimide III is a potent and selective inhibitor of protein kinase C (PKC).Bisindolylmaleimide III selectively …
Formula:
C23H20N4O2
Purity:
98.6%
Color and Shape:
Liquid
Molecular weight:
384.43
Ref: TM-T77628
| 5mg | 77.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 399.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
PKCiota-IN-2
CAS:2230055-52-2
PKCiota-IN-2 selectively inhibits PKC-ι (IC50=2.8nM) and also blocks PKC-α, ε (IC50s=71nM, 350nM).
Formula:
C24H21N5O
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
395.46
Ref: TM-T9863
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 775.00 € | ||
| 100mg | 1,040.00 € | ||
| 1mL*10mM (DMSO) | 278.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Cercosporin
CAS:35082-49-6
Cercosporin, produced by the plant pathogen Cercospora kikuchii and the elsinochromes, is a potent photosensitizer …
Formula:
C29H26O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
534.51
Ref: TM-T13605
| 5mg | To inquire |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Protein Kinase C (19-31) (TFA)(121545-65-1,free)
Protein Kinase C (19-31) TFA is a serine-modified PKCa-derived inhibitor for testing PKC activity.
Formula:
C69H119F3N26O18
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1657.84
Ref: TM-TP1052
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 7 Jan 2025
20-HETE
CAS:79551-86-3
20-HETE is a CYP450 product, vasoconstrictor, modulates K+ channels, affects NADPH, ROS, NF-κB, NO synthase, …
Formula:
C20H32O3
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
320.47
Ref: TM-T14021
| 1mg (312.04μM*10mL in Ethanol) | 1,107.00 € | ||
| 5mg (312.04μM*50mL in Ethanol) | 2,263.00 € | ||
| 100μg (312.04μM*1mL in Ethanol) | 460.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Psychosine
CAS:2238-90-6
Psychosine (Galactosylsphingosine) is a PKC inhibitor, and is highly cytotoxic, inducing cell death in a …
Formula:
C24H47NO7
Purity:
98%
Color and Shape:
White Powder
Molecular weight:
461.63
Ref: TM-T21260
| 1mg | 214.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
(8R)-8-Hydroxyepoxyboetirane A
(8R)-8-Hydroxyepoxyboetirane A is a neuroactivating compound that interacts with PKCδ-C1B. This compound binds into the …
Ref: TM-T200548
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 7 Jan 2025
