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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3180 products of "Endocrinology/Hormones"

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  • Estrone acetate
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    Estrone acetate

    CAS:
    <p>Estrone acetate (Hogival) is an estrogen derivative and an activator of estrogen receptors (ER). This compound can enhance breast development, stimulate the secretion of pituitary prolactin, and induce both the proliferation and activation of lactotrophs, evidenced by the reduction in prolactin storage granule size and the increase in the volume density of the rough endoplasmic reticulum and Golgi apparatus. Estrone acetate holds potential for endocrinological research and for investigating the mechanisms by which estrogen influences pituitary function, prolactin regulation, and breast tumor models.</p>
    Formula:C20H24O3
    Color and Shape:Solid
    Molecular weight:312.403

    Ref: TM-T206611

  • Androgen receptor degrader-5
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    Androgen receptor degrader-5

    CAS:
    <p>Androgen receptor degrader-5 (compound 14k) demonstrates superior capabilities, specifically in androgen receptor degradation and antiproliferative activity, showcasing its promising properties.</p>
    Formula:C29H25F4N5O2
    Color and Shape:Solid
    Molecular weight:551.53

    Ref: TM-T200197

  • ORIC-101
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    ORIC-101

    CAS:
    <p>ORIC-101 is a highly effective and selective glucocorticoid receptor antagonist (EC50: 5.6 nM). It also has anti-cancer activity.</p>
    Formula:C34H47NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:501.74

    Ref: TM-T16404

  • CymitQuimica logo
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    ERRγ agonist-1

    <p>ERRγ agonist-1 can be used in neuropsychological disorders research.</p>
    Formula:C17H21N5O
    Color and Shape:Solid
    Molecular weight:311.38

    Ref: TM-T60772

  • TRβ agonist 1
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    TRβ agonist 1

    CAS:
    <p>TRβ Agonist 1, a selective and mutation-sensitive thyroid hormone receptor β (TRβ) agonist, demonstrates an EC50 value of 21 nM.</p>
    Formula:C29H25FN2O8
    Color and Shape:Solid
    Molecular weight:548.52

    Ref: TM-T63876

  • Estrogen receptor antagonist 4
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    Estrogen receptor antagonist 4

    CAS:
    <p>Estrogen receptor antagonist 4 blocks ER, impacting cell growth and cancer research potential.</p>
    Formula:C23H29BF4N4O2
    Color and Shape:Solid
    Molecular weight:480.31

    Ref: TM-T63106

  • rel-SB-612111 hydrochloride
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    rel-SB-612111 hydrochloride

    CAS:
    <p>NOP receptor antagonist</p>
    Formula:C24H30Cl3NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.86

    Ref: TM-T23324

  • Androstatrione
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    Androstatrione

    CAS:
    <p>Androstatrione is an androgenic compound.</p>
    Formula:C19H26O3
    Color and Shape:Solid
    Molecular weight:302.41

    Ref: TM-T207371

  • JNJ-1250132
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    JNJ-1250132

    CAS:
    <p>JNJ-1250132 is a steroidal progesterone receptor modulator that inhibits binding of the receptor to DNA in vitro.</p>
    Formula:C33H41NO4
    Color and Shape:Solid
    Molecular weight:515.68

    Ref: TM-T27662

  • Metahexestrol
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    Metahexestrol

    CAS:
    <p>Metahexestrol is an inhibitor of the estrogen receptor (E2R) with antitumor activity. It significantly inhibits the proliferation of estrogen receptor-positive MCF-7 human breast cancer cell line with an ED50 of 1.0 μM. Additionally, Metahexestrol shows inhibitory activity in estrogen receptor-negative MDA-MB-231 cell lines, and its antiproliferative effect is not reversed by estrogen, suggesting that its mechanism may be partially independent of the E2R pathway. Metahexestrol is applicable in research on estrogen-dependent breast cancer.</p>
    Formula:C18H22O2
    Color and Shape:Solid
    Molecular weight:270.366

    Ref: TM-T206528

  • GC 14
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    GC 14

    CAS:
    <p>GC 14 is a selective thyroid hormone receptor antagonist, with IC50 values of 200 nM and 35 nM for hTRα and hTRβ, respectively.</p>
    Formula:C26H27NO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:449.5

    Ref: TM-T11376

  • LIT-001 free base
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    LIT-001 free base

    CAS:
    <p>LIT-001, a nonpeptide OT-R agonist, enhances mouse autism-like behavior, with EC50=55 nM and Ki=226 nM.</p>
    Formula:C28H33N7O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:531.67

    Ref: TM-T11856

  • GPR84 antagonist 3
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    GPR84 antagonist 3

    CAS:
    <p>Potent GPR84 antagonist 3 (compound 42), pIC50 8.28, inhibits GTPγS, with good pharmacokinetics.</p>
    Formula:C29H27N5O
    Color and Shape:Solid
    Molecular weight:461.56

    Ref: TM-T62918

  • Isotodesnitazene
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    Isotodesnitazene

    CAS:
    <p>Isotodesnitazene is an opioid compound that primarily targets the μ-opioid receptor (MOR). It exhibits EC50 values of 34.8 nM and 142 nM for MOR-βarr2 and MOR-mini-Gi, respectively. Isotodesnitazene can be utilized for research in opioid drugs.</p>
    Formula:C23H31N3O
    Color and Shape:Solid
    Molecular weight:365.51

    Ref: TM-T201840

  • Opioid receptor antagonist 1
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    Opioid receptor antagonist 1

    CAS:
    <p>Opioid receptor antagonist 1 (Compound 10) is an Orvinol-based antagonist of opioid receptors. It exhibits activity as an antagonist against the analgesic properties of morphine.</p>
    Formula:C24H29ClF3NO4
    Color and Shape:Solid
    Molecular weight:487.94

    Ref: TM-T204656

  • Sunobinop
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    Sunobinop

    CAS:
    <p>Sunobinop (S 117957) is an opioid receptor-like orphan receptor (ORL1) modulator.</p>
    Formula:C26H33N3O3
    Color and Shape:Solid
    Molecular weight:435.56

    Ref: TM-T62482

  • FL442
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    FL442

    CAS:
    <p>FL442 is an Androgen Receptor (AR) modulator. This compound exhibits potent inhibitory effects in AR-dependent prostate cancer cells, showing similar suppression efficiency to the traditional antiandrogen drugs Bicalutamide and Enzalutamide. It also maintains antiandrogen activity against the Enzalutamide-resistant AR mutant F876L. The pharmacokinetic properties of FL442 in mice reveal a longer half-life (8 hours), excellent targeting (prostate tissue), and metabolic stability. Additionally, it is effective at inhibiting LNCaP tumor growth at low plasma concentrations (30 ng/mL).</p>
    Formula:C15H13F3N2O
    Color and Shape:Solid
    Molecular weight:294.27

    Ref: TM-T200138

  • Anilopam
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    Anilopam

    CAS:
    <p>Anilopam is an opioid analgesic belonging to the benzazepine class and acts as an agonist at opioid receptors.</p>
    Formula:C20H26N2O
    Color and Shape:Solid
    Molecular weight:310.43

    Ref: TM-T201609

  • 22-Thiocyanatosalvinorin A
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    22-Thiocyanatosalvinorin A

    CAS:
    <p>22-Thiocyanatosalvinorin A (RB-64) is a potent selective agonist for the kappa-opioid receptor, exhibiting an EC50 value of 0.077 nM.</p>
    Formula:C24H27NO8S
    Color and Shape:Solid
    Molecular weight:489.54

    Ref: TM-T201845

  • CH5447240
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    CH5447240

    CAS:
    <p>CH5447240: potent hPTHR1 agonist, treats Hypoparathyroidism, EC50 12 nM, 55% oral bioavailability, raises rat serum calcium.</p>
    Formula:C26H39N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:517.68

    Ref: TM-T25234