Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(229 products)
- Annexin A(16 products)
- Aromatase(23 products)
- Estrogen/progestogen Receptor(66 products)
- GPR(1 products)
- Glucocorticoid Receptor(164 products)
- LHRH(2 products)
- Opioid Receptor(327 products)
- Prostaglandin Receptor(122 products)
- RAAS(89 products)
- Reductase(51 products)
- Somatostatin(57 products)
- Thyroid hormone receptor(THR)(34 products)
- Vasopressin Receptor(48 products)
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Found 3419 products of "Endocrinology/Hormones"
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LY2623091
CAS:LY2623091, a mineralocorticoid receptor antagonist, is utilized in treating refractory hypertension. It demonstrates CYP3A4-dependent clearance and exhibits synergistic effects when combined with CYP3A4 inhibitors.Formula:C30H30FN5O3Color and Shape:SolidMolecular weight:527.59pTH (1-37) (human)
CAS:pTH (1-37) human fragment boosts cAMP, alkaline phosphatase, growth, and BMD, potential for osteoporosis research.Formula:C195H316N58O54S2Color and Shape:SolidMolecular weight:4401.08BIBS 39
CAS:BIBS 39 is a new nonpeptide angiotensin II (AII) receptor antagonist.Formula:C32H36N4O3Purity:99.28%Color and Shape:SolidMolecular weight:524.65β-Lipotropin (61-69)
CAS:β-Lipotropin (61-69) is a potent opioid agonist [1] [2] .Formula:C45H66N10O15SMolecular weight:1019.13PL-017 TFA
PL-017 TFA: μ opioid agonist, IC50 5.5 nM, long-lasting analgesia in rats.Formula:C31H38F3N5O7Molecular weight:649.66(Tyr36)-pTH-Related Protein (1-36) (human, mouse, rat)
CAS:'(Tyr36)-pTH-Related Protein (1-36) (human, mouse, rat), a peptide, functions as a ligand for parathyroid hormone (PTH) receptors [1].'Formula:C194H303N59O53Molecular weight:4309.85PROTAC ERα Degrader-10
CAS:PROTACERα Degrader-10 (Compound 160a) is an orally bioavailable ERα degrader with a DC50 of 0.37-1.1 nM in MCF7, T47D, and CAMA-1 cells. It demonstrates antitumor activity in mouse models.Formula:C45H49N5O4Molecular weight:723.9Kalata B7
CAS:Kalata B7, a cyclotide isolated from Oldenlandia affinis DC (Rubiaceae), possesses membrane-permeating capabilities and acts as a partial agonist of oxytocin- and vasopressin V1a-receptors [1] [2].Formula:C128H196N36O40S6Molecular weight:3071.53Acetalin-3
CAS:Acetalin-3 (Ac-RFMWMT-NH2) is a hexapeptide that acts as a μ opioid receptor antagonist, displaying high affinity for μ and κ3 opioid receptors, weak affinity for κ1 receptors, and no affinity for κ2 receptors [1].Formula:C42H61N11O8S2Molecular weight:912.13Axelopran sulfate
CAS:Axelopran sulfate is used in Oral Therapies for Opioid-induced Bowel Dysfunction in Patients with Chronic Noncancer Pain.Formula:C26H41N3O8SColor and Shape:SolidMolecular weight:555.68ErSO
CAS:ErSO is a selective activator of anticipatory unfolded protein response (UPR) via ERα receptor. ErSO can be used in studies about anti-cancer.Formula:C22H13F6NO3Purity:98.36%Color and Shape:SolidMolecular weight:453.33Ref: TM-T39980
500mgTo inquire1mg71.00€5mg161.00€1mL*10mM (DMSO)172.00€10mg250.00€25mg411.00€50mg577.00€100mg772.00€N-Acetylthyroxine
CAS:N-Acetylthyroxine is a kind of Thyroxine analogue for the treatment of diagnosing and treating diabetes.Formula:C17H13I4NO5Color and Shape:SolidMolecular weight:818.91Gridegalutamide
CAS:Gridegalutamide exhibits anti-androgen and anti-tumor activities.Formula:C41H45F3N8O5SColor and Shape:SolidMolecular weight:818.91Isomer-Turosteride
Isomer-Turosteride, a novel 5α-reductase inhibitor, reduces prostate DHT and has anticancer properties without raising T levels.Formula:C27H45N3O3Purity:98.94%Color and Shape:SolidMolecular weight:459.67Latanoprost acid
CAS:Latanoprost acid is a prostanoid receptor agonist that blocks RANKL and can be used to reduce intraocular pressure.Formula:C23H34O5Purity:97.96%Color and Shape:Pale Yellow OilMolecular weight:390.51Ref: TM-T15718
1mg54.00€5mg138.00€1mL*10mM (DMSO)152.00€10mg215.00€25mg429.00€50mg637.00€100mg874.00€200mg1,161.00€Neuropeptide AF (human) acetate
Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative,
Purity:99.89%Color and Shape:SoildA 779
CAS:A 779 is a potent antagonist of the G-protein-coupled receptor Mas, the Ang1-7 receptor, which is distinct from conventional AngII.Formula:C39H60N12O11Purity:98%Color and Shape:SolidMolecular weight:872.97CIMBA hydrochloride
CIMBA hydrochloride is a selective antagonist of the G protein-coupled estrogen receptor (GPER). It can be utilized in research related to cholesterol gallstone disease in women.Color and Shape:Odour SolidTyr-W-MIF-1
CAS:Tyr-W-MIF-1, an opioid tetrapeptide, exhibits both opiate and antiopiate activities, and has been demonstrated to induce analgesia [1] [2] [5].Formula:C27H32N6O5Molecular weight:520.58SR-29065
CAS:SR-29065 is a REV-ERBα agonist that represses BMAL1 transcription and is used to study circadian regulation, cancer, and autoimmune disease mechanisms.Formula:C24H24F6N2O2SPurity:97.24% - 98.42%Color and Shape:Odour SolidMolecular weight:518.52XOMA-213
XOMA-213 (LFA-102; X213) is a human monoclonal antibody (mAb) that specifically targets the PRLR/Prolactin Receptor. It inhibits hPRL-dependent growth of BaF3/hPRLR cells with an EC50 of 0.5 μg/mL. In models such as the Nb2-11-luc xenograft mouse and the DMBA-induced rat breast cancer model, XOMA-213 effectively suppresses PRLR signaling and tumor growth. This compound is applicable in research focused on breast cancer, hyperprolactinemia, and prostate cancer.Nesvacumab
CAS:Nesvacumab (REGN910) is a fully human monoclonal antibody targeting Angiopoietin 2 (Ang2), which can be used for studying advanced solid tumors.Purity:98.7% (SDS-PAGE); 95.7% (SEC-HPLC) - 99.11% (SEC-HPLC)Color and Shape:LiquidMolecular weight:144.84 kDa3-Iodothyronamine hydrochloride
CAS:3-Iodothyronamine hydrochloride, Thyroid hormone derivative, activates TAAR1, induces hypothermia, for endocrine/metabolic research.Formula:C14H15ClINO2Color and Shape:SolidMolecular weight:391.63UFP-101 acetate
UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.
Formula:C84H142N32O23Purity:95.92%Color and Shape:SolidMolecular weight:1968.23difelikefalin acetate(1024828-77-0 Free base)
CAS:is a ketone and a building block.
Formula:C38H57N7O8Purity:96.94%Color and Shape:SolidMolecular weight:739.9OX04528
CAS:OX04528 is an orally active and potent GPR84 biased agonist.OX04528 inhibits cAMP signaling and may be useful in cancer research.Formula:C16H13F6NO2Purity:99.74%Color and Shape:SoildMolecular weight:365.27CTOP acetate
CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.Formula:C52H71N11O13S2Purity:99.87%Color and Shape:SoildMolecular weight:1122.32BMS-903452
CAS:BMS-903452: potent GPR119 agonist, EC50 = 14 nM, treats rodent diabetes, no P450 inhibition, safe for liver cells.Formula:C21H19Cl2FN4O4SPurity:98.69% - 99.76%Color and Shape:SolidMolecular weight:513.37Ref: TM-T67791
1mg95.00€5mg207.00€1mL*10mM (DMSO)244.00€10mg295.00€25mg444.00€50mg600.00€100mg810.00€200mg1,063.00€Nociceptin (1-13), amide
CAS:Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrainFormula:C61H100N22O15Purity:98%Color and Shape:SolidMolecular weight:1381.59Alunacedase alfa
CAS:Alunacedase alfa (APN-01) is an angiotensin-converting enzyme 2 with antiviral activity.Purity:99.1% (SDS-PAGE); 99.9% (SEC-HPLC) - 99.1% (SDS-PAGE); 99.9% (SEC-HPLC)Color and Shape:LiquidMolecular weight:85.03 kDaDuP 747 HCl
CAS:DuP 747 HCl is a selective kappa agonist with analgesic activity.DuP 747 consists of two conformations.Formula:C24H29Cl3N2O2Purity:99.85%Color and Shape:SoildMolecular weight:483.86Urotensin II, mouse TFA (9047-55-6 free base)
Urotensin II, mouse TFA is an endogenous ligand for the orphan GPR14 or SENR. It is a potent vasoconstrictor.Formula:C78H101N18F3O21S2Purity:98%Color and Shape:SolidMolecular weight:1747.88SNC 80
CAS:SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 nM), with analgesic and antidepressant potential.Formula:C28H39N3O2Purity:99.65%Color and Shape:SolidMolecular weight:449.63NH-3
CAS:NH-3, an orally active THR antagonist with a 55 nM IC50, blocks thyroid hormone binding and cofactor recruitment.Formula:C28H27NO6Purity:97.79% - 99.40%Color and Shape:SolidMolecular weight:473.52Ref: TM-T40548
1mg207.00€1mL*10mM (DMSO)467.00€5mg520.00€10mg750.00€25mg1,144.00€50mg1,521.00€100mg2,062.00€500mg4,159.00€GPCR agonist-2
CAS:GPCR agonist-2 (4-(Cyclopropylamino)-3-nitrobenzoic acid) is an agonist of the orphan human GPCR GPR109B.Formula:C10H10N2O4Purity:99.96%Color and Shape:SolidMolecular weight:222.215(R)-15-methyl Prostaglandin D2
CAS:15(R)-15-methyl Prostaglandin D2 (15(R)15methyl PGD2) is a synthetic analog of PGD2 and a CRTH2/DP2 receptor agonist.Formula:C21H34O5Color and Shape:SolidMolecular weight:366.49β-Endorphin (6-31), human
CAS:β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid receptors.Formula:C131H218N34O40Purity:98%Color and Shape:SolidMolecular weight:2909.38BPR1M97
CAS:BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.Formula:C18H18Cl2N2OPurity:98.78% - 99.95%Color and Shape:SolidMolecular weight:349.25LY255582
CAS:LY255582 is a selective centrally active opioid receptor antagonist with high affinity for mu, delta and kappa receptors with Ki of 0.4 nM, 5.2, 2.0 nM,Formula:C22H35NO2Purity:98%Color and Shape:SolidMolecular weight:345.52DPDPE
CAS:DPDPE is selective δ-opioid receptor agonist peptide.Formula:C30H39N5O7S2Purity:98%Color and Shape:SolidMolecular weight:645.79Deltorphin
CAS:Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.Formula:C44H62N10O10S2Purity:98.96%Color and Shape:SolidMolecular weight:955.15[D-Ala2]leucine-enkephalin acetate
[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study the signaling pathway ofFormula:C31H43N5O9Purity:98%Color and Shape:SolidMolecular weight:629.65β-Endorphin (1-27) (human) acetate
β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.
Formula:C141H221N33O42SPurity:96.52%Color and Shape:SolidMolecular weight:3082.52[Orn5]-URP acetate
[Orn5]-URP acetate is an effective and selective Urotensin-II receptor (UT) antagonist (pEC50 = 7.24). [Orn5]-URP exhibits no agonist activity.Formula:C50H66N10O12S2Purity:98.4300%Color and Shape:SolidMolecular weight:1063.25AT-121 hydrochloride
CAS:AT-121 hydrochloride: dual nociception/mu-opioid agonist, Ki 3.67/16.49 nM, safe, non-addictive pain reliever with analgesic effects.Formula:C24H39ClN4O3SPurity:97.28% - >99.99%Color and Shape:SolidMolecular weight:499.11Dermorphin
CAS:Dermorphin is agonist of μ-opioid receptor (MOR) agonist.Formula:C40H50N8O10Purity:98.82%Color and Shape:SolidMolecular weight:802.87[Orn8]-Urotensin II acetate
[Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.Formula:C65H87N13O20S2Purity:98.63%Color and Shape:SolidMolecular weight:1434.59[(pF)Phe4]Nociceptin(1-13)NH2 acetate
[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31.
Formula:C63H103FN22O17Purity:98.03%Color and Shape:SolidMolecular weight:1459.63(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin
CAS:(d(CH2)51,Tyr(Me)2, Orn8)-Oxytocin (OVT) is an antagonist of the oxytocin receptor that finds application in the study of neurological diseases [1].Formula:C48H74N12O12S2Purity:98%Color and Shape:SolidMolecular weight:1075.3Deltorphin acetate
Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioidFormula:C46H66N10O12S2Purity:98.93%Color and Shape:SolidMolecular weight:1015.21Ref: TM-T20166L
1mg175.00€5mg394.00€10mg590.00€25mg1,060.00€50mg1,591.00€100mg2,387.00€200mg3,580.00€Leumorphin, human
CAS:Leumorphin, human, is a potent agonist of the kappa opioid receptor (κ opioid receptor) and inhibits the contraction of the guinea pig ileum's myenteric plexus-Formula:C150H224N42O46Purity:98%Color and Shape:SolidMolecular weight:3351.64AH 7563
CAS:AH 7563 is structurally classified as an opioid compound with analgesic properties. In mice, its ED50 for pain relief was 15.3 mg/kg when administered orally in the Phenylquinone test, and 15.5 mg/kg when injected subcutaneously in the Hot plate test.Formula:C16H24N2OColor and Shape:SolidMolecular weight:260.38U-48520
CAS:U-48520 is an agonist of the μ-opioid receptor (μ-opioid receptor) with an EC50 of 1561 nM.Formula:C16H23ClN2OColor and Shape:SolidMolecular weight:294.82(-)-9-Hydroxycorynantheidine
CAS:(-)-9-Hydroxycorynantheidine (9-O-Desmethyl mitragynine) is a demethylated analog of Mitragynine, functioning as a selective and partial agonist for the μ-opioid receptor (μ-opioid receptor). This compound inhibits electrically stimulated twitch contractions in the guinea pig ileum.Formula:C22H28N2O4Color and Shape:SolidMolecular weight:384.47MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.Formula:C37H47Cl2N5O3Purity:98%Color and Shape:SolidMolecular weight:680.71WAY-298630
CAS:Fluorophenoxy benzimidazole, a CRTH2 blocker, IC50 < 10 μM for rhinitis, COPD, arthritis, eczema, conjunctivitis.Formula:C17H15FN2O3SPurity:97.84%Color and Shape:SolidMolecular weight:346.38Pro8-Oxytocin TFA
Pro8-Oxytocin TFA, a modified oxytocin (OXT) ligand, exhibits greater potency and efficacy than the standard mammalian OXT ligand, Leu8-Oxytocin, at primateFormula:C42H62N12O12S2·xC2HF3O2Purity:98%Color and Shape:SolidFluorphine
CAS:Fluorphine, an analog of Brorphine, binds to the μ-opioid receptor (MOR) with a Ki of 12.5 nM. It exhibits GTPγS binding activity with an EC50 of 75 nM and β-arrestin 2 recruitment activity with an EC50 of 377 nM, and it also has respiratory depressive effects.Formula:C20H22FN3OColor and Shape:SolidMolecular weight:339.41Orphine
CAS:Orphine is an opioid compound that can amplify the antinociceptive effects reduced by naloxone in mice.Formula:C20H23N3OColor and Shape:SolidMolecular weight:321.42PF-06478939 TFA
PF-06478939 TFA is a peptide that acts as a non-brain-penetrating agonist at the oxytocin (OT) and vasopressin receptors, exhibiting EC50 values of 0.01 nM andFormula:C78H134N14O22S2·xC2HF3O2Purity:98%Color and Shape:Solid(Val3,Pro8)-Oxytocin
CAS:(Val3,Pro8)-Oxytocin functions primarily as a Gq-dependent pathway agonist and exhibits secondary activity as a reduced efficacy agonist for β-arrestinFormula:C41H60N12O12S2Purity:98%Color and Shape:SolidMolecular weight:977.12CSD-CH2(1,8)-NH2
CSD-CH2(1,8)-NH2 is a selective and competitive kappa-opioid receptor (KOR) antagonist with a K i of 6.8 nM.Formula:C76H125N25O15S2Purity:98%Color and Shape:SolidMolecular weight:1693.09DALDA TFA
DALDA TFA is a potent, μ-opioid receptor agonist exhibiting high selectivity and an affinity constant (K i) of 1.69 nM.Formula:C30H45N9O5·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:611.74 (free base)AH 8529
CAS:AH 8529 is an orally active opioid compound with analgesic properties.Formula:C16H23ClN2OColor and Shape:SolidMolecular weight:294.82N-Phenethylnoroxymorphone
CAS:N-Phenethylnoroxymorphone is an opioid compound that can enhance morphine-induced analgesia in rats. It is used in the research of neurological disorders.Formula:C24H25NO4Color and Shape:SolidMolecular weight:391.46KOR agonist 3
KOR agonist 3 (Compound 5) is an agonist of the κ opioid receptor (κOR) with an EC50 of 0.88 nM. It also exhibits some activation of μOR, with an EC50 of 720 nM. However, KOR agonist 3 does not activate δOR at concentrations below 1 μM. Its ability to recruit β-Arrestin-2 is lower than that of U50488.Formula:C24H24N2O3Color and Shape:SolidMolecular weight:388.46Pro8-Oxytocin
CAS:Pro8-Oxytocin, a modified oxytocin (OXT) ligand, elicits more potent and efficacious responses at primate OXTR and induces stronger behavioral effects comparedFormula:C42H62N12O12S2Purity:98%Color and Shape:SolidMolecular weight:991.14Corynantheidine
CAS:Corynantheidine ((-)-Corynantheidine) is a partial agonist of the mu opioid receptor (MOR) and demonstrates MOR-dependent analgesic effects in mice.Formula:C22H28N2O3Color and Shape:SolidMolecular weight:368.47AH 7959
CAS:AH 7959 is an orally active N-substituted cyclohexylmethylbenzamide compound that exhibits analgesic properties. In mice, the ED50 for oral and subcutaneous administration of AH 7959 exceeds 100 mg/kg.Formula:C19H26Cl2N2OColor and Shape:SolidMolecular weight:369.33Dynorphin B (1-9)
CAS:Dynorphin B (1-9), a neuropeptide and the N-terminal cleavage product of dynorphin B, has its formation inhibited by N-ethylmaleimide (NEM), a non-selectiveFormula:C54H78N16O12Purity:98%Color and Shape:SolidMolecular weight:1143.3AP-238
CAS:AP-238 is a novel synthetic opioid (NSO) that acts as an agonist for the μ-opioid receptor (MOR), with an EC50 of 248 nM. Additionally, AP-238 exhibits analgesic properties.Formula:C18H26N2OColor and Shape:SolidMolecular weight:286.414-Hydroxy-1-(2-phenylethyl)piperidine
CAS:4-Hydroxy-1-(2-phenylethyl)piperidine is a synthetic ligand for muscarinic acetylcholine receptors (mAChR) or non-opioid intracellular sigma-1 receptors (σ1 receptors). It serves as a metabolite of the opioid compounds furanylfentanyl and 4-fluoroisobutyryl fentanyl (FIBF).Formula:C13H19NOColor and Shape:SolidMolecular weight:205.3β-Endorphin (1-27) (human)
CAS:β-Endorphin (1-27) (human) is an opioid antagonist that selectively binds to μ-, δ-, and κ-opioid receptors, with dissociation constants (Kis) of 5.31, 6.17,Formula:C139H217N33O40SPurity:98%Color and Shape:SolidMolecular weight:3022.47PF-06655075 TFA
PF-06655075 (TFA) is the trifluoroacetic acid (TFA) salt of PF-06655075, a novel, non-brain-penetrant oxytocin receptor agonist that exhibits enhancedPurity:98%Color and Shape:Odour Solid(1S,2R)-2-PCCA
(1S,2R)-2-PCCA is a novel and potent small molecule GPR88 receptor agonist with an EC50 value of 3 nM in the non-cellular system and 603 nM in the cellularFormula:C30H39Cl2N3OPurity:99.91%Color and Shape:SoildMolecular weight:528.56Piperidylthiambutene hydrochloride
CAS:Piperidylthiambutene hydrochloride is an opioid compound that exhibits analgesic effects in animal models.Formula:C17H22ClNS2Color and Shape:SolidMolecular weight:339.95DBPR116
CAS:DBPR116 is a prodrug of BPRMU191 that can penetrate the blood-brain barrier. It significantly enhances the delivery efficiency of drugs targeting the central nervous system. When combined with the antagonist Naltrexone, DBPR116 demonstrates superior safety and analgesic effects compared to morphine in various in vivo pharmacological studies, including thermal pain models, cancer pain models, constipation, sedation, psychological dependence, heart rate, and respiratory frequency. As a strategy for peripheral administration, DBPR116 effectively alleviates pain while reducing adverse effects, showing promise as a safer opioid analgesic.Formula:C19H18FNO3SColor and Shape:SolidMolecular weight:359.42PU-WS13 hydrobromide
PU-WS13 hydrobromide is a GRP94 inhibitor with anti-inflammatory activity and inhibits the proliferation of M2-like macrophages in mouse TNBC tumors.Formula:C17H21BrCl2N6SPurity:99.99%Color and Shape:SoildMolecular weight:492.26R-6890
CAS:R-6890 is an opioid compound with analgesic properties.Formula:C21H24ClN3OColor and Shape:SolidMolecular weight:369.89AH 8532
CAS:AH 8532 is an opioid compound with analgesic effects and is effective in inhibiting the quinone-induced writhing response in mice, with an oral ED50 of 16 mg/kg.Formula:C16H23ClN2OColor and Shape:SolidMolecular weight:294.82PF-06478939
PF-06478939 is a peptide that functions as an agonist at the oxytocin (OT) receptor and vasopressin receptor without crossing the blood-brain barrier.Formula:C78H134N14O22S2Purity:98%Color and Shape:SolidMolecular weight:1684.11[DPro10] Dynorphin A (1-11)acetate,porcine
[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.Formula:C65H107N21O15Purity:99.59%Color and Shape:SoildMolecular weight:1422.7PF-06655075
PF-06655075 is a novel, non-brain-penetrant oxytocin receptor agonist that demonstrates enhanced selectivity for the oxytocin receptor and substantially
Formula:C75H130N14O22S2Purity:98%Color and Shape:SolidMolecular weight:1644.05Bazedoxifene hydrochloride
CAS:Bazedoxifene hydrochloride (TSE 424 hydrochloride) is an estrogen receptor modulator and an inhibitor of IL-6/GP130 protein interaction.Formula:C30H35ClN2O3Purity:98.74%Color and Shape:SolidMolecular weight:507.06Ref: TM-T6404
1mg60.00€5mg138.00€10mg240.00€1mL*10mM (DMSO)240.00€25mg374.00€50mg673.00€100mg938.00€500mg1,872.00€Camizestrant TFA
Camizestrant TFA (AZD-9833 TFA) is a potent and orally active antagonist of estrogen receptor (ER).Formula:C26H29F7N6O2Purity:99.85%Color and Shape:SoildMolecular weight:590.54Ref: TM-T11237L
1mg65.00€5mg150.00€1mL*10mM (DMSO)158.00€10mg215.00€25mg338.00€50mg452.00€100mg662.00€200mg948.00€Valsartan Methyl Ester
CAS:Valsartan Methyl Ester is a potent angiotensin II receptor antagonist, IC50= 0.06uM.
Formula:C25H31N5O3Purity:99.54%Color and Shape:SolidMolecular weight:449.55ER ligand-2
ER ligand-2 is a ligand for ER. It can be used in the synthesis of PROTAC ER Degrader-11.Formula:C20H23BrOColor and Shape:SolidMolecular weight:359.3PROTAC ER Degrader-11
CAS:PROTA CER Degrader-11 (Example 26-1) is an effective degrader of PROTA CER with an IC50 of 0.66 nM. It plays a crucial role in cancer research.Formula:C43H53N5O4Color and Shape:SolidMolecular weight:703.914'-Hydroxytamoxifen TFA
4'-Hydroxytamoxifen TFA, a salt form of a metabolite of Tamoxifen, demonstrates higher affinity for ER compared to Tamoxifen itself. This compound induces non-apoptotic cytotoxicity in human endometrial adenocarcinoma cells.Formula:C28H30F3NO4Color and Shape:SolidMolecular weight:501.54ERD-1233
ERD-1233 is an effective oral PROTAC degrader of the estrogen receptor (estrogen receptor) with a DC50 of 0.9 nM. It plays a crucial role in research involving ER+ breast cancer.Formula:C49H53N5O6Color and Shape:SolidMolecular weight:807.986α-Methylprednisolone 21-hemisuccinate sodium salt
CAS:6α-Methylprednisolone 21-hemisuccinate sodium salt (Asmacortone), a water-soluble ester, is used for allergic, cardiac, and hypoxic emergencies.Formula:C26H33NaO8Purity:99.65%Color and Shape:Lyophilized PowderMolecular weight:496.53Protirelin Acetate
CAS:Protirelin Acetate (TRH Acetate) is a thyrotropin-releasing hormone, stimulating the release of thyrotropin and prolactin from the anterior pituitary.Formula:C16H22N6O4C2H4O2Purity:96.17%Color and Shape:SolidMolecular weight:452.46Dehydroisoandrosterone 3-acetate
CAS:Dehydroisoandrosterone 3-acetate (Prasterone acetate) is a primary C19 steroid generated by the adrenal cortex.Formula:C21H30O3Purity:>99.99%Color and Shape:SolidMolecular weight:330.46RD162
CAS:RD162 is a non-steroidal antiandrogen (NSAA) specifically binding to the androgen receptor (AR).Formula:C22H16F4N4O2SPurity:99.71%Color and Shape:SolidMolecular weight:476.45Ref: TM-T21740
1mg44.00€5mg113.00€1mL*10mM (DMSO)137.00€10mg177.00€25mg371.00€50mg553.00€100mg788.00€Premarin
CAS:Premarin (Estrone 3-sulfate) is an an estrogen sulfate with neuroprotective actions during traumatic brain injury.Formula:C18H22O5SPurity:99.74%Color and Shape:SoildMolecular weight:350.43Ref: TM-T36857L
1mg175.00€5mg394.00€1mL*10mM (DMSO)413.00€10mg582.00€25mg888.00€50mg1,243.00€100mg1,674.00€Benazeprilat
CAS:Benazeprilat(CGS 14831) is an orally active active metabolite of Benazepril.Benazeprilat has potent antihypertensive activity and can be used in combinationFormula:C22H24N2O5Purity:99.23%Color and Shape:Crystalline SolidMolecular weight:396.44Norethynodrel
CAS:Norethynodrel, a synthetic hormone, mimics progesterone, treats uterine bleeding/endometriosis, and is used with mestranol as a contraceptive.Formula:C20H26O2Purity:98%Color and Shape:Crystals From Aqueous Methanol SolidMolecular weight:298.42Estetrol
CAS:Estetrol (Donesta), a fetal liver-synthesized estrogen, selectively modulates estrogen receptors and may ease menopausal symptoms.Formula:C18H24O4Purity:99.93%Color and Shape:SolidMolecular weight:304.38Ref: TM-T15248
1mg39.00€5mg84.00€1mL*10mM (DMSO)93.00€10mg130.00€25mg268.00€50mg462.00€100mg773.00€200mg1,044.00€ARD-266
CAS:ARD-266 is a PROTAC degrader based on the von Hippel-Lindau E3 ligase that induces the degradation of AR proteins and is useful in prostate cancer research.Formula:C52H59ClN6O7Purity:99.89%Color and Shape:SolidMolecular weight:915.514,4'-(Cyclohexylidenemethylene)diphenol
CAS:4,4'-(Cyclohexylidenemethylene)diphenol (Compound 2) is a symmetrical cyclic non-steroidal estrogen. It exhibits high binding affinity to estrogen receptors ERα and ERβ.Formula:C19H20O2Color and Shape:SolidMolecular weight:280.36
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