Androgen Receptor
The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.
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JNJ-63576253
CAS:2110428-64-1
JNJ-63576253 is a Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate …
Formula:
C23H22ClF3N6O2S
Purity:
99.27%
Color and Shape:
Solid
Molecular weight:
538.97
Ref: TM-T9246
| 2mg | 46.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 547.00 € | ||
| 1mL*10mM (DMSO) | 83.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Ailanthone
CAS:981-15-7
Ailanthone (Δ13-Dehydrochaparrinone) is an effective inhibitor of both full-length androgen receptor (AR) (IC50: 69 nM) …
Formula:
C20H24O7
Purity:
99.71% - 99.78%
Color and Shape:
Solid
Molecular weight:
376.4
Ref: TM-TQ0209
| 1mg | 42.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
ARD-2128
CAS:2222111-87-5
ARD-2128: potent oral PROTAC that degrades AR, curbing prostate cancer growth with no toxicity.
Formula:
C45H50ClN7O6
Purity:
98.80%
Color and Shape:
Solid
Molecular weight:
820.37
Ref: TM-T39695
| 1mg | 213.00 € | ||
| 2mg | 319.00 € | ||
| 5mg | 540.00 € | ||
| 10mg | 777.00 € | ||
| 25mg | 1,180.00 € | ||
| 50mg | 1,570.00 € | ||
| 100mg | 2,133.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Boldenone Undecylenate
CAS:13103-34-9
Boldenone Undecylenate (Parenabol) is a synthetic steroid.
Formula:
C30H44O3
Purity:
99.39%
Color and Shape:
Light Yellow Oily Matter
Molecular weight:
452.67
Ref: TM-T3137
| 1mg | 35.00 € | ||
| 2mg | 47.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 138.00 € | ||
| 50mg | 241.00 € | ||
| 100mg | 388.00 € | ||
| 500mg | 918.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Triptophenolide
CAS:74285-86-2
Triptophenolide (Hypolide) is a compound isolated from Tripterygium wilfordii Hook with anti-inflammatory activity.
Formula:
C20H24O3
Purity:
98.07% - ≥95%
Color and Shape:
White Powder
Molecular weight:
312.4
Ref: TM-T3393
| 1mg | 35.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 132.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 270.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
AC-262536
CAS:870888-46-3
AC-262536 is a selective androgen receptor (SAR) modulator and exhibits potent agonist activity at the …
Formula:
C18H18N2O
Purity:
99.38%
Color and Shape:
Solid
Molecular weight:
278.35
Ref: TM-T26539
| 5mg | 44.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 232.00 € | ||
| 100mg | 346.00 € | ||
| 200mg | 492.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Enzalutamide
CAS:915087-33-1
Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist (IC50=36 nM in LNCaP).
Formula:
C21H16F4N4O2S
Purity:
100% - 99.67%
Color and Shape:
Solid
Molecular weight:
464.44
Ref: TM-T6002
| 5mg | 48.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 73.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 150.00 € | ||
| 200mg | 183.00 € | ||
| 500mg | 268.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
RU 58841
CAS:154992-24-2
RU 58841 (PSK-3841) is a specific androgen receptor antagonist or anti-androgen; RU 58841(PSK-3841) has a …
Formula:
C17H18F3N3O3
Purity:
99.31% - 99.77%
Color and Shape:
Solid
Molecular weight:
369.34
Ref: TM-T2236
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 106.00 € | ||
| 50mg | 141.00 € | ||
| 100mg | 197.00 € | ||
| 200mg | 170.00 € | ||
| 500mg | 480.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
EPI-001
CAS:227947-06-0
EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ～6 μM and a …
Formula:
C21H27ClO5
Purity:
99% - 99.28%
Color and Shape:
Solid
Molecular weight:
394.89
Ref: TM-T6829
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 75.00 € | ||
| 25mg | 125.00 € | ||
| 50mg | 199.00 € | ||
| 100mg | 296.00 € | ||
| 200mg | 440.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Clascoterone
CAS:19608-29-8
Clascoterone (CB-03-01) is a new topical and peripherally selective androgen antagonist.
Formula:
C24H34O5
Purity:
99.26% - 99.32%
Color and Shape:
Solid
Molecular weight:
402.52
Ref: TM-T3357
| 25mg | 50.00 € | ||
| 50mg | 62.00 € | ||
| 100mg | 88.00 € | ||
| 200mg | 130.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
DSRM-3716
CAS:58142-99-7
Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by …
Formula:
C9H6IN
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
255.06
Ref: TM-T8860
| 50mg | 49.00 € | ||
| 100mg | 78.00 € | ||
| 200mg | 94.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
p,p'-DDE
CAS:72-55-9
p,p'-DDE (p,p'-dichlorodiphenyldichloroethylene) is a metabolite and degradation product of the organochlorine pesticide DDT
Formula:
C14H8Cl4
Purity:
99.68%
Color and Shape:
White Crystalline Solid Physical Description White Crystalline Solid Or White Powder (Ntp 1992)
Molecular weight:
318.03
Ref: TM-T7440
| 100mg | 41.00 € | ||
| 500mg | 81.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
BMS-641988
CAS:1093276-09-5
BMS-641988 is a novel nonsteroidal androgen receptor antagonist for the treatment of prostate cancer.
Formula:
C20H20F3N3O5S
Purity:
100% - 100%
Color and Shape:
Soild
Molecular weight:
471.45
Ref: TM-T67818
| 1mg | 158.00 € | ||
| 5mg | 372.00 € | ||
| 10mg | 557.00 € | ||
| 25mg | 894.00 € | ||
| 50mg | 1,188.00 € | ||
| 100mg | 1,630.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
ONC1-13B
CAS:1351185-54-0
ONC1-13B, an androgen receptor antagonist, is used potentially for the treatment of prostate cancer.
Formula:
C22H16F4N4O3S
Purity:
99.45% - 99.85%
Color and Shape:
Solid
Molecular weight:
492.45
Ref: TM-T28238
| 1mg | 273.00 € | ||
| 5mg | 675.00 € | ||
| 10mg | 927.00 € | ||
| 25mg | 1,399.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,581.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
BMS-564929
CAS:627530-84-1
BMS-564929 is an agonist of androgen receptor (AR, Ki of 2.11±0.16 nM).
Formula:
C14H12ClN3O3
Color and Shape:
Solid
Molecular weight:
305.72
Ref: TM-T14675
| 50mg | 1,857.00 € | ||
| 100mg | 2,535.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
GLPG0492
CAS:1215085-92-9
GLPG0492 is a novel selective androgen receptor modulator.
Formula:
C19H14F3N3O3
Purity:
98.27%
Color and Shape:
Solid
Molecular weight:
389.33
Ref: TM-T11410L
| 1mg | 72.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 228.00 € | ||
| 25mg | 364.00 € | ||
| 50mg | 524.00 € | ||
| 100mg | 704.00 € | ||
| 200mg | 904.00 € | ||
| 1mL*10mM (DMSO) | 169.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Topterone
CAS:60607-35-4
Topterone (Win 17,665) is a potent topical antiandrogen that inhibits the stimulation of lumbar organ …
Formula:
C22H34O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
330.5
Ref: TM-T13187
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
Bifluranol
CAS:34633-34-6
Bifluranol (BX341) has anti-androgenic activity and has shown significant anti-prostatic activity in in vivo studies …
Formula:
C17H18F2O2
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
292.32
Ref: TM-T14843
| 1mg | 148.00 € | ||
| 5mg | 355.00 € | ||
| 10mg | 580.00 € | ||
| 25mg | 1,153.00 € | ||
| 50mg | 1,864.00 € | ||
| 100mg | 2,511.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
AZD3514
CAS:1240299-33-5
AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM and …
Formula:
C25H32F3N7O2
Purity:
96.6%
Color and Shape:
Solid
Molecular weight:
519.56
Ref: TM-T6400
| 5mg | 70.00 € | ||
| 1mL*10mM (DMSO) | 82.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
LGD-2226
CAS:328947-93-9
LGD-2226: selective oral androgen receptor modulator, EC50: 0.2nM, Ki: 1.5nM. Treats muscle loss, osteoporosis, sexual …
Formula:
C14H9F9N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
392.22
Ref: TM-T15749
| 25mg | 1,406.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Thursday 16 Jan 2025
