Androgen Receptor
The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.
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Darolutamide
CAS:1297538-32-9
Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 …
Formula:
C19H19ClN6O2
Purity:
99.14% - 99.62%
Color and Shape:
Solid
Molecular weight:
398.85
Ref: TM-T6915
| 1mg | 49.00 € | ||
| 2mg | 69.00 € | ||
| 5mg | 103.00 € | ||
| 10mg | 163.00 € | ||
| 25mg | 260.00 € | ||
| 50mg | 370.00 € | ||
| 100mg | 550.00 € | ||
| 500mg | 1,188.00 € | ||
| 1mL*10mM (DMSO) | 106.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Dimethylcurcumin
CAS:52328-98-0
Dimethylcurcumin (ASC-J9) (ASC-J9) is an androgen receptor degradation enhancer.
Formula:
C23H24O6
Purity:
95.77% - 98.96%
Color and Shape:
Solid
Molecular weight:
396.43
Ref: TM-TQ0214
| 20mg | 126.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Testosterone acetate
CAS:1045-69-8
Testosterone acetate (NSC-523836) is a hormone with in vitro antitumor activity.
Formula:
C21H30O3
Purity:
99.60%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
330.46
Ref: TM-TC0025
| 20mg | 54.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
GSK-2881078
CAS:1539314-06-1
GSK-2881078 is a selective androgen receptor modulato (SARM) that is being evaluated for effects on …
Formula:
C14H13F3N2O2S
Purity:
98.16% - 99.33%
Color and Shape:
Solid
Molecular weight:
330.33
Ref: TM-T3618
| 5mg | 44.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 123.00 € | ||
| 50mg | 193.00 € | ||
| 100mg | 321.00 € | ||
| 200mg | 459.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
MI-136
CAS:1628316-74-4
MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.
Formula:
C23H21F3N6S
Purity:
97.08% - 98.63%
Color and Shape:
Solid
Molecular weight:
470.51
Ref: TM-T6889
| 1mg | 46.00 € | ||
| 2mg | 62.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 145.00 € | ||
| 25mg | 274.00 € | ||
| 50mg | 494.00 € | ||
| 100mg | 716.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
CTK8A3536
CAS:926228-58-2
CTK8A3536 ((2-MORPHOLIN-4-YL-4-PHENYL-1,3-THIAZOL-5-YL)METHANOL) is an inhibitor of Androgen receptor.
Formula:
C14H16N2O2S
Purity:
99.62%
Color and Shape:
Solid
Molecular weight:
276.35
Ref: TM-T8592
| 1mg | 85.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € | ||
| 1mL*10mM (DMSO) | 163.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
YK11
CAS:1370003-76-1
YK11 is an androgen receptor partial agonist that activates androgen receptor transcriptional activity in HEK293 …
Formula:
C25H34O6
Purity:
98.91%
Color and Shape:
Soild
Molecular weight:
430.53
Ref: TM-T7358
| 1ml | 96.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
![3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile](https://static.cymitquimica.com/products/TM/thumb/T9752.jpg)
3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
CAS:2759137-87-4
3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.
Formula:
C18H14N4O
Purity:
98.15%
Color and Shape:
Solid
Molecular weight:
302.33
Ref: TM-T9752
| 1mg | 94.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 272.00 € | ||
| 25mg | 434.00 € | ||
| 50mg | 617.00 € | ||
| 100mg | 830.00 € | ||
| 1mL*10mM (DMSO) | 180.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
2-hydroxy Flutamide
CAS:52806-53-8
2-hydroxy Flutamide is competitive inhibition of androgen receptor (AR) for the treatment of prostate cancer
Formula:
C11H11F3N2O4
Purity:
98.53% - 99.45%
Color and Shape:
Solid
Molecular weight:
292.21
Ref: TM-T7690
| 5mg | 51.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 149.00 € | ||
| 50mg | 222.00 € | ||
| 100mg | 347.00 € | ||
| 200mg | 510.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Testosterone undecanoate
CAS:5949-44-0
Testosterone undecanoate is a metabolite of Testosterone, which is a promising androgen for male hormonal …
Formula:
C30H48O3
Purity:
99.45%
Color and Shape:
White Crystalline Powder
Molecular weight:
456.7
Ref: TM-T9035
| 1g | 87.00 € | ||
| 200mg | 41.00 € | ||
| 500mg | 60.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Apalutamide
CAS:956104-40-8
Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.
Formula:
C21H15F4N5O2S
Purity:
99.03% - 99.97%
Color and Shape:
Solid
Molecular weight:
477.43
Ref: TM-T2339
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 121.00 € | ||
| 25mg | 248.00 € | ||
| 50mg | 351.00 € | ||
| 100mg | 552.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
S-23
CAS:1010396-29-8
S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) is an oral selective androgen receptor modulator (
Formula:
C18H13ClF4N2O3
Purity:
98.55%
Color and Shape:
Solid
Molecular weight:
416.75
Ref: TM-T20789
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 123.00 € | ||
| 50mg | 183.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Bavdegalutamide
CAS:2222112-77-6
Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR).
Formula:
C41H43ClFN9O6
Purity:
97.17% - 99.04%
Color and Shape:
Solid
Molecular weight:
812.29
Ref: TM-T22263
| 2mg | 92.00 € | ||
| 5mg | 135.00 € | ||
| 10mg | 202.00 € | ||
| 25mg | 396.00 € | ||
| 50mg | 507.00 € | ||
| 100mg | 730.00 € | ||
| 200mg | 1,012.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
N-desmethyl Enzalutamide
CAS:1242137-16-1
N-desmethyl Enzalutamide (N-desmethyl MDV 3100) is the active Enzalutamide metabolite.It is the active metabolite of …
Formula:
C20H14F4N4O2S
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
450.41
Ref: TM-T19450
| 2mg | 34.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 133.00 € | ||
| 50mg | 247.00 € | ||
| 100mg | 362.00 € | ||
| 200mg | 512.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Enzalutamide carboxylic acid
CAS:1242137-15-0
Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .
Formula:
C20H13F4N3O3S
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
451.39
Ref: TM-T8217
| 1mg | 65.00 € | ||
| 2mg | 92.00 € | ||
| 5mg | 123.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 310.00 € | ||
| 50mg | 433.00 € | ||
| 100mg | 634.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Lupeol
CAS:545-47-1
Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.
Formula:
C30H50O
Purity:
98% - 99.31%
Color and Shape:
Needles From Alcohol Acetone White Powder
Molecular weight:
426.72
Ref: TM-T2895
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 72.00 € | ||
| 50mg | 113.00 € | ||
| 100mg | 183.00 € | ||
| 500mg | 454.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
VPC-13566
CAS:218464-59-6
VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and …
Formula:
C18H14N2
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
258.32
Ref: TM-T29111
| 1mg | 48.00 € | ||
| 2mg | 65.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 159.00 € | ||
| 25mg | 328.00 € | ||
| 50mg | 537.00 € | ||
| 100mg | 841.00 € | ||
| 500mg | 1,716.00 € | ||
| 1mL*10mM (DMSO) | 114.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Nandrolone decanoate
CAS:360-70-3
Nandrolone decanoate is an anabolic steroid similar to testosterone, stimulating muscle, bone growth, and red …
Formula:
C28H44O3
Purity:
98.43% - 99.03%
Color and Shape:
Solid
Molecular weight:
428.65
Ref: TM-T2556
| 25mg | 45.00 € | ||
| 50mg | 54.00 € | ||
| 100mg | 78.00 € | ||
| 200mg | 127.00 € | ||
| 500mg | 207.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
CLP-3094
CAS:312749-73-8
CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor.
Formula:
C15H13ClN2OS
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
304.79
Ref: TM-T9179
| 1mg | 53.00 € | ||
| 5mg | 114.00 € | ||
| 10mg | 188.00 € | ||
| 25mg | 331.00 € | ||
| 50mg | 496.00 € | ||
| 100mg | 705.00 € | ||
| 200mg | 572.00 € | ||
| 500mg | 1,385.00 € | ||
| 1mL*10mM (DMSO) | 125.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
JNJ-63576253 free base
CAS:2110426-27-0
JNJ-63576253 free base (TRC253) is a potent and orally active full antagonist of androgen receptor …
Formula:
C23H21F3N6O2S
Purity:
98.32%
Color and Shape:
Solid
Molecular weight:
502.51
Ref: TM-T8933
| 2mg | 39.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 161.00 € | ||
| 50mg | 248.00 € | ||
| 100mg | 365.00 € | ||
| 200mg | 520.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
