Androgen Receptor
The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.
Found 229 products of "Androgen Receptor"
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Darolutamide
CAS:Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).Formula:C19H19ClN6O2Purity:97.36% - >99.99%Color and Shape:SolidMolecular weight:398.85Ref: TM-T6915
1mg50.00€2mg66.00€5mg100.00€10mg158.00€25mg250.00€50mg358.00€100mg512.00€200mg732.00€1mL*10mM (DMSO)101.00€Dimethylcurcumin
CAS:Dimethylcurcumin (ASC-J9) (ASC-J9) is an androgen receptor degradation enhancer.Formula:C23H24O6Purity:97.36% - 98.96%Color and Shape:SolidMolecular weight:396.43Testosterone acetate
CAS:Testosterone acetate (NSC-523836) is a hormone with in vitro antitumor activity.Formula:C21H30O3Purity:99.6%Color and Shape:White To Off-White Crystalline PowderMolecular weight:330.46GSK-2881078
CAS:GSK-2881078 is a selective androgen receptor modulato (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting.Formula:C14H13F3N2O2SPurity:98.16% - 98.81%Color and Shape:SolidMolecular weight:330.33MI-136
CAS:MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.Formula:C23H21F3N6SPurity:98.63% - 99.12%Color and Shape:SolidMolecular weight:470.51Ref: TM-T6889
1mg44.00€5mg93.00€10mg140.00€25mg264.00€50mg447.00€100mg692.00€200mg964.00€1mL*10mM (DMSO)92.00€Nandrolone phenylpropionate
CAS:Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosisFormula:C27H34O3Purity:99.2% - 99.46%Color and Shape:White Or Milky Crystalline PowderMolecular weight:406.56YK11
CAS:YK11 is an androgen receptor partial agonist that activates androgen receptor transcriptional activity in HEK293 cells overexpressing androgen receptors when used at a concentration of 0.1 μM, with osteogenic activity.Formula:C25H34O6Purity:98.91%Color and Shape:SoildMolecular weight:430.53Androgen receptor-IN-4
CAS:3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.Formula:C18H14N4OPurity:98.41%Color and Shape:SolidMolecular weight:302.332-hydroxy Flutamide
CAS:2-hydroxy Flutamide is competitive inhibition of androgen receptor (AR) for the treatment of prostate cancerFormula:C11H11F3N2O4Purity:99.45% - 99.82%Color and Shape:SolidMolecular weight:292.21Testosterone undecanoate
CAS:Testosterone undecanoate is a metabolite of Testosterone, which is a promising androgen for male hormonal contraception.Formula:C30H48O3Purity:99.45% - 99.788%Color and Shape:White Crystalline PowderMolecular weight:456.7Apalutamide
CAS:Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.Formula:C21H15F4N5O2SPurity:99.03% - 99.91%Color and Shape:SolidMolecular weight:477.43AH-3960
CAS:AH-3960 是一种甲状腺激素受体 1 (PTHR1) 激动剂。Formula:C13H22N4O3Purity:98.44%Color and Shape:SolidMolecular weight:282.34VPC-13163
CAS:VPC-13566 inhibits growth in LNCaP, Enzalutamide-resistant MR49F, lowers AR gene, PSA, TMPRSS2 expression, but not in AR-independent PC3 cells.Formula:C16H14N2Purity:98.02%Color and Shape:SolidMolecular weight:234.3Ref: TM-T29110
1mg85.00€2mg111.00€5mg177.00€10mg269.00€25mg429.00€50mg610.00€100mg820.00€200mg1,071.00€1mL*10mM (DMSO)165.00€S-23
CAS:S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) is an oral selective androgen receptor modulator (Formula:C18H13ClF4N2O3Purity:99.55%Color and Shape:SolidMolecular weight:416.75Iprodione
CAS:Iprodione is a fungicide. Iprodione is also used in cannabis testing kits as a component of pesticide mixes.Formula:C13H13Cl2N3O3Purity:98.82%Color and Shape:Colorless Crystals Cream To Colorless Odorless PowderMolecular weight:330.17Bavdegalutamide
CAS:Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR).Formula:C41H43ClFN9O6Purity:97.17% - 99.04%Color and Shape:SolidMolecular weight:812.29N-desmethyl Enzalutamide
CAS:N-desmethyl Enzalutamide (N-desmethyl MDV 3100) is the active Enzalutamide metabolite.It is the active metabolite of Enzalutamide.Formula:C20H14F4N4O2SPurity:99.74%Color and Shape:SolidMolecular weight:450.41Ref: TM-T19450
2mg33.00€5mg50.00€10mg71.00€25mg131.00€50mg243.00€100mg355.00€200mg504.00€1mL*10mM (DMSO)55.00€Enzalutamide carboxylic acid
CAS:Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .Formula:C20H13F4N3O3SPurity:97.88%Color and Shape:SolidMolecular weight:451.39Ref: TM-T8217
1mg63.00€2mg88.00€5mg119.00€10mg177.00€25mg299.00€50mg416.00€100mg615.00€1mL*10mM (DMSO)133.00€Lupeol
CAS:Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.Formula:C30H50OPurity:98% - 99.96%Color and Shape:Needles From Alcohol Acetone White PowderMolecular weight:426.72VPC-13566
CAS:VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the
Formula:C18H14N2Purity:99.55%Color and Shape:SolidMolecular weight:258.32Galeterone
CAS:Galeterone (VN 124) is an oral androgen receptor modulator/CYP17 inhibitor with antiandrogen properties, targeting prostate cancer growth.Formula:C26H32N2OPurity:99.47% - 99.773%Color and Shape:SolidMolecular weight:388.55CLP-3094
CAS:CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor.Formula:C15H13ClN2OSPurity:99.84%Color and Shape:SolidMolecular weight:304.79JNJ-63576253 free base
CAS:JNJ-63576253 free base (TRC253) is a potent and orally active full antagonist of androgen receptor (AR). JNJ-63576253 can be used for the research of CRPC.Formula:C23H21F3N6O2SPurity:98.32%Color and Shape:SolidMolecular weight:502.51Ref: TM-T8933
2mg38.00€5mg50.00€10mg85.00€25mg159.00€50mg244.00€100mg359.00€200mg512.00€1mL*10mM (DMSO)86.00€CTK8A3536
CAS:CTK8A3536 ((2-MORPHOLIN-4-YL-4-PHENYL-1,3-THIAZOL-5-YL)METHANOL) is an inhibitor of Androgen receptor.Formula:C14H16N2O2SPurity:99.62%Color and Shape:SolidMolecular weight:276.35Ref: TM-T8592
1mg88.00€5mg170.00€10mg259.00€25mg425.00€50mg598.00€100mg810.00€200mg1,074.00€1mL*10mM (DMSO)169.00€Ailanthone
CAS:Ailanthone (Δ13-Dehydrochaparrinone) is an effective inhibitor of both full-length androgen receptor (AR) (IC50: 69 nM) and constitutively active truncated ARFormula:C20H24O7Purity:99.71% - 99.96%Color and Shape:SolidMolecular weight:376.4ARD-2128
CAS:ARD-2128: potent oral PROTAC that degrades AR, curbing prostate cancer growth with no toxicity.Formula:C45H50ClN7O6Purity:98.8%Color and Shape:SolidMolecular weight:820.37Boldenone Undecylenate
CAS:Boldenone Undecylenate (Parenabol) is a synthetic steroid.Formula:C30H44O3Purity:99.39%Color and Shape:Light Yellow Oily MatterMolecular weight:452.67Ref: TM-T3137
1mg35.00€2mg48.00€5mg52.00€10mg85.00€25mg140.00€50mg246.00€100mg396.00€500mg939.00€1mL*10mM (DMSO)52.00€Triptophenolide
CAS:Triptophenolide (Hypolide) is a compound isolated from Tripterygium wilfordii Hook with anti-inflammatory activity.Formula:C20H24O3Purity:98.07% - ≥95%Color and Shape:White PowderMolecular weight:312.40AC-262536
CAS:AC-262536 is a selective androgen receptor (SAR) modulator and exhibits potent agonist activity at the androgen receptor.Formula:C18H18N2OPurity:99.88%Color and Shape:SolidMolecular weight:278.35Ref: TM-T26539
5mg46.00€10mg74.00€25mg145.00€50mg240.00€100mg359.00€200mg510.00€1mL*10mM (DMSO)49.00€Enzalutamide
CAS:Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist (IC50=36 nM in LNCaP).Formula:C21H16F4N4O2SPurity:99% - 99.93%Color and Shape:SolidMolecular weight:464.44Ref: TM-T6002
5mg48.00€10mg56.00€25mg74.00€50mg96.00€100mg154.00€200mg187.00€500mg274.00€1mL*10mM (DMSO)52.00€RU 58841
CAS:RU 58841 (PSK-3841) is a specific androgen receptor antagonist or anti-androgen; RU 58841(PSK-3841) has a significant effect on hair regrowth.Formula:C17H18F3N3O3Purity:99.31% - 99.70%Color and Shape:SolidMolecular weight:369.34Ref: TM-T2236
5mg40.00€10mg63.00€25mg99.00€50mg130.00€100mg177.00€200mg245.00€500mg371.00€1mL*10mM (DMSO)48.00€EPI-001
CAS:EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ～6 μM and a selective PPAR-gamma modulator.Formula:C21H27ClO5Purity:99% - 99.67%Color and Shape:SolidMolecular weight:394.89Ref: TM-T6829
2mg34.00€5mg48.00€10mg73.00€25mg120.00€50mg192.00€100mg286.00€200mg425.00€1mL*10mM (DMSO)49.00€Clascoterone
CAS:Clascoterone (CB-03-01) is a new topical and peripherally selective androgen antagonist.Formula:C24H34O5Purity:99.2% - 99.72%Color and Shape:SolidMolecular weight:402.52DSRM-3716
CAS:Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery ofFormula:C9H6INPurity:97.28% - 99.785%Color and Shape:SolidMolecular weight:255.06p,p'-DDE
CAS:p,p'-DDE (p,p'-dichlorodiphenyldichloroethylene) is a metabolite and degradation product of the organochlorine pesticide DDTFormula:C14H8Cl4Purity:99.68%Color and Shape:White Crystalline Solid Physical Description White Crystalline Solid Or White Powder (Ntp 1992)Molecular weight:318.03CSRM617 hydrochloride
CAS:CSRM617 hydrochloride: selective OC2 inhibitor, Kd 7.43 uM, binds OC2-HOX, induces apoptosis, tolerable in mouse prostate cancer.Formula:C10H14ClN3O5Purity:99.59%Color and Shape:SoildMolecular weight:291.69LY2452473
CAS:LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer activity for the study of prostate cancer.Formula:C22H22N4O2Purity:99.72%Color and Shape:SolidMolecular weight:374.44Ref: TM-T15804
1mg34.00€5mg67.00€10mg96.00€25mg133.00€50mg170.00€100mg253.00€200mg386.00€1mL*10mM (DMSO)73.00€Masofaniten
CAS:Masofaniten (EPI-7386) is an orally active androgen receptor (AR) inhibitor with antitumor activity for the study of prostate and breast cancer.Formula:C24H24Cl2N4O4SPurity:98.42% - 98.66%Color and Shape:SolidMolecular weight:535.44Estromustine
CAS:Estromustine, an active metabolite of estramustine phosphate, is used to treat prostate cancer.Formula:C23H29Cl2NO3Color and Shape:SolidMolecular weight:438.39GDC-2992
CAS:GDC-2992 is a selective androgen receptor (AR) degradator that degrades AR and inhibits proliferation in VCaP cells,CRPC.Formula:C45H51ClN8O5Purity:99.82%Color and Shape:SoildMolecular weight:819.39AR antagonist 6
CAS:AR antagonist 6 (compound 6i), a diphenyl ether androgen receptor (AR) antagonist, binds to the AR with an affinity of 120 nM. It demonstrates low toxicity and effective in vitro activity in the golden Syrian hamster ear model. [19] [1]Formula:C16H12F3NO2Color and Shape:SolidMolecular weight:307.27Procymidone
CAS:Procymidone is a broad-spectrum fungicide that inhibits fungal glycerol triester synthesis, thereby disrupting hyphal growth. androgen receptor (AR) antagonistFormula:C13H11Cl2NO2Purity:99.86%Color and Shape:Colorless SolidMolecular weight:284.14JNJ-37654032
CAS:JNJ-37654032: orally active, nonsteroidal SARM. Mixed AR agonist/antagonist. Selective for muscle, grows levator ani, max at 3mg/kg, ED(50) 0.8mg/kg.Formula:C11H7Cl2F3N2OColor and Shape:SolidMolecular weight:311.09Androgen receptor antagonist 4
CAS:Compound AT2 is an AR inhibitor with anticancer effects, blocking DHT action and AR nuclear translocation (IC50=0.15μM).Formula:C22H18ClNColor and Shape:SolidMolecular weight:331.84Chlormadinone (free base)
CAS:Chlormadinone: synthetic hormone, treats BPH and PCOS, blocks androgen/estrogen, boosts bone cell growth.Formula:C21H27ClO3Color and Shape:SolidMolecular weight:362.89Bifluranol
CAS:Bifluranol (BX341) has anti-androgenic activity and has shown significant anti-prostatic activity in in vivo studies for the treatment of benign prostaticFormula:C17H18F2O2Purity:99.86%Color and Shape:SolidMolecular weight:292.32Gumelutamide
CAS:Gumelutamide, a tetrahydropyridopyrimidine compound, functions as both an antiandrogen and an antineoplastic agent by acting as an androgen antagonist.Formula:C22H21ClN6OColor and Shape:SolidMolecular weight:420.89AZD3514
CAS:AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM and has ability of reducing AR protein expression.Phase 1.
Formula:C25H32F3N7O2Purity:98.09%Color and Shape:SolidMolecular weight:519.56Honokiol DCA
CAS:Honokiol DCA inhibits DRP1, enhances respiration via mitochondrial repair, and is active against Vemurafenib-resistant melanoma.Formula:C22H18Cl4O4Color and Shape:SolidMolecular weight:488.19Prochloraz
CAS:Prochloraz: broad-spectrum imidazole fungicide; blocks placental aromatase (IC50=40nM), estrogen/androgen receptors; activates aryl hydrocarbon receptors.Formula:C15H16Cl3N3O2Purity:99.75% - 99.79%Color and Shape:Colorless SolidMolecular weight:376.67
