Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(229 products)
- Annexin A(16 products)
- Aromatase(23 products)
- Estrogen/progestogen Receptor(66 products)
- GPR(1 products)
- Glucocorticoid Receptor(164 products)
- LHRH(2 products)
- Opioid Receptor(327 products)
- Prostaglandin Receptor(122 products)
- RAAS(89 products)
- Reductase(51 products)
- Somatostatin(57 products)
- Thyroid hormone receptor(THR)(34 products)
- Vasopressin Receptor(48 products)
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Found 3419 products of "Endocrinology/Hormones"
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Deltorphin
CAS:Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.Formula:C44H62N10O10S2Purity:98.96%Color and Shape:SolidMolecular weight:955.15[D-Ala2]leucine-enkephalin acetate
[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study the signaling pathway ofFormula:C31H43N5O9Purity:98%Color and Shape:SolidMolecular weight:629.65β-Endorphin (1-27) (human) acetate
β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.
Formula:C141H221N33O42SPurity:96.52%Color and Shape:SolidMolecular weight:3082.52[Orn5]-URP acetate
[Orn5]-URP acetate is an effective and selective Urotensin-II receptor (UT) antagonist (pEC50 = 7.24). [Orn5]-URP exhibits no agonist activity.Formula:C50H66N10O12S2Purity:98.4300%Color and Shape:SolidMolecular weight:1063.25AT-121 hydrochloride
CAS:AT-121 hydrochloride: dual nociception/mu-opioid agonist, Ki 3.67/16.49 nM, safe, non-addictive pain reliever with analgesic effects.Formula:C24H39ClN4O3SPurity:97.28% - >99.99%Color and Shape:SolidMolecular weight:499.11Dermorphin
CAS:Dermorphin is agonist of μ-opioid receptor (MOR) agonist.Formula:C40H50N8O10Purity:98.82%Color and Shape:SolidMolecular weight:802.87[Orn8]-Urotensin II acetate
[Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.Formula:C65H87N13O20S2Purity:98.63%Color and Shape:SolidMolecular weight:1434.59[(pF)Phe4]Nociceptin(1-13)NH2 acetate
[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31.
Formula:C63H103FN22O17Purity:98.03%Color and Shape:SolidMolecular weight:1459.63(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin
CAS:(d(CH2)51,Tyr(Me)2, Orn8)-Oxytocin (OVT) is an antagonist of the oxytocin receptor that finds application in the study of neurological diseases [1].Formula:C48H74N12O12S2Purity:98%Color and Shape:SolidMolecular weight:1075.3Deltorphin acetate
Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioidFormula:C46H66N10O12S2Purity:98.93%Color and Shape:SolidMolecular weight:1015.21Ref: TM-T20166L
1mg175.00€5mg394.00€10mg590.00€25mg1,060.00€50mg1,591.00€100mg2,387.00€200mg3,580.00€Leumorphin, human
CAS:Leumorphin, human, is a potent agonist of the kappa opioid receptor (κ opioid receptor) and inhibits the contraction of the guinea pig ileum's myenteric plexus-Formula:C150H224N42O46Purity:98%Color and Shape:SolidMolecular weight:3351.64AH 7563
CAS:AH 7563 is structurally classified as an opioid compound with analgesic properties. In mice, its ED50 for pain relief was 15.3 mg/kg when administered orally in the Phenylquinone test, and 15.5 mg/kg when injected subcutaneously in the Hot plate test.Formula:C16H24N2OColor and Shape:SolidMolecular weight:260.38U-48520
CAS:U-48520 is an agonist of the μ-opioid receptor (μ-opioid receptor) with an EC50 of 1561 nM.Formula:C16H23ClN2OColor and Shape:SolidMolecular weight:294.82(-)-9-Hydroxycorynantheidine
CAS:(-)-9-Hydroxycorynantheidine (9-O-Desmethyl mitragynine) is a demethylated analog of Mitragynine, functioning as a selective and partial agonist for the μ-opioid receptor (μ-opioid receptor). This compound inhibits electrically stimulated twitch contractions in the guinea pig ileum.Formula:C22H28N2O4Color and Shape:SolidMolecular weight:384.47MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.Formula:C37H47Cl2N5O3Purity:98%Color and Shape:SolidMolecular weight:680.71WAY-298630
CAS:Fluorophenoxy benzimidazole, a CRTH2 blocker, IC50 < 10 μM for rhinitis, COPD, arthritis, eczema, conjunctivitis.Formula:C17H15FN2O3SPurity:97.84%Color and Shape:SolidMolecular weight:346.38Pro8-Oxytocin TFA
Pro8-Oxytocin TFA, a modified oxytocin (OXT) ligand, exhibits greater potency and efficacy than the standard mammalian OXT ligand, Leu8-Oxytocin, at primateFormula:C42H62N12O12S2·xC2HF3O2Purity:98%Color and Shape:SolidFluorphine
CAS:Fluorphine, an analog of Brorphine, binds to the μ-opioid receptor (MOR) with a Ki of 12.5 nM. It exhibits GTPγS binding activity with an EC50 of 75 nM and β-arrestin 2 recruitment activity with an EC50 of 377 nM, and it also has respiratory depressive effects.Formula:C20H22FN3OColor and Shape:SolidMolecular weight:339.41Orphine
CAS:Orphine is an opioid compound that can amplify the antinociceptive effects reduced by naloxone in mice.Formula:C20H23N3OColor and Shape:SolidMolecular weight:321.42PF-06478939 TFA
PF-06478939 TFA is a peptide that acts as a non-brain-penetrating agonist at the oxytocin (OT) and vasopressin receptors, exhibiting EC50 values of 0.01 nM andFormula:C78H134N14O22S2·xC2HF3O2Purity:98%Color and Shape:Solid
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