Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(230 products)
- Annexin A(16 products)
- Aromatase(23 products)
- Estrogen/progestogen Receptor(66 products)
- GPR(1 products)
- Glucocorticoid Receptor(165 products)
- LHRH(2 products)
- Opioid Receptor(327 products)
- Prostaglandin Receptor(126 products)
- RAAS(89 products)
- Reductase(51 products)
- Somatostatin(57 products)
- Thyroid hormone receptor(THR)(34 products)
- Vasopressin Receptor(48 products)
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Found 3421 products of "Endocrinology/Hormones"
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KOR agonist 3
KOR agonist 3 (Compound 5) is an agonist of the κ opioid receptor (κOR) with an EC50 of 0.88 nM. It also exhibits some activation of μOR, with an EC50 of 720 nM. However, KOR agonist 3 does not activate δOR at concentrations below 1 μM. Its ability to recruit β-Arrestin-2 is lower than that of U50488.Formula:C24H24N2O3Color and Shape:SolidMolecular weight:388.46Pro8-Oxytocin
CAS:Pro8-Oxytocin, a modified oxytocin (OXT) ligand, elicits more potent and efficacious responses at primate OXTR and induces stronger behavioral effects comparedFormula:C42H62N12O12S2Purity:98%Color and Shape:SolidMolecular weight:991.14Corynantheidine
CAS:Corynantheidine ((-)-Corynantheidine) is a partial agonist of the mu opioid receptor (MOR) and demonstrates MOR-dependent analgesic effects in mice.Formula:C22H28N2O3Color and Shape:SolidMolecular weight:368.47AH 7959
CAS:AH 7959 is an orally active N-substituted cyclohexylmethylbenzamide compound that exhibits analgesic properties. In mice, the ED50 for oral and subcutaneous administration of AH 7959 exceeds 100 mg/kg.Formula:C19H26Cl2N2OColor and Shape:SolidMolecular weight:369.33Dynorphin B (1-9)
CAS:Dynorphin B (1-9), a neuropeptide and the N-terminal cleavage product of dynorphin B, has its formation inhibited by N-ethylmaleimide (NEM), a non-selectiveFormula:C54H78N16O12Purity:98%Color and Shape:SolidMolecular weight:1143.3AP-238
CAS:AP-238 is a novel synthetic opioid (NSO) that acts as an agonist for the μ-opioid receptor (MOR), with an EC50 of 248 nM. Additionally, AP-238 exhibits analgesic properties.Formula:C18H26N2OColor and Shape:SolidMolecular weight:286.41Nesvacumab
CAS:Nesvacumab (REGN910) is a fully human monoclonal antibody targeting Angiopoietin 2 (Ang2), which can be used for studying advanced solid tumors.Purity:98.7% (SDS-PAGE); 95.7% (SEC-HPLC) - 99.11% (SEC-HPLC)Color and Shape:LiquidMolecular weight:144.84 kDaTetrahydro Aldosterone
CAS:Tetrahydro Aldosterone is a steroidal compound that inhibits the adrenal angiotensin II receptor, with an IC50 of 10 μM.Formula:C21H32O5Color and Shape:SolidMolecular weight:364.48PRL 2915
CAS:PRL 2915 is a potent antagonist of the human somatostatin subtype 2 receptor (hsst 2), exhibiting a binding affinity (K_i) of 12 nM [1].Formula:C59H71ClN12O8S2Color and Shape:SolidMolecular weight:1175.85PRO20
PRO20 is a specific and competitive antagonist of the (pro)renin receptor (PRR). It inhibits the calcium influx induced by Proproin with an IC50 value of 81 nmol/L. By blocking the binding of Prorenin to PRR, PRO20 inhibits the activation of the renin-angiotensin system (RAS), reducing the production of angiotensin II (Ang II) and exerting antihypertensive effects. PRO20 holds promise for research in antihypertensive agents.
Color and Shape:Odour SolidProtirelin Acetate
CAS:Protirelin Acetate (TRH Acetate) is a thyrotropin-releasing hormone, stimulating the release of thyrotropin and prolactin from the anterior pituitary.Formula:C16H22N6O4C2H4O2Purity:96.17%Color and Shape:SolidMolecular weight:452.46DPC-AJ1951 TFA
DPC-AJ1951 TFA is a 14 amino acid peptide, potent PTH/PPR agonist, tested in bone resorption assays.Formula:C78H128F3N23O21Color and Shape:SolidMolecular weight:1781.024-Hydroxy-1-(2-phenylethyl)piperidine
CAS:4-Hydroxy-1-(2-phenylethyl)piperidine is a synthetic ligand for muscarinic acetylcholine receptors (mAChR) or non-opioid intracellular sigma-1 receptors (σ1 receptors). It serves as a metabolite of the opioid compounds furanylfentanyl and 4-fluoroisobutyryl fentanyl (FIBF).Formula:C13H19NOColor and Shape:SolidMolecular weight:205.3(Glu2)-TRH
CAS:(Glu2)-TRH: Stable TRH analog; reduces TRH's cholinergic action; no thyroliberinase metabolism; neuroprotective with antidepressant, anticonvulsant effects.Formula:C15H22N4O6Color and Shape:SolidMolecular weight:354.36Osteostatin
CAS:Osteostatin, derived from parathyroid hormone-related protein (PTHrP) 107-111, has demonstrated properties conducive to bone repair in animal models presentingFormula:C27H41N9O8Color and Shape:SolidMolecular weight:619.677α-(Thiomethyl)spironolactone
CAS:7α-(Thiomethyl)spironolactone is a steroid receptor antagonist and major spironolactone metabolite, steroid metabolism, nuclear receptor, and coronavirus.Formula:C23H32O3SPurity:>99.99%Color and Shape:SolidMolecular weight:388.56β-Endorphin (1-27) (human)
CAS:β-Endorphin (1-27) (human) is an opioid antagonist that selectively binds to μ-, δ-, and κ-opioid receptors, with dissociation constants (Kis) of 5.31, 6.17,Formula:C139H217N33O40SPurity:98%Color and Shape:SolidMolecular weight:3022.473-Iodothyronamine hydrochloride
CAS:3-Iodothyronamine hydrochloride, Thyroid hormone derivative, activates TAAR1, induces hypothermia, for endocrine/metabolic research.Formula:C14H15ClINO2Color and Shape:SolidMolecular weight:391.63PF-06655075 TFA
PF-06655075 (TFA) is the trifluoroacetic acid (TFA) salt of PF-06655075, a novel, non-brain-penetrant oxytocin receptor agonist that exhibits enhancedPurity:98%Color and Shape:Odour SolidUFP-101 acetate
UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.
Formula:C84H142N32O23Purity:95.92%Color and Shape:SolidMolecular weight:1968.23
