Androgen Receptor
The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.
Found 229 products of "Androgen Receptor"
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VPC-14449
CAS:VPC-14449 is a selective androgen receptor DNA-binding domain (AR-DBD) inhibitor, useful in prostate cancer research.Formula:C10H10Br2N4OSPurity:99.56%Color and Shape:SolidMolecular weight:394.09BMS-564929
CAS:BMS-564929 is an AR agonist that upregulates the expression and activity of fat-producing enzymes, reducing VAT content and lipid levels.Formula:C14H12ClN3O3Purity:98.17%Color and Shape:SolidMolecular weight:305.72VPC-13789
CAS:VPC-13789: potent, selective oral antiandrogen for CRPC with 0.19 μM IC50 in LNCaP cells.Formula:C21H16F3N3OColor and Shape:SolidMolecular weight:383.37Androgen receptor antagonist 3
CAS:Androgen receptor antagonist 3 (Compound C18) has anticancer activities that is an antagonist of androgen receptor (AR) (IC 50 = 2.4 μM) [1].Formula:C22H18ClNColor and Shape:SolidMolecular weight:331.84(R)-UT-155
CAS:(R)-UT-155 is a selective androgen receptor degrader (SARD) ligand.Formula:C20H15F4N3O2Color and Shape:SolidMolecular weight:405.35Lubabegron fumarate
CAS:Lubabegron (LY591281, LY488756 fumarate) is a beta-agonist approved in 2018 to lower ammonia in cattle waste, aiding environment and health.Formula:C29H29N3O3SC4H4O4Color and Shape:SolidMolecular weight:557.66MK-4541
CAS:MK-4541: oral, selective AR modulator, blocks 5α-reductase, curbs AR+ prostate cancer growth, effective in mouse model.Formula:C22H31F3N2O3Color and Shape:SolidMolecular weight:428.49HG122
CAS:HG122 promotes AR degradation via proteasome, inhibiting castration-resistant prostate cancer.Formula:C15H13N5O5Color and Shape:SolidMolecular weight:343.29LGD-2226
CAS:LGD-2226: selective oral androgen receptor modulator, EC50: 0.2nM, Ki: 1.5nM. Treats muscle loss, osteoporosis, sexual issues.Formula:C14H9F9N2OPurity:98%Color and Shape:SolidMolecular weight:392.22Dimethomorph
CAS:Dimethomorph is a fungicide and sterol biosynthesis inhibitor that inhibits fungal cell wall formation,. inhibits androgen receptor (AR) .Formula:C21H22ClNO4Purity:99.20%Color and Shape:Solid CrystallineMolecular weight:387.86CSRM617
CAS:CSRM617: selective ONECUT2 inhibitor, Kd 7.43 uM, binds OC2-HOX, induces apoptosis, tolerable in mouse prostate cancer model.Formula:C10H13N3O5Purity:98%Color and Shape:SolidMolecular weight:255.23MK-3984
CAS:MK-3984 is a selective androgen receptor modulator, used in the study of conditions caused by androgen deficiency.Formula:C17H12F7NO2Purity:99.91%Color and Shape:SolidMolecular weight:395.27TFM-4AS-1
CAS:androgen receptor modulatorFormula:C27H33F3N2O2Purity:98%Color and Shape:SolidMolecular weight:474.56VPC-3033
CAS:VPC-3033 is an antagonist of the androgen receptor. It acts by inhibiting the LNCaP cell line as well as cell lines with the wild-type androgen receptor.Formula:C21H14O2Purity:98%Color and Shape:SolidMolecular weight:298.33Topterone
CAS:Topterone (Win 17,665) is a potent topical antiandrogen that inhibits the stimulation of lumbar organ development by testosterone and dihydrotestosterone inFormula:C22H34O2Purity:>99.99%Color and Shape:SolidMolecular weight:330.5Ar-V7-IN-1
CAS:Ar-V7-IN-1 (compound 47) is a potent inhibitor of Ar-V7,associated with resistance to AR-targeted therapy with desmoplasia-resistant prostate cancer (mCRPC).Formula:C10H10Br2N4OSColor and Shape:SolidMolecular weight:394.09Carbazole derivative 1
CAS:Carbazole derivative 1 is used to reduce androgen or oestrogen levels in mammals.Formula:C18H13FN2Purity:98%Color and Shape:SolidMolecular weight:276.31Seviteronel
CAS:Seviteronel (VT-464) is a novel CYP17 cleavage enzyme inhibitor and androgen receptor antagonist for the study of breast and prostate cancer.Formula:C18H17F4N3O3Purity:99.67% - 99.98%Color and Shape:SolidMolecular weight:399.34BMS-641988
CAS:BMS-641988 is a novel nonsteroidal androgen receptor antagonist for the treatment of prostate cancer.Formula:C20H20F3N3O5SPurity:99.3% - 99.92%Color and Shape:SoildMolecular weight:471.45Rosolutamide
CAS:Rosolutamide (ALZ-003) is a curcumin analog, an Nrf1 and Nrf2 activator.Formula:C28H32O6Purity:95.48% - 99.15%Color and Shape:SolidMolecular weight:464.55
