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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3183 products of "Endocrinology/Hormones"

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  • Zankiren
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    Zankiren

    CAS:
    <p>Zankiren is a renin inhibitor. Zankiren can reduce blood pressure, plasma renin activity, and angiotension II.</p>
    Formula:C35H55N5O6S2
    Color and Shape:Solid
    Molecular weight:705.97

    Ref: TM-T29204

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    D3R/MOR antagonist 1

    <p>Compound 114 (D3R/MOR antagonist 1) exhibits dual antagonistic activity at dopamine D3 receptors (D3R) and mu-opioid receptors (MOR), with K i values of 46.5 nM</p>
    Formula:C22H27Cl2N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:420.38

    Ref: TM-T78778

  • PROTAC ERα Degrader-8
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    PROTAC ERα Degrader-8

    CAS:
    <p>PROTAC ERα Degrader-8 (compound ii-56), a highly potent degrader of Erα, achieves a DC50 of just 0.000006 μM in MCF7 cells [1].</p>
    Formula:C47H51N5O4
    Color and Shape:Solid
    Molecular weight:749.94

    Ref: TM-T87265

  • ICI 174,864
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    ICI 174,864

    CAS:
    <p>Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.</p>
    Formula:C38H53N5O7
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:691.87

    Ref: TM-TP2013

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    KOR agonist 4

    <p>KOR agonist 4 (compound 39) is an agonist targeting the κ opioid receptor (Kappa Opioid Receptor) and activates G protein signaling. It has an EC50 of 14 nM and an Emax of 83% for binding to GTPγS. This compound demonstrates moderate to high intrinsic clearance in human liver cells and shows selectivity for the κ opioid receptor over the μ (MOR) and δ (DOR) opioid receptors by factors of 60 and 810, respectively. KOR agonist 4 is useful for research into central nervous system (CNS) disorders.</p>
    Formula:C21H25N3
    Color and Shape:Solid
    Molecular weight:319.44

    Ref: TM-T205240

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    Vasopressin Dimer (anti-parallel) (TFA)

    <p>Vasopressin Dimer (anti-parallel) TFA, an anti-parallel dimer form of vasopressin, has the capability to activate four G protein-coupled receptors: V1aR, V1bR,</p>
    Formula:C94H131F3N30O26S4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2282.49

    Ref: TM-T80198

  • Nociceptin(1-7)
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    Nociceptin(1-7)

    CAS:
    <p>Bioactive metabolite of nociceptin, antagonist of nociceptin-induced hyperalgesia</p>
    Formula:C31H41N7O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:655.709

    Ref: TM-T23076

  • MT-7716 free base
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    MT-7716 free base

    CAS:
    <p>MT-7716: selective NOP agonist, potential in preventing alcohol abuse/relapse.</p>
    Formula:C27H28N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.54

    Ref: TM-T12120L

  • Raloxifene 4'-glucuronide
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    Raloxifene 4'-glucuronide

    CAS:
    <p>Raloxifene 4'-glucuronide is a primary metabolite of Raloxifene.</p>
    Formula:C34H35NO10S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:649.71

    Ref: TM-T12686

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    4A7C-301

    <p>4A7C-301, a Nurr1 agonist, exhibits potent neuroprotective effects in vitro and markedly mitigates neuropathological abnormalities while enhancing motor and</p>
    Color and Shape:Odour Solid

    Ref: TM-T83328

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    [Nphe1]Nociceptin(1-13)NH2 TFA

    <p>[Nphe1]Nociceptin(1-13)NH2 is a selective nociceptin receptor antagonist with potential analgesic properties, pKi=8.4, pA2=6.0.</p>
    Formula:C63H101F3N22O17
    Color and Shape:Solid
    Molecular weight:1495.61

    Ref: TM-T75909

  • CJ-15208
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    CJ-15208

    CAS:
    <p>CJ-15208: κ-opioid antagonist, IC50: 47 nM kappa, 260 nM mu, 2600 nM delta, reverses asimadoline effects in rabbits (ED50 1.3 µM).</p>
    Formula:C34H35N5O4
    Color and Shape:Solid
    Molecular weight:577.67

    Ref: TM-T27027

  • Orphanin FQ(1-11)
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    Orphanin FQ(1-11)

    CAS:
    <p>Nociceptin peptide fragment (1-11) with potent ORL1/KOR-3 receptor agonism (Ki = 55 nM), no opioid receptor affinity, and analgesic in mice.</p>
    Formula:C49H75N15O14
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1098.2

    Ref: TM-TP1882

  • SNIPER(ER)-87
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    SNIPER(ER)-87

    CAS:
    <p>SNIPER(ER)-87 is a chemical compound composed of a derivative of the inhibitor of apoptosis protein (IAP) ligand LCL161 conjugated to the estrogen receptor α (</p>
    Formula:C59H73N5O10S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1044.32

    Ref: TM-T18697

  • Triphenylethylene
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    Triphenylethylene

    CAS:
    <p>Compound PDK0283, with CAS No. 58-72-0, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0283 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>
    Formula:C20H16
    Color and Shape:White Powder
    Molecular weight:256.34

    Ref: TM-PDK0283

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    Angiotensin II (1-4), human TFA

    <p>Angiotensin II is a potent direct vasoconstrictor, causing arteries and veins to constrict, so leading to an increase in blood pressure.</p>
    Formula:C26H38F3N7O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:665.62

    Ref: TM-TP1661

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    KOR agonist 5

    <p>KOR agonist 5 (Compound 10a) is both a KOR/MOR modulator, exhibiting agonistic effects on KOR and antagonistic effects on MOR. It effectively blocks morphine-induced antinociception and gastrointestinal motility inhibition. KOR agonist 5 is applicable in research related to substance use disorder (SUD).</p>
    Formula:C38H38N2O5
    Color and Shape:Solid
    Molecular weight:602.72

    Ref: TM-T205351

  • Inocoterone acetate
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    Inocoterone acetate

    CAS:
    <p>Inocoterone acetate is a nonsteroidal antiandrogen that binds to the androgen receptor and possesses antiandrogenic activity in animal models.</p>
    Formula:C18H26O3
    Color and Shape:Solid
    Molecular weight:290.40

    Ref: TM-T25536

  • RS 21314
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    RS 21314

    CAS:
    <p>RS 21314 is a thiol ester corticosteroid that is topical.</p>
    Formula:C24H30F2O5S
    Color and Shape:Solid
    Molecular weight:468.55

    Ref: TM-T34410

  • 18-Oxocortisol
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    18-Oxocortisol

    CAS:
    <p>18-Oxocortisol, a naturally occurring mineralocorticoid and adrenal biomarker, is produced by CYP11B2.</p>
    Formula:C21H28O6
    Color and Shape:Solid
    Molecular weight:376.449

    Ref: TM-T39991