Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(208 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(48 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(297 products)
- Prostaglandin Receptor(119 products)
- RAAS(86 products)
- Reductase(52 products)
- Somatostatin(46 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
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Found 3180 products of "Endocrinology/Hormones"
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GPR88 agonist 2
<p>GPR88 agonist 2 (compound 53) serves as a potent, brain-penetrant agonist of GPR88, exhibiting an EC50 of 14 µM in the GPR88 cAMP functional assay [1].</p>Color and Shape:Odour SolidTD-802
CAS:<p>TD-802, an AR-targeting PROTAC with microsomal stability, shows promise for castration-resistant prostate cancer.</p>Formula:C52H61ClN10O6Color and Shape:SolidMolecular weight:957.56MT-7716 hydrochloride
CAS:<p>MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)</p>Formula:C27H29ClN4O2Purity:98%Color and Shape:SolidMolecular weight:477ODM-204
CAS:<p>ODM-204 is novel nonsteroidal dual inhibitor of both androgen receptor and CYP17A1 enzyme(IC50s of 80 nM and 22 nM, respectively).</p>Formula:C20H21F3N4Purity:98%Color and Shape:SolidMolecular weight:374.40(S,S)-J-113397
CAS:<p>(S,S)-J-113397 is an isomer of J-113397 . J-113397 is an Opioid Receptor antagonist [1] .</p>Formula:C24H37N3O2Color and Shape:SolidMolecular weight:399.57Myrciacetin
CAS:<p>Myrciacetin from Rhododendron inhibits rat aldose reductase with IC50 of 13 μM.</p>Formula:C17H16O6Color and Shape:SolidMolecular weight:316.309Nurr1 agonist 12
<p>Nurr1 agonist 12 (Compound 37) acts as an agonist of the nuclear receptor-related protein 1 (Nurr1), enhancing its transcriptional activity with an EC50 of 0.06 μM. It stimulates human response elements NBRE, NurRE, and DR5 with EC50 values of 0.07 μM, 0.027 μM, and 0.014 μM, respectively. Additionally, Nurr1 agonist 12 induces the expression of neurotrophic genes regulated by Nurr1, such as tyrosine hydroxylase (TH), SOD1/2, BDNF, Sestrin 3, and BIRC5 (Survivin). The compound also demonstrates neuroprotective effects against neurotoxicity caused by Paraquat.</p>Formula:C18H12ClN3OColor and Shape:SolidMolecular weight:321.76GNE-502
CAS:<p>GNE-502 is an orally active and potent estrogen receptor (ER) degrader, specifically designed for research on breast cancer.</p>Formula:C25H30FN3O3SColor and Shape:SolidMolecular weight:471.59Retosiban
CAS:<p>Retosiban is an effective and selective oxytocin antagonist (Ki: 0.65 nM).</p>Formula:C27H34N4O5Purity:98%Color and Shape:SolidMolecular weight:494.58Antidiabetic agent 15
<p>Antidiabetic agent 15 (compound 1B15) acts as a dual inhibitor of AT1R and NEP, reducing oxidative stress and restoring mitochondrial membrane potential.</p>Formula:C26H23NO5Color and Shape:SolidMolecular weight:429.15762Epi-Cryptoacetalide
<p>Epi-Cryptoacetalide is a useful organic compound for research related to life sciences and the catalog number is T126054.</p>Formula:C18H22O3Color and Shape:SolidMolecular weight:286.371N-Acetyl-α-Endorphin
CAS:N-Acetyl-α-Endorphin is a chemical compound consisting of α-Endorphin that has been acetylated at the N-terminal.Formula:C79H122N18O27SPurity:98%Color and Shape:SolidMolecular weight:1787.98Valorphin
CAS:<p>Valorphin (Valorphin TFAsalt) has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.</p>Formula:C44H61N9O11Purity:98%Color and Shape:SolidMolecular weight:892.01R-6890
CAS:<p>R-6890 is an opioid compound with analgesic properties.</p>Formula:C21H24ClN3OColor and Shape:SolidMolecular weight:369.89Inocoterone acetate
CAS:<p>Inocoterone acetate is a nonsteroidal antiandrogen that binds to the androgen receptor and possesses antiandrogenic activity in animal models.</p>Formula:C18H26O3Color and Shape:SolidMolecular weight:290.40RLA-4842
<p>RLA-4842: iron-based anti-androgen; inhibits mCRPC cell proliferation.</p>Formula:C42H46F3N5O8SColor and Shape:SolidMolecular weight:837.9AM-5262
CAS:<p>AM-5262 is a potent GPR40 Full Agonist with improved rat PK profile and general selectivity profile.</p>Formula:C33H35FO4Color and Shape:SolidMolecular weight:514.63rac-1,2-bis-Palmitoyl-3-chloropropanediol
CAS:<p>3-MCPD ester found in edible oils, highest in olive pomace; toxic to mouse kidneys and spermatids.</p>Formula:C35H67ClO4Color and Shape:SolidMolecular weight:587.37Betamethasone acibutate
CAS:<p>Betamethasone acibutate, a glucocorticoid, is derived from Betamethasone.</p>Formula:C28H37FO7Purity:98%Color and Shape:SolidMolecular weight:504.59Bexirestrant
CAS:<p>Bexirestrant is an orally active ER-α degrader commonly employed in the research of antiestrogen and antineoplastic therapies.</p>Formula:C29H26F3NO2Color and Shape:SolidMolecular weight:477.527
