Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(207 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(49 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(296 products)
- Prostaglandin Receptor(119 products)
- RAAS(86 products)
- Reductase(52 products)
- Somatostatin(46 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
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Found 3178 products of "Endocrinology/Hormones"
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PROTAC ERRα ligand 1
CAS:<p>PROTAC ERRα ligand 1 is an α (ERRα) antagonist of estrogen-related receptor (IC50s of 0.04 and 2.8 μM for ERRα and ERRγ, respectively).</p>Formula:C19H11F3N2O4SPurity:99.45%Color and Shape:SolidMolecular weight:420.36(R)-Equol
CAS:<p>(R)-Equol ((+)-Equol) is an ERα and ERβ agonist with Kis of 27.4 and 15.4 nM, respectively.</p>Formula:C15H14O3Purity:99.59%Color and Shape:SolidMolecular weight:242.27CHF-4227
CAS:<p>CHF-4227 is a novel, potent and selective estrogen receptor modulator that reduces cholesterol and LDL cholesterol concentrations.</p>Formula:C30H33NO4Purity:98.32%Color and Shape:SolidMolecular weight:471.59Ethisterone
CAS:<p>Ethisterone (17α-Ethynyltestosterone) is a progestogen hormone.</p>Formula:C21H28O2Purity:97.96% - 99.50%Color and Shape:Off-White PowderMolecular weight:312.45SK33
CAS:<p>SK33 is a potent and tissue selective anti-androgen agent. SK33 reduces androgen receptor (AR) transcriptional activity.</p>Formula:C20H13F9N2O3Purity:99.55%Color and Shape:SolidMolecular weight:500.31Bicalutamide
CAS:<p>Bicalutamide (ICI-176334), a synthetic, nonsteroidal antiandrogen, competitively binds to cytosolic androgen receptors in target tissues, thereby inhibiting the</p>Formula:C18H14F4N2O4SPurity:98% - 99.87%Color and Shape:Off-White Crystalline SolidMolecular weight:430.37Pomisartan 2HCl
<p>Pomisartan 2HCl (BIBR363 2HCL) is a small molecule AT1R antagonist used to study heart failure and hypertension.</p>Formula:C31H32Cl2N4O2Purity:99.88%Color and Shape:SoildMolecular weight:563.52Flutamide
CAS:<p>Flutamide (SCH 13521) is an antiandrogen with about the same potency as cyproterone in rodent and canine species.</p>Formula:C11H11F3N2O3Purity:99.6% - 99.96%Color and Shape:SolidMolecular weight:276.21ZT 52656A hydrochloride
CAS:<p>ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.</p>Formula:C19H26ClF3N2OPurity:98.78%Color and Shape:SolidMolecular weight:390.87Meptazinol hydrochloride
CAS:<p>Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.</p>Formula:C15H23NO·HClPurity:99.75%Color and Shape:White SolidMolecular weight:269.81Mirtazapine
CAS:<p>Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.</p>Formula:C17H19N3Purity:99.98%Color and Shape:SolidMolecular weight:265.35FTBMT
CAS:<p>FTBMT is a selective GPR52 agonist (EC50: 75 nM) and it also has antipsychotic and procognitive properties.</p>Formula:C19H16F4N4OPurity:99.56%Color and Shape:SolidMolecular weight:392.35Naltrexone hydrochloride
CAS:<p>Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.</p>Formula:C20H24ClNO4Purity:98.72% - 99.65%Color and Shape:White Crystalline PowderMolecular weight:377.862Loteprednol etabonate
CAS:<p>Loteprednol etabonate (Lotemax) is an ophthalmic analog of the corticosteroid prednisolone with anti-inflammatory activity.</p>Formula:C24H31ClO7Purity:99.19%Color and Shape:SolidMolecular weight:466.95NE 52-QQ57
CAS:<p>NE 52-QQ57 is a selective, and orally available antagonist of GPR4(IC50 : 70 nM),with anti-inflammatory activity.</p>Formula:C24H28N6OPurity:98.63%Color and Shape:SolidMolecular weight:416.52Samidorphan HCl
CAS:<p>Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.</p>Formula:C21H27ClN2O4Purity:96.79% - 97.85%Color and Shape:SoildMolecular weight:406.9Topilutamide
CAS:<p>Topilutamide (Fluridil) is a topical nonsteroidal antiandrogen.</p>Formula:C13H11F6N3O5Purity:98.77% - 99.24%Color and Shape:SolidMolecular weight:403.23Hydrocortisone acetate
CAS:<p>Hydrocortisone acetate (Cortisol 21-acetate) is the synthetic acetate salt form of hydrocortisone, a corticosteroid with anti-inflammatory and immunosuppressive</p>Formula:C23H32O6Purity:98.89% - 99.22%Color and Shape:White To Off-White Crystalline PowderMolecular weight:404.5Halcinonide
CAS:<p>Halcinonide (Halciderm), a high-efficiency corticosteroid, is served as an anti-inflammatory agent used in topical preparations.</p>Formula:C24H32ClFO5Purity:99.32% - 99.93%Color and Shape:SolidMolecular weight:454.96Allylestrenol
CAS:<p>Allylestrenol (Gestanin) is a synthetic steroid with progestational activity.</p>Formula:C21H32OPurity:>99.99%Color and Shape:White Crystalline PowderMolecular weight:300.48Glucagon (1-29), bovine, human, porcine hydrochloride
CAS:<p>Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. Glucagon increases HNF4α phosphorylation.</p>Formula:C153H225N43O49S·ClHPurity:95.65% - 98.03%Color and Shape:SolidMolecular weight:3519.21Resorcinolnaphthalein
CAS:<p>Resorcinolnaphthalein is a specific enhancer of angiotensin-converting enzyme 2 (ACE2) (EC50 value of 19.5 μM).</p>Formula:C24H14O5Purity:98.18%Color and Shape:SolidMolecular weight:382.36Betamethasone dipropionate
CAS:<p>Betamethasone Dipropionate, a synthetic glucocorticoid, modulates gene expression to manage inflammation and autoimmune activity.</p>Formula:C28H37FO7Purity:98.13% - 99.59%Color and Shape:PowderMolecular weight:504.59Clobetasol propionate
CAS:<p>Clobetasol propionate (CGP9555) exerts its effect by binding to cytoplasmic glucocorticoid receptors and subsequently activates glucocorticoid receptor-mediated</p>Formula:C25H32ClFO5Purity:99.41%Color and Shape:White Crystalline PowderMolecular weight:466.97Betamethasone acibutate
CAS:<p>Betamethasone acibutate, a glucocorticoid, is derived from Betamethasone.</p>Formula:C28H37FO7Purity:98%Color and Shape:SolidMolecular weight:504.59Biphalin TFA
CAS:<p>Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.</p>Formula:C46H56N10O10·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:909.00 (free base)Remikiren
CAS:<p>Remikiren is a highly specific renin inhibitor with oral activity for the treatment of hypertensio.</p>Formula:C33H50N4O6SColor and Shape:SolidMolecular weight:630.84ARCC-4
CAS:<p>ARCC-4: A VHL-recruiting, low-nanomolar (DC50=5nM) AR degrader; outshines enzalutamide; degrades AR mutants resistant to therapy.</p>Formula:C53H56F3N7O7S2Purity:98%Color and Shape:SolidMolecular weight:1024.18Parathyroid hormone (1-34) (rat)
CAS:<p>Parathyroid hormone (PTH) receptor agonist. Increases serum PTH levels and bone mass in rats.</p>Formula:C180H291N55O48S2Purity:98%Color and Shape:SolidMolecular weight:4057.742-Ethylhexyl trans-4-methoxycinnamate
CAS:<p>2-Ethylhexyl trans-4-methoxycinnamate is a sunscreen agent.</p>Formula:C18H26O3Purity:98.92%Color and Shape:Pale Yellow LiquidMolecular weight:290.4U-54494A hydrochloride
CAS:<p>U-54494A hydrochloride is a benzamide derivative related to kappa opioid receptor agonists. U-54494A hydrochloride has anticonvulsant activity.</p>Formula:C18H25Cl3N2OColor and Shape:SolidMolecular weight:391.764A7C-301
<p>4A7C-301, a Nurr1 agonist, exhibits potent neuroprotective effects in vitro and markedly mitigates neuropathological abnormalities while enhancing motor and</p>Color and Shape:Odour SolidRLA-4842
<p>RLA-4842: iron-based anti-androgen; inhibits mCRPC cell proliferation.</p>Formula:C42H46F3N5O8SColor and Shape:SolidMolecular weight:837.918-Oxocortisol
CAS:<p>18-Oxocortisol, a naturally occurring mineralocorticoid and adrenal biomarker, is produced by CYP11B2.</p>Formula:C21H28O6Color and Shape:SolidMolecular weight:376.449T4-ATA (S-isomer)
<p>T4-ATA S-isomer, the active form of the thyroid hormone, represents the S-isomer of T4-ATA.</p>Formula:C19H15I4NO6SPurity:98%Color and Shape:SolidMolecular weight:893.01[Sar1, Ile8]-Angiotensin II TFA
<p>[Sar1,Ile8]-Angiotensin II (TFA) contracts arteries and affects cell growth in vascular muscle.</p>Formula:C48H74F3N13O12Purity:98%Color and Shape:SolidMolecular weight:1082.18PROTAC AR-V7 degrader-1
CAS:<p>Potent, oral AR-V7 degrader (Compound 6); DC50: 0.32µM; targets AR-DBD via VHL E3; EC50: 0.88µM in 22Rv1 cells.</p>Formula:C41H52N6O6S2Color and Shape:SolidMolecular weight:789.02HINT1-IN-1
<p>HINT1-IN-1 (compound 8) is an inhibitor of histidine triad nucleotide-binding protein 1 (HINT1) with a Ki of 1.14 μM. It influences the cross-regulation between μ-opioid receptors (MOR) and NMDA receptors (NMDAR).</p>Formula:C23H24N8O5Color and Shape:SolidMolecular weight:492.49BI 653048 phosphate
CAS:<p>BI 653048 phosphate is a selective and orally active agonist of nonsteroidal glucocorticoid (GC)(IC50 : 55 nM).</p>Formula:C23H28F4N3O8PSPurity:98%Color and Shape:SolidMolecular weight:613.52PROTAC AR Degrader-4 TFA
<p>PROTAC AR Degrader-4: IAP ligand, linker, AR binder; it's a SNIPER that degrades AR non-genetically.</p>Formula:C45H68F3N3O11Color and Shape:SolidMolecular weight:884.03KOR agonist 4
<p>KOR agonist 4 (compound 39) is an agonist targeting the κ opioid receptor (Kappa Opioid Receptor) and activates G protein signaling. It has an EC50 of 14 nM and an Emax of 83% for binding to GTPγS. This compound demonstrates moderate to high intrinsic clearance in human liver cells and shows selectivity for the κ opioid receptor over the μ (MOR) and δ (DOR) opioid receptors by factors of 60 and 810, respectively. KOR agonist 4 is useful for research into central nervous system (CNS) disorders.</p>Formula:C21H25N3Color and Shape:SolidMolecular weight:319.44Enclomiphene-d4
<p>Enclomiphene-d4 is the deuterium-labeled analog of Enclomiphene. Enclomiphene functions as a potent and orally active estrogen receptor antagonist, exhibiting antiestrogenic properties.</p>Color and Shape:Odour SolidAngiotensin amide
CAS:<p>Angiotensin amide, an octapeptide amide, can be used to increase blood pressure by vasoconstriction.</p>Formula:C49H70N14O11Purity:98%Color and Shape:SolidMolecular weight:1031.17Cgp 29287
CAS:<p>Cgp 29287 is a primate-specific renin inhibitor. It also has a prolonged duration of action.</p>Formula:C72H110N20O15Color and Shape:SolidMolecular weight:1495.77Orphanin FQ(1-11)
CAS:<p>Nociceptin peptide fragment (1-11) with potent ORL1/KOR-3 receptor agonism (Ki = 55 nM), no opioid receptor affinity, and analgesic in mice.</p>Formula:C49H75N15O14Purity:98%Color and Shape:SolidMolecular weight:1098.2Urotensin II (114-124), human TFA
<p>Urotensin II (114-124), human TFA, is an 11-amino acid peptide and potent vasoconstrictor, acting as GPR14 agonist.</p>Formula:C66H86F3N13O20S2Purity:98%Color and Shape:SolidMolecular weight:1502.59Zavacorilant
CAS:<p>Zavacorilant is capable of modulating glucocorticoid receptor (GR).</p>Formula:C25H26FN7O3S2Color and Shape:SolidMolecular weight:555.65ARD-2051
CAS:<p>ARD-2051 is a potent, orally active proteolysis-targeting chimera degrader of the androgen receptor (AR), exhibiting DC50 values of 0.6 nM in degrading AR</p>Formula:C43H45ClN8O5Purity:98%Color and Shape:SolidMolecular weight:789.32UFP-101
CAS:<p>Strong, selective NOP receptor antagonist with pKi=10.24; >3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.</p>Formula:C82H138N32O21Purity:98%Color and Shape:SolidMolecular weight:1908.19Herkinorin
CAS:<p>Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.</p>Formula:C28H30O8Color and Shape:SolidMolecular weight:494.53
