Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(209 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(49 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(298 products)
- Prostaglandin Receptor(120 products)
- RAAS(87 products)
- Reductase(52 products)
- Somatostatin(49 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
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Found 3184 products of "Endocrinology/Hormones"
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Desketoraloxifene
CAS:<p>Desketoraloxifene is a selective estrogen receptor modulator, inhibiting mammalian PLD (PLD1 and PLD2).</p>Formula:C27H27NO3SPurity:98%Color and Shape:SolidMolecular weight:445.57HG122
CAS:<p>HG122 promotes AR degradation via proteasome, inhibiting castration-resistant prostate cancer.</p>Formula:C15H13N5O5Color and Shape:SolidMolecular weight:343.29Aldose reductase-IN-2
CAS:<p>Aldose reductase-IN-2 (5f) inhibits AR with antioxidant effects; potential anti-diabetic drug.</p>Formula:C25H28N4O5Color and Shape:SolidMolecular weight:464.51FK-739 free acid
CAS:<p>FK-739, an angiotensin II receptor blocker, inhibits rat aorta binding (IC50=8.6 nM) but not bovine cerebellum.</p>Formula:C24H23N7Purity:98%Color and Shape:SolidMolecular weight:409.49GSK706
CAS:<p>GSK706 is a novel effective agonist of the GPR119.</p>Formula:C23H29N5O4SPurity:98%Color and Shape:SolidMolecular weight:471.57Lubabegron fumarate
CAS:<p>Lubabegron (LY591281, LY488756 fumarate) is a beta-agonist approved in 2018 to lower ammonia in cattle waste, aiding environment and health.</p>Formula:C29H29N3O3SC4H4O4Color and Shape:SolidMolecular weight:557.66Viminol
CAS:<p>Viminol is an opioid analgesic. Viminol is based on the α-pyrryl-2-aminoethanol structure, unlike any other class of opioids.</p>Formula:C21H31ClN2OPurity:98%Color and Shape:SolidMolecular weight:362.94JTC-801 free base
CAS:<p>JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).</p>Formula:C26H25N3O2Purity:98%Color and Shape:SolidMolecular weight:411.5(R)-DPN
CAS:<p>estrogen receptor (ER) β agonist</p>Formula:C15H13NO2Purity:98%Color and Shape:SolidMolecular weight:239.27Estrogen receptor β antagonist 2
CAS:<p>Estrogen receptor β antagonist 2 is a selective, potent estrogen receptor β (ERβ) antagonist that acts on Erα (IC50: 109.10 μM) and Erβ (IC50: 0.63 μM).</p>Formula:C23H26N2O6Color and Shape:SolidMolecular weight:426.46Zuclomiphene citrate
CAS:<p>Zuclomiphene citrate, a cis isomer of Clomiphene, has stronger antiestrogenic effects and better inhibits LH secretion.</p>Formula:C32H36ClNO8Purity:98%Color and Shape:SolidMolecular weight:598.08SIM-688
CAS:<p>SIM-688 is a selective and orally active estrogen receptor inhibitor of NF-κB transcriptional activity (IC50 = 122 nM in HAECT-1 cells).</p>Formula:C34H31F3N2O2Purity:99.56%Color and Shape:SolidMolecular weight:556.62Olmesartan methyl ester
CAS:<p>Olmesartan methyl ester: an intermediate for synthesizing Olmesartan medoxomil, a strong AT1 receptor blocker.</p>Formula:C25H28N6O3Color and Shape:SolidMolecular weight:460.53Aldose reductase-IN-6
CAS:<p>AR inhibitor Aldose reductase-IN-6: IC50 3.164 μM, Ki 0.018 μM, non-toxic to normal cells.</p>Formula:C20H16N4O2SColor and Shape:SolidMolecular weight:376.43Aldose reductase-IN-4
CAS:<p>Aldose reductase-IN-4 (compund IIc) is an inhibitor of aldose reductase with IC50s of 11.70 μM and 0.98 μM for ALR1 and ALR2, respectively [1].</p>Formula:C14H10FNO3SColor and Shape:SolidMolecular weight:291.3Cyprodinil
CAS:<p>Cyprodinil is a fungicide blocking methionine synthesis in fungi and hinders B. cinerea, P. herpotrichoides, H. oryzae growth; it's also an AR agonist.</p>Formula:C14H15N3Color and Shape:SolidMolecular weight:225.29Idoxifene
CAS:<p>Idoxifene is a tissue-specific selective estrogen receptor modulator.</p>Formula:C28H30INOColor and Shape:SolidMolecular weight:523.45LY 281217
CAS:<p>LY 281217, an organic opioid agonist, can produce analgesic effects in mice.</p>Formula:C32H42N4O6Purity:98%Color and Shape:SolidMolecular weight:578.7Dehydro Olmesartan
CAS:<p>Dehydro Olmesartan, from Olmesartan, is an AT1R blocker for researching hypertension.</p>Formula:C24H24N6O2Color and Shape:SolidMolecular weight:428.49FERb 033
CAS:<p>ERβ receptor agonist</p>Formula:C13H9ClFNO3Purity:98%Color and Shape:SolidMolecular weight:281.67Chlorothalonil
CAS:<p>Chlorothalonil (DAC 2787): Broad-spectrum, efficient, low-toxicity fungicide for fruits, vegetables, rice, wheat, cotton.</p>Formula:C8Cl4N2Purity:98.01% - 98.71%Color and Shape:Colorless Crystals SolidMolecular weight:265.91LY285434
CAS:<p>LY285434 is a suitable angiotensin II receptor antagonist.</p>Formula:C23H25N5O2Purity:98%Color and Shape:SolidMolecular weight:403.48(R,R)-THC
CAS:<p>agonist at ERα receptor and antagonist at ERβ receptor</p>Formula:C22H24O2Purity:98%Color and Shape:SolidMolecular weight:320.42ATC0065 HCl
CAS:<p>ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.</p>Formula:C25H31BrCl2F3N5OColor and Shape:SolidMolecular weight:625.35SB 706375
CAS:<p>urotensin-II (UT) receptor antagonist</p>Formula:C20H22BrF3N2O5SPurity:98%Color and Shape:SolidMolecular weight:539.36FSHR agonist 1
CAS:<p>FSHR agonist 1: high-affinity, allosteric FSHR activator, pEC50 of 7.72, interacts with TMD.</p>Formula:C26H33N3O3SColor and Shape:SolidMolecular weight:467.62SB-568849
CAS:<p>SB-568849 is a melanin-concentrating hormone receptor 1 antagonist (pKi: 7.7).</p>Formula:C28H31F3N2O3Purity:98%Color and Shape:SolidMolecular weight:500.55DK3
CAS:<p>DK3 is a potent and selective agonist of estrogen-related receptor alpha (ERRα). ERRα is a potential drug target for cancer and metabolic diseases [1].</p>Formula:C16H14N2O2Color and Shape:SolidMolecular weight:266.29Nitromifene
CAS:<p>Nitromifene is the estrogen receptor antagonist.</p>Formula:C27H28N2O4Purity:98%Color and Shape:SolidMolecular weight:444.52Levormeloxifene
CAS:<p>Levormeloxifene is a selective modulator of the estrogen receptor. It inhibits the production of vaginal tropoelastin and transforming growth factor-beta 1.</p>Formula:C30H35NO3Purity:98%Color and Shape:SolidMolecular weight:457.6Glucocorticoid receptor-IN-2
CAS:<p>Glucocorticoid receptor-IN-2 selectively targets GR with anti-inflammatory effects (IC50: 0.171 nM) and activates MMTV (EC50: 0.94 nM).</p>Formula:C25H20F4N6O2Color and Shape:SolidMolecular weight:512.46AT1R antagonist 1
CAS:<p>AT1R Antagonist 1 (compound 10) serves as a potent, selective ligand for AT1R with considerable affinity, demonstrated by a K i value of 8.5 nM [1].</p>Formula:C28H32F3N5O4S2Color and Shape:SolidMolecular weight:623.71ALR2-IN-2
<p>ALR2-IN-2 inhibits ALR2 (27 nM IC50) & ALR1 (228 nM IC50), used in diabetes complication research.</p>Formula:C17H11FN2O2S2Color and Shape:SolidMolecular weight:358.41Aldose reductase-IN-5
CAS:<p>Aldose reductase-IN-5 inhibits ALR2, boosts inhibitory response and antioxidants, slowing diabetes complications.</p>Formula:C18H15NO5Color and Shape:SolidMolecular weight:325.32Gumelutamide
CAS:<p>Gumelutamide, a tetrahydropyridopyrimidine compound, functions as both an antiandrogen and an antineoplastic agent by acting as an androgen antagonist.</p>Formula:C22H21ClN6OColor and Shape:SolidMolecular weight:420.89GSK1104252A
CAS:<p>GSK1104252A is a potent and selective agonist of GPR119.</p>Formula:C22H27FN4O5SPurity:98%Color and Shape:SolidMolecular weight:478.54Estrogen receptor antagonist 1
CAS:<p>"Potent estrogen receptor blocker with promise for breast cancer treatment per WO2021249533A1."</p>Formula:C28H33F4N5Color and Shape:SolidMolecular weight:515.59Xelaglifam
CAS:<p>Xelaglifam is a potent agonist of G protein-coupled receptor 40 (GPR40) and exhibits hypoglycemic effects.</p>Formula:C30H28FNO5Color and Shape:SolidMolecular weight:501.55Estrogen receptor antagonist 2
CAS:<p>ER antagonist 2 selectively suppresses ERα, a key breast cancer driver, with research potential in the disease.</p>Formula:C26H31F4N5Color and Shape:SolidMolecular weight:489.55ML138
CAS:<p>ML138 is a probe for MLPCN, an agonist of the κ opioid receptor.</p>Formula:C19H14Cl2N4OSColor and Shape:SolidMolecular weight:417.31FFA1 agonist-1
CAS:<p>FFA1 agonist-1 (Compound 17a) is an orally active fatty acid receptor (FFA1) agonist (EC50: 0.75 μM).</p>Formula:C27H36ClNO3Color and Shape:SolidMolecular weight:458.04TFM-4AS-1
CAS:<p>androgen receptor modulator</p>Formula:C27H33F3N2O2Purity:98%Color and Shape:SolidMolecular weight:474.56RU 752
CAS:<p>RU 752 is an antagonist of mineralocorticoid receptor that inhibits aldosterone synthesis.</p>Formula:C22H30O4Purity:98%Color and Shape:SolidMolecular weight:358.47Androgen receptor antagonist 4
CAS:<p>Compound AT2 is an AR inhibitor with anticancer effects, blocking DHT action and AR nuclear translocation (IC50=0.15μM).</p>Formula:C22H18ClNColor and Shape:SolidMolecular weight:331.84Liothyronine HCl
CAS:<p>Liothyronine is a T3 thyroid hormone normally synthesized and secreted by the thyroid gland in much smaller quantities than thyroxine.</p>Formula:C15H13ClI3NO4Purity:98%Color and Shape:SolidMolecular weight:687.43TCS 3035
CAS:<p>GPR35 agonist 4 (compound 10), pEC50 5.86, potent in human/rat but inactive with R3.36 mutation.</p>Formula:C12H9NO5SColor and Shape:SolidMolecular weight:279.27EMD 66684
CAS:<p>angiotensin AT1 receptor antagonist</p>Formula:C28H31ClN8O2Purity:98%Color and Shape:SolidMolecular weight:547.06ALR2-IN-3
<p>ALR2-IN-2 inhibits ALR2 strongly (IC50: 22 nM) and ALR1 less (IC50: 116 nM), used in diabetes complication studies.</p>Formula:C17H12N2O3S2Color and Shape:SolidMolecular weight:356.42AS1907417
CAS:<p>AS1907417 is a GPR119 agonist.</p>Formula:C19H27N3O4SColor and Shape:SolidMolecular weight:393.5ATC0065
CAS:<p>ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.</p>Formula:C25H29BrF3N5OColor and Shape:SolidMolecular weight:552.43
