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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3178 products of "Endocrinology/Hormones"

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  • PD 123177
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    PD 123177

    CAS:
    <p>PD 123177 is an inhibitor of Nonpeptide angiotensin AII-2.</p>
    Formula:C29H28N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:480.56

    Ref: TM-T28322

  • Ac-RYYRIK-NH2
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    Ac-RYYRIK-NH2

    CAS:
    <p>NOP site high affinity ligand (Ki=1.5 nM); blocks nociceptin effects in rat brain/heart; agonist in vivo, reduces mouse movement.</p>
    Formula:C44H70N14O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:939.12

    Ref: TM-TP1940

  • OX04528
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    OX04528

    CAS:
    <p>OX04528 is an orally active and potent GPR84 biased agonist.OX04528 inhibits cAMP signaling and may be useful in cancer research.</p>
    Formula:C16H13F6NO2
    Purity:99.74%
    Color and Shape:Soild
    Molecular weight:365.27

    Ref: TM-T84313

  • Raloxifene 4'-glucuronide
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    Raloxifene 4'-glucuronide

    CAS:
    <p>Raloxifene 4'-glucuronide is a primary metabolite of Raloxifene.</p>
    Formula:C34H35NO10S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:649.71

    Ref: TM-T12686

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    Antitumor agent-195

    <p>Antitumor agent-195 (compound 16c) is a dual-targeting agent that simultaneously targets STAT3 and NQO1. At a concentration of 1 μM, it significantly inhibits the phosphorylation of STAT3 at the Tyr705 site and effectively induces apoptosis in MDA-MB-231 and MDA-MB-468 breast cancer cells. As a substrate of NQO1, Antitumor agent-195 markedly increases ROS production, causing severe DNA damage in a dose-dependent manner. It also demonstrates strong antitumor properties in MDA-MB-231 xenograft models.</p>
    Formula:C22H22N2O4
    Color and Shape:Solid
    Molecular weight:378.42

    Ref: TM-T205391

  • Axelopran
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    Axelopran

    CAS:
    <p>Axelopran (TD-1211) treats opioid constipation; it's a potent, selective peripheral opioid blocker.</p>
    Formula:C26H39N3O4
    Color and Shape:Solid
    Molecular weight:457.61

    Ref: TM-T30236

  • PD 125967
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    PD 125967

    CAS:
    <p>PD 125967 is a renin inhibitor, which represents a group of pharmaceutical drugs used primarily to treat essential hypertension.</p>
    Formula:C51H67N5O4
    Color and Shape:Solid
    Molecular weight:814.11

    Ref: TM-T28324

  • Nocistatin
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    Nocistatin

    CAS:
    <p>Nocistatin, a neuropeptide, blocks Nociceptin effects and inhibits 5-HT release, acting on an opioid-related receptor.</p>
    Formula:C32H56N10O12
    Color and Shape:Solid
    Molecular weight:772.85

    Ref: TM-T76420

  • [Orn8]-Urotensin II
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    [Orn8]-Urotensin II

    CAS:
    <p>[Orn8]-Urotensin II is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.</p>
    Formula:C63H83N13O18S2
    Color and Shape:Solid
    Molecular weight:1374.55

    Ref: TM-T37527

  • Cgp 44099
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    Cgp 44099

    CAS:
    <p>Cgp 44099 is a potent plasma renin inhibitor from all subprimate species.</p>
    Formula:C69H104N14O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1337.676

    Ref: TM-T25230

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    Alunacedase alfa

    CAS:
    <p>Alunacedase alfa (APN-01) is an angiotensin-converting enzyme 2 with antiviral activity.</p>
    Purity:99.1% (SDS-PAGE); 99.9% (SEC-HPLC) - 99.1% (SDS-PAGE); 99.9% (SEC-HPLC)
    Color and Shape:Liquid

    Ref: TM-T80587

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    (rel)-PROTAC ERRα Degrader-1

    <p>(rel)-PROTAC ERRα Degrader-1 is a relative configuration of PROTAC ERRα Degrader-1, which is an estrogen-related receptor alpha (ERRa) degrader.</p>
    Formula:C54H49Cl2F6N7O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1108.91

    Ref: TM-T18651

  • CymitQuimica logo
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    HINT1-IN-1

    <p>HINT1-IN-1 (compound 8) is an inhibitor of histidine triad nucleotide-binding protein 1 (HINT1) with a Ki of 1.14 μM. It influences the cross-regulation between μ-opioid receptors (MOR) and NMDA receptors (NMDAR).</p>
    Formula:C23H24N8O5
    Color and Shape:Solid
    Molecular weight:492.49

    Ref: TM-T205282

  • PROTAC ER Degrader-4
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    PROTAC ER Degrader-4

    CAS:
    <p>PROTAC ER Degrader-4 is a PROATC degrader of estrogen receptor (ER)(IC50 of 0.8 nM).</p>
    Formula:C53H67F3N6O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1005.2

    Ref: TM-T13839

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    PTP1B/AKR1B1-IN-1

    <p>PTP1B/AKR1B1-IN-1 is a dual inhibitor targeting protein tyrosine phosphatase 1B (PTP1B) and aldose reductase (AKR1B1), exhibiting inhibitory potency with IC50s</p>
    Formula:C22H21NO4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:427.54

    Ref: TM-T78702

  • SNIPER(ER)-110
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    SNIPER(ER)-110

    <p>SNIPER(ER)-110 links cIAP1 and estrogen ligands. SNIPER(ER)-51 degrades ER protein; DC50 &lt;3 nM at 4h, 7.7 nM at 48h.</p>
    Formula:C66H83N5O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1122.39

    Ref: TM-T18696

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    ST-CY14

    <p>ST-CY14 is an inhibitor of the Nur77-PPARγ interaction with an EC50 of 3.15 μM. It binds to Nur77 (Kd=32 nM) to prevent its ubiquitination and degradation by PPARγ, reducing fatty acid uptake and mitochondrial respiration, and inhibiting the transcription of CD36 and FABP4. ST-CY14 suppresses proliferation and migration of MCF7 and MDA-MB-231 cancer cells and impedes tumor growth and bone metastasis in mouse models.</p>
    Formula:C139H237N57O31S2
    Color and Shape:Solid
    Molecular weight:3266.86

    Ref: TM-TP3109

  • DAMGO (TFA)
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    DAMGO (TFA)

    CAS:
    <p>DAMGO is a selective peptide agonist of the µ-opioid receptor .</p>
    Formula:C28H36F3N5O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:627.61

    Ref: TM-TP1607

  • OT-R antagonist 2
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    OT-R antagonist 2

    CAS:
    <p>OT-R antagonist 2 is a nonpeptide low molecular weight antagonist of OT-R .</p>
    Formula:C28H29N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:471.55

    Ref: TM-T12331

  • (d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin
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    (d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin

    CAS:
    <p>(d(CH2)51,Tyr(Me)2, Orn8)-Oxytocin (OVT) is an antagonist of the oxytocin receptor that finds application in the study of neurological diseases [1].</p>
    Formula:C48H74N12O12S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1075.3

    Ref: TM-T80126