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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3178 products of "Endocrinology/Hormones"

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  • Angiotensin amide
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    Angiotensin amide

    CAS:
    <p>Angiotensin amide, an octapeptide amide, can be used to increase blood pressure by vasoconstriction.</p>
    Formula:C49H70N14O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1031.17

    Ref: TM-TP2446

  • PROTAC ER Degrader-3
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    PROTAC ER Degrader-3

    CAS:
    <p>PROTAC ER Degrader-3 from patent WO2017201449A1 is a PAC synthesis intermediate for ADC/PROTAC antibody conjugates, boosting ERα degradation.</p>
    Formula:C71H77N7O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1220.434

    Ref: TM-T18607

  • UFP-101
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    UFP-101

    CAS:
    <p>Strong, selective NOP receptor antagonist with pKi=10.24; &gt;3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.</p>
    Formula:C82H138N32O21
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1908.19

    Ref: TM-TP2105

  • Biphalin TFA
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    Biphalin TFA

    CAS:
    <p>Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.</p>
    Formula:C46H56N10O10·xC2HF3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:909.00 (free base)

    Ref: TM-T80074

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    Antitumor agent-195

    <p>Antitumor agent-195 (compound 16c) is a dual-targeting agent that simultaneously targets STAT3 and NQO1. At a concentration of 1 μM, it significantly inhibits the phosphorylation of STAT3 at the Tyr705 site and effectively induces apoptosis in MDA-MB-231 and MDA-MB-468 breast cancer cells. As a substrate of NQO1, Antitumor agent-195 markedly increases ROS production, causing severe DNA damage in a dose-dependent manner. It also demonstrates strong antitumor properties in MDA-MB-231 xenograft models.</p>
    Formula:C22H22N2O4
    Color and Shape:Solid
    Molecular weight:378.42

    Ref: TM-T205391

  • TRV055 acetate
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    TRV055 acetate

    <p>TRV055 acetate is a ligand of angiotensin II type 1 receptor and stimulates cellular Gq-mediated signaling.</p>
    Formula:C44H61N9O11
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:892.01

    Ref: TM-T40220L

  • ARD-2585
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    ARD-2585

    CAS:
    <p>ARD-2585 is an orally active and selective androgen receptor PROTAC degrader with anticancer activity for the study of prostate cancer.</p>
    Formula:C41H43ClN8O5
    Color and Shape:Solid
    Molecular weight:763.28

    Ref: TM-T74141

  • BigLEN(mouse)
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    BigLEN(mouse)

    CAS:
    <p>GPR171 agonist from ProSAAS controls mouse appetite, reduces glutamate in paraventricular neurons via G protein.</p>
    Formula:C78H130N24O22
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1756.03

    Ref: TM-TP2073

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    (rel)-PROTAC ERRα Degrader-1

    <p>(rel)-PROTAC ERRα Degrader-1 is a relative configuration of PROTAC ERRα Degrader-1, which is an estrogen-related receptor alpha (ERRa) degrader.</p>
    Formula:C54H49Cl2F6N7O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1108.91

    Ref: TM-T18651

  • PROTAC ER Degrader-4
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    PROTAC ER Degrader-4

    CAS:
    <p>PROTAC ER Degrader-4 is a PROATC degrader of estrogen receptor (ER)(IC50 of 0.8 nM).</p>
    Formula:C53H67F3N6O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1005.2

    Ref: TM-T13839

  • GNE-274
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    GNE-274

    CAS:
    <p>GNE-274, akin to GDC-0927 but non-degrading, is a partial ER agonist in breast cancer, enhancing chromatin at ER sites, inhibiting ER-LBD.</p>
    Formula:C29H31NO4
    Color and Shape:Solid
    Molecular weight:457.57

    Ref: TM-T39916

  • 3-epi-25-hydroxy Vitamin D3
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    3-epi-25-hydroxy Vitamin D3

    CAS:
    <p>3-epi-25-hydroxy Vitamin D3 lowers serum PTH in male weanling rats at 0.5 and 1 IU/g doses; doesn't affect females.</p>
    Formula:C27H44O2
    Color and Shape:Solid
    Molecular weight:400.64

    Ref: TM-T35500

  • U-54494A hydrochloride
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    U-54494A hydrochloride

    CAS:
    <p>U-54494A hydrochloride is a benzamide derivative related to kappa opioid receptor agonists. U-54494A hydrochloride has anticonvulsant activity.</p>
    Formula:C18H25Cl3N2O
    Color and Shape:Solid
    Molecular weight:391.76

    Ref: TM-T36372

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    Antihypertensive agent 3

    <p>Antihypertensive agent 3 (compound 4a), an angiotensin II receptor 1 antagonist, demonstrates antihypertensive activity in spontaneously hypertensive rats (SHRs</p>
    Formula:C16H13NO4S
    Color and Shape:Solid
    Molecular weight:315.34

    Ref: TM-T79267

  • Methylprednisolone Acetate
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    Methylprednisolone Acetate

    <p>Methylprednisolone Acetate(Depo-Medrate) has the ability to inhibit oxygen free radicals and can be used to treat acute spinal cord injuries.</p>
    Formula:C24H32O6
    Purity:99.74%
    Color and Shape:Off-White Solid
    Molecular weight:416.51

    Ref: TM-T21338

  • Axelopran
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    Axelopran

    CAS:
    <p>Axelopran (TD-1211) treats opioid constipation; it's a potent, selective peripheral opioid blocker.</p>
    Formula:C26H39N3O4
    Color and Shape:Solid
    Molecular weight:457.61

    Ref: TM-T30236

  • SL910102
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    SL910102

    CAS:
    <p>SL910102 is a nonpeptide angiotensin antagonist of the AT1 receptor.</p>
    Formula:C30H30N6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:490.60

    Ref: TM-T16895

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    PTP1B/AKR1B1-IN-1

    <p>PTP1B/AKR1B1-IN-1 is a dual inhibitor targeting protein tyrosine phosphatase 1B (PTP1B) and aldose reductase (AKR1B1), exhibiting inhibitory potency with IC50s</p>
    Formula:C22H21NO4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:427.54

    Ref: TM-T78702

  • Myrciacetin
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    Myrciacetin

    CAS:
    <p>Myrciacetin from Rhododendron inhibits rat aldose reductase with IC50 of 13 μM.</p>
    Formula:C17H16O6
    Color and Shape:Solid
    Molecular weight:316.309

    Ref: TM-T39435

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    HINT1-IN-1

    <p>HINT1-IN-1 (compound 8) is an inhibitor of histidine triad nucleotide-binding protein 1 (HINT1) with a Ki of 1.14 μM. It influences the cross-regulation between μ-opioid receptors (MOR) and NMDA receptors (NMDAR).</p>
    Formula:C23H24N8O5
    Color and Shape:Solid
    Molecular weight:492.49

    Ref: TM-T205282