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Androgen Receptor

Androgen Receptor

The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.

Found 207 products of "Androgen Receptor"

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  • LGD-2226
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    LGD-2226

    CAS:
    <p>LGD-2226: selective oral androgen receptor modulator, EC50: 0.2nM, Ki: 1.5nM. Treats muscle loss, osteoporosis, sexual issues.</p>
    Formula:C14H9F9N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.22

    Ref: TM-T15749

  • S-40503
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    S-40503

    CAS:
    <p>S-40503 is an investigational selective androgen receptor modulator (SARM).</p>
    Formula:C15H23N3O3
    Color and Shape:Solid
    Molecular weight:293.36

    Ref: TM-T28650

  • Cyprodinil
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    Cyprodinil

    CAS:
    <p>Cyprodinil is a fungicide blocking methionine synthesis in fungi and hinders B. cinerea, P. herpotrichoides, H. oryzae growth; it's also an AR agonist.</p>
    Formula:C14H15N3
    Color and Shape:Solid
    Molecular weight:225.29

    Ref: TM-T41331

  • BMS-641988
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    BMS-641988

    CAS:
    <p>BMS-641988 is a novel nonsteroidal androgen receptor antagonist for the treatment of prostate cancer.</p>
    Formula:C20H20F3N3O5S
    Purity:99.57% - 99.92%
    Color and Shape:Soild
    Molecular weight:471.45

    Ref: TM-T67818

  • GLPG0492
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    GLPG0492

    CAS:
    <p>GLPG0492 is a novel selective androgen receptor modulator.</p>
    Formula:C19H14F3N3O3
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:389.33

    Ref: TM-T11410L

  • ONC1-13B
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    ONC1-13B

    CAS:
    <p>ONC1-13B, an androgen receptor antagonist, is used potentially for the treatment of prostate cancer.</p>
    Formula:C22H16F4N4O3S
    Purity:99.36% - 99.85%
    Color and Shape:Solid
    Molecular weight:492.45

    Ref: TM-T28238

  • Ralaniten triacetate
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    Ralaniten triacetate

    CAS:
    <p>Ralaniten triacetate (EPI-506) is a precursor of Ralaniten, an AR-NTD inhibitor, which can be used in the study of prostate and breast cancer.</p>
    Formula:C27H33ClO8
    Purity:98.69%
    Color and Shape:Solid
    Molecular weight:521.00

    Ref: TM-T36375

  • Androgen receptor-IN-5
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    Androgen receptor-IN-5

    CAS:
    <p>Androgen receptor-IN-5 is a potent inhibitor of the androgen receptor with anticancer properties.</p>
    Formula:C22H10Cl2F4N4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:525.31

    Ref: TM-T79024

  • (rel)-BMS-641988
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    (rel)-BMS-641988

    CAS:
    <p>(rel)-BMS-641988, a relative configuration of the potent nonsteroidal androgen receptor antagonist BMS-641988, holds potential for prostate cancer research.</p>
    Formula:C20H20F3N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:471.45

    Ref: TM-T71670

  • LGD-2941
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    LGD-2941

    CAS:
    <p>LGD-2941 is an androgen receptor modulator. LGD-2941 is used for the treatment of hypogonadism, female sexual dysfunction and menopausal syndrome.</p>
    Formula:C17H16F6N2O2
    Color and Shape:Solid
    Molecular weight:394.31

    Ref: TM-T27826

  • Androgen receptor degrader-1
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    Androgen receptor degrader-1

    CAS:
    <p>Androgen Receptor Degrader-1 (Compound 18) is a potent agent for androgen receptor degradation, applicable in cancer research [1].</p>
    Formula:C15H14ClN3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:335.74

    Ref: TM-T80633

  • Androgen receptor degrader-2
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    Androgen receptor degrader-2

    CAS:
    <p>Androgen Receptor Degrader-2 (Compound 9) is a potent degrader of androgen receptors, with potential application in cancer research [1].</p>
    Formula:C16H16ClN3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:349.77

    Ref: TM-T80647

  • N-Nitrosodicyclohexylamine
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    N-Nitrosodicyclohexylamine

    CAS:
    <p>N-Nitrosodicyclohexylamine (NDCHA), an N-nitrosocompound, exhibits anti-androgenic activity by competitively binding to the androgen receptor (AR) in opposition</p>
    Formula:C12H22N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:210.32

    Ref: TM-T81662

  • Celiprolol hydrochloride
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    Celiprolol hydrochloride

    CAS:
    <p>Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.</p>
    Formula:C20H33N3O4·HCl
    Color and Shape:White Crystalline Solid
    Molecular weight:415.96

    Ref: TM-T1244

  • Androgen receptor antagonist 5
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    Androgen receptor antagonist 5

    CAS:
    <p>AR antagonist 5 blocks AR (IC50: 6.17 μM), hinders LNCaP cell growth, and has anti-tumor effects in mouse models.</p>
    Formula:C21H15F4N5O3S
    Color and Shape:Solid
    Molecular weight:493.43

    Ref: TM-T63324

  • Trimegestone
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    Trimegestone

    CAS:
    <p>Trimegestone, a highly effective oral progestogen, is used for endometrial protection, all doses inducing secretory endometrial transformation.</p>
    Formula:C22H30O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:342.47

    Ref: TM-T20755

  • JJH260
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    JJH260

    CAS:
    <p>JJH260, a N-hydroxy hydantoin carbamate, inhibits AIG1 and ADTRP with IC50 values of 0.57 μM and 8.5 μM, respectively, and targets ABHD6, LYPLA1/2.</p>
    Formula:C29H34ClN5O5
    Color and Shape:Solid
    Molecular weight:568.06

    Ref: TM-T38107

  • JNJ-26146900
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    JNJ-26146900

    CAS:
    <p>JNJ-26146900 is a nonsteroidal androgen receptor (AR) ligand with tissue-selective activity in rats. JNJ-26146900 binds to the rat AR with a K(i) of 400nM.</p>
    Formula:C15H15F3N2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:360.35

    Ref: TM-T27671

  • VPC-14228
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    VPC-14228

    CAS:
    <p>VPC-14228 is a specific AR-DBD inhibitor that acts by inhibiting both Y594A and Q592A mutants.</p>
    Formula:C13H14N2OS
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:246.33

    Ref: TM-T24943

  • PLK1/BRD4-IN-1
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    PLK1/BRD4-IN-1

    CAS:
    <p>PLK1/BRD4-IN-1 (9b) is an orally active dual inhibitor of PLK1 (IC50: 22 nM) and BRD4 (IC50: 109 nM).</p>
    Formula:C31H43N9O2
    Color and Shape:Solid
    Molecular weight:573.73

    Ref: TM-T64058