Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(229 products)
- Annexin A(16 products)
- Aromatase(23 products)
- Estrogen/progestogen Receptor(66 products)
- GPR(1 products)
- Glucocorticoid Receptor(165 products)
- LHRH(2 products)
- Opioid Receptor(327 products)
- Prostaglandin Receptor(122 products)
- RAAS(89 products)
- Reductase(51 products)
- Somatostatin(57 products)
- Thyroid hormone receptor(THR)(33 products)
- Vasopressin Receptor(48 products)
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Found 3420 products of "Endocrinology/Hormones"
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PD 117302
CAS:PD 117302: nonpeptide, kappa-opioid agonist, anti-arrhythmic, anticonvulsant, impacts locomotion, diuresis.Formula:C21H28N2OSColor and Shape:SolidMolecular weight:356.52THR-β agonist 3
CAS:THR-β agonist 3 is a potent agonist of THR-β.Formula:C29H32ClO5PColor and Shape:SolidMolecular weight:526.99Androgen receptor-IN-5
CAS:Androgen receptor-IN-5 is a potent inhibitor of the androgen receptor with anticancer properties.Formula:C22H10Cl2F4N4OSPurity:98%Color and Shape:SolidMolecular weight:525.31LY303336
CAS:LY303336 is an antagonist of AT1 receptor.Formula:C30H37N4O11PSPurity:98%Color and Shape:SolidMolecular weight:692.67MCHR1 antagonist 3
CAS:MCHR1 antagonist 3, a potent antagonist of the melanin-concentrating hormone receptor-1 (MCHR1), is employed for the regulation of energy metabolism.Formula:C29H36N4O2Purity:98%Color and Shape:SolidMolecular weight:472.6210β,17β-dihydroxyestra-1,4-dien-3-one
CAS:10β,17β-dihydroxyestra-1,4-dien-3-one (DHED) has neuroprotective effects, can improve cognitive dysfunction, and can be used to study brain injury.Formula:C18H24O3Color and Shape:SolidMolecular weight:288.38GPR120 Agonist 1
CAS:GPR120 Agonist 1 selectively activates human/mouse GPR120 with EC50 of 42/77 nM in HEK293 cells.Formula:C20H12ClF6NO3SPurity:98%Color and Shape:SolidMolecular weight:495.82CYT-1010
CAS:CYT-1010, a mu-opioid receptor agonist; EC50: β-arrestin, 13.1 nM; cAMP, 0.0053 nM. Extracted from patent WO2013173730A2.Formula:C35H40N6O5Purity:98%Color and Shape:SolidMolecular weight:624.73N-Demethyl Mifepristone
CAS:N-Demethyl Mifepristone (RU 42633), an active metabolite of Mifepristone, exhibits 61% of the affinity for the glucocorticoid receptor relative to Mifepristone'Formula:C28H33NO2Purity:98%Color and Shape:SolidMolecular weight:415.57Firuglipel
CAS:Firuglipel is an orally available and selective agonist of GPR119.Formula:C25H26FN3O5Purity:98%Color and Shape:SolidMolecular weight:467.49MCHR1 antagonist 2
CAS:MCHR1 antagonist 2 is an antagonist of melanin-concentratin hormone receptor 1(MCH1-R, IC50 = 65 nM) and also inhibits hERG.Formula:C23H21FN2O5Purity:98.29%Color and Shape:SolidMolecular weight:424.42Ref: TM-T11966
2mg43.00€5mg66.00€1mL*10mM (DMSO)80.00€10mg100.00€25mg210.00€50mg334.00€100mg537.00€200mg710.00€Halobetasol
CAS:Halobetasol (Ulobetasol), a corticosteroid, is utilized in the research of severe localized psoriasis [1].Formula:C22H27ClF2O4Purity:98%Color and Shape:SolidMolecular weight:428.9μ opioid receptor agonist 3
CAS:Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.Formula:C22H28N2O2Purity:98%Color and Shape:SolidMolecular weight:352.47TA-606
CAS:TA-606 is an angiotensin type 1 receptor antagonist with antihypertensive activity.Formula:C33H40ClN7O6Color and Shape:SolidMolecular weight:666.17AMG 837 sodium salt
CAS:AMG 837 sodium salt: potent GPR40 agonist, EC50=13 nM; enhances insulin secretion; superior pharmacokinetics.Formula:C26H21F3NaO3Purity:98%Color and Shape:SolidMolecular weight:461.436GPR139 agonist-2
CAS:GPR139 agonist-2 (compound 20a), a potent GPR139 agonist with an EC50 of 24.7 nM, has demonstrated efficacy in rescuing social interaction deficits andFormula:C17H15F3N4O3Color and Shape:SolidMolecular weight:380.32Fulvestrant (R enantiomer)
CAS:Fulvestrant R enantiomer is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.Formula:C32H47F5O3SPurity:98%Color and Shape:SolidMolecular weight:606.77Encaleret
CAS:Encaleret( JIT-305) is an antagonist of oral calcium-sensing receptor (CaSR), it is used for the treatment of osteoporosis.Formula:C29H33ClFNO4Color and Shape:SolidMolecular weight:514.03THR-β modulator-1
CAS:THR-β Modulator-1 (Compound 1a) is a potent modulator of the thyroid hormone receptor β, utilized in the study of thyroid hormone receptor-associated disordersFormula:C17H14Cl2N6O4Color and Shape:SolidMolecular weight:437.24Fosdagrocorat
CAS:Fosdagrocorat is an agonist of the dissociated glucocorticoid receptor.Formula:C29H30F3N2O5PColor and Shape:SolidMolecular weight:574.53Epelsiban besylate
CAS:Epelsiban Besylate is an oral drug that is a highly selective anamol oxytocin receptor antagonist.Formula:C36H44N4O7SColor and Shape:SolidMolecular weight:676.83Glucocorticoid receptor agonist
CAS:Glucocorticoid receptor agonist is an effective glucocorticoid receptor agonist.Formula:C20H20F4N2O2Purity:98%Color and Shape:SolidMolecular weight:396.38GPR119 agonist 2
CAS:GPR119 agonist 2 (compound 43), an orally active agonist of GPR119, exhibits favorable pharmacokinetic properties in rodents and has demonstrated efficacy inFormula:C23H24FN5O4S2Color and Shape:SolidMolecular weight:517.6EPI-7170
CAS:EPI-7170: Ralaniten analogue, blocks androgen receptor, inhibits transcription in AR & variants, fights enzalutamide-resistant prostate cancer.Formula:C22H28Cl3NO6SColor and Shape:SolidMolecular weight:540.88Androgen receptor degrader-3
CAS:Androgen Receptor Degrader-3 (ARD-3) is a compound that inhibits androgen receptor signaling and promotes the degradation of the receptor, with potentialFormula:C45H51ClN8O5Purity:98%Color and Shape:SolidMolecular weight:819.39Biotin-cholesterol
CAS:Biotin-cholesterol, a biotinylated derivative of cholesterol, serves as a precursor in the manufacturing of biotin-conjugated liposomes and micelles, which are utilized in drug delivery systems [1].Formula:C37H60N2O3SColor and Shape:SolidMolecular weight:612.9520α-dihydro Prednisolone
CAS:"20α-Dihydro Prednisolone, a prednisolone metabolite, is detected in cattle urine post-adrenocorticotropic hormone (ACTH) administration but absent in both naturally stressed and non-stressed cattle."Formula:C21H30O5Color and Shape:SolidMolecular weight:362.466N-Benzylnaltrindole hydrochloride
CAS:δ2 opioid receptor antagonistFormula:C33H33ClN2O3Purity:98%Color and Shape:SolidMolecular weight:541.08R-84760 hydrochloride
CAS:R-84760, a potent κ-opioid receptor agonist, relieves tonic pain via supraspinal/spinal pathways, activating noradrenergic descent.Formula:C19H25Cl3N2OSColor and Shape:SolidMolecular weight:435.84AKR1C3-IN-6
CAS:AKR1C3-IN-6: Strong AKR1C3 inhibitor (IC50: 0.31 μM); weak on AKR1C2 (IC50: 73.23 μM); shows antitumor effects.Formula:C18H15F3N4O3Color and Shape:SolidMolecular weight:392.33ES 936
CAS:ES 936 is a potent and selective NQO1 inhibitor, inhibiting more than 95% of NQO1 100 nM, with a cell line-dependent inhibition duration.Formula:C18H16N2O6Purity:98%Color and Shape:SolidMolecular weight:356.33GPR88-IN-1
CAS:GPR88-IN-1 is a GPR88 antagonist that may be utilized for the study of central nervous system disorders [1].Formula:C25H28N4O2Color and Shape:SolidMolecular weight:416.52Prodilidine hydrochloride
CAS:Prodilidine hydrochloride is an opioid analgesic.Formula:C15H22ClNO2Color and Shape:SolidMolecular weight:283.79LX-039
CAS:LX-039: Selective oral estrogen receptor degrader with EC50 of 2.99 nM, antitumor activity, C-3 indole chloride, and robust mouse pharmacokinetics.Formula:C27H20Cl2FNO2Color and Shape:SolidMolecular weight:480.36Trap-101 hydrochloride
CAS:nociceptin/orphanin FQ (NOP) receptor antagonistFormula:C24H36ClN3O2Purity:98%Color and Shape:SolidMolecular weight:434.02DPP-4/GPR119 modulator 2
CAS:DPP-4/GPR119 modulator 2 is an inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 0.22 μM) and an agonist of GPR119 (EC50: 0.95 μM).Formula:C30H40N8O3Color and Shape:SolidMolecular weight:560.69Fulvestrant (S enantiomer)
CAS:Fulvestrant S enantiomer is the less active S enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.Formula:C32H47F5O3SPurity:98%Color and Shape:SolidMolecular weight:606.77THRβ receptor agonist-1
CAS:THRβ receptor agonist-1 is an agonist for the THRβ receptor [1].Formula:C18H12Cl2N6O4Color and Shape:SolidMolecular weight:447.23Nylestriol
CAS:Nylestriol (LY 49825) is an agonist of estrogen receptor.Formula:C25H32O3Purity:98.88%Color and Shape:SolidMolecular weight:380.52Ref: TM-T20744
2mg34.00€5mg50.00€1mL*10mM (DMSO)54.00€10mg71.00€25mg104.00€50mg152.00€100mg219.00€200mg310.00€DuP-532
CAS:DuP-532, an angiotensin type 1 receptor antagonist, is used potentially for the treatment of hypertension and heart failure.Formula:C23H19F5N6O2Color and Shape:SolidMolecular weight:506.43Dagrocorat
CAS:Dagrocorat is a novel and dissociated agonist of glucocorticoid receptor.Formula:C29H29F3N2O2Purity:98%Color and Shape:SolidMolecular weight:494.55CL-329167
CAS:CL-329167 (compound 12) is an orally active, competitive angiotensin II receptor antagonist (IC50=6 nM) suitable for hypertension research.Formula:C30H32N6O2Purity:99.08% - 99.42%Color and Shape:SolidMolecular weight:508.61Etiroxate
CAS:Etiroxate (CG-635) is a lipid-lowering agent utilized in hyperlipoproteinemia studies [1].Formula:C18H17I4NO4Color and Shape:SolidMolecular weight:818.95MR2034
CAS:MR2034 is an agonist of kappa-Opioid receptor. MR2034 stimulates hypothalamic-pituitary-adrenal axis.Formula:C19H27NO2Color and Shape:SolidMolecular weight:301.42TRβ agonist 3
CAS:TRβ agonist 3 (Compound 3) is a potent TRβ agonist that is a new potential TRβ-selective thyromimetics.Formula:C20H25NO3Color and Shape:SolidMolecular weight:327.42Zopolrestat
CAS:Zopolrestat (CP 73850) is a potent inhibitor of aldose reductase (IC50 = 3.1 nM).Formula:C19H12F3N3O3SPurity:99.74%Color and Shape:SolidMolecular weight:419.38Nurr1 agonist 4
CAS:Nurr1 agonist 4 (compound 8) serves as a potent Nurr1 agonist, exhibiting an EC50 value of 2.1 μM [1].Formula:C12H10O4Purity:98%Color and Shape:SolidMolecular weight:218.21Estrogen receptor antagonist 3
CAS:ER antagonist 3 degrades ER, crucial in cell regulation; ER antagonist 4 may aid cancer research. (Patent WO2021213358A1, compound 7)Formula:C26H29BF6N4O2Color and Shape:SolidMolecular weight:554.34RU 58668
CAS:Pure antiestrogen that downregulates estrogen receptor expressionFormula:C34H43F5O5SPurity:98%Color and Shape:SolidMolecular weight:658.76JNJ-17148066
CAS:JNJ-17148066 is an agonist of estrogen receptor ESR1.Formula:C30H31NO5Purity:98%Color and Shape:SolidMolecular weight:485.57
