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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3183 products of "Endocrinology/Hormones"

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  • (±)-AC 7954 hydrochloride

    CAS:
    <p>(±)-AC 7954 hydrochloride is a urotensin-II (UT) receptor activator.</p>
    Formula:C19H21Cl2NO2
    Purity:99.42%
    Color and Shape:White Solid
    Molecular weight:366.28
  • DK3

    CAS:
    <p>DK3 is a potent and selective agonist of estrogen-related receptor alpha (ERRα). ERRα is a potential drug target for cancer and metabolic diseases [1].</p>
    Formula:C16H14N2O2
    Color and Shape:Solid
    Molecular weight:266.29
  • SHR1653

    CAS:
    <p>SHR1653 is a highly potent, selective and brain penetrated antagonist of oxytocin receptor (OTR)(IC50 of 15 nM for hOTR).</p>
    Formula:C21H21ClFN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:429.88
  • Capesaris

    CAS:
    <p>Capesaris (GTX-758) is an oral estrogen receptor α agonist, used in prostate cancer research.</p>
    Formula:C19H13F2NO3
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:341.31
  • Androgen receptor antagonist 1

    CAS:
    <p>Androgen receptor antagonist 1, an oral full AR antagonist (IC50 59 nM), for PROTAC synthesis, reducing AR protein by 24–47% in LNCaP cells at 1–10 μM.</p>
    Formula:C21H25ClN4O3
    Purity:99.054%
    Color and Shape:Solid
    Molecular weight:416.9
  • PF-4455242 HCl

    CAS:
    <p>PF-4455242 HCl is a selective and orally available κ-opioid receptor antagonist that exhibiting antidepressant effects.</p>
    Formula:C21H29ClN2O2S
    Purity:99.59%
    Color and Shape:Solid
    Molecular weight:408.99
  • SB-568849

    CAS:
    <p>SB-568849 is a melanin-concentrating hormone receptor 1 antagonist (pKi: 7.7).</p>
    Formula:C28H31F3N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:500.55
  • Dimethomorph

    CAS:
    <p>Dimethomorph is a fungicide and sterol biosynthesis inhibitor that inhibits fungal cell wall formation,. inhibits androgen receptor (AR) .</p>
    Formula:C21H22ClNO4
    Purity:99.2%
    Color and Shape:Solid Crystalline
    Molecular weight:387.86
  • FSHR agonist 1

    CAS:
    <p>FSHR agonist 1: high-affinity, allosteric FSHR activator, pEC50 of 7.72, interacts with TMD.</p>
    Formula:C26H33N3O3S
    Color and Shape:Solid
    Molecular weight:467.62
  • MCH-1 antagonist 1

    CAS:
    <p>MCH-1 antagonist 1 also inhibits CYP3A4 (IC50: 10μM).MCH-1 antagonist 1 is a potent melanin concentrating hormone (MCH-1) antagonist (Ki: 2.6 nM).</p>
    Formula:C25H26N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.5
  • CP-866087

    CAS:
    <p>CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.</p>
    Formula:C24H28N2O2
    Purity:99.56% - >99.99%
    Color and Shape:Soild
    Molecular weight:376.49
  • SB 706375

    CAS:
    <p>urotensin-II (UT) receptor antagonist</p>
    Formula:C20H22BrF3N2O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:539.36
  • ATC0065 HCl

    CAS:
    <p>ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.</p>
    Formula:C25H31BrCl2F3N5O
    Color and Shape:Solid
    Molecular weight:625.35
  • GPR84 antagonist 8

    CAS:
    <p>GPR84 antagonist 8 is a selective GPR84 antagonist applicable for investigating inflammatory and fibrotic diseases.</p>
    Formula:C23H23N3O5
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:421.45
  • VPC-3033

    CAS:
    <p>VPC-3033 is an antagonist of the androgen receptor. It acts by inhibiting the LNCaP cell line as well as cell lines with the wild-type androgen receptor.</p>
    Formula:C21H14O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:298.33
  • Camizestrant

    CAS:
    <p>Camizestrant (Estrogen receptor antagonist 2) is an antagonist of the estrogen receptor and can be used in studies about ER+ HER2-advanced breast cancer[1].</p>
    Formula:C24H28F4N6
    Purity:97.25% - 99.57%
    Color and Shape:Solid
    Molecular weight:476.51
  • L 366682

    CAS:
    <p>L 366682 is an oxytocin antagonist.</p>
    Formula:C40H53N9O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:755.91
  • OT antagonist 1

    CAS:
    <p>OT antagonist 1 is a potent and selective antagonist of Oxytocin(Ki of 50 nM)</p>
    Formula:C22H22N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:390.44
  • VPC-13789

    CAS:
    <p>VPC-13789: potent, selective oral antiandrogen for CRPC with 0.19 μM IC50 in LNCaP cells.</p>
    Formula:C21H16F3N3O
    Color and Shape:Solid
    Molecular weight:383.37
  • Dup 747

    CAS:
    <p>Dup 747 is an analgesic that binds with high affinity and selectivity to the kappa-opioid receptor.</p>
    Formula:C24H28Cl2N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:447.4
  • (R,R)-THC

    CAS:
    <p>agonist at ERα receptor and antagonist at ERβ receptor</p>
    Formula:C22H24O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:320.42
  • LY285434

    CAS:
    <p>LY285434 is a suitable angiotensin II receptor antagonist.</p>
    Formula:C23H25N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:403.48
  • Chlorothalonil

    CAS:
    <p>Chlorothalonil (DAC 2787): Broad-spectrum, efficient, low-toxicity fungicide for fruits, vegetables, rice, wheat, cotton.</p>
    Formula:C8Cl4N2
    Purity:98.01% - 98.71%
    Color and Shape:Colorless Crystals Solid
    Molecular weight:265.91
  • D36

    CAS:
    <p>D36 is an androgen receptor allosteric antagonist. It also has inverse agonist properties.</p>
    Formula:C21H24N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:336.43
  • FERb 033

    CAS:
    <p>ERβ receptor agonist</p>
    Formula:C13H9ClFNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:281.67
  • BTI-A-404

    CAS:
    <p>BTI-A-404 is a potent and selective competitive inverse agonist of human GPR43.</p>
    Formula:C22H26N4O2
    Color and Shape:Solid
    Molecular weight:378.47
  • MK-4541

    CAS:
    <p>MK-4541: oral, selective AR modulator, blocks 5α-reductase, curbs AR+ prostate cancer growth, effective in mouse model.</p>
    Formula:C22H31F3N2O3
    Color and Shape:Solid
    Molecular weight:428.49
  • SCH 221510

    CAS:
    <p>SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.</p>
    Formula:C28H31NO
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:397.55
  • Fenhexamid

    CAS:
    <p>Fenhexamid (Elevate), a sterol biosynthesis inhibitor, shows antifungal activity against the plant pathogenic fungus.</p>
    Formula:C14H17Cl2NO2
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:302.20
  • Dehydro Olmesartan

    CAS:
    <p>Dehydro Olmesartan, from Olmesartan, is an AT1R blocker for researching hypertension.</p>
    Formula:C24H24N6O2
    Color and Shape:Solid
    Molecular weight:428.49
  • KB-130015

    CAS:
    <p>KB-130015, a activator of hERG1 potassium channels, blocks native and recombinant hERG1 channels at high voltages.</p>
    Formula:C18H14I2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:548.11
  • RU 43044

    CAS:
    <p>RU 43044 is a selective glucocorticoid receptor antagonist that has exhibited an antidepressant-like effect.</p>
    Formula:C29H34O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.58
  • LY 281217

    CAS:
    <p>LY 281217, an organic opioid agonist, can produce analgesic effects in mice.</p>
    Formula:C32H42N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:578.7
  • Idoxifene

    CAS:
    <p>Idoxifene is a tissue-specific selective estrogen receptor modulator.</p>
    Formula:C28H30INO
    Color and Shape:Solid
    Molecular weight:523.45
  • L-366509

    CAS:
    <p>L-366,509 is an antagonist of oxytocin.</p>
    Formula:C25H33NO5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:459.6
  • Cyprodinil

    CAS:
    <p>Cyprodinil is a fungicide blocking methionine synthesis in fungi and hinders B. cinerea, P. herpotrichoides, H. oryzae growth; it's also an AR agonist.</p>
    Formula:C14H15N3
    Color and Shape:Solid
    Molecular weight:225.29
  • DDD028

    CAS:
    <p>DDD-028 is a potential non-opioid and non-cannabinoid analgesic. It was used for treating neuropathic and inflammatory pain.</p>
    Formula:C20H20N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:288.39
  • Androgen receptor antagonist 3

    CAS:
    <p>Androgen receptor antagonist 3 (Compound C18) has anticancer activities that is an antagonist of androgen receptor (AR) (IC 50 = 2.4 μM) [1].</p>
    Formula:C22H18ClN
    Color and Shape:Solid
    Molecular weight:331.84
  • J9

    CAS:
    <p>J9 is an inhibitor of Glucocorticoid resistance. J9 reverses Dexamethasone Resistance in T-cell Acute Lymphoblastic Leukemia.</p>
    Formula:C12H12N4
    Color and Shape:Solid
    Molecular weight:212.25
  • Aldose reductase-IN-4

    CAS:
    <p>Aldose reductase-IN-4 (compund IIc) is an inhibitor of aldose reductase with IC50s of 11.70 μM and 0.98 μM for ALR1 and ALR2, respectively [1].</p>
    Formula:C14H10FNO3S
    Color and Shape:Solid
    Molecular weight:291.3
  • Aldose reductase-IN-6

    CAS:
    <p>AR inhibitor Aldose reductase-IN-6: IC50 3.164 μM, Ki 0.018 μM, non-toxic to normal cells.</p>
    Formula:C20H16N4O2S
    Color and Shape:Solid
    Molecular weight:376.43
  • BMS-819881

    CAS:
    <p>BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM and it also is selective and potent for</p>
    Formula:C24H21ClN2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:468.95
  • Olmesartan methyl ester

    CAS:
    <p>Olmesartan methyl ester: an intermediate for synthesizing Olmesartan medoxomil, a strong AT1 receptor blocker.</p>
    Formula:C25H28N6O3
    Color and Shape:Solid
    Molecular weight:460.53
  • GPR40 agonist 1

    CAS:
    <p>GPR40 agonist 1 is an effective new GPR40 agonist (EC50s: 17 nM and 2 nM for rGPR40 and hGPR40).</p>
    Formula:C27H30FN3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:479.54
  • Endomorphin 1 acetate

    CAS:
    <p>Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can be used to study neurological diseases.</p>
    Formula:C36H42N6O7
    Color and Shape:Solid
    Molecular weight:670.75
  • SIM-688

    CAS:
    <p>SIM-688 is a selective and orally active estrogen receptor inhibitor of NF-κB transcriptional activity (IC50 = 122 nM in HAECT-1 cells).</p>
    Formula:C34H31F3N2O2
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:556.62
  • ORL1 antagonist 1

    CAS:
    <p>ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).</p>
    Formula:C20H22ClN5
    Purity:98.92%
    Color and Shape:Solid
    Molecular weight:367.88
  • Opioid receptor modulator 1

    CAS:
    <p>Opioid receptor modulator 1 is a modulator of opioid receptor.</p>
    Formula:C18H23NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:285.38
  • BMS-986124

    CAS:
    <p>BMS-986124 is an allosteric modulator of the μ-Opioid Receptor.</p>
    Formula:C16H15BrClNO3S2
    Color and Shape:Solid
    Molecular weight:448.78
  • Estrogen receptor-IN-1

    CAS:
    <p>Estrogen receptor-IN-1 (compound 16) is an effective estrogen receptor (ER) inhibitor with IC 50 s of 13, 5μM for ERα and Erβ, respectively [1].</p>
    Formula:C14H16OSi
    Color and Shape:Solid
    Molecular weight:228.36