Androgen Receptor
The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.
Found 207 products of "Androgen Receptor"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
MI-136
CAS:<p>MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.</p>Formula:C23H21F3N6SPurity:98.63% - 99.12%Color and Shape:SolidMolecular weight:470.51Apalutamide
CAS:<p>Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.</p>Formula:C21H15F4N5O2SPurity:99.03% - 99.91%Color and Shape:SolidMolecular weight:477.43S-23
CAS:<p>S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) is an oral selective androgen receptor modulator (</p>Formula:C18H13ClF4N2O3Purity:99.55%Color and Shape:SolidMolecular weight:416.75Iprodione
CAS:<p>Iprodione is a fungicide. Iprodione is also used in cannabis testing kits as a component of pesticide mixes.</p>Formula:C13H13Cl2N3O3Purity:98.82%Color and Shape:Colorless Crystals Cream To Colorless Odorless PowderMolecular weight:330.17Testosterone undecanoate
CAS:<p>Testosterone undecanoate is a metabolite of Testosterone, which is a promising androgen for male hormonal contraception.</p>Formula:C30H48O3Purity:99.45% - 99.788%Color and Shape:White Crystalline PowderMolecular weight:456.7CLP-3094
CAS:<p>CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor.</p>Formula:C15H13ClN2OSPurity:99.84%Color and Shape:SolidMolecular weight:304.79AC-262536
CAS:<p>AC-262536 is a selective androgen receptor (SAR) modulator and exhibits potent agonist activity at the androgen receptor.</p>Formula:C18H18N2OPurity:99.88%Color and Shape:SolidMolecular weight:278.35Triptophenolide
CAS:<p>Triptophenolide (Hypolide) is a compound isolated from Tripterygium wilfordii Hook with anti-inflammatory activity.</p>Formula:C20H24O3Purity:98.07% - ≥95%Color and Shape:White PowderMolecular weight:312.4Boldenone Undecylenate
CAS:<p>Boldenone Undecylenate (Parenabol) is a synthetic steroid.</p>Formula:C30H44O3Purity:99.39%Color and Shape:Light Yellow Oily MatterMolecular weight:452.67JNJ-63576253 free base
CAS:<p>JNJ-63576253 free base (TRC253) is a potent and orally active full antagonist of androgen receptor (AR). JNJ-63576253 can be used for the research of CRPC.</p>Formula:C23H21F3N6O2SPurity:98.32%Color and Shape:SolidMolecular weight:502.51Dimethylcurcumin
CAS:<p>Dimethylcurcumin (ASC-J9) (ASC-J9) is an androgen receptor degradation enhancer.</p>Formula:C23H24O6Purity:97.36% - 98.96%Color and Shape:SolidMolecular weight:396.43Nandrolone phenylpropionate
CAS:<p>Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosis</p>Formula:C27H34O3Purity:99.2% - 99.46%Color and Shape:White Or Milky Crystalline PowderMolecular weight:406.56JNJ-63576253
CAS:<p>JNJ-63576253 is a Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC).</p>Formula:C23H22ClF3N6O2SPurity:98.71%Color and Shape:SolidMolecular weight:538.97Ailanthone
CAS:<p>Ailanthone (Δ13-Dehydrochaparrinone) is an effective inhibitor of both full-length androgen receptor (AR) (IC50: 69 nM) and constitutively active truncated AR</p>Formula:C20H24O7Purity:99.71% - 99.96%Color and Shape:SolidMolecular weight:376.43-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
CAS:<p>3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.</p>Formula:C18H14N4OPurity:98.41%Color and Shape:SolidMolecular weight:302.33ARD-2128
CAS:<p>ARD-2128: potent oral PROTAC that degrades AR, curbing prostate cancer growth with no toxicity.</p>Formula:C45H50ClN7O6Purity:98.8%Color and Shape:SolidMolecular weight:820.372-hydroxy Flutamide
CAS:<p>2-hydroxy Flutamide is competitive inhibition of androgen receptor (AR) for the treatment of prostate cancer</p>Formula:C11H11F3N2O4Purity:99.45% - 99.82%Color and Shape:SolidMolecular weight:292.21AH-3960
CAS:<p>AH-3960 是一种甲状腺激素受体 1 (PTHR1) 激动剂。</p>Formula:C13H22N4O3Purity:98.44%Color and Shape:SolidMolecular weight:282.34DSRM-3716
CAS:<p>Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery of</p>Formula:C9H6INPurity:97.28% - 99.785%Color and Shape:SolidMolecular weight:255.06Bavdegalutamide
CAS:<p>Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR).</p>Formula:C41H43ClFN9O6Purity:97.17% - 99.04%Color and Shape:SolidMolecular weight:812.29N-desmethyl Enzalutamide
CAS:<p>N-desmethyl Enzalutamide (N-desmethyl MDV 3100) is the active Enzalutamide metabolite.It is the active metabolite of Enzalutamide.</p>Formula:C20H14F4N4O2SPurity:99.74%Color and Shape:SolidMolecular weight:450.41Enzalutamide carboxylic acid
CAS:<p>Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .</p>Formula:C20H13F4N3O3SPurity:97.88%Color and Shape:SolidMolecular weight:451.39Clascoterone
CAS:<p>Clascoterone (CB-03-01) is a new topical and peripherally selective androgen antagonist.</p>Formula:C24H34O5Purity:99.2% - 99.64%Color and Shape:SolidMolecular weight:402.52LY2452473
CAS:<p>LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer activity for the study of prostate cancer.</p>Formula:C22H22N4O2Purity:99.72%Color and Shape:SolidMolecular weight:374.44Masofaniten
CAS:<p>Masofaniten (EPI-7386) is an orally active androgen receptor (AR) inhibitor with antitumor activity for the study of prostate and breast cancer.</p>Formula:C24H24Cl2N4O4SPurity:98.42% - 98.66%Color and Shape:SolidMolecular weight:535.44AR antagonist 6
CAS:<p>AR antagonist 6 (compound 6i), a diphenyl ether androgen receptor (AR) antagonist, binds to the AR with an affinity of 120 nM. It demonstrates low toxicity and effective in vitro activity in the golden Syrian hamster ear model. [19] [1]</p>Formula:C16H12F3NO2Color and Shape:SolidMolecular weight:307.27GDC-2992
CAS:<p>GDC-2992 is a selective androgen receptor (AR) degradator that degrades AR and inhibits proliferation in VCaP cells,CRPC.</p>Formula:C45H51ClN8O5Purity:99.82%Color and Shape:SoildMolecular weight:819.39Estromustine
CAS:<p>Estromustine, an active metabolite of estramustine phosphate, is used to treat prostate cancer.</p>Formula:C23H29Cl2NO3Color and Shape:SolidMolecular weight:438.39Procymidone
CAS:<p>Procymidone is a broad-spectrum fungicide that inhibits fungal glycerol triester synthesis, thereby disrupting hyphal growth. androgen receptor (AR) antagonist</p>Formula:C13H11Cl2NO2Purity:99.86%Color and Shape:Colorless SolidMolecular weight:284.14JNJ-37654032
CAS:<p>JNJ-37654032: orally active, nonsteroidal SARM. Mixed AR agonist/antagonist. Selective for muscle, grows levator ani, max at 3mg/kg, ED(50) 0.8mg/kg.</p>Formula:C11H7Cl2F3N2OColor and Shape:SolidMolecular weight:311.09BMS-564929
CAS:<p>BMS-564929 is an AR agonist that upregulates the expression and activity of fat-producing enzymes, reducing VAT content and lipid levels.</p>Formula:C14H12ClN3O3Purity:98.17%Color and Shape:SolidMolecular weight:305.72(R)-Bicalutamide
CAS:<p>(R)-Bicalutamide, an AR antagonist with antitumor properties, is crucial in prostate cancer research.</p>Formula:C18H14F4N2O4SColor and Shape:SolidMolecular weight:430.37LG-121071
CAS:<p>LG-121071: oral SARM, high-affinity AR full agonist, Ki=17 nM.</p>Formula:C15H15F3N2OPurity:98%Color and Shape:SolidMolecular weight:296.29Honokiol DCA
CAS:<p>Honokiol DCA inhibits DRP1, enhances respiration via mitochondrial repair, and is active against Vemurafenib-resistant melanoma.</p>Formula:C22H18Cl4O4Color and Shape:SolidMolecular weight:488.19Lubabegron fumarate
CAS:<p>Lubabegron (LY591281, LY488756 fumarate) is a beta-agonist approved in 2018 to lower ammonia in cattle waste, aiding environment and health.</p>Formula:C29H29N3O3SC4H4O4Color and Shape:SolidMolecular weight:557.66Gumelutamide
CAS:<p>Gumelutamide, a tetrahydropyridopyrimidine compound, functions as both an antiandrogen and an antineoplastic agent by acting as an androgen antagonist.</p>Formula:C22H21ClN6OColor and Shape:SolidMolecular weight:420.89TFM-4AS-1
CAS:<p>androgen receptor modulator</p>Formula:C27H33F3N2O2Purity:98%Color and Shape:SolidMolecular weight:474.56HG122
CAS:<p>HG122 promotes AR degradation via proteasome, inhibiting castration-resistant prostate cancer.</p>Formula:C15H13N5O5Color and Shape:SolidMolecular weight:343.29Androgen receptor antagonist 4
CAS:<p>Compound AT2 is an AR inhibitor with anticancer effects, blocking DHT action and AR nuclear translocation (IC50=0.15μM).</p>Formula:C22H18ClNColor and Shape:SolidMolecular weight:331.84AZD3514
CAS:<p>AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM and has ability of reducing AR protein expression.Phase 1.</p>Formula:C25H32F3N7O2Purity:98.09%Color and Shape:SolidMolecular weight:519.56AR antagonist 2
CAS:<p>AR antagonist 2 (compound 58) is a potent inhibitor of the androgen receptor (AR) (IC50: 0.95 μM).</p>Formula:C22H17ClFN5O2SColor and Shape:SolidMolecular weight:469.92AR antagonist 5
CAS:<p>Compound 30a, known as AR Antagonist 5, is a selective androgen receptor (AR) antagonist that demonstrates an IC 50 value of 134.8 nM. It exhibits favorable pharmacokinetic properties, characterized by high skin exposure and low plasma exposure [1].</p>Formula:C23H21F3N6O2Color and Shape:SolidMolecular weight:470.45CSRM617
CAS:<p>CSRM617: selective ONECUT2 inhibitor, Kd 7.43 uM, binds OC2-HOX, induces apoptosis, tolerable in mouse prostate cancer model.</p>Formula:C10H13N3O5Purity:98%Color and Shape:SolidMolecular weight:255.23MK-4541
CAS:<p>MK-4541: oral, selective AR modulator, blocks 5α-reductase, curbs AR+ prostate cancer growth, effective in mouse model.</p>Formula:C22H31F3N2O3Color and Shape:SolidMolecular weight:428.49(R)-UT-155
CAS:<p>(R)-UT-155 is a selective androgen receptor degrader (SARD) ligand.</p>Formula:C20H15F4N3O2Color and Shape:SolidMolecular weight:405.35Carbazole derivative 1
CAS:<p>Carbazole derivative 1 is used to reduce androgen or oestrogen levels in mammals.</p>Formula:C18H13FN2Purity:98%Color and Shape:SolidMolecular weight:276.31VPC-3033
CAS:<p>VPC-3033 is an antagonist of the androgen receptor. It acts by inhibiting the LNCaP cell line as well as cell lines with the wild-type androgen receptor.</p>Formula:C21H14O2Purity:98%Color and Shape:SolidMolecular weight:298.33Androgen receptor antagonist 3
CAS:<p>Androgen receptor antagonist 3 (Compound C18) has anticancer activities that is an antagonist of androgen receptor (AR) (IC 50 = 2.4 μM) [1].</p>Formula:C22H18ClNColor and Shape:SolidMolecular weight:331.84RU 58642
CAS:<p>RU 58642 is an effective systemic antiandrogen for androgen-dependent disorders.</p>Formula:C15H11F3N4O2Purity:98%Color and Shape:SolidMolecular weight:336.27VPC-13789
CAS:<p>VPC-13789: potent, selective oral antiandrogen for CRPC with 0.19 μM IC50 in LNCaP cells.</p>Formula:C21H16F3N3OColor and Shape:SolidMolecular weight:383.37
![3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT9752.webp&w=3840&q=75)
