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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3183 products of "Endocrinology/Hormones"

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  • PROTAC ER Degrader-3

    CAS:
    <p>PROTAC ER Degrader-3 from patent WO2017201449A1 is a PAC synthesis intermediate for ADC/PROTAC antibody conjugates, boosting ERα degradation.</p>
    Formula:C71H77N7O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1220.434
  • T4-ATA (S-isomer)


    <p>T4-ATA S-isomer, the active form of the thyroid hormone, represents the S-isomer of T4-ATA.</p>
    Formula:C19H15I4NO6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:893.01
  • TRV-120027

    CAS:
    <p>TRV120027: β-arrestin-1-biased agonist, angiotensin II type 1 receptor, reduces vasoconstriction, boosts heart muscle contraction.</p>
    Formula:C43H67N13O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:926.09
  • Frakefamide TFA


    <p>Frakefamide TFA: potent, peripherally active μ-opioid agonist; doesn't cross blood-brain barrier.</p>
    Formula:C32H35F4N5O7
    Color and Shape:Solid
    Molecular weight:677.64
  • Herkinorin

    CAS:
    <p>Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.</p>
    Formula:C28H30O8
    Color and Shape:Solid
    Molecular weight:494.53
  • Locicortolone

    CAS:
    <p>Locicortolone is a synthetic glucocorticoid corticosteroid which was never marketed.</p>
    Formula:C22H28Cl2O3
    Color and Shape:Solid
    Molecular weight:411.36
  • AL-438

    CAS:
    <p>AL-438 is a non-steroidal selective glucocorticoid receptor modulator.</p>
    Formula:C23H25NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:347.45
  • Linuron

    CAS:
    <p>Linuron herbicide disrupts photosynthesis and acts as an androgen receptor antagonist.</p>
    Formula:C9H10Cl2N2O2
    Purity:99.08%
    Color and Shape:White Crystalline Solid Linuron Is A Colorless Crystals Non Corrosive Used As An Herbicide
    Molecular weight:249.09
  • ERRγ agonist-2

    CAS:
    <p>ERRγ agonist-2 is a potent and selective ERRγ inverse agonist with a K d value of 6.5 μM.</p>
    Formula:C27H21N5O2
    Color and Shape:Solid
    Molecular weight:447.49
  • Ditekiren

    CAS:
    <p>Ditekiren is a renin inhibitor with orally active.</p>
    Formula:C50H75N9O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:930.19
  • β-Endorphin, equine TFA


    <p>β-Endorphin, equine TFA, an endogenous opioid peptide, demonstrates high affinity binding to μ/δ opioid receptors and possesses analgesic properties [1] [2] [3</p>
    Formula:C156H249F3N42O46S
    Color and Shape:Solid
    Molecular weight:3537.96
  • RTI-13951-33 hydrochloride


    <p>RTI-13951-33 HCl: potent, selective GPR88 agonist; brain-penetrant; EC50 = 25nM; curbs rat alcohol behaviors.</p>
    Formula:C28H35Cl2N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:532.5
  • GLL 398

    CAS:
    <p>GLL 398 is an orally active and selective degrader of estrogen receptor with an IC50 of 1.14 nM. GLL 398 blocks tumor growth in xenograft breast cancer models.</p>
    Formula:C25H23BO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:398.26
  • OT antagonist 1 demethyl derivative


    <p>OT antagonist 1 demethyl derivative is the demethyl derivative of OT antagonist 1. OT antagonist 1 is a selective Oxytocin antagonist (Ki of 50 nM. )</p>
    Formula:C21H20N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.41
  • ST-CY14


    <p>ST-CY14 is an inhibitor of the Nur77-PPARγ interaction with an EC50 of 3.15 μM. It binds to Nur77 (Kd=32 nM) to prevent its ubiquitination and degradation by PPARγ, reducing fatty acid uptake and mitochondrial respiration, and inhibiting the transcription of CD36 and FABP4. ST-CY14 suppresses proliferation and migration of MCF7 and MDA-MB-231 cancer cells and impedes tumor growth and bone metastasis in mouse models.</p>
    Formula:C139H237N57O31S2
    Color and Shape:Solid
    Molecular weight:3266.86
  • THR-β agonist 2 diacetate


    <p>THR-β agonist 2 diacetate (Compound 3) is a potent THR-β agonist with potential applications in researching metabolic disorders such as obesity, hyperlipidemia, hypercholesterolemia, and diabetes, as well as other conditions like steatosis and non-alcoholic steatohepatitis (NASH), atherosclerosis, and other related diseases and conditions.</p>
    Color and Shape:Odour Solid
  • PROTAC ERα Degrader-8

    CAS:
    <p>PROTAC ERα Degrader-8 (compound ii-56), a highly potent degrader of Erα, achieves a DC50 of just 0.000006 μM in MCF7 cells [1].</p>
    Formula:C47H51N5O4
    Color and Shape:Solid
    Molecular weight:749.94
  • Antihypertensive agent 2


    <p>Antihypertensive agent 2 (Compound 4g) exhibits effective antagonistic activities against angiotensin II receptor 1 and reduces blood pressure with equal or</p>
    Formula:C22H15NO3
    Color and Shape:Solid
    Molecular weight:341.36
  • OT antagonist 3 analog


    <p>OT antagonist 3 analog is an analog of OT antagonist 3.</p>
    Formula:C20H18N6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:374.4
  • Dynorphin B (1-13) (TFA)


    <p>Dynorphin B (1-13) TFA acts as an agonist on opioid κ-receptor .</p>
    Formula:C76H116N21F3O19
    Color and Shape:Solid
    Molecular weight:1684.86