Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(208 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(48 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(297 products)
- Prostaglandin Receptor(119 products)
- RAAS(86 products)
- Reductase(52 products)
- Somatostatin(46 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
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Found 3180 products of "Endocrinology/Hormones"
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VPC-13566
CAS:<p>VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the</p>Formula:C18H14N2Purity:99.55%Color and Shape:SolidMolecular weight:258.32Alvimopan monohydrate
CAS:<p>Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.</p>Formula:C25H34N2O5Purity:98%Color and Shape:SolidMolecular weight:442.55AH-7614
CAS:<p>AH-7614 (AH 7614) is a selective and potent free fatty acid receptor 4 (FFA4/GPR120) antagonist.</p>Formula:C20H17NO3SPurity:98.05%Color and Shape:SolidMolecular weight:351.42EST73502 HCl
CAS:<p>EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.</p>Formula:C19H27ClF2N2O2Purity:99.96%Color and Shape:SolidMolecular weight:388.88[D-Ala2]leucine-enkephalin
CAS:<p>[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.</p>Formula:C29H39N5O7Purity:98.06%Color and Shape:SolidMolecular weight:569.65Nafoxidine HCl(1845-11-0 Free base)
CAS:<p>Nafoxidine is a partial estrogen antagonist.</p>Formula:C29H32ClNO2Color and Shape:SolidMolecular weight:462.03ARV-471
CAS:<p>ARV-471 (Vepdegestrant) is a orally active Cereblon -based estrogen receptor (ER) PROTAC degrader. ARV-471 is developed for the research of breast cancer.</p>Formula:C45H49N5O4Purity:97.15% - >99.99%Color and Shape:SolidMolecular weight:723.9Methylprednisolone succinate
CAS:<p>Methylprednisolone succinate (Methylprednisolone hemisuccinate) is a synthetic glucocorticoid and is widely used as an anti-inflammatory agent.</p>Formula:C26H34O8Purity:98.41% - 99.82%Color and Shape:White Or Almost-White Solid PowderMolecular weight:474.54Testosterone undecanoate
CAS:<p>Testosterone undecanoate is a metabolite of Testosterone, which is a promising androgen for male hormonal contraception.</p>Formula:C30H48O3Purity:99.45% - 99.788%Color and Shape:White Crystalline PowderMolecular weight:456.7Methylnaltrexone bromide
CAS:<p>Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.</p>Formula:C21H26BrNO4Purity:99.02%Color and Shape:SolidMolecular weight:436.35Ac-RYYRWK-NH2 acetate
<p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>Formula:C51H73N15O11Purity:98.59%Color and Shape:SolidMolecular weight:1072.22MBX-2982
CAS:<p>MBX-2982 is a selective, orally-available GPR119 agonist, used for the treatment of diabetes.</p>Formula:C22H24N8OSPurity:98% - 99.96%Color and Shape:SolidMolecular weight:448.54AS1269574
CAS:<p>AS1269574 is a potent, orally available GPR119 agonist. AS1269574(AS 1269574) has the potential for the research of type 2 diabetes.</p>Formula:C13H14BrN3OPurity:99.99%Color and Shape:SolidMolecular weight:308.17Adrenorphin 3TFA(88377-68-8(free base))
<p>Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Formula:C50H72N15O15SPurity:>99.99%Color and Shape:SolidMolecular weight:1326.26Ulipristal
CAS:<p>Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.</p>Formula:C28H35NO3Purity:99.82%Color and Shape:SolidMolecular weight:433.58Urotensin II (114-124), human acetate
<p>Urotensin II (114-124), human acetate is an 11-amino acid residue peptide, is a potent vasoconstrictor and agonist for the orphan receptor GPR14.</p>Formula:C66H89N13O20S2Purity:>99.99%Color and Shape:SolidMolecular weight:1448.63PW0787
CAS:<p>PW0787 is a potent, selective, orally active, and brain-penetrant GPR52 agonist (EC50=135 nM).</p>Formula:C23H20F4N4O2Purity:98.42%Color and Shape:SolidMolecular weight:460.42JNJ-63576253
CAS:<p>JNJ-63576253 is a Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC).</p>Formula:C23H22ClF3N6O2SPurity:98.71%Color and Shape:SolidMolecular weight:538.97SSAA09E2
CAS:<p>SSAA09E2 is a new SARS-CoV replication inhibitor, acting by blocking early interactions of SARS-S with the receptor for SARS-CoV, Angiotensin Converting Enzyme-</p>Formula:C16H20N4O2Purity:99.41%Color and Shape:SolidMolecular weight:300.36N-Acetyl-Ser-Asp-Lys-Pro
CAS:<p>Acetyl Ser-Asp-Lys-Pro, derived from thymosin β4 in bone marrow, blocks stem cell cycle progression and shields mice from Ara-C toxicity.</p>Formula:C20H33N5O9Purity:99.85%Color and Shape:SolidMolecular weight:487.5Palosuran hydrochloride 540769-28-6(free base)
<p>Palosuran hydrochloride 540769-28-6(free base)(ACT-058362 hydrochloride) is a new potent and specific antagonist of the human UT receptor with an IC50 of 3.6±0.</p>Formula:C25H31ClN4O2Purity:99.75%Color and Shape:SolidMolecular weight:454.99Hemorphin-7 acetate(152685-85-3 free base)
<p>Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.</p>Formula:C51H68N12O13Purity:99.66%Color and Shape:SolidMolecular weight:1057.16Alamandine TFA
<p>Alamandine TFA, a RAS peptide, binds MrgD receptors, has anti-hypertensive effects, and protects heart and kidneys.</p>Formula:C42H63F3N12O11Purity:99.62%Color and Shape:SoildMolecular weight:969.02Acein acetate
<p>ACE ligand with Kd 2.79 nM, inactive on ACE up to 500 nM. Boosts NMDA/D-serine-induced dopamine release in striatum.</p>Formula:C45H72N10O15Purity:99.43%Color and Shape:SolidMolecular weight:993.11Azilsartan Medoxomil
CAS:<p>Azilsartan Medoxomil (TAK-491) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults</p>Formula:C30H24N4O8Purity:99.83%Color and Shape:SolidMolecular weight:568.53b-Casomorphin (1-3) Acetate
<p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>Formula:C25H31N3O7Purity:98.99%Color and Shape:SolidMolecular weight:485.53Trans-Tranilast
CAS:<p>Trans-Tranilast is an antiallergic drug developed by Kissei Pharmaceuticals. It has been used for the treatment of allergic disorders such as atopic dermatitis.</p>Formula:C18H17NO5Purity:99.41% - ≥95%Color and Shape:SolidMolecular weight:327.33DAMGO
CAS:<p>DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.</p>Formula:C26H35N5O6Purity:98.83% - 99.92%Color and Shape:SolidMolecular weight:513.59Velsecorat
CAS:<p>Velsecorat (AZD7594) is an effective and selective nonsteroidal glucocorticoid receptor modulator (IC50: 0.9 nM).</p>Formula:C32H32F2N4O6Purity:99.35%Color and Shape:SolidMolecular weight:606.62Sobetirome
CAS:<p>Sobetirome (IACS-010759) is a selective agonist of thyroid hormone receptor β (TRβ) and binds selectively to TRβ-1 (EC50: 0.16 μM).</p>Formula:C20H24O4Purity:98.08% - 98.25%Color and Shape:SolidMolecular weight:328.4H-Val-Pro-Pro-OH
CAS:<p>H-Val-Pro-Pro-OH is an inhibitor of Angiotensin I converting enzyme (ACE)( IC50 : 9 μM).</p>Formula:C15H25N3O4Purity:98.23%Color and Shape:SolidMolecular weight:311.38Tranilast
CAS:<p>Tranilast (SB 252218), an antiallergic drug, suppresses lipid mediator and cytokine release from inflammatory cells, therefore utilized in the treatment of</p>Formula:C18H17NO5Purity:99.67% - >99.99%Color and Shape:White With Light Yellow Crystalline PowderMolecular weight:327.334-CMTB
CAS:<p>4-CMTB is a selective agonist of FFA2 and GPR43.It also is a positive allosteric modulator (pEC50=6.38).</p>Formula:C14H15ClN2OSPurity:99.59%Color and Shape:SolidMolecular weight:294.8MS21570
CAS:<p>MS21570 as a GPR171 antagonist based on its ability to block,with an IC50 of 220 Nm,that reduces anxiety-like behavior and fear conditioning in mice.</p>Formula:C10H11N3S2Purity:97.79%Color and Shape:SolidMolecular weight:237.34Nalmefene hydrochloride
CAS:<p>Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.</p>Formula:C21H26ClNO3Purity:98% - 99.85%Color and Shape:SolidMolecular weight:375.89Timapiprant
CAS:<p>Timapiprant (OC000459) is a potent and selective D prostanoid receptor 2 (DP2) antagonist (IC50: 13 nM).</p>Formula:C21H17FN2O2Purity:97.44% - 99.51%Color and Shape:SolidMolecular weight:348.37Angiotensin I/II (1-6)
CAS:<p>Angiotensin I/II (1-6) is a peptide (ASP-ARG-VAL-TYR-ILE-HIS) that contains the amino acids 1-6 and is converted from Angiotensin I/II peptide.</p>Formula:C36H55N11O10Purity:99.44%Color and Shape:SolidMolecular weight:801.893-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
CAS:<p>3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.</p>Formula:C18H14N4OPurity:98.41%Color and Shape:SolidMolecular weight:302.33Bisphenol B
CAS:<p>Bisphenol B has a binding affinity for estrogen receptors.</p>Formula:C16H18O2Purity:97.35% - 99.62%Color and Shape:Crystal Or Tan Granules Odorless Slightly Brown SolidMolecular weight:242.31AZD1981
CAS:<p>AZD1981: selective CRTh2 antagonist, IC50 4 nM, 1000x specificity over 340+ enzymes/receptors, tested in asthma and other trials.</p>Formula:C19H17ClN2O3SPurity:98.87% - 99.67%Color and Shape:SolidMolecular weight:388.87Lasofoxifene
CAS:<p>Lasofoxifene (CP-336156) is a selective oestrogen receptor modulator/antagonist that reduces serum IL-6 levels and inhibits joint inflammation and osteoporosis.</p>Formula:C28H31NO2Purity:99.6%Color and Shape:SolidMolecular weight:413.55CTK8A3536
CAS:<p>CTK8A3536 ((2-MORPHOLIN-4-YL-4-PHENYL-1,3-THIAZOL-5-YL)METHANOL) is an inhibitor of Androgen receptor.</p>Formula:C14H16N2O2SPurity:99.62%Color and Shape:SolidMolecular weight:276.35Finerenone
CAS:<p>Finerenone (BAY-948862) is a selective and orally nonsteroidal antagonist of the mineralocorticoid receptor (MR). Cost effective and quality assured.</p>Formula:C21H22N4O3Purity:99.45% - 99.91%Color and Shape:SolidMolecular weight:378.42CVN424
CAS:<p>CVN424 is a selective and novel GPR6 Inverse agonist effective in models of Parkinson Disease.</p>Formula:C24H29F2N5O3Purity:99.02%Color and Shape:SolidMolecular weight:473.52Tyr-Gly-Gly-Phe-Met-OH
CAS:<p>Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.</p>Formula:C27H35N5O7SPurity:≥95%Color and Shape:White Lyophilised SolidMolecular weight:573.66TC-O 9311
CAS:<p>TC-O 9311 (TCO-9311) is an effective agonist of GPR139 (EC50 = 39 nM in CHO-K1 cells expressing human GPR139).</p>Formula:C20H19N3O4Purity:99.24% - 99.84%Color and Shape:SolidMolecular weight:365.38Chlorotrianisene
CAS:<p>Chlorotrianisene, a synthetic SERM, is orally active, lipophilic, and has estrogenic and antiestrogenic effects.</p>Formula:C23H21ClO3Purity:98.88% - 99.03%Color and Shape:Crystals From Methanol Physical Description Small White Crystals Or White Powder Softens At 226°F Odorless (Ntp 1992)Molecular weight:380.86H3B-5942
CAS:<p>H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).</p>Formula:C31H34N4O2Purity:99.21% - ≥95%Color and Shape:SolidMolecular weight:494.63Kisspeptin-10, human (TFA)(374675-21-5,FREE)
<p>Kisspeptin-10 TFA: vasoconstrictor, inhibits angiogenesis & metastasis; key in kidney development & osteoblast differentiation via GPR54 & NFATc4/BMP2.</p>Formula:C63H83N17O14·C2HF3O2Purity:>99.99%Color and Shape:SolidMolecular weight:1416.46Ferrous Bisglycinate
CAS:<p>Ferrous Bisglycinate (Bisglycine iron(II) salt) is used in the fortification of infant formulations and foods.</p>Formula:C4H8FeN2O4Purity:≥95%Color and Shape:SolidMolecular weight:203.96
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