Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(229 products)
- Annexin A(16 products)
- Aromatase(22 products)
- Estrogen/progestogen Receptor(55 products)
- GPR(1 products)
- Glucocorticoid Receptor(167 products)
- LHRH(1 products)
- Opioid Receptor(322 products)
- Prostaglandin Receptor(122 products)
- RAAS(90 products)
- Reductase(50 products)
- Somatostatin(54 products)
- Thyroid hormone receptor(THR)(30 products)
- Vasopressin Receptor(46 products)
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Found 3359 products of "Endocrinology/Hormones"
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Tamoxifen-PEG-Clozapine
Tamoxifen-PEG-Clozapine is an estrogen receptor α (ERα) PROTAC degrader. It targets ERα for degradation through the ubiquitin-proteasome system by utilizing the E3 ubiquitin ligase component N-recognin 5. This compound is applicable in cancer research. (Pink: ERα inhibitor; Black: linker; Blue: CRBN Ligand)Formula:C54H63ClN6O7Color and Shape:SolidMolecular weight:943.567AR ligand-33
<p>AR ligand-33 is a ligand for the androgen receptor (AR), and it can be used as a target protein ligand for the synthesis of PROTAC AR Degrader-8.</p>Formula:C25H28N2O3Color and Shape:SolidMolecular weight:404.501RU26988
CAS:RU26988 is a bioactive chemical.Formula:C22H26O3Color and Shape:SolidMolecular weight:338.44Paramethasone
CAS:Parametasone is a glucocorticoid with the general properties of corticosteroids.Formula:C22H29FO5Color and Shape:SolidMolecular weight:392.46GPR88 agonist 2
GPR88 agonist 2 (compound 53) serves as a potent, brain-penetrant agonist of GPR88, exhibiting an EC50 of 14 µM in the GPR88 cAMP functional assay [1].Color and Shape:Odour SolidGalloylalbiflorin
CAS:Galloylalbiflorin, an AR antagonist with IC50 53.3μM, is sourced from Paeonia lactiflora roots, exhibiting anti-androgenic properties.Formula:C30H32O15Color and Shape:SolidMolecular weight:632.57TD-802
CAS:TD-802, an AR-targeting PROTAC with microsomal stability, shows promise for castration-resistant prostate cancer.Formula:C52H61ClN10O6Color and Shape:SolidMolecular weight:957.56Human PTHrP-(1-36)
CAS:Human PTHrP-(1-36) is a secreted form of parathyroid hormone-related protein that exhibits anticalciuric effects and promotes beta cell function andFormula:C191H305N59O52Molecular weight:4259.83Demoxytocin
CAS:Demoxytocin, oxytocin analog, enhances smooth muscle contraction by increasing calcium ion permeability. Used in labor research.Formula:C43H65N11O12S2Molecular weight:992.17GNE-502
CAS:GNE-502 is an orally active and potent estrogen receptor (ER) degrader, specifically designed for research on breast cancer.Formula:C25H30FN3O3SColor and Shape:SolidMolecular weight:471.59Clocinnamox mesylate
CAS:Clocinnamox mesylate: irreversible μ-opioid blocker; Ki: 0.7 nM (mouse μ), 1.9 nM (δ), 5.7 nM (κ).Formula:C30H33ClN2O7SColor and Shape:SolidMolecular weight:601.11CP 85339
CAS:CP 85339 is an aspartic acid protease inhibitor for X-ray analysis of peptide-renin complexes.Formula:C31H49ClN4O6SColor and Shape:SolidMolecular weight:641.26PROTAC ER Degrader-12
PROTACER Degrader-12 (Compound 70) is an estrogen receptor PROTAC degrader with a degradation concentration (DC50) of less than 10 nM. It inhibits the proliferation of MCF-7 cells at a DC50 of under 10 nM and exhibits anticancer properties.Formula:C47H48F3N5O5Molecular weight:819.36075Angiotensin II (3-8), human TFA
Angiotensin II (3-8), human (TFA) is an angiotensin AT1 receptor agonist with less activity.Formula:C42H55F3N8O10Purity:98%Color and Shape:SolidMolecular weight:888.93β-Endorphin (1-27) (human) acetate
<p>β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.</p>Formula:C141H221N33O42SPurity:96.52%Color and Shape:SolidMolecular weight:3082.52β-S-ARCA triammonium
β-S-ARCA (triammonium) is an analog of the mRNA7-methylguanosine (m7G) cap structure, featuring a thio-phosphorylated segment. When bound to mRNA, β-S-ARCA (triammonium) extends the cellular half-life and enhances protein expression. This compound is utilized in research for mRNA-based cancer vaccines.Formula:C22H40N13O17P3SColor and Shape:SolidMolecular weight:883.62PSDalpha
PSDalpha, a conjugate of PS, TB, and 17β-estradiol, degrades ERα with peak absorption at 465 nm, effectively inhibiting MCF-7 cell growth.Formula:C44H39N3O2SColor and Shape:SolidMolecular weight:673.86K-Opioid receptor agonist-1
CAS:K-Opioid receptor agonist-1 (Compound 5a) acts as an agonist for the κ-Opioid receptor, exhibiting a K_i of 0.25 nM and an EC_50 of 2 nM. This compound is capable of crossing the blood-brain barrier (BBB), evidenced by brain/plasma ratios ranging from 0.50 to 0.65. Additionally, K-Opioid receptor agonist-1 demonstrates anti-inflammatory effects in dermatitis models induced by either Arachidonic acid or oxazolidinone.Formula:C22H29Cl2N3O3Molecular weight:454.39[Orn5]-URP acetate
[Orn5]-URP acetate is an effective and selective Urotensin-II receptor (UT) antagonist (pEC50 = 7.24). [Orn5]-URP exhibits no agonist activity.Formula:C50H66N10O12S2Purity:98.4300%Color and Shape:SolidMolecular weight:1063.25Bufrolin
CAS:Bufrolin is a potent GPR35 agonist, mast cell stabilizer, and anti-inflammatory research agent.Formula:C18H16N2O6Color and Shape:SolidMolecular weight:356.33
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